PT105459B - MECHANICAL DEVICE FOR CONVERSION OF KINETIC ENERGY OF MARINE OR FLUVIAL CURRENTS IN ELECTRICAL ENERGY - Google Patents

Abstract

The device disclosed herein relates to a mechanical system converting the kinetic energy contained in the marine or fluvial currents into electrical energy. It is composed of three operating units, called Kinetic Energy Capture Unit (1), Gravity Energy Recovery Unit (2) and Electric Power Conversion Unit (3) which, connected through a traction cable (4) , are synchronized and conditioned in a two-way cyclic movement of some of their mechanical components. This process is activated from the kinetic energy collection unit (1) which, submerged and exposed to the kinetic force of the fluid (54), has a system of floodgates (12) with rotational axes (13) positioned in the support structure (5), said gates (12) opening and closing through an opening and closing system of the gates (6) comprising: a fixed opening / closing system of the fixed gates (7), connected to the support structure (5); ); a system for opening and closing the movable floodgates (8) connected in its front zone, to the traction cable (4) and connected in the zone posterior to the gates (12), through a hinged system (14); a damper and movement conditioner system (9) which, simultaneously with a system of slides (17) with damping stops (18), damp and condition the movement of the opening / closing system of the movable sluices (8); an engaging / disengaging system (10) situated between the fixed opening / closing system of the fixed gates (7) and the opening / closing system of the movable gates (8). The kinetic energy collection unit 1, by closing or opening its gates 12, acquires a drag force greater than or less than the gravitational force 55 of the weights 40 placed on the hoist 39, (39) being conditioned in its upward and downward movement by rails (38) and by a lower damper system (41) and its upper (42). The Electric Power Conversion Unit 3, which, like the Gravitic Energy Recovery Unit 2, is positioned on a dry platform 37, captures the bi-directional movement of the traction cable 4, electrical power from one or more generators (52).

Description

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In the; xx, xxx, xxx, xxx, xxx, xxx, xxx, xxx, xxx, xxxx, xxxxxxxxxxxx, xxxxxxxxxxxxxxx, 7753 P3P7G7I GP5 ••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• " .alpha., .delta. ca a'íap '.; L d. gt; gogo âCC-G Ç: C; ·.). at 7.0 sec. 5.57: 7.7. . 135: 5 - &quot; the blade was 5: 754.7 DC. to 10 S's: G, • ÇÇ; , 577P piGG i 737 3 Gp5: 37 ': 3555 57. G 3 7 3 75 035 DC hl te: d C' e G-quot; 7; 7.575 g Gdppp 1 c i.p., 55 755 | • CDC: CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC CDC g.p.5 5777 GO G5. :: 3.: 5 Gp.Cv.Cc sd pi. C · CO · c re 7575 GG of 5 CS and ': P · 1 g DiDiP5 G53 ijGvid: cc-: 7 p. 5757: 7 G-575 r-g. to '535.5 3 ·: 5. &lt; ίΡ P; 7 çÇ iÇ; 35557; &lt; i57i qm: &lt; C 70 77 3375: &quot; GO: 7.7: &dt; 11 d; 7g5: â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ- &lt;  € ƒâ € ƒâ € ƒ355: â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ7.77 (c) 7.75 (s, 1H), 7.75 (d, J = 8.4 Hz, 1H). CD 37 57G · ':. ·; C of r:> x d ···-D 'colao oCDS: d: G? 7 77 G5G7 53557.77377 Rob. i. 553555 d.75 55:75 V5G · 'and · 5-y .. GCCv Par :; 557 Cd; C, 5.8; N, 5.8. -: C aaci. 7d G: G3P.3.7? '3555: Cdvx r3G? 5 ·': '&quot;lt; / RTI &gt; c · -G dG 533: 77: 77: CtO of VACC 555 57357 55 '55 7: C: ia.i 5:33 7.5.5: 3: 3 (33 rc 3 a Γ .; GO 7: 3 DCD / Î ± CÎ ± 5; C.C.V .; 757 G p33333G: cb> 3337, dGdP ene: 3 G 7. • C D d b adito kú i 77555: 575 ·; 73 573 G: C = 55% Cd: d i.G br. V: SJC JC id LGd: G:. : i. .7 &quot; ' 5.355 (d, 1H); '3' '; C.D., or 575 DEG-55 DEG. D d op'G; G7G, Glycine Glycerol. Çi ap ida; , Mp: 75755 55575.5 7.55 51.3557 i: CC: cc 575753: 3 3555 .57035 1, - 1 tsl &amp;W; C 0 Ca dC ;. : 7 7: P7 xppoaiP GP57 3G 35: 5.57 37; s' d 57 P3 :. 5, 7: 1. of: 5.1 g. 55: a: 377pl; GTdxp ivi; 7: 7 75 GG G3. 55 55 G a 53 7. p C: pi 5357 5: 7: 33G: 5575: 3553:! ;; 11 TÇ 57 jiovi? (D): [delta]; r: G: 7GpGC: dG: 5355 ....... &lt; 35: 5: ... 5353 553 3 D 3373: QC Dx &gt; '.1.7 ·: GC 7: 557 OD 75 5557777 C: eC: χχχ 55.5: .75 3 7: 335555 3 --- 3 < 55375 and CpV Cd d S. i; J VCS S and i5a GU 5G5: 5r:. C gI gives DD5-.55: diVyGa to G1 .i5 P575 to pG5 5: 5G7 57753 55 eq: CGG 5.77. 5 * 1a; : 30 d .; C-GOC: G77A. : ·. 57G P55 3: C; cC; (3) (2) (2) (2) (2) (2) (2) (2) (2) (3) 7537 '6p: S1157 5 jpd? 8: 5 06 C 7 Wx.KX ··· 5 1 ia 533 a a; 7 * gpcx 77 C St: G p.55 53555.73 lo 3: t P: .5-5 3.7 : 357: 35535375500: 5: 575: 575: 575: 575: 575: : 7.37 (1H, d, J = 7.5 Hz), 7.55 (1H, d, J = : 575: 57533: W: d 5553 373575573 C: d: 5373: VP: 1 7.8% C-5% C-5% C-5% C-5% C-5% 1, 2, 3, 4, 7, 7, 5, 6, 7, 7, 7, 7, 7, 7, 7, 7, 7, 7, 7, pdpdddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddddfddddddddddddddddddddddddddddddddddddddddddddddddddddddddd ; &lt; Ç &quot; G555 &quot; and &quot; tb______________________________________ tb 55.5 tb______________________________________ tb 55.5 tb______________________________________ tb______________________________________ tb______________________________________ tb______________________________________ tb______________________________________ tbC: : &gt; · &lt;5; : r'V of da:. CDCl3). G: 73357: 757 and 53 dx C: ix 7.5: 573 5577 Ρ53 5757! ?: 333 1 3 θ 'Λ i 1 &gt; 7: 55-35: 53: 57-55.). - p - p - at. DCI-p 57 07.72 0 0 i &gt;; -05 4 3 6 Sc. at 00 and 70 ° C: • V ti. 0 37533: C ·: p. Calc'd: C, 75.33; Cc: 773 Idd d; US Pat. No. 3,353,543 and US Pat. No. 3,353,585 and US Pat. 7:: 7575535 P; P: IACCC 5:33 capioa :: P0 the s-C: o gV · ''! of 33757. D. 5.5; 73 555: C 1 57'7: 5 55 3 7ΪΟ 33: 33 05: 7 çr: .5773 G DC 5353.7.0755, C; ; P: 5.3 x 107; ? i.li &lt; 75735-755: nc: PCD 555: 3. : G335 37335 5.CD G7 · Di &gt; c: a 3 05373: gives 5737 3.77 GO 3 3577: 57 and 57735: 1 &quot; : -11 C: CD CcC c 037735 73d3 33 57 57 5 35: 5555.7; C: 53: O: Cc O: C 35: 133753757 57 CCT: 5, 507 555: 57: 57 (POG 55: 57-77 ° C (c) (c) (c): (a) (b): (c) diac. 37357: 555, 5, pp. 3575-705, pp. 355-703; ............................ 553753.53 a. G 5557 Pi. D 53 3.53. (c) 3,3,3,3,3,7,7- r and P .; 355 00.5557 p yi: 73 73 or 05577 Varius .. 7.73 CCi 5350:::. ; v.> 3033: .5: 7. ; 3'37.55 '57 1113377 cr; rcr 703 f.P:::::::::::::::::::::::::::. 75: 5: 3373: 5753 7730 v.a. 57 a.a. D-5-rax 77.5 5: 3 &amp; '' Ci 0: 0373 d 5 5 5700; iaaavs act: spevalg d &gt; S &gt; : 10: U iodine pav. to goxodorx; .0, -Pó P at these '0.0 <0: 133: 33i33 PP2-31, · ogxsaaav t so • Vi .0 Ti TiO vi iv 0 Ti i Ti. to cs.pt. ada iir. • s o; (ps), as well as the first and second sentences, are shown in the figure below. osd a Pav vss vssda v s.ipsxsads ps the minutes v; soara osta ata, Eo a: o: S rasada ~ S: s es ss and 11 ad es 3, .00: 00: 1 .. , adoa PP oo .se assa cxbs · sss ss srvaov saess: uo use ·, ca s &gt; χ.χχο &gt;: axs: ts-s: s The results are shown in Table 3. The results are shown in Table 2. The results are shown in Table 2. The results are shown below: '', '' '' '' '' '' '' '' '' '' '' '' '' '' '' ' Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ (v0): v0: c0: c0: c0: c0: c0: c0: c0: c0: c0: : 0 Ti vagas vvvvs * i '· pPP 0Ti 00: 002 0 O'0t t043 drias' 000000 0 0 0 | i> gvvvvv Go P VP0 .0., Sv \ 3.- d.S - ττόρΡ avieres ds SPSS To T, 0. •. ·. ·. : d. The. gaaà : &gt;. · v: »· vads. , as: d: 0 to svss: v to d-Td: id ass 'V fvV.OgV.V st if, X0' Ti 0 OS: voitol. (1), (2), (3) and (4) and (4). Γ0 VSd p 'd 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0. aivoaoa, ta ii sViva Ό 0: < r V; P a p o v e: V | S è VV ap ·; d V: Opales te: 0i, 0: i The vis ivtap looks; of the .1 00 - avaSev apapí ps V 0 0 a.l: d: a vis dias, i: a 0.i. i T iv 00 0 0 i i i i i i i i i i ti i i iiii: c ap 000 0 The Ti ta 00 ϊ ........ 00 v av: ai e ....... .Çl00L | 0.3 0 sv a v sv aorso vpiv.a 0s: di sV -y ....... a: a? V: va tosava a ........ t 011 'Í00 · 0 v sa: In this case, the following equation is used: : .oq • 0Γ; 00T: at this vvvt assa svs s: .os asseei: o <

Qt &gt; a · 0 0:00: nivs p: toa> ss to so. i.e. 000: 0/0 PT) 154., soissrs. ssvi.a svpisv: SS vasa as: S VtOS .V: OSS O t aso: 10 .1.0 T. &gt; The following table shows the results of the present study. The results are summarized in the following table. The results are summarized in the following table. s t r srss da: t-ass ciada: avs: aci Vl.vv, svvtts ss fs gg: ò p:: d: V; SP X: S S a ta sssaaa at: St:; ii00'Ti: S V SV.V 0 0 0100 flgv.vtsg: aced ... dO: e. 0 0 ': ss p.;. Tas ds: ss.t. ssvt Î'0: 0 &gt; 0 Iso sa.sp. -, This iss is T = 0V: O: S; it is. to-pdrrt .0: 0. ssw; 00 r vas sv.aao.tf ls, SO: 00 0 '. 0 -00. In this case, the results can be summarized in the following table. vOsi:: 0.00010 3 ... T) 0 ..... 'aovss ivvvaasas the &lt; I \ '' gt;: i Oá / Và &lt;; isa i'0.0.0 0 0 ·. to St: a vi s S: as s v: sa visa: V · ν: · -O; ssgt vsrsasais:,: asipataos oo 0 &lt; i 0: TO 0 sa: siat SS. : avst ta- i.-ads: s; &quot;; and wings to: o :. 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 rs; 0 'iarrpo vasa :::;. '00' V0 \ 00: 'Ti 0 0: 0: o vi i. : i.vs, V :: aavv. s St 00 ps v isa. t '0 &gt; : 3: lvvp: lvvp: lvvp: lvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvvv T. VS: SS V0: 0: life would be 0 is pa ss j âd. «, Taa spdsv a Oisv tsva ss ss ss sceps p vs <: vss 330- 1 0 0 <St: 0 aast agi.s this st. The results are shown in Table 2. The results are shown in Table 1. Table 2 shows the results obtained in the present study. gev: v.

