RU92016232A - DERIVATIVES OF 13- (SUBSTITUTED TIO) -ACETOXYMILBEMICINE, METHOD FOR THEIR PRODUCTION AND AGRICULTURAL COMPOSITION - Google Patents
DERIVATIVES OF 13- (SUBSTITUTED TIO) -ACETOXYMILBEMICINE, METHOD FOR THEIR PRODUCTION AND AGRICULTURAL COMPOSITIONInfo
- Publication number
- RU92016232A RU92016232A RU92016232/04A RU92016232A RU92016232A RU 92016232 A RU92016232 A RU 92016232A RU 92016232/04 A RU92016232/04 A RU 92016232/04A RU 92016232 A RU92016232 A RU 92016232A RU 92016232 A RU92016232 A RU 92016232A
- Authority
- RU
- Russia
- Prior art keywords
- acetoxymilbemicine
- derivatives
- production
- agricultural composition
- substituted
- Prior art date
Links
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 2
- 125000000623 heterocyclic group Chemical group 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- 125000000217 alkyl group Chemical group 0.000 claims 1
- 230000000507 anthelmentic Effects 0.000 claims 1
- 125000006615 aromatic heterocyclic group Chemical group 0.000 claims 1
- 125000003710 aryl alkyl group Chemical group 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000004981 cycloalkylmethyl group Chemical group 0.000 claims 1
- 238000003898 horticulture Methods 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000004435 hydrogen atoms Chemical class [H]* 0.000 claims 1
- 239000002917 insecticide Substances 0.000 claims 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 239000011780 sodium chloride Substances 0.000 claims 1
- 125000004149 thio group Chemical group *S* 0.000 claims 1
Claims (1)
где R1 представляет метил, этил или изопропил; R2 - алкил, аралкил, циклоалкил, циклоалкилметил, арил, гетероциклическую группу или тио группу, замещенную гетероциклической группой; R3 представляет водород, метил или этил; или R2 вместе с R3 представляет -(CH2)n-, где n представляет 3, 4 или 5; А представляет ароматическую гетероциклическую группу; и их соли, которые являются ценными в сельском хозяйстве и садоводстве антигельминтными, аскарицидными и инсектицидными агентами.Describes compounds having the formula:
where R 1 represents methyl, ethyl or isopropyl; R 2 is alkyl, aralkyl, cycloalkyl, cycloalkylmethyl, aryl, a heterocyclic group or a thio group substituted by a heterocyclic group; R 3 represents hydrogen, methyl or ethyl; or R 2 together with R 3 is - (CH 2 ) n -, where n is 3, 4 or 5; A represents an aromatic heterocyclic group; and their salts, which are valuable in agriculture and horticulture anthelmintic, ascaricidal and insecticidal agents.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP3-334650 | 1991-12-18 | ||
| JP33465091 | 1991-12-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU92016232A true RU92016232A (en) | 1996-03-20 |
| RU2086552C1 RU2086552C1 (en) | 1997-08-10 |
Family
ID=18279733
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU92016232/04A RU2086552C1 (en) | 1991-12-18 | 1992-12-17 | Derivatives of 13-(substituted thio)acetoxymilbemycine, method for their production, insecticide composition and method for protection of plants |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US5276033A (en) |
| EP (1) | EP0549273B1 (en) |
| JP (1) | JP3087987B2 (en) |
| KR (1) | KR0171426B1 (en) |
| CN (1) | CN1039645C (en) |
| AT (1) | ATE163419T1 (en) |
| AU (1) | AU658037B2 (en) |
| CA (1) | CA2085703C (en) |
| DE (1) | DE69224508T2 (en) |
| DK (1) | DK0549273T3 (en) |
| EG (1) | EG19869A (en) |
| ES (1) | ES2114551T3 (en) |
| HK (1) | HK1007658A1 (en) |
| HU (1) | HU217303B (en) |
| IL (1) | IL104171A (en) |
| LV (1) | LV12132B (en) |
| MX (1) | MX9207464A (en) |
| NZ (1) | NZ245533A (en) |
| RU (1) | RU2086552C1 (en) |
| UA (1) | UA44886C2 (en) |
| ZA (1) | ZA929882B (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2554074C1 (en) * | 2014-04-18 | 2015-06-27 | Игорь Викторович Заварзин | Antiparasitic agent |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3767560D1 (en) * | 1986-03-25 | 1991-02-28 | Sankyo Co | MACROLIDE CONNECTIONS, THEIR PRODUCTION AND USE. |
| JP2622197B2 (en) * | 1990-03-01 | 1997-06-18 | 三共株式会社 | 13-ether substituted milbemycin derivative |
| US5614470A (en) * | 1994-04-01 | 1997-03-25 | Sankyo Company, Limited | 13-substituted milbemycin derivatives, their preparation and their use |
