RU2016143415A - RECOMBINANT PEPTIDE OF LONG-TERM ACTION, INHIBITING HIV FUSION WITH TARGET CELL - Google Patents

RECOMBINANT PEPTIDE OF LONG-TERM ACTION, INHIBITING HIV FUSION WITH TARGET CELL Download PDF

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Publication number
RU2016143415A
RU2016143415A RU2016143415A RU2016143415A RU2016143415A RU 2016143415 A RU2016143415 A RU 2016143415A RU 2016143415 A RU2016143415 A RU 2016143415A RU 2016143415 A RU2016143415 A RU 2016143415A RU 2016143415 A RU2016143415 A RU 2016143415A
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RU
Russia
Prior art keywords
recombinant peptide
target cell
long
inhibiting hiv
hiv fusion
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RU2016143415A
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Russian (ru)
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RU2016143415A3 (en
Inventor
Вагиф Али оглы Гасанов
Александр Федорович Шевалье
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Общество С Ограниченной Ответственностью "Биохарт"
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Priority to RU2016143415A priority Critical patent/RU2016143415A/en
Publication of RU2016143415A publication Critical patent/RU2016143415A/en
Publication of RU2016143415A3 publication Critical patent/RU2016143415A3/ru

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Claims (5)

1. Рекомбинантный пептид, ингибирующий слияние ВИЧ с клеткой-мишенью, характеризующийся тем, что имеет аминокислотную последовательность SEQ ID: 1: TTWMEWDREINNYTSLIHSLIEESQNQQEKNEQELLELAFLEKENALLRQEVVALRQELSHLRAVLSRYQASFTTFTVTKYWFYRLLSALFGIPMALIWGIYFAILSFLHIVA1. Recombinant peptide that inhibits the fusion of HIV with a target cell, characterized in that it has the amino acid sequence of SEQ ID: 1: TTWMEWDREINNYTSLIHSLIEESQNQQEKNEQELLELAFLEKENALLRQEVVALRQELSHLRAVLSRYQASFTTFTVTKALWFILFILFYFLF 2. Рекомбинантный пептид по п. 1, в котором в качестве участка, способствующего димеризации пептида, содержится любая аминокислотная последовательность, обладающая способностью образовывать димеры параллельных альфа-спиралей.2. The recombinant peptide according to claim 1, wherein any amino acid sequence containing the ability to form dimers of parallel alpha helices is contained as a region facilitating dimerization of the peptide. 3. Рекомбинантный пептид по п. 1, в котором в качестве последовательности, обеспечивающей сродство с холестерином на мембране клетки, выступает последовательность, содержащая холестерин-связывающий консенсусный мотив Leu/Val-X(1-5)-Tyr-X(1-5)-Arg/Lys3. The recombinant peptide according to claim 1, in which the sequence containing the cholesterol-binding consensus motif Leu / Val-X (1-5) -Tyr-X (1-5 ) -Arg / Lys 4. Штамм-продуцент Е. coli, экспрессирующий рекомбинантный пептид SEQ ID: 1.4. The producer strain E. coli expressing the recombinant peptide SEQ ID: 1. 5. Фармацевтическая композиция на основе пептида SEQ ID: 1 для подкожного, внутримышечного или ректального введения.5. Pharmaceutical composition based on the peptide SEQ ID: 1 for subcutaneous, intramuscular or rectal administration.
RU2016143415A 2016-11-03 2016-11-03 RECOMBINANT PEPTIDE OF LONG-TERM ACTION, INHIBITING HIV FUSION WITH TARGET CELL RU2016143415A (en)

Priority Applications (1)

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RU2016143415A RU2016143415A (en) 2016-11-03 2016-11-03 RECOMBINANT PEPTIDE OF LONG-TERM ACTION, INHIBITING HIV FUSION WITH TARGET CELL

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
RU2016143415A RU2016143415A (en) 2016-11-03 2016-11-03 RECOMBINANT PEPTIDE OF LONG-TERM ACTION, INHIBITING HIV FUSION WITH TARGET CELL

Publications (2)

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RU2016143415A true RU2016143415A (en) 2018-05-03
RU2016143415A3 RU2016143415A3 (en) 2019-06-06

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020139116A1 (en) * 2018-12-28 2020-07-02 Общество С Ограниченной Ответственностью "Биохарт" Recombinant inhibitor of hiv entry
RU2753191C2 (en) * 2019-09-26 2021-08-12 Федеральное государственное бюджетное учреждение науки Институт Биологии Развития им. Н.К. Кольцова Российской Академии Наук New recombinant growth hormone analogue with prolonged activity

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020139116A1 (en) * 2018-12-28 2020-07-02 Общество С Ограниченной Ответственностью "Биохарт" Recombinant inhibitor of hiv entry
RU2753191C2 (en) * 2019-09-26 2021-08-12 Федеральное государственное бюджетное учреждение науки Институт Биологии Развития им. Н.К. Кольцова Российской Академии Наук New recombinant growth hormone analogue with prolonged activity

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RU2016143415A3 (en) 2019-06-06

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