RU2002110295A - Factor Xa Inhibitors - Google Patents

Factor Xa Inhibitors Download PDF

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RU2002110295A
RU2002110295A RU2002110295/04A RU2002110295A RU2002110295A RU 2002110295 A RU2002110295 A RU 2002110295A RU 2002110295/04 A RU2002110295/04 A RU 2002110295/04A RU 2002110295 A RU2002110295 A RU 2002110295A RU 2002110295 A RU2002110295 A RU 2002110295A
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inhibitors
factor
text
formula
graphic part
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RU2002110295/04A
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Russian (ru)
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Бинг-Йан ЖУ (US)
Бинг-Йан ЖУ
Жаозхонг Джон ДЖИА (US)
Жаозхонг Джон ДЖИА
Венронг ХУАНГ (US)
Венронг ХУАНГ
Йонгхонг СОНГ (US)
Йонгхонг Сонг
Джеймс КЭНТЕР (US)
Джеймс КЭНТЕР
Роберт М. СКАРБОРУ (US)
Роберт М. Скарбору
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Милленниум Фармасьютикалс, Инк. (Us)
Милленниум Фармасьютикалс, Инк.
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Publication of RU2002110295A publication Critical patent/RU2002110295A/en

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    • C07—ORGANIC CHEMISTRY
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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Текст формулы в факсимильном виде (см. графическую часть)The text of the formula in facsimile form (see graphic part)
RU2002110295/04A 1999-09-17 2000-09-15 Factor Xa Inhibitors RU2002110295A (en)

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