<P> <p> <p> </ p> SOS ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ (i.e., cso: x eavrovo / age). doxrosvsae. s ieaeeastsntãia CíM5ações Sass of the tat-vpao ISAs, ον :, svasos: the outputs have been entered durto aspsvso: the atevspo, C'Oà step oas s esterases are asseaSSsxaeaSsa sa &gt;: v.:, si.aasv'S: svsi.va .. A ss o va s 3. avo ds se so rvvoa.v so: vs; si: as. s, a p sets' d; These are just: s. s aras s ss droplets, ον.ρ: ο χ vass ,. aaesxva avessa xs-Otas rata cosa as taasdSi oav à so a sova v. vu vsvasaesa; ': asaxaavaav wings to χ: ν.νχνορ,:. The invention relates to a method for the preparation of a pharmaceutical composition comprising a pharmaceutical composition comprising a pharmaceutical composition and a pharmaceutical composition. .. ·. (I.e. ν / ρ. ·· Α A cie 00 aa st 00 C0: t r a a nt. -or-. T O. to CisSciCtIon :: AA 0 < The present invention relates to a method for the preparation of a compound of the formula: ## STR2 ## wherein R 1 and R 2 are as defined above. The invention relates to a method for the preparation of a compound of the formula (I): i.e., in the range of 0 to .00% by weight. r t 0. eaccd: &quot; v ... bbV-rcpA V 'AA 0.:-. V; 0- <0 0 bar. iAA. r < 00 i 1 to A. &lt; The results are shown in Fig. The following table shows the results of the analysis of the results of the analysis of the results obtained in the present study. be r tctieca to rim

d; V -0 b- f Ç A '&quot; V, V, V, V, V; &gt; ·. b \ _i p 0 '\ ·· -0 \. The reaction mixture is cooled to 0 ° C. i. 0: 0 early: a cc o gocç: i. the cross-sectional view of the cross-sectional view shows a cross-sectional view of the cross-sectional view of the pouch. A C.:. . ib: 0: 0 -c. ceascaerste 0 0 0:00 'b &lt; . Cr, J. Biol. ..................... 000 CSCi::. Ui 0:. a, d.acccib &lt; i.e. 0-A b c C 0 O: A A A A C A C C P A C C C C A C C C C C C C C C C C C C C C : O: C: OO: 1,: 0: A b c c Ο · 0: A.:. 0, 000:: coauthority. ai bp ac ar a ta ca i a a .A n -a \ - <· · a a a:::::::::::::. you c a. The apc -000: 0: .0. \ '. iviiiii: i ';. '0 0 -: 000 <0 Aip the breeding Ca A A i. (a) and (b), and (b). In addition, p-pv-s. ab. 000 to F: i: i to i. b-V ·· scra s ··: - 1 C vi Óli Ça d0- 00; 0i.b 0.0. A: · '-' · 'c t r d. 00; cc A. 0: sv V: -0. The invention relates to a method for the preparation of a compound of formula (I). a ?: 0 ..:. 1. ecctc cr ..... <0 Vi: di ic -i: .0: 0.1 ii icedt: a 'dvpá <: - .. v -.- Vv. (c) (a) (c) (c) (c) (c). v; A '0000' 00 i &quot; The reaction mixture was cooled to 0 ° C. cci: cCs. Λ0ρ .; 000 J cr 0.0 or adi: .. C.! , &lt; / RTI &gt; . ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ AV AV AV AV AV AV AV AV AV. . to fall Acidac. d: s: 0: 00 A.Vi V 'to C d · tadaa aat ^ PV: -V:,: 00i'. up until ; v; i.e., 0: 0. i. ccr.cri.ctas a? adr-s to Cp; p; .b to: cc; ibl.A. . 0 0 OV; 1: -0-. : 0: 0C.:. ... ••: • Vb.: 0: c. f 000 0A- b &lt; i 0.00 0.00 0 ib bv qc.co OO 0 ·. cd bi cbic ar a: parc i T '0-0. 0.01-0.001. In the case of cc-cc-cc-cc. ............ . c 00 A vi, 0y 0 Oi'i'V'00 0 'b · .0 of: Ad v. Amino Acids. THE . i. Cí: ad &lt; i.e. CcC oct bi i v. In the present invention, the compounds of the present invention may be prepared by the following steps: (a) preparing a compound of formula (I): (a) In addition, the composition of the present invention relates to the preparation of a compound of the formula: ## STR1 ## ..a.bbb.bc .. .b <V: .0 O 0 .r 0.b çA i • ç.pt y-γ A poado: .cear soe; pç.at 0 <lt; '&quot; (A) and (b), (c) and (c), and (c) 03. 00 00 • V ib i - - dba, the archaic toacca 0a ipcccc 0.00Ç bv \ a - A c: 0, 0, 0, 0, 0, 0, 0, 0, 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 A, i................ CVVd 0.0 V ': ii 0': '0 aac &quot;; i''i -' 'ccp; tccct Ο &quot; 0θ: ib:; 0i ca 000: ·: 0 A; , where: (b) (b) (b) (b): (b) (c): (c) ............................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................... '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' ' d: C ': cs abccs Pope CeCiai abab: A0 A 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 • A v: b if AV &quot; 0 &quot; 0 &quot; 0 &quot; • &quot; 0 &quot; In the preferred embodiment of the present invention, the present invention relates to a method for the preparation of a compound of the general formula (I) of the general formula (I): in the presence of a pharmaceutically acceptable carrier, the pcaatmei, gives way to the tensions of the tension and facilitate the removal of the molecule is always the same as the caces and the amount of ammonia in the tea law would be expected to be achieved in a similar manner as would have been achieved in the present invention. fast plasti &lt; - P system. mechanic · dose be of tantamount,. It measures the melior aà: to adapt to the different conditions in which it will enccrmrará eraatmidc, thus, it is easy to stick to your efficiency. and the wetting of the material is carried out. to give, to present, and to melize the difference between the iseus coe coefficients of the coffers too - The mechanism of the merger would give the micríma of raldo posai mel, so as to imitate tanio: gcact poses: i: The x-ketotic system dose functionally functions from an anteroglyte to an inert medium with the nozzle as shown in Fig. mechanical mechanic:.:. propomide. let me be able to take advantage of: an efficient way may be the energy density present in the ocean currents, This deposit is made only from the parent to the parent child, and the child is in the same condition as the other parent child, and the child is the parent of the child.

Summary of the report d ninth i. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 10, 10, 10, 10, 10, 10, 10, 10, 10, i millstone directed to: a: denrersám the kinetic energy present in .marimbes esxrrentee or fluciais am symmetrical energy, To loa cg oentuga the acgáo of olfereatea stetemaa mecâxxicoa fce, sujeitos1 áo read Fridge tis the ore to a fear of splinters? Acknowledgments. as follows: o: Container of ebé-rgla oiPdtioaf: peteneia acamitiea c eiástioCí friction and inertia; they are acquiring a cease-and-desist in the United States of America; The provision is for three units: functional? eoc xmrrve: r: sci: .onnmoa Paeiqaxxr port dnidede d Captapáe x? e Imic.: fie

CdnC: 11, as? Yes? 1 diene peroxidase data exrcmiii as; The present invention further relates to a method of controlling the risk of injury to the injured person. ρ Dilution rate of water, solvent and subject to ferqe

Ci ly 3 ca s is. cerr ssciaic; d G-emes a is; S-ams 1 • d i ν '· siararra &lt; GlO1 Glidlpl., Where: 1 is L ã V G G; yyc 'f &quot;; eeee etid: G · GG?::; d;:; IG XI IG-1 to CCS. at the same time, See, e.g., c. ice, cee is; 'P yi G; '' '' '' '' '' '' '' '' '' '' '' '' :P. diyl] 1 .1. GG3: G, v-terma-amin and B 'GGI. a. C.-C'G p.ds: o < 11 pâ 'Gd Cl and> gt; and CSC, GG, G, G, G, G, G, G Ρ < &gt; : d · Λ-- ·. ' poe Ce.dicdi ;: e.sy ': da a a a i d; : A.aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa W ·.·. Pd 1.:. d • 1 • may be the same as that of G3 SC. dp .1: paie eoTids. C i GT dd Gd SCREW R e ra ra m e ra tio ns of the C e d e c c e d ix e g e dvc> of f d \> g and p ms): $ C ss r; C: air, C: + 1: G: 1: amemf re of: ': Over there. •1. U G &lt; A ssion of Cdd: p yyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyy yyyyyyyyyyyyyyyyyyyyyyyy &lt; / RTI &gt; &lt; / RTI &gt; &lt; / RTI &gt; 1 G: di G .1 G: 'i yy 1) ν 1, P tl SO: • '• • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • r 'ρry: c :: y. çp; : a cc s s GG G C C C C C C C C C C C C C C C C G y · 1 .. ab srempcrr ta a yy; v BB GG m, i ceedcit ca d 'quot; 3! G B, lG dC C USi d ;; &gt; .:W. (1) (1) (1) (1) (1) (1) ICC · s ϊ ·:., νχ ca p. · '·': '.;. yy HGG 'a / lC'G -; BB G Ϋ 'no: lnt <: read from the PC 1 1 lyi; :W; • SS; a a; 'd'; &quot; 1 &quot;, &quot; &quot; yy art ?. / Gt and Gd and X: yrdy: d '> X XGi s ce ce ΡΝ P'> Hi b Mamma a r [po rc G o ......... Qyy: CSC and .1. and dm.CC is ·. and if GdCG; iesc ssasiaec 133 GG ta \\\ a to L; The following information is available on the basis of the following information: loves 3i Λ r. BB and G]. C and. C 'S' .; &gt; G e. air-liquid. smirecie 1.GGG c; fall • V - · v ν -: &lt; Ρ & acaacvi &lt; yue you are Cd yyyeiy y y G-: Cie; And I have been able to assure that I will be able to do so. eur-lex.europa.eu eur-lex.europa.eu iciss v-i ci ·: Idi ccecl de s &quot; d: ciaerpi e Cirét i ea: : casyypi &quot; PP and. , and in the following cases: (a) the following: (a) - g.gg ;; sms, and the srira-arac er Ul p. (c): (c) (c): (c) (c): (b) (c) (b) to be able to see this situation. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - (1), and (2), and (2), respectively. &lt; / RTI &gt; &lt; / RTI &gt; &lt; / RTI &gt; The invention relates to a process for the preparation of a compound of the formula: ## STR2 ## in which R @ 1 is as defined in formula (I). ..... G be ÇG! .......: LP sis rca assa Ce Ce .......... : ••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• " s ΐ ΐ ΐ ΐ s s s s s s s s s s s ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ + ; &gt; &lt; / RTI &gt; (1) and (2) and (2), respectively. ICC: CID V Ii GEMI GEMI and i; cyy c. &lt; G '111 without cysimetry; CS ripse • is ;; rPctcdCd dd 1; and-i-ild · sia-Par. gt; g &lt; / RTI &gt;gt; &lt; / RTI &gt; 3111 I sar bceWá: C; art id! ytyy: s and .GG s; id.G &quot; i.e., d: 1: i. and m c; asm; ebaips &gt;. : .m G1 it m.s t cr Í.5 Tiidcad.,; g. 1, 3, 4, and 5, p ·. '&lt; CG mear G-GS v ees::. 1: 11131; G: 1H-NMR (DMSO-d6):? - t 3 • and v.- t: : C, · · <· ':' • Pic'-; : · &Quot; dGG. G is the number of cells in the cell. g d a; : g. c-read and CGG: di .Cl and Ga GC ie r s IGc Si: If it GG; im ,. Paec, G tmll G -il ssm α · bt v L; ; 3 scea cs; dCcid. C 1 -C 8 -alkyl; C 1 -C 8 -alkyl; 1.: at the same time if asp aess: ae GB 33 d: y &gt; C Ldd 'iVy: iC SC S: p O Çy &gt; it was a hundred and thirty-two; p and p t esc abc, · am sb: · G λ. gives an a and a a csr a ta yu .vv pP Ϊ iGG 1V .G P GGG i GG; s; eaCa Gt 1.-i i, · G y> y yy q ':>' T: cyGyicCs cs. to the feet. . . .. m &gt; GG * to cim; i; G ai rs; ·. ·. and (c) cc ...... G ....... and yr. : ·· - · y ..... dy · s; y and c < without d i y>: P GGG mea to cmampacs and to 1.13:. . V PC 'v.; I; β .e? Yy;' d çscedc: i.m :; . Gy; esar is d lr a G aed to ο dislama sse B &lt;. : JL'j 'cyy and BB \' c.: e s; and GCdt'GV. c G v.c: y.l and ...; d. L; g G &quot; GiGil GGB at c 1 years c 0 ·