| NO317090B1 (en) * | 1995-09-29 | 2004-08-02 | 13-substituted milbemycin-5-oxime derivatives, anthelmistic, mite-killing and insecticidal preparations comprising such a compound, methods for protecting plants against parasite damage and using the compounds to prepare | |
| MXPA04003854A (en) * | 2001-10-25 | 2005-02-17 | Sankyo Lifetech Company Ltd | Anthelmintic composition. |
| EP1849363A1 (en) * | 2006-03-09 | 2007-10-31 | Cheminova A/S | Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3950360A (en) * | 1972-06-08 | 1976-04-13 | Sankyo Company Limited | Antibiotic substances |
| US4206205A (en) * | 1977-10-03 | 1980-06-03 | Merck & Co., Inc. | Monosaccharide and aglycone derivatives of C-076 |
| US4201861A (en) * | 1977-10-03 | 1980-05-06 | Merck & Co., Inc. | Acyl derivatives of C-076 compounds |
| US4171314A (en) * | 1977-12-19 | 1979-10-16 | Merck & Co., Inc. | 13-Halo and 13-deoxy C-076 compounds |
| US4173571A (en) * | 1977-12-19 | 1979-11-06 | Merck & Co., Inc. | 13-Halo and 13-deoxy derivatives of C-076 compounds |
| US4203976A (en) * | 1978-08-02 | 1980-05-20 | Merck & Co., Inc. | Sugar derivatives of C-076 compounds |
| JPS5632481A (en) * | 1979-08-23 | 1981-04-01 | Sankyo Co Ltd | Antibiotic b-41d, its preparation, and acaricide and anthelminthic agent and repellent containing the same as active constituent |
| US4289760A (en) * | 1980-05-02 | 1981-09-15 | Merck & Co., Inc. | 23-Keto derivatives of C-076 compounds |
| US4457920A (en) * | 1981-09-03 | 1984-07-03 | Merck & Co., Inc. | 4a-Substituted avermectin compounds |
| US4423209A (en) * | 1982-02-26 | 1983-12-27 | Merck & Co., Inc. | Processes for the interconversion of avermectin compounds |
| JPS59108785A (en) * | 1982-11-25 | 1984-06-23 | Sankyo Co Ltd | 5-oxime derivative of milbemycins |
| US4579864A (en) * | 1984-06-11 | 1986-04-01 | Merck & Co., Inc. | Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives |
| US4547491A (en) * | 1984-07-18 | 1985-10-15 | Merck & Co., Inc. | C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use |
| US4696922A (en) * | 1984-11-26 | 1987-09-29 | Ciba-Geigy Corporation | 5-azolylacetoxymilbemycins as ecto- and endoparasites |
| JPS6289685A (en) * | 1985-05-31 | 1987-04-24 | Sankyo Co Ltd | 13-halogenomilbemycin derivative |
| DE3767560D1 (en) * | 1986-03-25 | 1991-02-28 | Sankyo Co | MACROLIDE CONNECTIONS, THEIR PRODUCTION AND USE. |
| JPH0826026B2 (en) * | 1986-06-13 | 1996-03-13 | 三共株式会社 | 13-ester derivative of milbemycin and its use |
| JPH085894B2 (en) * | 1990-03-01 | 1996-01-24 | 三共株式会社 | Milbemycin ether derivative |
| JP2622197B2 (en) * | 1990-03-01 | 1997-06-18 | 三共株式会社 | 13-ether substituted milbemycin derivative |
-
1992
- 1992-12-17 US US07/992,865 patent/US5276033A/en not_active Expired - Fee Related
- 1992-12-17 RU RU92016232/04A patent/RU2086552C1/en not_active IP Right Cessation
- 1992-12-17 EG EG78792A patent/EG19869A/en active
- 1992-12-17 CA CA002085703A patent/CA2085703C/en not_active Expired - Fee Related
- 1992-12-17 KR KR1019920024697A patent/KR0171426B1/en not_active IP Right Cessation
- 1992-12-18 ZA ZA929882A patent/ZA929882B/en unknown
- 1992-12-18 IL IL10417192A patent/IL104171A/en not_active IP Right Cessation
- 1992-12-18 DK DK92311581T patent/DK0549273T3/en active
- 1992-12-18 CN CN92115349A patent/CN1039645C/en not_active Expired - Fee Related
- 1992-12-18 AU AU30312/92A patent/AU658037B2/en not_active Ceased
- 1992-12-18 DE DE69224508T patent/DE69224508T2/en not_active Expired - Fee Related
- 1992-12-18 ES ES92311581T patent/ES2114551T3/en not_active Expired - Lifetime
- 1992-12-18 EP EP92311581A patent/EP0549273B1/en not_active Expired - Lifetime
- 1992-12-18 JP JP04338308A patent/JP3087987B2/en not_active Expired - Fee Related
- 1992-12-18 NZ NZ245533A patent/NZ245533A/en unknown
- 1992-12-18 MX MX9207464A patent/MX9207464A/en unknown
- 1992-12-18 HU HU9204023A patent/HU217303B/en not_active IP Right Cessation
- 1992-12-18 AT AT92311581T patent/ATE163419T1/en not_active IP Right Cessation
-
1993
- 1993-06-18 UA UA93003130A patent/UA44886C2/en unknown
-
1998
- 1998-06-25 HK HK98106679A patent/HK1007658A1/en not_active IP Right Cessation
- 1998-07-02 LV LVP-98-140A patent/LV12132B/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2554074C1 (en) * | 2014-04-18 | 2015-06-27 | Игорь Викторович Заварзин | Antiparasitic agent |
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