RU2002118334A - Pyrazolecarboxamide and pyrazolthioamide derivatives as fungicides - Google Patents

Pyrazolecarboxamide and pyrazolthioamide derivatives as fungicides

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Publication number
RU2002118334A
RU2002118334A RU2002118334/04A RU2002118334A RU2002118334A RU 2002118334 A RU2002118334 A RU 2002118334A RU 2002118334/04 A RU2002118334/04 A RU 2002118334/04A RU 2002118334 A RU2002118334 A RU 2002118334A RU 2002118334 A RU2002118334 A RU 2002118334A
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RU
Russia
Prior art keywords
formula
alkyl
compound
haloalkyl
denotes
Prior art date
Application number
RU2002118334/04A
Other languages
Russian (ru)
Other versions
RU2259356C2 (en
Inventor
Харальд Вальтер
Original Assignee
Зингента Партисипейшнс Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9929163.5A external-priority patent/GB9929163D0/en
Priority claimed from GBGB9929563.6A external-priority patent/GB9929563D0/en
Application filed by Зингента Партисипейшнс Аг filed Critical Зингента Партисипейшнс Аг
Publication of RU2002118334A publication Critical patent/RU2002118334A/en
Application granted granted Critical
Publication of RU2259356C2 publication Critical patent/RU2259356C2/en

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Claims (10)

1. Пиразолкарбоксамид формулы I1. Pyrazolecarboxamide of the formula I
Figure 00000001
Figure 00000001
 где X обозначает кислород или серу;where X is oxygen or sulfur; R1 обозначает C1-С3алкил, C1-С3галоалкил, С1-С3алкокси-С1-С3алкил или C1-С3галоалкокси-С1-С3алкил;R 1 is C 1 -C 3 alkyl, C 1 -C 3 haloalkyl, C 1 -C 3 alkoxy-C 1 -C 3 alkyl or C 1 -C 3 haloalkoxy-C 1 -C 3 alkyl; R2 обозначает C1-С3галоалкил;R 2 is C 1 -C 3 haloalkyl; R3 обозначает галоген, при условии, что если R1 обозначает СН3, R2 обозначает CF3 и Х обозначает кислород, то R3 обозначает бром или йод.R 3 is halogen, provided that if R 1 is CH 3 , R 2 is CF 3 and X is oxygen, then R 3 is bromine or iodine. 2. Соединение формулы I по п.1, в котором Х обозначает кислород.2. The compound of formula I according to claim 1, in which X is oxygen. 3. Соединение формулы I по п.1, в котором Х обозначает серу.3. The compound of formula I according to claim 1, in which X is sulfur. 4. Соединение по п.2 или 3, в котором R1 обозначает C1-С3алкил, и R3 обозначает фтор, хлор или бром.4. The compound according to claim 2 or 3, in which R 1 denotes C 1 -C 3 alkyl, and R 3 denotes fluorine, chlorine or bromine. 5. Соединение формулы I по п.4, в котором R2 обозначает CF3, CF2H, CFH2, CF2CF3, CCl3, CH2CF3, СН2CCl3 или CF2CF2CF3.5. The compound of formula I according to claim 4, in which R 2 is CF 3 , CF 2 H, CFH 2 , CF 2 CF 3 , CCl 3 , CH 2 CF 3 , CH 2 CCl 3 or CF 2 CF 2 CF 3 . 6. Соединение по п.2 или 3, в котором R1 обозначает C1-С3галоалкил, и R3 обозначает фтор, хлор или бром.6. The compound according to claim 2 or 3, in which R 1 denotes C 1 -C 3 haloalkyl, and R 3 denotes fluorine, chlorine or bromine. 7. Способ получения соединений формулы I, предусматривающий взаимодействие исходных продуктов согласно7. A method of obtaining compounds of formula I, involving the interaction of the starting products according to а) схемеa) scheme
Figure 00000002
Figure 00000002
 где X, R1, R2 и R3 имеют значения, указанные для формулы I в п.1; илиwhere X, R 1 , R 2 and R 3 have the meanings indicated for formula I in claim 1; or б) согласно схемеb) according to the scheme
Figure 00000003
Figure 00000003
 в) согласно схемеc) according to the scheme
Figure 00000004
Figure 00000004
 где R1, R2 и R3 имеют значения, указанные для формулы I в п.1, a R4 обозначает хлор, бром или йод.where R 1 , R 2 and R 3 have the meanings indicated for formula I in claim 1, and R 4 denotes chlorine, bromine or iodine. 8. Композиция для борьбы с микроорганизмами и предупреждения их нападения и поражения ими растений, в которой действующее вещество представляет собой соединение по п.1 в сочетании с приемлемым носителем.8. A composition for controlling microorganisms and preventing their attack and damage to plants, in which the active substance is a compound according to claim 1 in combination with an acceptable carrier. 9. Способ борьбы с фитопатогенными организмами или предупреждения поражения ими культурных растений путем нанесения соединения формулы I по п.1 на растения, их части или места их обитания.9. A method of controlling phytopathogenic organisms or preventing their defeat of cultivated plants by applying the compounds of formula I according to claim 1 on plants, their parts or their habitats. 10. Соединение формулы V10. The compound of formula V
Figure 00000005
Figure 00000005
 где X обозначает кислород или серу;where X is oxygen or sulfur; R1 обозначает C1-С3алкил, C1-С3галоалкил, С1-С3алкокси-С1-С3алкил или C1-С3галоалкокси-С1-С3алкил;R 1 is C 1 -C 3 alkyl, C 1 -C 3 haloalkyl, C 1 -C 3 alkoxy-C 1 -C 3 alkyl or C 1 -C 3 haloalkoxy-C 1 -C 3 alkyl; R2 обозначает C1-С3галоалкил;R 2 is C 1 -C 3 haloalkyl; R3 обозначает хлор, бром или йод.R 3 is chloro, bromo or iodo.
RU2002118334/04A 1999-12-09 2000-11-11 Pyrazolcarboxamide and pyrazolthioamide derivatives as fungicides RU2259356C2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9929163.5A GB9929163D0 (en) 1999-12-09 1999-12-09 Organic compounds
GB9929163.5 1999-12-09
GB9929563.6 1999-12-14
GBGB9929563.6A GB9929563D0 (en) 1999-12-14 1999-12-14 Organic compounds

Publications (2)

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RU2002118334A true RU2002118334A (en) 2003-12-20
RU2259356C2 RU2259356C2 (en) 2005-08-27

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EP (1) EP1235811B1 (en)
JP (1) JP2003516395A (en)
KR (1) KR20020058089A (en)
CN (1) CN1227235C (en)
AR (1) AR026915A1 (en)
AT (1) ATE296806T1 (en)
AU (1) AU771389B2 (en)
BR (1) BR0016203A (en)
CA (1) CA2382921A1 (en)
CZ (1) CZ20021890A3 (en)
DE (1) DE60020598T2 (en)
ES (1) ES2241676T3 (en)
HU (1) HUP0203624A3 (en)
IL (1) IL149191A0 (en)
MX (1) MXPA02004237A (en)
NZ (1) NZ518051A (en)
PL (1) PL354102A1 (en)
PT (1) PT1235811E (en)
RU (1) RU2259356C2 (en)
WO (1) WO2001042223A1 (en)

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