C is the SSC and the SSC is the same. DETAILED DESCRIPTION OF THE INVENTION eep, 1 pdvd · aaip psí a; Cd: ai. A: .d: dd ::: dC; i tida sis aaa P t t t t t t t t t t t. : Α.βϊ *: t i. The results are shown in Fig. • t; rp PP a st a 0 iet A ;; ddd to aaa, Ό. '. :.: ν.ν>. '.' dd prsPts; dU: d d Sstt d: ........... Assa V '' so; OC to psp tasca roa v;. ·; , ·. • a: d.d-. at 111 aA ·. d: • d Cd · lati. s-r pd · Α · \ '·; A d dd-rp Pow D At Vi: ppsp â † 'AA C At 00 ta to & aaeJ. the results are shown in the following table. A ssstt P: V. CDCl3 .delta. and in the following cases: a a a a a a a - - - - - - Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ Ϊ. Isaar. ? ............ Pt. t ta a Ett · ris an sta ::; p x · &gt; · D · r; SP dst prati a - ã ã ã ã ã ã Ad • A D:; ·; p ', v' '' 'sv Ai d-dd aV-s'> <s; C-OC dC λ -x and ax; x-A ··· 'of O; • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • t hi dd A; Ep dd '· dalal. ct; • SSPT SSP t tc V V \ •• v sdraaés; of the isrsp ssasia :: A r &gt; dd &gt; d &gt; d &gt; d &gt; d &gt; d &gt; d &gt; d &gt; d &gt; d &gt; d AiA &gt; 'Ρ sai ist sasb rt tapíSis. . tv a siss stcsas-or Vd.Vd a Yes;; · SV Í. S; 1 st a t a dló iaAr x. ·, .r v.v p- PP S P ita · HS SP Ssa. ρρ. sta ie yCIDÁCAA st aaa VP: XO CâI A «O; , p A d 'd dd-Oddd •' A> • The value of the value of the value of the value is given by: O: t: ts: P; a. d-t: d of Pf d 0 COOlCO · * '< tassta5 •. · &gt;.; &lt; RTI ID = 0.0 &gt; &lt; / RTI &gt; to: &quot; A j-P; '; a) Cd aádP.sub.a Va; ..... tCO Cd tsta i'd C. &lt;; A: A: A: V: V: V: V::::::::::::::::::::::::::::::::: Tddd C.sub.a ddd: v.v.v.C.Cd.Cd.C.S. S.: P.S. Stat. pOCadd 'oer c aaa drs.it at v c :: · < · A A.À Ststtaria Cddd. PPf idOidd 'V dCOdO Cd • d A; • d d';: iAcptr 'C V' 'C !: si ss- d'Cdd) .A't.dÇ. V t ΐ t t t t t t t t t t t t t t t t t t (c), (d), (d), (d) and (d). the &lt; a &gt; &gt; ttsr &lt; P &lt; R &gt; 1 p.t to a ...: p -A s: .r a tu a aaddd d a rai; 'CAd. A A. o .V a Ά a Cd it 0 pss. psar píssaatt. • V app P 00 sfr • 0 'aa tsa. A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A PSS CiOs: 's »r going to Asia. a. a. V idit., Dp aa, - V, - ts di.tsasasti. % dAd. d. p .. · a assa γχ · i · · CAA a dd 0 ' &lt; Cd of the Cd if the CdOid is the same as that of the rat. -st if you want to do it. ! d d. ·% ·% ···.:. bake; : r-a.i.s. s p .ta, Sés sra; £ qlks da tvácogi a

This Lsa would make Father P ossa eaesaida dspracte. and the. n. aaaarctea s ·; p &gt;·; p · a ir i r 0: ts a ritaia t d'AA'A: A.d..t.: ·. X. ratt st dcrs t, Eat st CddÇ.d: 'P X ··· X. OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO OO ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... •THE. Cd · aaa iiqsstp: s stitiita ssàa 0 tssrar st: - wing A dai ispsa h OOOtOdO; .A asked A .. if pst.P dp st-alrs ipptr asir Cd apstr istpss t, 0 .t sta: (; ssrsasiai ts S: S'ss saras par atlsait a: χΆΐ apasai C. -; A dis Apr dd AddOd.daa at P Pa to dCCAa 0 tarara 0: cr trasassad .Cd dC dddd dd The apt stds S5PP Èx A atiat ãs. '. ·' · · · · · ..i X. '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' IOO: dC 0 spstí.SPar xdt V: daOç:; ·· '; P &lt; s raistc 0 ia ata' ii '.Αi 00.0. OCd; Ο.Α, Α Co ... The following table shows the results of the analysis of the results obtained in the present study. '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '. ooc C CC. 000 P o rd o rd o rd C o rt C o rt P a rt: However, (x, y, y, y, y, ..., ...). sp. ............ ptS X t XvS A; ; t C.A AA &gt; C ': iv; r dCOdddO; dAÇDa 00 SstrP Aatstar Ps.srtaaa. s: .i. A A A d. (d). 0- at 1 a iavr ortapta qr Pstst ddO 'Adi:: A: 0 dd · 0 CddiOà t sia ·'. , n ·. (I.e. .1; &gt; PP coo c. t Clddd Odd; .d.: dC .dd SP S P r 1 pa

035 toa aap 0 70 n C i Ge Ge V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V V. 3 V 00555 0 (tipi 70:07). This is the case of the 80:85 phase of this thesis. tb: 5: 557: 558 Ο |3535 pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe pe Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Go Γ S t t And that is to say that the sara is the V-a. W ith: Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò: 35 35 35 Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò: and the lactic acid content of lactic acid was determined by the following equation: (1) (b) (b) (b) 6 Vip7 v7 0 \ 7 V Sdpo .st, ίιΓν t 088 to ao ai va 1 to 850 c PS at .G -ò- • U.iÇi ÕOy aríp.:. :: a é.c · 7: i0 30 5 to 30::::::::::::::::::::::::::::: : 5 .t: 75.5'7; 7: 7 1 &quot; '··························································································· Λ l l l l l l l l l l l l l l l l l l l l Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ Χ 3d ': i.dada - ·: d.: · Rodúporáç 085: 55; and XX-Gr ala. 1, 2, 3, 4, 5, 8, 8, 8, 8, 10, 10, 10, 10, 10, 0, 0355075710: 0 UCE £ 4 '' - 37.33a ................. -i .................. &gt; 7 _w 3.01 ru ta,;.?: 'aa; Ed. aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa d.i.a.i.i.i.i.i.q.t. 000: 075800: / 0558 088 O: give 800: 07500-7000; pp ·; ·: Here G · &quot; ata 70:00 to 00800 50,500 / .7 5008880 {pic: &lt;: 5: 850050 55 7 0 0: .55050 58 3 dS.H NMR (DMSO-d6): γ7 and oodoar The composition of the present invention comprises a compound of the formula: ## STR1 ## in which the amount of the compound of formula (I) ................ -0 '' • ay .................. 33- iàao to-oo too 0 MC • V7-V00000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000 0.8 g of the title compound. S75 &lt; i75s: &quot; Î'855: 550: 3: 3. : aa. : 58 0 0: aaa: to 0 5 5.55: 55 750 i: d, 5 3 · '' ait: .555875 5: 5057: 05: 51 057 0: 8 -ep Ge 3 8:50 o : i; 53: available. V '; ; : · Ν ν ν ν ν ν ν β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β β ν β β ν ν ν ν: .1. 5: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1. d /; 85, 533; of the title compound was prepared as a white solid. p = 5.07, p = 3.07, p = 3.07, p = 0.05, p = 0.05, p = 0.05, p = 75 ° F (3 ° C), 5% by weight, 1% by weight, The compound of the formula: ## STR8 ## wherein R is as defined in claim 1, wherein R 1 and R 2 are as defined in claim 1, 1 to 55: 1 to 55: 1 to 55: 1 to 55: 1 to 55: 1 to 55: 5 to 0: / Θ Θ Θ Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π. : 55555 .....: 0 75075 SO 5-.sup.3 ': action: at CT 3 5 3 · 0 · 0 t 50> Xa: 3: i C <0 5; 0 50: 5,555: 1: 3x07 and .55: 577-: 55555: 00: 1: 1: 73: 0 .0 aa 000050 775: 0.775: 75857: - 55575: 5 - - - - - - - - - - - - - - - : p7: δ :: ·:> · · & & & & ap ap ap ap ap ap ap ap ap ap ap ap ap ap ap 57 57 57 57 57 57 57 57 57 57 57 57 57 57 57 57 57 57 57 8 8 SOS.c. poat, that of 005550.ovae J j. 5: .....; 550 5.55555.0075- "Ό-ρί G 5: 5 5 55 0 55: 5: 5: 5: 5: 5 a: 3:; A:> 5 pa ..... o ^ .. ... ii; ..... io. O-P / Op; ....................... 5 'to 5'. : 55.55: Îμ 8855: 558 Î "Î ± βâ, † â, † â, † â, € â, <â, € â, <â, € 43; .3 ··; ·. pop 337 7 0: 5505 0 · 55 U 550 00.0 7 - · ... 0: 5508-5755 a. the 55: t: 5 Was: J pod, 3 · &gt; i.e. er: 5.85.0 0.55 1.0: 0.5555 0.555550. 7875 &quot; Op: d: · ν,. ·. '. 3: ···· 3 5: 5: 7: 057: ptotem 55: 5550 po: 7 173.5 l XX .0: 07 c 07 073 8575 ......... Q 55 35 li: 5755.5 '555.5:. i.e. 55. Γΐ; 0 xi-> 7 &quot;7;0; 55: t.t5.5 5-: 7:: S: .7.7: 55 55: 000: .5775, 8550.0: 33: p-GGao 33.55 v G-a-07 5: 000 Q :. · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · : 55 0 0 t / 3; t X p 3 5 ..: 3:: ap: V it x. p-5,500; Si 5; Î »X-O-λ X: 5555: S 5 to 10: 5580 of

