RU2002102009A - Optically active amides of 1- (4-chlorobenzoyl) -5-methoxy-2-methylindole-3-acetic acid with derivatives of (S) amino acids - Google Patents

Optically active amides of 1- (4-chlorobenzoyl) -5-methoxy-2-methylindole-3-acetic acid with derivatives of (S) amino acids

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Publication number
RU2002102009A
RU2002102009A RU2002102009/04A RU2002102009A RU2002102009A RU 2002102009 A RU2002102009 A RU 2002102009A RU 2002102009/04 A RU2002102009/04 A RU 2002102009/04A RU 2002102009 A RU2002102009 A RU 2002102009A RU 2002102009 A RU2002102009 A RU 2002102009A
Authority
RU
Russia
Prior art keywords
amino acids
methylindole
chlorobenzoyl
methoxy
derivatives
Prior art date
Application number
RU2002102009/04A
Other languages
Russian (ru)
Inventor
Галина Львовна Левит
Виктор Павлович Краснов
Олег Николаевич Чупахин
Валерий Николаевич Чарушин
Татьяна Викторовна Матвеева
Александр Михайлович Дёмин
Марина Анатольевна Королёва
Валентин Абдулхаевич Сафин
Лада Владимировна Аникина
Юрий Борисович Вихарев
Александр Генрихович Толстиков
Original Assignee
Государственное учреждение Институт технической химии Уральского отделения РАН
Учреждение Институт органического синтеза Уральского отделения РАН
Filing date
Publication date
Application filed by Государственное учреждение Институт технической химии Уральского отделения РАН, Учреждение Институт органического синтеза Уральского отделения РАН filed Critical Государственное учреждение Институт технической химии Уральского отделения РАН
Publication of RU2002102009A publication Critical patent/RU2002102009A/en

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Claims (2)

1. Оптически активные амиды 1-(4-хлорбензоил)-5-метокси-2-метилиндол-3-уксусной кислоты с производными (S)-аминокислот общей формулы1. Optically active amides of 1- (4-chlorobenzoyl) -5-methoxy-2-methylindole-3-acetic acid with derivatives of (S) -amino acids of the general formula
Figure 00000001
Figure 00000001
 где R1 - остаток (S)-аминокислот: аланин, серин, метионин, фенилаланин, гистидин; γ-этиловый эфир глутаминовой кислоты;where R 1 is the residue of (S) -amino acids: alanine, serine, methionine, phenylalanine, histidine; glutamic acid γ-ethyl ester; R2 - метил или этил.R 2 is methyl or ethyl. 2. Индивидуальные стереоизомеры соединений по п.1, в качестве противовоспалительного средства.2. Individual stereoisomers of the compounds according to claim 1, as an anti-inflammatory agent.
RU2002102009/04A 2002-01-21 Optically active amides of 1- (4-chlorobenzoyl) -5-methoxy-2-methylindole-3-acetic acid with derivatives of (S) amino acids RU2002102009A (en)

Publications (1)

Publication Number Publication Date
RU2002102009A true RU2002102009A (en) 2003-08-27

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