PT71721B - Process for preparing a composition for treatment of pain,feverand inflammations with compositions containing 2-(substituted- piperidinomethyl)propane and propene nitriles - Google Patents

Process for preparing a composition for treatment of pain,feverand inflammations with compositions containing 2-(substituted- piperidinomethyl)propane and propene nitriles

Info

Publication number
PT71721B
PT71721B PT71721A PT7172180A PT71721B PT 71721 B PT71721 B PT 71721B PT 71721 A PT71721 A PT 71721A PT 7172180 A PT7172180 A PT 7172180A PT 71721 B PT71721 B PT 71721B
Authority
PT
Portugal
Prior art keywords
feverand
piperidinomethyl
inflammations
propene
nitriles
Prior art date
Application number
PT71721A
Other languages
English (en)
Portuguese (pt)
Other versions
PT71721A (en
Inventor
Nathaniel Grier
Richard A Dybas
Bruce A Witzel
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of PT71721A publication Critical patent/PT71721A/pt
Publication of PT71721B publication Critical patent/PT71721B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/145Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/26Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/38Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT71721A 1979-08-21 1980-08-21 Process for preparing a composition for treatment of pain,feverand inflammations with compositions containing 2-(substituted- piperidinomethyl)propane and propene nitriles PT71721B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/068,376 US4254131A (en) 1979-08-21 1979-08-21 Treatment of pain, fever, and inflammation with compositions containing 2-(substitutedpiperidinomethyl)propane and propene nitriles

Publications (2)

Publication Number Publication Date
PT71721A PT71721A (en) 1980-09-01
PT71721B true PT71721B (en) 1983-08-24

Family

ID=22082165

Family Applications (1)

Application Number Title Priority Date Filing Date
PT71721A PT71721B (en) 1979-08-21 1980-08-21 Process for preparing a composition for treatment of pain,feverand inflammations with compositions containing 2-(substituted- piperidinomethyl)propane and propene nitriles

Country Status (6)

Country Link
US (1) US4254131A (enExample)
EP (1) EP0024356A1 (enExample)
JP (1) JPS5636417A (enExample)
ES (1) ES8106294A1 (enExample)
GR (1) GR69837B (enExample)
PT (1) PT71721B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59176743A (ja) * 1983-03-26 1984-10-06 Daikin Ind Ltd 現像液

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3101340A (en) * 1960-07-18 1963-08-20 Searle & Co 4-tertiary-butyl-, 4-diphenylmethyl-, and 4-diphenylhydroxymethyl - piperidinopropionitriles
FR1451180A (fr) * 1962-05-17 1966-01-07 Heinz Haury Chem Fab Fa Dr Procédé pour la préparation d'amines tertiaires
US3262936A (en) * 1965-07-19 1966-07-26 Sterling Drug Inc Ring substituted-1-cyanolower-alkylpiperidines
GB1420759A (en) * 1972-07-12 1976-01-14 Wyeth John & Brother Ltd Piperidine derivatives

Also Published As

Publication number Publication date
US4254131A (en) 1981-03-03
ES494400A0 (es) 1981-08-01
GR69837B (enExample) 1982-07-19
PT71721A (en) 1980-09-01
JPS5636417A (en) 1981-04-09
EP0024356A1 (en) 1981-03-04
ES8106294A1 (es) 1981-08-01

Similar Documents

Publication Publication Date Title
DE3062467D1 (en) Process for the preparation of 4,1',6'-trichloro-4,1',6'-trideoxy-galactosucrose
CS420091A3 (en) Derivatives of carbazol-4-yloxy-propanol amine, process of their preparation and medicament containing these compounds
DE3060330D1 (en) Azolyloxy-acetamides, process for their preparation and their use as herbicides
PH16099A (en) Guanidinothiazole compounds,process for preparing them and medical composition containing them
DE3063937D1 (en) Hair treatment composition
JPS5627265A (en) Blade for bat of pinggpong
DE3065077D1 (en) Composition and process for stabilizing soil
ZA80667B (en) A mixture of stereoisomers of a-cyano-3-(4-halo-genophenoxy)-benzyl 2-(4-chlorophenyl)isovalerate, a process for producing the same, and a composition containing the same
GR60791B (en) 2',3',6'-trichlor-4-cyano-4'-benzoylureido-diphenylether,preparation process and use thereof as insecticides
IL57416A0 (en) Nitro compounds,process for preparing them and compositions containing them
PT71210A (en) Process for the preparation of a fungicidal composition containing hydroxyalkyl-triazoles
GB2048868B (en) Preparation of 2',6'-dialkyl - n - alkoxymethyl - 2 - chloroacetanilides
PT71721B (en) Process for preparing a composition for treatment of pain,feverand inflammations with compositions containing 2-(substituted- piperidinomethyl)propane and propene nitriles
IL57415A0 (en) Nitro compounds,process for preparing them and compositions containing them
ZA807964B (en) Process for the preparation of 4,1,6-trichloro -4,1'6-trideoxy galactosucrose
PT70039A (en) Process for preparation of 1(2,6-dihalobenzoyl)-3-(5-substituted-2-pyridinyl) ureias and their use as insecticides
DE3060617D1 (en) Process for the preparation of 1,3,5-trichlorobenzene
PT72029A (en) Process for the preparation of cationic compounds of the naphthalimid series
JPS5634613A (en) Hair treatment composition
IL59211A0 (en) Selected 3-trichloromethyl-5-cyclic amine-1,2,4-thiadiazole compounds and their use as ammonium nitrification inhibitors
IL56854A (en) Preparation of 2-(2,2-dimethyl-3-buten-1-yl)-2-oxazolines,2-alkoxy-2-alkyl-3-methylbutenyl oxazolidine derivatives employed therein and their preparation
DE3063201D1 (en) Guanidinium compounds, process for their preparation and their use as microbicides
DE3066124D1 (en) Substituted aromatic biologically active compound, a process for its preparation and its use as biocide
ZA80970B (en) Useful guanidinothiazole compounds,process for preparing them and medical compositions containing them
DE2960313D1 (en) N-(o-ethyl-s-n-propyl-(di)thiophosphoryloxy)-naphtalimides, process for their preparation, pesticidal compositions containing them, their preparation and use