WWWWWWWWHHWBWWW-WWW WWWWWWWHHWBWWW-WWW 8 X) ΒΟΧΧΧΟΟ). SSIAO 880008: 808 ° C. from the dps of the d) r s to the d) aaif) dr!:. '' '' '' '' '' '' '' '' '' '' '' '' '' '' '. xyloxiodi o · .. d 88. ; Cb: - p-C b. -¾ C-CCCOCUb dtvHd; ·; ν ο ϊ: ·; ··: t &gt; Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â Â : i a; U, U d, X IB ^ Baa OCa-Vd ra dax]: · d a < l Utpd; (b) Xs / t: adt). : U pCtt) tCC ¢: ¾ taa d · s-. , s, and d · d-dl and d - Bd: v - B B 'UC at dpi Ϊ: 0 ························································· dsX ·) 't t: att ato xtcaxito ipu: a o? The aio; r &gt; db, d, d, d, and dc. (a) and (b), (b) and (b) a, C a da): d; , 'Χό d' dd atix yvimt ΪΟΪ 'v · S &lt; &lt; . X.vv Λ Oc · Ú} o B a% c- Uú atttt: t XX): at 8 X.XG8 dra: ó acdia .Latia. there; • • • • • • • • • • • • • • • • • • • • • • • • • a day at da ·· d; : · S d taa r d :, x> x: x a taaa andoti • i); t &quot; X XB 4 1:. &Quot; ν ': i ooa O-d. dB or '· ti. d. ; i.1.a a: B; L 08 UrÇ: y..y <d ·· C; x d ‡. b Xt.BO.) αa.Ba U Xp Otx UiC X'C ·, s.:· · sXaaot (X): iS v: 8aad Γ.Ί B, · · a a a a a a,,, C, ·· dQ. 005): '' '' '' '' '' '' '' '' '' '' '' ' of B., d ::; lue.tid: 0 X. Ud C d:, C aa Cd aaxap xo) x to a pa:.: xt.8 ·. ···: s · /.&gt;, d: - 'v 0 . idí-d .; axtaa x .1¾ • X d x: a :; U U 'd; td Β.Οί :: Χ: · 3 fi; di:. .: &Gt; V: CU i i U .d; . U i '; dddd; a: aa CGf: '; it will be brought to this point in the following sentence: , a). UoU :: v C U; I saw: ·:) ...... v tdà8 · B'i \ y'dB B.,:; D yd \ d y. d- - tB: a ta B.: ¾. C U: aaB) E- X): ata. oxapropion r? • ÓB B aaid CXX. &Lt; iU C 1¾. 1JC Ή · € (Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή Ή i.e., BIA; saa: d. ; B &quot; \ d; (i). · Xda. ................... to BtBD 10 Xa vC; ata b.ax: ......... d- '' Va.pt> u 1 ·: ·. · \ Β) ·, χ · yd d ....... B: &quot; :. 0 d tapot to o-aio U · λ ':' '' '' '' '' '' '' '' '' '' '' '' '' '' '' :) &gt; to .1. id Odddd: • there is Updat Β;; · d / / Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi Bi. X '); C ·;;; (I.e. : Good; 1 to xBBoaaxtaion ΓΒ7 X 8 ut B .8 dst Ba itta a: p &lt; .................. -. .. '.'. 1 d; Cd: t 8: at: aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa .1 loa paax d. axaa òs .¾: ···; ; 1a). A-B adi) Ba Btd; Q. • B &gt;. V 'lsd 8: t.P ti dl a aio x st a: CC atatatsa cie ·: ¾¾) QX v; -d ...... BX3B ...... d;:. 'd %%' .. · · · .. · a · · .. M tiU b; ..... Cd '; -i :. ¹H-NMR; ; ...... XO P: ... ... x) 8.api aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa aa xetax oada t C tp. aatatd. X d. a-boa eu, (c) a x 0 Op a.B • d a, and t: a: a: cB .. s.d.aa: X1BBL) X &gt;. (a) (b), (b), (b), (b) and (c). , BI C'Q. How useful are you? • s.vv < ) B of the xBCBC i 1 :: cx.aa xtsaapo · r tos will drop the t12 a; 1 to 1a, 1a to 1a, and 2a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to 1a to as in the case of OO.aC.a.Sub. of the BiBEC x x) o xa. xxx. toes; B.ixdd xxTXttxá a.8 aaaapo t. iv. 8 a B: 0 a.ia8 d a a 112b x a t χχοοοχ'ΧΒΟχ: X1 PP 1 axaxtaa; : ap a. : x) x;: xpprtxas xtstSbbBd.aadaavas xtlíBoB, BB · &quot; Eaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa &gt; B 3 'yyyy ai a cx) axpx.x8xvxss

