RU2007143336A - PHARMACEUTICAL COMPOSITION BASED ON A PEPTIDE NORMALIZING URINATION AND METHOD OF APPLICATION - Google Patents

PHARMACEUTICAL COMPOSITION BASED ON A PEPTIDE NORMALIZING URINATION AND METHOD OF APPLICATION Download PDF

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Publication number
RU2007143336A
RU2007143336A RU2007143336/15A RU2007143336A RU2007143336A RU 2007143336 A RU2007143336 A RU 2007143336A RU 2007143336/15 A RU2007143336/15 A RU 2007143336/15A RU 2007143336 A RU2007143336 A RU 2007143336A RU 2007143336 A RU2007143336 A RU 2007143336A
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Russia
Prior art keywords
glutamyl
glu
asp
seq
sequence
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RU2007143336/15A
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Russian (ru)
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RU2367467C2 (en
Inventor
Владимир Хацкелевич Хавинсон (RU)
Владимир Хацкелевич Хавинсон
Владимир Викторович Малинин (RU)
Владимир Викторович Малинин
Галина Анатольевна Рыжак (RU)
Галина Анатольевна Рыжак
Ленар Васильевич Козлов (RU)
Ленар Васильевич Козлов
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Закрытое акционерное общество "Эксесс Байосаинс" (RU)
Закрытое акционерное общество "Эксесс Байосаинс"
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Priority to RU2007143336/15A priority Critical patent/RU2367467C2/en
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Abstract

1. Фармацевтическая композиция, нормализующая мочеиспускание, характеризующаяся тем, что в качестве действующего вещества содержит эффективное количество пептида глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1] и фармацевтически приемлемый носитель. ! 2. Фармацевтическая композиция по п.1, отличающаяся тем, что находится в форме, подходящей для парентерального введения. ! 3. Пептид глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1]. ! 4. Пептид глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1], обладающий биологической активностью, проявляющейся в нормализации мочеиспускания путем регуляции функции детрузорно-сфинктерной системы мочевого пузыря. ! 5. Способ регуляции функции детрузорно-сфинктерной системы мочевого пузыря, заключающийся во введении пациенту фармацевтической композиции, содержащей в качестве действующего вещества эффективное количество пептида глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1] в дозе от 0,01 до 100 мкг/кг массы тела однократно ежедневно в течение 10 дней. ! 6. Способ по п.5, отличающийся тем, что введение осуществляют внутримышечно.1. A pharmaceutical composition that normalizes urination, characterized in that the active substance contains an effective amount of a glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1] and a pharmaceutically acceptable carrier. ! 2. The pharmaceutical composition according to claim 1, characterized in that it is in a form suitable for parenteral administration. ! 3. The glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1]. ! 4. The glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1], which has a biological activity that manifests itself in normalizing urination by regulating the function of the detrusor-sphincter system of the bladder. ! 5. A method for regulating the function of the detrusor-sphincter system of the bladder, which consists in administering to the patient a pharmaceutical composition containing, as active substance, an effective amount of a glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1] at a dose of 0.01 to 100 mcg / kg body weight once daily for 10 days. ! 6. The method according to claim 5, characterized in that the introduction is carried out intramuscularly.

Claims (6)

1. Фармацевтическая композиция, нормализующая мочеиспускание, характеризующаяся тем, что в качестве действующего вещества содержит эффективное количество пептида глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1] и фармацевтически приемлемый носитель.1. A pharmaceutical composition that normalizes urination, characterized in that the active substance contains an effective amount of a glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1] and a pharmaceutically acceptable carrier. 2. Фармацевтическая композиция по п.1, отличающаяся тем, что находится в форме, подходящей для парентерального введения.2. The pharmaceutical composition according to claim 1, characterized in that it is in a form suitable for parenteral administration. 3. Пептид глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1].3. The glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1]. 4. Пептид глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1], обладающий биологической активностью, проявляющейся в нормализации мочеиспускания путем регуляции функции детрузорно-сфинктерной системы мочевого пузыря.4. The glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1], which has a biological activity that manifests itself in normalizing urination by regulating the function of the detrusor-sphincter system of the bladder. 5. Способ регуляции функции детрузорно-сфинктерной системы мочевого пузыря, заключающийся во введении пациенту фармацевтической композиции, содержащей в качестве действующего вещества эффективное количество пептида глутамил-аспарагиновая кислота общей формулы: H-Glu-Asp-OH последовательности 1 [SEQ ID NO:1] в дозе от 0,01 до 100 мкг/кг массы тела однократно ежедневно в течение 10 дней.5. A method for regulating the function of the detrusor-sphincter system of the bladder, which consists in administering to the patient a pharmaceutical composition containing, as active substance, an effective amount of a glutamyl-aspartic acid peptide of the general formula: H-Glu-Asp-OH sequence 1 [SEQ ID NO: 1] at a dose of 0.01 to 100 mcg / kg body weight once daily for 10 days. 6. Способ по п.5, отличающийся тем, что введение осуществляют внутримышечно.6. The method according to claim 5, characterized in that the introduction is carried out intramuscularly.
RU2007143336/15A 2007-11-26 2007-11-26 Peptide pharmaceutical composition normalising urination, and method of application thereof RU2367467C2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
RU2007143336/15A RU2367467C2 (en) 2007-11-26 2007-11-26 Peptide pharmaceutical composition normalising urination, and method of application thereof

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Application Number Priority Date Filing Date Title
RU2007143336/15A RU2367467C2 (en) 2007-11-26 2007-11-26 Peptide pharmaceutical composition normalising urination, and method of application thereof

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RU2007143336A true RU2007143336A (en) 2009-06-10
RU2367467C2 RU2367467C2 (en) 2009-09-20

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