RU93005335A - ANTOGONISTS OF TACHYKININ RECEPTOR, ISOHINOLINE AND METHOD FOR THEIR RECOVERY - Google Patents

ANTOGONISTS OF TACHYKININ RECEPTOR, ISOHINOLINE AND METHOD FOR THEIR RECOVERY

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Publication number
RU93005335A
RU93005335A RU93005335/14A RU93005335A RU93005335A RU 93005335 A RU93005335 A RU 93005335A RU 93005335/14 A RU93005335/14 A RU 93005335/14A RU 93005335 A RU93005335 A RU 93005335A RU 93005335 A RU93005335 A RU 93005335A
Authority
RU
Russia
Prior art keywords
substituted
tachykinin receptor
isohinoline
antogonists
recovery
Prior art date
Application number
RU93005335/14A
Other languages
Russian (ru)
Inventor
Нацугари Хидеаки
Сирафудзи Хидео
Дои Такаюки
Original Assignee
Такеда Кемикал Индастриз, Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Такеда Кемикал Индастриз, Лтд. filed Critical Такеда Кемикал Индастриз, Лтд.
Publication of RU93005335A publication Critical patent/RU93005335A/en

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Claims (1)

Предложена новая композиция, представленная формулой, указанной в описании, где циклы А и В каждый представляет собой бензольные кольца, возможно имеющие заместители; R - атом водорода или алкильная группа, которая может быть замещена; R1 - атом водорода или алкильная группа, которая может быть замещена; R2 - углеводородная или гетероциклическая группа, каждая из которых может быть замещена, или R1 и R2, взятые вместе с атомом азота, к которому они присоединены, образуют цикл, который может быть замещен, или его фармацевтически приемлемую соль, которая является полезной в качестве антагониста рецептора тахикинина.A new composition is proposed, represented by the formula specified in the description, where cycles A and B each represent benzene rings, possibly having substituents; R is a hydrogen atom or an alkyl group which may be substituted; R 1 is a hydrogen atom or an alkyl group which may be substituted; R 2 is a hydrocarbon or heterocyclic group each of which may be substituted, or R 1 and R 2 taken together with the nitrogen atom to which they are attached form a cycle which may be substituted or its pharmaceutically acceptable salt which is useful as a tachykinin receptor antagonist.
RU93005335/14A 1993-04-15 1993-04-14 ANTOGONISTS OF TACHYKININ RECEPTOR, ISOHINOLINE AND METHOD FOR THEIR RECOVERY RU93005335A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP04-095291 1993-04-15

Publications (1)

Publication Number Publication Date
RU93005335A true RU93005335A (en) 1996-06-20

Family

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