C. CU &gt; d y'i O U id U CC \ J; d.:. r'j.t ',. ·: pstaiat a a: aspo a; t attex ') a a οοηοχχχη .a t a a d ,? the a .ia -a v a a ·. S · &quot; B &quot; &quot; 3: ¾¾¾¾¾¾ a: ¾¾¾¾¾¾ ia ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ ρ. The title compound was prepared according to the procedure described in Example 1. -aa ds t d oateaoo x Bt a); : â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ: . B &quot; baxpi) .alpha., p. Hello to Di: (C) (d): (d) to (a): (a) (a): (b): (b); 12, 80ppm; Oiilit: VÓ C; CIO o C &gt; &gt; Ρ, ΙϊΡ:; p .; polyamide; C (CHCl3):? R 1 is hydrogen; O? 20 3PF V? 0 t}: 2:: c; 000 bp ': 1525 (2 boi 801 (0 * ib the dummy Morta: PP P: .X> C :. r: tl: .e; l: 2.¾;. (S): ••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• 5 to 10: 1: 1: 1 to 2: 1 to 2: 1 to 2: 1 to 2: 1 to 2: 1 to 1: 1, 2, 3, 4, 5, 7, 8, 10, 10, 10, 10, 10, 20, 20, 20, 20, 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 10, 12 of 8 &quot;20; 2 &quot; 20 pbop02 all 0- &quot;p'1'0; DD &quot;, &quot; i.e., pbO2, pb02, pb2, pb2, pb2, pb2, pb2, pb2, pb2, pb2, pb2. (12.5%) of the compound of formula (I) in the presence of a compound of formula (I): wherein: , c: 8 provided · polo or rcorocti, corito? :: ooboo lo pop (8 d) (Only, PosP (1: 0) 0:22 p.i.q., p. 5i: â € ƒâ € ƒâ € ƒXDX biVa iq ion; (1): 1515 80 i 8 ρ 3; .i: 520 b:............... PiO2 O5: 5,500; Padd :::: PO 50 bi-ib-1; (2) (2): (2): (2): (2): (2):. (d V 0 to A CC V. Π; wire OP 2: 2 (i (V ».5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5 .5) bl b b & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & & b b b b b b b b b b 2: 121 3.02 1 aã PP 13 x; 1, if 3 3 (.311 (3: dl c 02212 02 22 OO 05 ;; OS ': bv O (i λ if p ;: \ / · ϊ, (b): bb: ibid ii:::::::::::::::: <P i0;: 2. p b0 0 22: v ..... OOP i ..... ...................... 1 2 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 1, 2, 3, 4, 5, 6, 7, 8, 2 'to (b) (b) (b) (b) (b) (b) (b) (b) (b) ). &gt; And 2: 2: 15-23: 2: 2: 2: 2: 1: p ...... p Olp (1001200b: 0: 20 (0bi 2 Ò-: 115 00: OOP 0 c <1? 0:52 (&quot; is lop C-2-ν ...... PCipa (2 00 (: 00): 1: 1: 55p: 01: 50: 55: 081 oo p = 020; O2 = 200; 2: 122; 205; 25 (00); (0, 1, 2, 3, 4, 5, 6, 7, 10, 10, 10, 10, 10, 10, 10, 10, 3, PC Pb CC q: 50002 0.2 OO: 1 H-1 Pb: (2 (b) (5) (1: 51: 2: 1: 51: (b) A compound according to claim 1, wherein the compound of formula (II): wherein R1, R2, R3 and R4 are as defined above. 02: ilo &quot; 82: &quot; 2 &quot;, &quot; 2 PO &quot; 0.1, 20 POI: i 0: tp db: 0: 8; (2), 2 ', 2, 1, 2, 3, 4, 5, 6, 5, 5, 11 (b) (b) (b) (b) (i.e., b). i: P3 &quot; Pb ibt 2 db; (51: 8: 18-80) Pb (3 Sb 1 .0 4 ': 5: 05500 (tb) of bi * 25.5; - :::: 00210 5: 3 13}, B &quot; given i '; 3p C: trac vrii P ·' P ': ········································································ The reaction was carried out in a similar manner to that described in Example 1, but the reaction mixture was evaporated under reduced pressure to give the title compound as a white solid. SO2-O2-O2-O-O-O-O-O-O-O-O-O-O-O-O-O-; at the end of the reaction, at the end of the reaction. As shown in FIG. 3, the composition of claim 1, wherein the compound of formula (33) comprises a compound of formula (33). 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a to 3a : 22 ii gold 5 20 ra CdCoi1i1i '' '-' '' '' '' '' '' ' a. ata- SC ·· :: o • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • : &gt;; Χ 2:. 1 021> 000 a a V lc Pd aa stsípra ç d d a 101 assoi a a; 1: 0 C. paa. (a) (b) and (b). (d) is added to the compound (i); P acification: 2:: 2- -: alt &gt; r coca cola 2s. v \ 33 Vv; '&quot; 1: 5: 0. : d &quot; 2: 2: 1: 1: 0: 0: 0: 0: 0: 0: 0. O; ii 3 Π ·. to. p o of • 0 • p; N &quot;:; (A), (b) and (b). 0000 If aaidct '1 s; a or ν-ΙΟ d < Λ '' '' 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 1,3 Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ. i; 11.2: 0.0 0 0 ii 00.0 Hi: 0 ii &quot; 'p ar> 0 p; Diffraction of the ICG: a ρ < s? per c. The title compound was prepared as a white powder. i 1 02a ΐ = ¾ 1.} i &gt; 3 to: C ci C ci a a a a Γ Γ Γ Γ Γ: lp 'ip ip: l: lOO; : .0. 1, 2, 3, 4, 5, 11 to &quot; &quot; 02: If i '. id '' 2. 2, 3, 4, 5, 6, ·. V -Î ± -, β- i. Bad.; aaa - i 0 '0 d 3 0: 0 03: Qp> cs pOOC at Î'.5: 0 of the color ____: &gt; The invention relates to a method for the preparation of a compound of the formula: wherein: â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ A further preferred embodiment of the present invention is the use thereof. 1: 1, p. erraa &quot; P: the icaPC; : 1 · · * · &gt; ·. (2), (2), (2), (3) and (4) are as defined in claim 1, (121 roasted roasted breadcrumbs): 0331 d * S: οο, οο ή \ .2 ': &gt;: i: 3 ϋ ip'; ρ;: i; à · 'urt &quot; id .; the given; id '& a': sc: 00: 1 loas • .Oq. SC is wires Ps ll> 30 'ss i • j.avàaspa> s.Ur; of the oil: 2 after 2 years of production, at the end of the second half of the year. The reaction mixture is filtered and the filtrate is evaporated to dryness. The filtrate is then evaporated to dryness, dried, and evaporated to dryness. 3 Ò Ò Ò '' Ci Ci Ci Ci Ci Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò · · · · · · · · · · · · · · · · · · · · · · · · · · · ·. The following table shows the results of the analysis of the results obtained in the literature: 1.11 ai The title compound was prepared from the title compound as a white solid, mp 218 DEG- · ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... ..... 2 2 2 2 2 2 2 2 Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό. 3Q. . 1 C Si Ui Mc á C v · · ··············································· 4: 3, 4, 5, 8, of the following: (a) R a la: C aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa (I.e. : l '·; .P: '.i .; 11: 0 .08. The wing VN V · d .O; : ';. &Gt;: o i00: i. ................... . : 0 to 10,000; ciao a ddp 's 51 1 v (of ira.dcat 130 i 37') coi ...... i li a ...... dc: ...... aa; po rsc &quot; 2: i Co ') ....... Oi OO1 adrá · d 1! i M c .... ata dtSíÍ ...... ... t ....... ccltstart &quot; ad OCoXa Sn C l i no: 1 day OO. &gt; B- 1 '' -o &lt; aa. • r'1 '&quot; dl. ct &lt; a.l. The results are shown in Table 1 below. rc ia: &gt; p .; The reaction is carried out; C sac-C sac-C sac-C dd-alkyl; 3 '-thiadiazoline. c. .ala to 1. O.t. In addition, the compounds of the present invention may also be prepared by the following methods: (a) The compounds of formula (I) , and in the presence of a compound of the formula: ## STR1 ## in which R 2 is as defined in claim 1, : ••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• (1), (2), (2), (2), (2) and (4). 0-3 Π O O v Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò θ'-: V: '' '' '' '' '' '' '' '' '' '' '' '' ''. Ο li: OC aar ed ap: aís í < rac pc i'iO 0'd'O ãv í S: S asppsaascicca p, ·. 1 to 3: 3: 3: 3: 3: 1: 1: 1: In the case of the present invention, the present invention relates to the preparation of the compounds of formula (I): 2: 1 to 2: 1 to 2: 1 to 3: 1 to 2: 1 to 2: 1 to 2: 1 to 2: 1 to 2: The reaction was carried out in a similar manner to that described in Example 1 (a) and (b). ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta ta. A and B are the same as those for the first two years of the year. 0: 0: 0: 0: 0: 0: 0: 0: 0: 0: 0: 0: 0: 0: 0: and the number of cells in the cell is equal to the number of cells in the cell. '- • Ν Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό Ό. iso. SSCi. :  € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ ti pc ϋ da Ui OOOO -0:; . (1), (2) and (3). CSC .1 CS. and c. iOOxOOC 0: b 0 of the epsilon eps ccfsc: c X · X M s 0 Y &gt; Pb '&gt;A1b; ' Oli assa - at 0 ° C. B:. s. The reaction is carried out in a similar manner to that described in Example 1 (b). SpSSSSS :: 11 Ό Ο. Γ0 and:: d &gt; Γ p. 0 and y 0; . (C) (b). 5 ° C t.O; tascbsis S P saia ds. a cc: cs 1 i ii .1: i:: s: ss sca sb svs ji; ai .000 The a-c, 'lea ia a bÒb ΟΟρ'ί, ΟνΟ. ·. CpPtCSC; ·::: saaib CC: abf ssasf; a c te et aça, -day 0: .0¾ saa asá. is, i.e., from 0 to 0; ::: en en C C C C,,,,,,,,,,,,. (I): (i) (i). .............. ............................. ·· of iasap Hi, 1, ·: aeaat 'is {: ps &gt; . ftd. ds IpOTOO xi <b H if: aca c: 10 0 b; (i.e. yN béi ·············································································································· 0 ; Si-C tlssi of &gt; 13-d: C: q a a: cs this is the CCS) is added to the XS. OOO; 00 • a a ti 1 ό YiyOl O 'a <t O-d. 70 0: · '·· &gt; v ··: '.? - 0 0: 00.0 .. ocd C s, ct Çi: sssea cd Ssc 0 'a sla ps. • &lt;: a b; B; . &Gt;: &lt; / RTI &gt; (b) (b) (b) (b). s & c. XOOObS -0 aac s &lt; yc: 000 'cc cc v vc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc cc sSTCi s.bes ice, ··: '.' v ãh; tddc w;: 1 ossal ia iCS; (s): 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, s.ca · &gt; ' . &lt; b &gt; bsl dV: s d. d; : 0; i v < 0, .0000. the. (S tc '<1 pc QO 0.,: 000; 11 • bp and O-OO dSi t: dda ees tC: Ai.C.SS;: CSC or baa aesf ao do cabe The '00 .00 · Π.ΟίΟ 'λ aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç aç b b b b b b b b b b b b b b b b b b b b b b b: The present invention relates to a process for the preparation of the compositions of the invention in which the compositions of the present invention are suitable for the preparation of the compositions of the invention. OCXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXX ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí 000 000 000 000 000 000 000 ¾ ¾ ¾ ¾ ¾ ¾ ¾. M. B........................... 7) OaSiC - V · '' · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · Lip i pdb} Tsa Ό l: ba: -:. 10 v> O Tida al (a), (b) and (c) and (c) and (b). 14- 00 acra assa dl iSCS ..... 0: .00 'sscplse ....... o. .C ......... c ps ,; this is the result of the reduction of the amount of the oil. : .0 'Hi &quot; 'riU> 100: 0 biss. Od. \: a / ia: dSfs.edf:; cc '0.0001 · 01; O: ; ip: found: C, 70.0; ; l e; : A: o, ···:: \ fs.i: X. .b cXOXOy Ob &gt; 0 doo •• OiiOii CiOiO · ΐ>: ······································································································· aalea: aunt's age: i'P · ρ; Ϊ S.. Y À À À À À "" "" "VI 0 0 0 0 0 0 0 0 0 0 0 0 0 0 B B B B. over there. &lt; for example, days 1, 2, and 3 days. ; Sb ga.i.s d-¾. . i ç / Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ. li Pd is asides to:;: 0c and icca.sf at 0.00 .00 ': C 00 &gt;; CA. : 0 &gt; 0s: prot ac: o: si (S; O • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • ; and (b), the compounds of the present invention may be prepared by the following methods: (a) the compounds of formula (I): (1) and (2) and (3) and (4) and (4) and (4) and (4). i ΐ ba ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ ΐ 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 7 '', '' ',' '' '' '' '' '' '' '' '' '' '' ' , Ss.a. .. SS.CS ssial .......... 0 0: '0; ..... 1. vi cf, c. Sa::; b sia ssba ccssl csa .1 0 &lt; θ V Xc: 1 cd: Ispests • 11 11.1 • dsi: ΐ: ΐ · 1 · · 0 0 0 0 0 0:::::::: oets is aac biOO: ••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• x> g: xO'x si: b, proa eaC: í si 0: 0> 001 o · ca Ό esc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc sc. (I.e. g. 22000053 eda; b.22 rb-r .2.0: 52-5-2 22 f ·.:? The reaction mixture was stirred at room temperature for 30 minutes. Ci v 1. a a pii ί'.ι.ν. x. 1 2 po b á.â: a a a a Γ; · 3023 v. · · · · · · · · · · · · · · · · · · · · · · · C Cri; iis · sd &gt; Ilo. '1 b' re, and Oa> 0 own '0.00 of 0 200 T; 1 bl 3 552 2 5.25 0 1 2 3 4 5 5 5 5 5 5 5 5 5 6 7 8 9 or 1: 500: 0 22 52503 dspee c lede do.v ti. 1 pi <b aaaaa 0: 3,3; of the compound of formula (II): ???????????????????????????????????????????? 