PT90563A - Processo para a preparacao de 3-(n-meterociclil)-2,6-diaminopiridinas e de -n-oxidos substituidos e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de 3-(n-meterociclil)-2,6-diaminopiridinas e de -n-oxidos substituidos e de composicoes farmaceuticas que os contem

Info

Publication number
PT90563A
PT90563A PT90563A PT9056389A PT90563A PT 90563 A PT90563 A PT 90563A PT 90563 A PT90563 A PT 90563A PT 9056389 A PT9056389 A PT 9056389A PT 90563 A PT90563 A PT 90563A
Authority
PT
Portugal
Prior art keywords
meterocyclyl
diaminopyridines
oxides
substituted
contain
Prior art date
Application number
PT90563A
Other languages
English (en)
Inventor
Juergen Engel
Bernd Nickel
Istvan Szelenyi
Peter Emig
Original Assignee
Asta Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asta Pharma Ag filed Critical Asta Pharma Ag
Publication of PT90563A publication Critical patent/PT90563A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT90563A 1988-05-16 1989-05-15 Processo para a preparacao de 3-(n-meterociclil)-2,6-diaminopiridinas e de -n-oxidos substituidos e de composicoes farmaceuticas que os contem PT90563A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3816629 1988-05-16

Publications (1)

Publication Number Publication Date
PT90563A true PT90563A (pt) 1989-11-30

Family

ID=6354463

Family Applications (1)

Application Number Title Priority Date Filing Date
PT90563A PT90563A (pt) 1988-05-16 1989-05-15 Processo para a preparacao de 3-(n-meterociclil)-2,6-diaminopiridinas e de -n-oxidos substituidos e de composicoes farmaceuticas que os contem

Country Status (8)

Country Link
US (1) US4923858A (pt)
EP (1) EP0343429A1 (pt)
JP (1) JPH0217186A (pt)
AU (1) AU3481989A (pt)
DK (1) DK232689A (pt)
MC (1) MC2029A1 (pt)
PT (1) PT90563A (pt)
YU (1) YU99889A (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69209576D1 (de) * 1991-05-10 1996-05-09 Takeda Chemical Industries Ltd Pyridinderivate, deren Herstellung und Anwendung
DE4200259A1 (de) * 1992-01-08 1993-07-15 Asta Medica Ag Neue 1,2,4-triaminobenzol-derivate und verfahren zu deren herstellung
US20050089559A1 (en) 2003-10-23 2005-04-28 Istvan Szelenyi Combinations of potassium channel openers and sodium channel inhibitors or sodium channel-influencing active compounds for treating pains
FI20045369A (fi) * 2004-10-01 2006-04-02 Avantone Oy Suojatun mikrorakennealueen käsittävä tuote sekä menetelmä ja laite sen tuottamiseksi
US7960436B2 (en) 2006-06-05 2011-06-14 Valeant Pharmaceuticals International Substituted arylamino-1,2,3,4-tetrahydro naphthalenes and-2,3-dihydro-1H-indenes as potassium channel modulators
US8993593B2 (en) 2006-08-23 2015-03-31 Valeant Pharmaceuticals International N-(4-(6-fluoro-3,4-dihydroisoquinolin-2(1H)-yl)-2,6-dimethylphenyl)-3,3-dimethylbutanamide as potassium channel modulators
EP2061465B1 (en) 2006-08-23 2013-04-10 Valeant Pharmaceuticals International Derivatives of 4-(n-azacycloalkyl) anilides as potassium channel modulators
US8722929B2 (en) 2006-10-10 2014-05-13 Valeant Pharmaceuticals International N-[2-amino-4-(phenylmethoxy)phenyl] amides and related compounds as potassium channel modulators
US8030518B2 (en) 2006-11-28 2011-10-04 Valeant Pharmaceuticals International 1,4 diamino bicyclic retigabine analogues as potassium channel modulators
US8367684B2 (en) 2007-06-13 2013-02-05 Valeant Pharmaceuticals International Derivatives of 4-(N-azacycloalkyl) anilides as potassium channel modulators
US8563566B2 (en) 2007-08-01 2013-10-22 Valeant Pharmaceuticals International Naphthyridine derivatives as potassium channel modulators
US7786146B2 (en) 2007-08-13 2010-08-31 Valeant Pharmaceuticals International Derivatives of 5-amino-4,6-disubstituted indole and 5-amino-4,6-disubstituted indoline as potassium channel modulators

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE764362R (en) * 1966-05-12 1971-09-16 Degussa Subst amino pyridienes production
DE1670522C3 (de) * 1966-05-12 1978-08-31 Deutsche Gold- Und Silber-Scheideanstalt Vormals Roessler, 6000 Frankfurt Neue Benzylaminopyridine
ES368093A1 (es) * 1968-07-16 1971-07-16 Degussa Procedimiento para la preparacion de bencilaminas n-hetero-ciclicamente sustituidas.
DE3337593A1 (de) * 1982-10-27 1984-05-03 Degussa Ag, 6000 Frankfurt 2-amino-3-acylamino-6-benzylamino-pyridin-derivate mit antiepileptischer wirkung
WO1987001706A2 (en) * 1985-09-12 1987-03-26 The Upjohn Company C20 through c26 amino steroids
ES2078890T3 (es) * 1986-10-09 1996-01-01 Upjohn Co Amino esteroides en c20 a c26.