5: 1: 2: 3 U-2 .1 0.3. biatá · ò · Xrt: -i 52 ó iCi: .a .fát 22 0 2310, · · ρ &quot; 3 s 3 1C; 5525: 5.1 P.1 c. The product is a copolymer. mp. ; to t. ca alone · 0.1 Cp '; 1: 2, 2: 2, 2: 2, 2: 2, 2: 2, 2: 2, 2: 2, erpipv loO; • Dc two 2033 Cp :; C and d; r &gt; 8 20 p i ν 'r ·; 1 to 2 is 2 to 2: 1 to 2: 1 to 3: 1 to 2: 1 to 2: 1 to 2: s.2dP 0 1: 3 b ί o lie Pr Pr &quot; 0.025 123.253 P2 530 52.1 ode Pd3 Cb · Ce 253; ipiie; C-O-2.02; b; c 2 c -1 to c 2202; UC · &gt; ,. p &quot;-d:; b &b; V. 521 cc-pro. at: :·.,;. 1a. ............... 0 :, 1 '&quot;' rp 1. eccer and e: iapoaé 20030: 205 5.55 pr? • C14 H25 N2 O2: 532.55 5'-i: 5: 23.5: v; d: 0 C: v v;. ·., b-C. c. V. '. The title compound was prepared from the title compound as a white powder, mp 218-221øC. 1 H-NMR (CDCl3):? ΧΌ C ir; .55TT; l .; • 2, 3, 4, 5, 6, 8, 10, dceert; : 2), p2 &quot;rC; s P 'b' b.rrc 550032 fj, 3 25 1 ':' 1 23 3 CC li li 0 · ,. 3: 03-2: 30250 and aa to v. (b) a compound of the formula: ## STR1 ## C? D 5 '? C ix C d: - v bpt if it affects it e8.1 ........ aaa a cr ... .p.yi-p.ya: 3 3 :: 52í 'M ... ... . γ p χΤ'ϊ: '. ......... 3:22: ca: ················································ The reaction mixture was cooled to 0 ° C. Fig. 1 or V. ic · ρί ': ϊ. ··; · Ctl ;. Ci-CX ii. (COCH), and (C (OCH)). appoints Òp; l2 < .P; &lt; 3 '' &lt; VV ·?. 2.21: 22; Fig. 502 S.S253C 51202: 5, s. 0? rCiCoCB 2535 32 '2.2 ac &gt; a a. · a cc. c.c. •••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• at 2 ° C. 2030 Od bbv'V çu; . 3: 23: 00: 00: 0; The composition of formula (I): a) C-1. (C) 1 3322: 5: 1: to Tu 1. d ·: 'A Blt &quot; ¥ i: 3 t a d. C2 30H₂ :Cl₂: C₂CH₂ :Cl₂: C₂CH₂ :Cl₂: C₂CH₂ plCl₂: C₂CH₂ plCl₂: C₂CH₂ plCl₂: C₂CH₂₂Cl₂: C₂CH₂₂Cl₂: C₂CH₂₂Cl₂: C, 50.22; :  € ƒâ € ƒâ € ƒ30 dp: e; 25: 5322; yl] -1,3- Vd ara .1.251.03: C:. : Î »max 2: 1 1513 PCoC: 3 jdi 2525; :; 1-Î ± -cyclohexanecarboxylic acid; 552 52 555 555 e.t ib ili Ç. o .a; 3.2 is; Cl &gt;C2-C6-C6-alkyl; 3? 01323 52.52 5.55 ?? 5 dc -O; W; (c) C 221: C 221: C 221: C 221: C 221: 1, 2, 3, 4, 5, 6, 7, 8, 8, 9, 10, 15, 15, 16, 16, 16, 16, sesic and 32 2 2253 ol Irp r 2.52 50 1 b OOP 5? 52 2?: OP &lt; 5000 C? The invention relates to a method for the preparation of a compound of the general formula (I): wherein: X is an integer from 1 to 10; , 2: 2: 2: 1: 1: 2: 3: 2: 3: 2: 3: 2: 25 :: 0 rb: o O: 2: 3: t22: dr3iO X ...... r; Cl ······························: 5, 5, 5, 5, 5, 5, 6, 5, 5, 5, 5, 5, 5, 5, 5, 5, C 3 H 6 O 3 O 2 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 3 O 2 O ., nc οό and C; 02; 21 s. · V a 5355325 25.2 P pO ? · ': X' '.tc &gt; of' ν'ré C j p; i and ^ 2 poíí'i: Ti: ¥ Gs' der CSR. . 1: 3: 15: 1: 2: 1: 1: 1: 1: 1: 1: 1: 1: 1. tr: 12552; .25 p25bac ir A11C1C, ccC pbCiCi CCC: &gt; (c) (b) (b) (b) (b) (b) 232530 2: yl 3 &gt; P a ca. elo · '&gt; (C) (b) and (b) in the presence of a compound of the formula: ## STR8 ## up to 02:. ;; ........... • R 1: 1: 1: 2: 2: 1: 0: 0: 0: 0: 0: 0: 015: (1), (2), (2), (2), (2) and (2) and (2) and (2) and (2). X; ic &lt; 2 &gt; 53205 &lt; 23 &gt; pp. of ...... 2x r.VrC ·. ^ ..... 0.2.555Ó525 ΐ; 3.2 ,. 25.1 '2 552 to 2: 2: 2: 1: 2: 2: 2: A suspension according to any of claims 1 to 4, 32.10 3 .iod 25 ?? The. or? 3b5ba; 35 2 ri-C r a Χ: Πΐ Ira- -Gi GC rata of the p j à ja V V V V V p p V V V V V V V. ·; a a; settled ata; OOOX &gt;, &lt;:1; (Χ ΧΡΓ ΧΡΓ ΧΡΓ 0 tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot tot :: :: :: :: :: :: :: :: :: :: :: :: : θ rafer-êre 0.0, 0-0. 0xxx: <a: tiae: ap S: tXX '&quot; a: p: cr: ixaaaa.l.ds; t 0 The tl it: cr ... Psx xtas x P r xxx ti * dd. d ·, ·,; a prxxtaax, ·: i: a xis; dxa: aaxai tix: xxá .axax.xa: xrx. '• • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • xaaa flx CGOG 1; pi G xa: rl.aixo; xx xxa: □ .dr 0: Xx xxx .xxxxXxXx 0, ÍtC aX XX a C: ap priaiá ia O xta qÍO arare-axx1 1 · 0, COO, &lt; tb &gt; &numsp; &numsp; &numsp; & numsp & numsp & numsp & numsp & numsp & numsp & numsp & numsp GCCoGOTl, Accordingly, the present invention relates to a method for the preparation of a compound of the formula (I): wherein X is as defined in formula (I): wherein X is as defined in formula (I) : O, &gt; 0 ca ·: d. And Xaa is the number of cells in each cell, and the number of cells in each cell is equal to the number of cells in the cell. , ¾ Ti t .O .O .O pa pa pa pa pa pa. . ·. a. G tao &quot; Pi.â, "â," Oâ, "â, ... Oâ," Oâ,,. ; rx. r xx. XX.XT: TXÍXP. a; xxxxax: to 1; 0.8. a.aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa GO · á · d ':; ; · &Lt; x '' '' '' Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ ΙΚΙΡΡ. to CP; p &gt; xx-xt XPX a: apasxa ria a: · .... ::: ': Cd coo; • axaax.t oo prx ssanae aa.xj ααχχ ..... ft |; ... ato: OTO as txxxpaa • d <p ·; arppp pxxa. 0-01 S S- · ·. S-V, - s-x ·. ·. . ·. : :: :!s. ······························································ 0 • d i xa px.x; 01 t -0 0 i · á:>: XuxS-a-axais-o χχα a 1.1 ', .1 axaaxs iC-. stxa pt-r iOG. 0 .rsxtapxa 1Cl .... · &Gt; . ·. Ό xxid Gi .d .. \ aO αχχ *! to the e c i d i, · x: td, 1 wool v < • 0 ataax das; c O; 0 '01) XXII; it is the same as in the other. '' '' '' '' '' '' '' '' '' '' '' '' '' '' or 0 ax-xx 1:: p / .Op_; 1 i; axx G xalrda cfc-xraexapaa • 0 C-'a dd G .d'Ο .: '! daxa ΨΪ ti a tsÀPpí; 1: '' '' • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • (x, y) = 0 (x, y) = 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, xx xx xxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxXxxxxxxxxxxxxxxxxxxxxxxxxxxxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxxxxxxxXxxxxxxxxxxxxxxxxxxxxxxxxxxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxxxxxxxxxxxXxxxxxXxXxXxXxXxXxXxXxXxXxxxxxxxxxxxxXxXxXxXxXxXxXxXxXxXxxxxxxxXxxxxxxxxXxxxxxXxXxXxXxXxXxXxXxXxXxxxxxxxXxxxxxXxXxXxXxXxXxxxxxXxxxxxxxxxxxxxx (x, y, x, y, x, y), dx 0x0, xx, xx, xx, t-O-O-COO-xa> P 0 dt: P: 0 0 0 d X_ 1 xx cx pb at xxx Px: xxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxixxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxXxxxxxxxxxxxxxxxXxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxxx, (x, y, x, y, x, y, x, y) 51 x 0.1 x 10 x 10 x 1 x x x x x 2 x 1 x 2 x 1 x 2 x 2 x x 2 x x 2 x x 2 x x 2 x x 2 x x x x x x x x x x x x xx (1): C0 χχ, χαί .. 0 Cdd Pst '- s: xícXd ittx Pd' <adrt ;, 0.0 xial'-1 1 ····························································· to O.Gd 1.0 ax X 1 X 2 X 2 X 2 X 2 X 2 X 2 X 2: . 1 &gt; '11} COG 0 ρθ o as' Γ 4 0 li xsa d: x GO 0 &quot; OGOG'07............. , · '· Χ; xdp ΡΧΧΡ. X xa X dxd XX Oi .d IP I 0 0 O t sx-: xcax: xxx.5Pi. x; x.itx.a x: áa. xxaaxxx The Pt, PPP i. (O) O: C (O) O; a tx |: p; you are ipEP .O) and vdd lx P. x rhes ida xpr. O.G-dp'10 aiil 0 xx: aaix O d; ÇC CO: apoat xa for χ.χ.χχ The XX rc &quot; It-O dO: C G 00: '- d d ΟΙ 1. &lt; v '; 1 1 qxsa a 0 CO xaa a XXX O'G 1. XXX O.Ç .: c: aa <rs xpl.di rarc. , td axxax 1 v. &lt; (1 g., 1 g., g. x g. iaa: YesXXX aO? S! ! ; -0.alpha.-oxo-1-oxo. to X XX X X X.X. G.Ç, OÇ ,. OGlGiCd. 1G0:. ; G p. a xaxxx o ... a .. XXX d O x.àx; x. in .xx "OGoo i. i-it, and .1 dxxuxx: G GO x axxax: xxaxxs.t xx; xxxxx; OCi xaa the Q Pd · d · xp xi r: p: SxS 5! T; .XXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXxXXxXxXxXxXxXxXxxXxXxXxxXxXxxXxXxxXXxxXxxXxXxxXxxXxxXXxXxxXxxXXxXxxXXxXxxXXxXxxXxxXXxXxxXxxXXxXxxXxXxxXxXxxXxXXxXxXxXxxXXXxXxXxXxxXXxXxXxxXxxXXxXxxXxXxXxxXxXxxXXxXxxXxXxxXXxXxxXxXxxXxXxxXxXxxXxxXxxXxXxxXXxXxxXxxXXxXxxXXxXxxXXxXxxXxxXXxXXxXxxXxxXXxXxXxxXXxXxxXxX :. d. .................... Ix pis txlrax.l sx xxa S; | xs. , qi.xx ΧϊχχΧ, ρΙ.Χϊ..1χχ :: ρ χχχα ap ;: dsax a xxa xx .faces; CctHCHCHalkyl: the atxpaxy. aty a .1 xxxxxpl-xxsad I; χ. ..f cxaxxxpxlxx: xi. tb 10: 1. CG, axxxra tare. -from my father Pa | S; . there.; cox: áti.t: .al'da pair jx..xxxadee; x pp; ... ap; .... X.r a. x x pá ..... í | ax ..... aqaá: .... s.aú.a. X.xxx:aax:pxrx.p a at χχχχχχρρ i. atxsra to axs. s t 1 .t xx l.de · p &lt; &gt; r sx; a ta xx x ai xxa atai. ta. &gt; The ratio of 1 PP to TXG is 1 to 6; (1), and (2), and (2), and (2). XTC X is the same as PPt i. HPr; i; d iW: T .0 GpYa; Χ; Χ Χ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^ ^: id &lt; RTI ID = 0.0 &gt; &lt; / RTI &gt; &lt; tb &gt; &lt; tb &gt; (i.e., gt: gt; gt; gt; gt; gt; gt; gt; to stop the action of the atherosclerotic arthritis of the artery. a. (a) and (b), and (b). Xaa: Y aaa tdrtPam p; ada aar X GiC Y 'Y. Λ dp-G at; aar ariai aoap \, -pa pi, G ·; T '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' and dd: i.rtríato (3 i id G -dl a GT .1 i a ar :; a spdet. itr: d.do ae:: ogG err e? 'G γ; i (X, X, X, X, X, X, X, X, X, X, Y) t: r ds dT d ica a '·'. · 'YY £ ar G to in ΐόΓρθΓ ·· Χ.'Γr rai: -da-it • γ · γγ i -G ip C : CXD O TTXd ': G iX to aaa i: · acxaa <acaa or apa ja ra: .ipd 1. (X) Y. aat:: a &gt; air i Pa a: raaaaaida of the V. ot χ a at pi • ^ Y i; T γ; v ': GCi'GiG: U'-Y-.ti t' s: · Υ: Pt lar pp''i :: pa .. s- 'V ;; · · · ·. N. γ GG /, T w r a sa uteiterate: Γ: &quot; d &gt;: Y Y d -d of the GGG aa:. O: X 1.1¾¾ - '' 'Xy-yy ..... XiXG :: ρΥχθΡΧ: · Ρί' r Y Λ rttra: .0 '' SP; : rtde rtde a de parrt: ta a \ ·· < ·. (a), (b), (c), (c), (c), and (c) • GOX a .1 there is now a P GGG a PG ri ta rt of the arid atart aT XT a> gt; ; Y \% a G i γ G aaradiar of Pd a γ ······································ - YY of PCS ΟΠ ΟΠ G G G G G G G G G G G G G G G. G. G. G. G. G. G. G. G. G. G. G. G. G. G. G. G.. · The torso of the gypsy gypsum gypsum gypsumum gypsumum gypsum gypsumum gypsumum gypsum The present invention relates to a process for the preparation of a compound of formula (I): A compound of the formula: ## STR1 ## wherein R 1 and R 2 are as defined in formula (I). GT: r ... ;. GG t &lt; raaa eatat X, C- G o: G r urta i, · ad γ &gt; · Y that ar ar to art, t PÓ Y'P; G of trrd G pi G t G: ar Po adac pX · γ · γγ given to G-d 3 D ra> ... aat: t.ri ar ..... occ GG .... γ ····················································· C .1 0 ad X a rd: a: aa of r ··. * · R; ? pitia .t • dl, r ': ·. . X G G G t T t t t t t t t t t t t t t t t t t t t t t t t t t t t. Y ad} pa: datriatura \ G.d Gli r.i. d: a p. roaa ta t taro rdat G: 10: lid .i Ϋ; ' (A) and (b), respectively. parra, r U: Y; i YG: a ai Λ d.j < The title compound was prepared as a white powder. and d to X., as a function of temperature. Jaitarraa of XGG .lha v Pd X • .d ·: roataat, ·>: artà t a; . PS:: Y ·; r a γ ::. γγό · 'rtt a a a apor da rlsp; v. And a.l b -a Y: · a Ts a jtarta: í a d; S Pít r apt a orr Τ: ata: ti. The ! Siatilate, G. to VY · g of the PP diU ················································································ ; The invention relates to a process for the preparation of a compound of the formula: ## STR1 ## in which R 1 and R 2 are as defined in formula (I). d r'Y to the tora; · ÍY: i Pd r qda}> d-aetr aar c a γ; to X • d a a aa γ ·: γΡ · Ρ> ·: ·> d i a: i :: γ r: ar; p Par t; G: o For d: v: .t.r: pa.ír,:::;; sr, G pa r 11 r d v> The following table shows the graph of the graph of the graph of the graph. ργΐ. (I). ·. The; G d yyG-GG a; tf d: p oa; : Ytd O.iX 1Y C: G X r. · A sweet potato to be added to: YdYy 1 from GG d: GG ata. C aa Y '' p Γ d Υ.Ϊ Pi- to give a a i., D :: e .; , p Υ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ 3.. of the aCld i; d: d. er d-p there aY-: r d a ..... &gt; . • • • • • • • • • • • • • • • • • • • • • • • • • • and (b) a compound of the formula: dY · &gt; rstaa ·; aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa g. g. g. ata · - &gt; · O asra dotaa da ptaa dd:. ). The present invention relates to a process for the preparation of a compound of formula (I). Y.; i i Q 0 '; sv'C'Y: and X. • ·, Υ. · ΝΥ; . And t.G · tt: d. ; • G G G Gy Υ.,. ΓΟ t IPI E G i}

$ X

Ni: &gt;Go; or from the 20th to the 11th century, to the arsenicals: rd. ; · 'Ao: · &gt;; (I.e. 8 (t 1 f COSO; in the pao t of the d. -> a and bj: on the corsoa siso ΧΧΧ ti: d 8: ld aa l qa o ij a; The following table shows the results of the analysis of the results of the two experiments. or V: o .to o: ad: a XX 7: 7 1: ai: 1 'd!' y''il \ <ab: srPdr :: s / .ba; y: hi>: (1), (1), (2), (2) and (3). X ': X': X '' '' '' '' '' '' '' '' '' '' '' '' '' '' ' In order to be able to do this, we must: • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO: ISO / IEC Or drt ote 0 dolly X1 yacht: Ροό: Ρ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ d d d d d d d d d d d d d d d Λ Λ Λ Λ Λ Λ Λ Λ Λ Λ Γ Γ Γ Γ Γ Γ Γ Γ • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - the tail ayy i-did or iiyyy.dt ta a i. '; Lrs.il. 0 S, ΧίοΧΙΧΧΧ II X IX X O P oot X! ' Ί. and d; ) ibd .v.v.d · t.v. · :. 0.7.0 .si · r: dd i ·. . · ;. The compound according to any one of claims 1 to 4, wherein the compound of formula (I): wherein: PS S; c. 'd' i - la, incidentally: ssoaon. d; 0 ° C. CtOrO id: li doct 1 oo &gt; In the case of &lt; tb &gt; (I) rao sd.isoata; 5 xc; ; C &gt; d: · dl. to-ooi orrod X. Λ ti (¾: ¾. and OO 'O-F l t t t dr V V V V V V V V V V V V V V ..vibli 11 {.; · a; 1, - · ·; · / 0. a sill ad 'i. · &quot;: S. -s-, -.1 v &gt; i &gt; And X-ray diffraction (X-ray diffraction), and (X-ray diffraction) of the OrO 0 .XadidiXy: .................. 1,100: 0% of the total number of copies: > by andrOi::::::::::::::::::::::::::::::: \ l.la: \\ \\ \\ \\ \\ \\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\\ ' d: ·; &gt; 05 5 st Γΐϋ: O · / Ο. -Λ ·! 'to aisoot yv ^ iXidii lÍ dy: Sy- ....... ao; d y'i &gt; &Gt; o: 8M} &quot; ..............: 1 p1 '.p lo O ........ o a: o t OOS osodoa db qy (1), (2), (3) and (4) and (4) dy.V.iivv òy powder and fo, br.i C · ydOti qq- v ·········································································································································································· Oli laito; 1: 0.1: 5 :: 0 .l.o.r. d a:. ::: d .. · qy.iyt. oo yy oldlao vi.O t aoso y sipl 0 'ip; i and d: ···: lioi 0 'i &quot; and v i f i d d f o o o o o o o o · · · · · · · · ·. . Amino Acids: 50,000 to 50,000,000; ;; And; &lt;: i: o; op iiy. · '; The present invention relates to the use of a radiopharmaceutical according to the present invention. d &gt; .àv.t y: .11 la; 1 &quot; &quot; and &quot; &quot; yyy yyy.r · 'Sr y: · Cyt lia cx s: s pro CM · 0 ... tod} ....: 11,0 ΟΙΙ, Ρ.Ο; 1. 0? »: --- (0 and: ..... ao ..... 1: yy;: d · '' -l • Ot d tò: 'Ο' ··:! Iy: opt .0; ν '-θ'; 'θ (. ···: y; 0: 0 r: io toç r-lX-y 1 to aror 1: 0: y.yyyyyyo y y; The composition of the present invention relates to a process for the preparation of a compound of the formula: ## STR1 ## wherein R 1 and R 2 are independently selected from the group consisting of halogen, halogen, and halogen; , and (c) (1): (1): (1): (1): (1) The d-dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt dt Eitto ili OdM 5 S; i> g>: Oi .VO .1? T and y; (1) and (2) and (2) and (2) and (2) and (3) and (4) , and p-r &lt; yyyy: O;; and y): &lt; and X ioy liter r: d: '························································· : rs 0 ariorslri ιιι, ΐιϋι sírto {22} id; ot tt and Cy i; yi: ΐ a poot: o. (81%), or 3% (2%) of the population. spin and y ·>: 1 ardqa: Ϊ &quot; and y: [li; : yy y.:L .1 and odo. and y yy: \ * - 'd' ·: ·. da sst. sdp: t: assa and y. o · iOP c · S.yy and ...; X4 dr: pOptl ..... boot ....... Hi: 0iO &lt; O d: dlppdM [3] ao; aitqa · pp yuy p; r · o ·; (i.e. 0 The rotopi i ct ΙΙΙο'ρι ΓίΟ indo d. .8. \ s' .0 \ d: gives -. . . y ispo V 'V; (i). Î ±, β, Î ± 1: 1: 1: 1. : ·. v. i .; Λ ·: il srsm: il. yy and idro-aa d: -d; soo: po • .s · 0- or •: x! the &amp; 1: r yyy {il. and to λ qc di oo to Ota 0; 0: 01: 0 oilsi .0; 1 dl yy yy y y c y i. roo r. .i: O: ·· ·; ; ta (s): y: y: y: y: y: y: y: y: i, p and p: p i p i p i p i p i p i p i p i p i p i p i p i p i In the present invention, the present invention relates to a process for the preparation of a compound of formula (I): (i) 0, 2, 3, 4, 5, 6, 7, 8, 8, 9, 10, p C ta ta 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33 33: • 4B κ <0 and a .: 8333: 0 v 3bl: ciac: ataa ais • G: apX • 3 bl-3 3; G-Cl 1: 3 CO 3 substrate; 3p G-: 3 scries Pd: H ca 3i 3> a cibo ca: bi, '0': 3 · v '·. Λ · · and 3. A sspara 3a b a c e 3 3 • V ': x3 xy.G:; &gt; p &lt; a: a. 3 to 3: 3: 1: 3: 3: 3: 3: 1: 3: 1: 1: 1. (3): 3, 4, 5, 6, 7, 8, 9, 9, 10, 11, 12, 13, 13, 13, 13, 13, 13, 13, . · &Gt;·; .303 to its o r ter abocaa V: '': '' 3: Π: Vb- \ ', sbi J sa: a. as follows: Spsu 3. -G33 ac C-3 -mp fM t-1. G: 3 reet ae C GlvhG a • 3 ta; X Ο: sa sa '' '' '' Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο. 1 ac: l.ca: d 13 3c i.sys 3 x 1 0 c 3338- a ah aa: • G àç 3 &quot;: i'à alaar &lt; 3333, a. Çk 3 &lt; χ: ii. ϊ tea 3 1 ·> 333 cm í Q----------o o o o o o o o o o o. bi-G3 &gt; aisatl 3:13 vi 0.0 3 3 -3 3 c 3 <xib .: .11 ia · s: .pcsa: O -ts b h Po • Cb d. Glu aq. G CpS Ge. 8. G G a a w. Çp i &gt; : ab) la YÍ ·· &quot; 1 &quot; p. G · ΐ sar: lio pulls Paa aas a a; 03 Sapsaavt 330 ee M V 8, 3 aeraa i · a paaaa: ϊ < The results are summarized in the following table. : βCl-dβ3 -:; Λ '. 83: a: a.a ;: aiiç ϊ. ' 3: 33-33. ; s u Gt; CX.3 b- of 3-0 GVG: 1a 0: 3333333 3'ii: a · · i · .0. 3 '. 3 β: &lt; (cc): CEC s 11 '3 31 abc X 8 - b bar aaai': 0 - £ λ £ b csa - c3 - - - - 33333-33-33 r Cd-SH? G 3 G x. 3: 1: 1: 3: 1: 1. Î ±, β3, β: 5 ashes. '' 1 'Λ>' '. ··. ala bavisi bar el e; a at 0 ° C Gi-C GtOG hGG; 1 v '< Example 1: xtb psa CHO 3 &gt; bpx. The invention relates to a method for the preparation of polyethylene glycols and polyvinylpyrrolidone in the form of polyvinyl alcohol, polyvinylpyrrolidone, polyvinylpyrrolidone, polyvinylpyrrolidone and polyvinylpyrrolidone. 3: 3 to 3: 1 ssa abPib 1333; 3: SCIENCE: G to a '3 3 acha ce 3 ar 1 f i a χϊΐχ a ic a. 30.1 'ssah s sssss iiu &gt; pesr csisr. b. 33 ai: face to face; C A S A S S S: coss a cie saasdass id cb rrsss 3.GG33: iai color; wings:; .b. a-b. · 3 air coras -recaa lo 11. '3' C; aa CS .ac t 333 C aO a • 3 0: aob ta Π 33 O -> EC 3 '3' r; r; r; a -: ai - x - b.i b - s tb ..k.i. 1.0 ΓΚ3 3 aa:: s < (5 hg) dairy. &gt;. ¹³C. G.l 3-3 b-OIC of s) C: Ethylpyridine; :::::::: t £ 1: 3 ... rs. Aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa (I.e. G: 3: 1. .3 · &lt; EIA pc 'CG &gt;. 3 G cdisp dk PCO: .ssar Pd •: 3t G '; &gt; -> &gt; CTl. b: 'Õ a cp st aa o: ao pcsc. 333 CC. b-330 He; : 33 i. ^ pt} .......... abi; Also . .b: x saa &quot; cii bêa scasd a ...... l: x 3 a ca a i 333: s: do: ....... asa 3 J: 3: bGG &gt; 3: 8.3 &gt; &lt; / RTI &gt; &gt; &gt; &gt; · &Gt; ' . bc: .iCs: G a sprue:. as is the bi-asbs. . ·. .s... . rb sb.r .1 i3G becomes P S: Ei b; tb G 'Π t &quot; thi. a. VCIB a .13: SS., S.D. 3: 13133 b331 Gb &gt; weighing ca 1 bb ·; to 333G. x \ · &quot; :. . asara r C33 CGb: p xn. cir: 3. 33> 13 secs of bis. .13-3 '. •••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• .He cccac: ti · &quot; nb. 3 'CIO:; Ρρ: ορ: ρο ...... ybj; of .Hbb; IH1, SE: SE3: 3 adsorbed to pbbGix I0; csssaa laalc .π G- 3: 0 MC 3: p: COOà i c; daacts to asparagus: vdC: CSC '. 13 cc calssssss.ssd. The invention relates to a process for the preparation of a compound of the formula: ## STR1 ## in which: p: scacccc Cai .p &gt;:u;; parts • ICH.j. shat of it 1 aa ....... HH p £ cSSis ϊ ϊ ip / sp b ': 33.333 3: 3 3> : 3. : 0: 0: aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa 333-3-3: 3.00 Gly-3-ol: 1: 3 GG G; &lt; Ehta: 83,383.33 from GG'33 &gt;. -3: 13: 3 hexanes; , 3.3, 33: 30G, 333d '. 3vb 1H sssa; P; air dessat: rs.s i.dc c sosss s:: sc s isa a η ¥ j. P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P P &lt; RTI ID = 0.0 &gt; PP &lt; / RTI &gt; &lt; / RTI &gt; · -Ast r Pt rtr. ' (i) i i i i i PP PP PP PP PP PP PP PP PP PP PP. Hi, PP, I, IXr-Xa. r ΤΧΧΧ · d ·············································· d- f. eur-lex.europa.eu eur-lex.europa.eu p. tXXcd iXi ar. : .PJ ΡΤίΡ, Ρ 1; Clamp I I Γ ;: 1 - - ¾. I χχ Pds, p ΡΡΡΟΡ ΡΡΡΟΡ β ΡΡΡΟΡ 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1. C PH₂O: C P PH₂O: C₂ ;H₂O: C PH₂O: it will give £ 1 Pt paat d '' '' '' '' '' '' '' '. ai i a a pu r íu PP :; Pp. pPiPPiPjpi ii ·· 'So .. .P.v .. ... .Ca; ρρΐρρρςρρρ ..... ·:. ¥ · ΐίΐ '..... PP': Ργ> · P PP Π ci ¥; for example, v; c-x td aCl Q + a ppppp. (1: 1). X; &gt;1; i.e. ..pppo pp tparr tiç; XI c j c c 1 t> W; j PPC; . &Gt; r :; tc &gt; \ P '; aP. pd. : a t a :; (i) PPi QVi: t X; d d; Υγ pppf Xdo dictate: í dcd l. · Χ · d pp: S a: · &gt;! no PPC . Π; # ¥: i: IvSX • Ç;.; c and ....... ii:!;: dd: ...... &lt; Pd: P? Pppi XXZ Pi at i-il &quot; data &lt; / RTI &gt; &lt; / RTI &gt;; -d PP; : rp: t £ prx r * p: · ': · gt; PP-PP-PP-PP-PP-PP-PP-PP-PP-PP-PP-PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP pp. 0; Pâ, â, â, â,,; ip Civix ti 0 PyC'a s'. v., vCXc a; • rvtic da ρρρρ; 'Pta ari c' · i .dc.l ss at; of t .PP P Ρ: Ρ; ΡΡί} PDP .sv d .s. P X X Pp. S ': X i. . . <d. ··. S.SS. ·; ¥. &gt;. C: a .: iYXci # pcp # xJ aà 1 U.tpp o aaarentc; V.y. &lt; d &lt; Ç T; &gt;::; pis prppl: prpC # 1. ii. 1. x atip ΥΛΥ # i # .ci b; Γ X: '& ic 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1. S and rhexe: Cpd. .11 to &quot; : ¾ ta ra; (I.e. s. cation PP; C Yd PP χά P d P P: de! PPSP t.a.n &quot; 'λ' 'PP, pp. ppppp:;. ra-aip tPP: PP; ci d, 1. Ol OlVi p xao: rid;!. Txiii vi; ..... C.1 tátar í '< ·; dvid! λ • X fV: Ux οχ: X C i i, P 1 rii '... p; P 'Ρ P; t; p upap: of y .0 ¥ li Oiyii to iPcasiPit: ·; The following information is given in the following pages: PP:

Saqnapp:. the year-to-year changeover to the year-on- Eur-lex.europa.eu eur-lex.europa.eu iV ': iii.C lapa · cd t # C ·· s arip; Typically, (i), (ii), (c), (d), (c) and (c) : aa atara iv iv-1 &gt; ,, P P P IpOP; P1 rPia p a t P; PX 5t: p P; Pt 2: D # 1: i; P; pt: tp ;; to give · 11 ;. the PP: • Ί11 &gt;. 'V. , C ...... # p p pa t radp d P tPP i p :; X ρ Π a itPP; ; c.:. | X; Χ, Ρ, ΡίΡί ida dai; :.... .... .... .... .... .... ....::::: S-itiPP; .delta.: 1 to 5% by weight; PiP pX # β # .Πχ &gt; ¥ of PP:. (2-methoxyphenyl) -1-piperazin-1-one; A method according to any of the preceding claims, characterized in that the method of claim 1, further comprising the steps of: (a) reacting a compound of formula (I) with a compound of formula (I): 0 PP? idividdX a :: P P: ppu paibil iplpdp; Dr Xá d ¥ c ici ity: p a.apari.aa:: t; ai ... i> iCv \ d op r papear opipp; s: ρ.ρΡ.Ρ; θ: Χρρ: .ρΡχϊ ta .;. aPrppP: tr Pd rlPippíp ρηχό;., Ροη dpppppipppp P; pS pPPPPpiS PndPdiP PPPP; ΡΡΡΡί Ppippyp: p pppxpp; pp &gt; ,

Id.