Also Published As

Publication number Publication date
YU99889A (en) 1990-12-31
EP0343429A1 (de) 1989-11-29
DK232689D0 (da) 1989-05-12
MC2029A1 (fr) 1990-04-25
JPH0217186A (ja) 1990-01-22
AU3481989A (en) 1989-11-16
US4923858A (en) 1990-05-08
DK232689A (da) 1989-11-17

Similar Documents

Publication Publication Date Title
PT93094A (pt) Processo para a preparacao de 1,3-oxatiolanos substituidos e de composicoes farmaceuticas que os contem
PT81007B (pt) Processo para a preparacao de derivados de 1,2-benzoisotiazolil-3-piperazina com accao analgesica e de composicoes farmaceuticas que os contem
PT92497A (pt) Processo para a preparacao de derivados de ureia de dipeptideos inibidores de enzimas, e de composicoes farmaceuticas que os contem
PT99671A (pt) Processo para a preparacao de heparosanos-n,o-sulfatados e de composicoes farmaceuticas que os contem
PT89661A (pt) Processo para a preparacao de compostos pirrolicos substituidos e de composicoes farmaceuticas que os contem
PT84549B (pt) Processo para a preparacao de compostos macrolidos e de composicoes anti-helminticas, acaricidas e insecticidas que os contem
PT84449B (pt) Processo para a preparacao de novos derivados 3,5-dissubstituidos do pirocatecol e de composicoes farmaceuticas que os contem
PT98369A (pt) Processo para a preparacao de azois substituidos e de composicoes farmaceuticas que os contem
PT89497A (pt) Processo para a preparacao de compostos piperidinilicos 1,4-dissubstituidos e de composicoes farmaceuticas que os contem
PT80921B (pt) Processo para a preparacao de derivados de 3-acilaminometil-imidazo {1,2-a} piridinas e de composicoes farmaceuticas que os contem
PT87201A (pt) Processo para a preparacao de novos derivados de cefalosporina 3,7-substituida e de composicoes farmaceuticas que os contem
PT84460B (pt) Processo para a preparacao de derivados de ciclopropano 1,1-dissubstituidos e de composicoes farmaceuticas que os contem
PT84828B (pt) Processo para a preparacao de compostos heterociclicos triciclicos fundidos e de composicoes farmaceuticas que os contem
PT93067A (pt) Processo para a preparacao de derivados de 2-hidroxiacidos alifaticos e de eteres de 1-benzil-3-hidroximetilindazol, e de composicoes farmaceuticas que os contem
PT90563A (pt) Processo para a preparacao de 3-(n-meterociclil)-2,6-diaminopiridinas e de -n-oxidos substituidos e de composicoes farmaceuticas que os contem
PT90017A (pt) Processo para a preparacao de derivados de arilpiperazinilalcoxi de imidas ciclicas e de uma composicao farmaceutica que os contem
PT84478B (pt) Processo para a preparacao de derivados de pirazolo-{3,4-d}-pirimidina e de composicoes farmaceuticas que os contem
PT89715A (pt) Processo para a preparacao de novos derivados de 1,4-benzoxazina e 1,4-benzotiazina e de composicoes farmaceuticas que os contem
PT88351A (pt) Processo para a preparacao de derivados de isoxazol-beta-carbolina e de composicoes farmaceuticas que os contem
PT92264A (pt) Processo para a preparacao de 14alfa, 17alfa-etano-estratrienos e de composicoes farmaceuticas que os contem
PT94629A (pt) Processo para a preparacao de derivados de cromado e de composicoes farmaceuticas que os contem
PT91787A (pt) Processo para a preparacao de tienopiranos substituidos e de composicoes farmaceuticas que os contem
PT91215A (pt) Processo para a preparacao de antagonistas de bombesina e de composicoes farmaceuticas que os contem
PT81955B (pt) Processo para a preparacao de derivados de all-cis-1,3,5-triamino-2,4,6-trihidroxi-ciclohexano e de composicoes farmaceuticas que os contem
PT85916A (pt) Processo para a preparacao de glicosidos de antraciclina, de compostos intermedios e de composicoes farmaceuticas que os contem

Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940621