Prarteara f aoe &quot; the real angry. by PCaC Cl)

Pa rttl T; ooa: 01 gdd • O; to t; t 0: 1 1.00. V, as shown in Fig. . iV-dd) where: VVC:: 1) 0: 1). Asparagus was the first isolate of OC; 1: 1). The title compound was prepared according to the procedure described in Example 1. r Idd ds ...... <1: Islam MO: WHO ..... Cio .dial ms: v OC VV islll siidi 1 ... .da ....... dd) S .. S: td: i - - ·; i ... ... pS, S: V &gt; : ii &lt;1; V &gt; &gt; &gt; &gt; VcCcC O) s- ·? · _> EXAMPLE 1 A compound of the formula: t: ar: ···; dl das a · tos • V and; OS id) &gt; t-toaster C-Vd- to 4'or. ds = 100; d CCC &lt; 0 .. · XCC CC IMS 13.0 C. V M :: s; : G dt: -¾ poi)): 0 i 4: v} s VC ··. I ottrrdos MO BG ί'οΡ.ί dsIG pray? the .V CVC d &quot; dd.id .... :: P ixCi CC CC 1.: 0, rra soo: ao, a dpã lo ... v V: V; ...... Cd: j (;. Md C 3.) &lt; d. V C C a C r r a Ms Ms Ms Ms;; V C 'atoa U): t aroslraar; 1-0 10 Ss of all; tis \ -p); yes. c V; WE ARE t | t 5 s o. t a OK. s t CCCC 0--V dc EC Md ors. C dt d d d d d d d d d d d d d d d d d d d d d d d d d d d a &quot; 1 &quot; 1 &quot; &quot; &quot; &quot; ida ': &gt; (b) (b) (b) (b) (b) (b) (b) (b) (V) (V) (5)). o '' t t.rtso; doa di saodo sota cl.vi is t. :) is · .0; A · x ... t SOMOU. 11:.:; or, The compounds of formula (I) The invention relates to a process for the preparation of a compound of formula (XIII). to O) to D take; ; 1: 0 to 1: 1. s. to the do · ..- V. &quot; i 4 Ot. id < to attriaot:. V C C CC C V V ‡ T ‡ ‡ ‡ † † † † † † † † † † † † † † † † † ttoto; .tO; ) r 13 :; from oCoC, ..., ..., ..., &gt; I sis) &gt; . x.d.s ....... v. &quot; Eur-lex.europa.eu eur-lex.europa.eu . Λ. . . . It is: it sounds like the one ... ai ........ to jam Ci-CV of the .......... of the attractiveness of the. . Vi 'to rsad :). . (a) to (c), (c) to (c) i.e., i. .......... iCO C C < c. : C: D: C: D: D: D: D: D: D: D: D: D: (3, 4, 5, 6, 8, 10, 10, 10, 10, 10, 10, 10, 10, 10, 10, 10, 10, C Ord td; vv.c ViVCd rotates; The present invention relates to a process for the preparation of a compound of the formula: ## STR1 ## wherein R 1 is as defined above. &gt; 1) to: 1 to 1 p: other; : i.ii - aii to::::::::::::::::::::: (d) tb______________________________________ tb______________________________________ tb______________________________________ tb______________________________________ tb______________________________________ tb tb______________________________________ tb tb______________________________________ tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb : a; t PMITIM C: i), t.asrbá:. ts s rts: tlOtl: stii. sado. &gt; 1 il's d dv.;:. I-dõC; ; to a asa r a rd r v d ti; ): 0: 1: 1: 1. Cdi:: ir a; i d: i. a. po: y-, s ·· r \ ld.t to ........ to oc ll lt: V να: cc c ·: · Χ ·· .a: ·. - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - i &gt;; ! (i.e. .VV: δ;.: V; '; The CCVC dC i C VC i tract is not a a i. to the cvo cc cial SABotaí IS; shovel to face aa xt · 2 λ vs

Pa UISSC ξ 1}, ITP: p: Csaarporoao Π F t, color tot vane ara pfOPPS &gt; enPP r aocl} PP cot crowding AUA abacctaaed, shallow CDA qq optao, duck: sweetened of: e ásroeavb cat herein ooapasacttse al . otota pLs appaaa-P popoís ae tote-eae · $ cd, · c arao css ae eoaroric tac ;. .ia.ge.aae the o.occia (go ρρρρρρρρ cesium piatpop orax Estia the wool {ίρρ only the i: U aotaroa &lt; -'oPP p · p i aaoaaa; IJI i • Co, px; paxít dcaui td.r ... íappqppd .PXÍ2 V pa t :. SAR would ciiilPa: until the CPM:: the .s '. iitda read AA ay ci.t the boy DCP: rt r i XXR .: &gt;' IPP IX Xr x .t px i; 2 2; P22: iV; 2,1 aa to Pt ox.xv. 2 Q.0 &lt; a &gt; Odette's point of view::::::::::::::::::::::::: {{{{{{{{{{{{{{{{{{{{ 2. The CP: (4) P PC d; aa 22 2 .- s s 2: s SS: ·, d d d ad ad ad ad ad ad ad 2.2 2.2 2.2 2.2 2.2 2.2 2.2 2.2 2.2 2.2? > 2> 2> 2 <2 <2 <2 <2 <2 <2 <2 <2 <<< ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ ΧΒΒ CP CP CP CP CP CP CP CP CP CP. ; ••••••••••••••••••••••••••••••••••••••••••••••••••••• 2 •••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• " (a) and (b). P oc aso:::::::::::::::::::::::: ...... ...... ...... ...... ...... ...... ....... .................... Aa It is important to note that in the present case, s2 :: 2 P t bi bi. In the case of the invention, the invention relates to a process for the preparation of a compound of formula (I): (a) Compounds of formula (I): (a) Compounds of formula (I): (CDCl3) Î'(CDCl3) Î'(CDClâ,ƒ) â, C.àXd uu ipO: b V ·. '. pot PP atooriá tiipdQpg. P PC v. (c) OPC (OP.1) will be ready for air-to-air operation::> .Cpi &quot; dd ..... ai pd ο ;;;; a 2.V cdr ccpcia . aa t ·; s 'Vs' 0 ap p Γ.- X. a. ia: a la: a. : xXpc.iPi. â &gt; The following table shows the results of the analysis of the results obtained in the present study. :: a: p cl t S.2 atcpac PPPO &lt; &gt; 2.0 &quot; 2, 3, 4, 5, 6, 8, under denada &lt;. P ac p: ¾. OiB at tfig ppsX c ap: Cp CP cP, p: P a. p epio 0: icaappstoa d 10 u: X :. : U2 'X;' X. 'cpo. open to the paca qua P: idpii: i dCP iaaa utpr fa rpgp dtf: 2 = ar a p t P-itpaa.iosa i P Cgr. CiV. to aa ac idp aaa:.: i.ca mop; 2. oo o o oo ..... MC ..... i ' 9 ^ ...... &gt; VCV VCV VVcV xxoa a. PC OC ....... (et adq.) X0: C tl Ôx XXU pow. 2 xvacta Ptot et al., 1540 from the supp., Pp.: S-oc ... to ... · &gt; / .X &gt; .c Xviidd U X2>: .i .. to air: Uxxa o SC B'Cid ibu = 2) <: &gt; •. â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ Pd p. di PPO.P O 0 ss, · ν ia 00; (a) the following steps: (a) reacting a compound of the formula: i.ip oUoto pd vcccpti &quot; soocttooit? ato aac as isspoe • 2 &gt; . i v: a Idvpr d v; d SO 2:; The. 2. to 2. XIXX. (X, y, x, y), where x is the number of x, y, x, y, (X, y, x), x, y, x, y, x, y, : U. 22. A compound according to claim 1, wherein the compound of formula (I) is in the form of a compound of formula (I). Okay C--C₂-C ·-C v-C de-C de-C de-C de-C de-C de-C de-C de-C de-C de-C de-C de-C de- · Χχ XV à c itX: Ci ra (iaol, 0222: ·; Χ X · ρ :. '&quot; iv. Budget: t, 2 .X. , sq -v 2 Ss * '': '' '' '' '' '' '' '' '' '' '' '' '' '' ' (2) and (2) and (2) and (2) and (2) and (2) and (2). (1), and (2), and (2), where X is the number of points X, X, X, X, , S, C, and C respectively. the cot is the i ii iViX.aiiV p i plt.Odd. for example. The. the following is an example: V Ρ'ΡΡ 'araactuated U. X.'; dtttbc ...... gives: air rrc the goose: popdoa cd. acosta • V .. S. · ____ V.N ..:. 2X. The invention relates to a method for the preparation of a compound of the formula: ## STR1 ## wherein X is as defined in formula (I). . of the title compound of formula (I): ................ ; 22 ° C: 2 ° C; . 20 sdaaaati titan a; (a) (b) (b) (b) (b) (b) (b) (b) (b)

Idsrsser. (36) tt aat 'Ç - · SB aOSld d, aã as ci ··· ;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;; and r ·. •• ircpp:., A: at 5 Uu.a.i. Xa ian M: i na. donates 0.8 C OS; na i. · · · · · ·. . t aaert; .1; S I. 11: - G? :. . aas; Xyl • * S · · · X · &quot; 7.SV, &lt; pAi tai t i ast C · Vã p St P ytl · SOM of the flow to the .0. X-t-C &gt;: P. air to .¾ ·: s; ; r; A. TAC of the minutes: • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • oét. / i. aq: aq; i Pu Pdu € 5¾¾: 001: 0.1. β: thiol; Fraction: ata st ti eido ff P p p V: j. a if * MM; Then, read the following sections. at least • VXis a XV: sar Cl ti os os X X X X X X X X V;;;;. c: P. Thereby the invention is carried out in a manner similar to that of the present invention. CU c.0 a i Via V. ça l_ã V áT: X ialaa •: M. iX x l · .. ·· iã; The results of the present invention are shown in Figures 1 and 2 of the accompanying drawings in which: FIG. ; air to 1 dCBC; C G gives '1': X '' ''. • d: t: &gt; V> g: V; 5 to 10% by weight. 6 Is) • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • x, v, c, d, e). ...... j: Pi'1 ads d _, ···; EXAMPLE 4 OXOr CO: . and G iPl is.O Mi \ iàv; , wherein: (i) '' '' '', s Md a a; ada: ¾. cSO vi: i. SCS: aslaei i.n.òy: x. ' jTip; Rf: 0; Ϊ 'Γ; 6a. PO i ;; e.p; thi; Fig. ça aà vs M. y. . and · &gt;. ,· OK; ui a f 1s. i XP ia. pa < The composition of the present invention is shown in FIG. t .1,0001: aã and XaV p. a a a :: PPix · '; ·: Λ P P X s Or dl il i XX li li i ;; a. 0: of st .. · ΡΡ! Ρ: dt 'and Pib T3 to act UlP i. P Xã 'Ϊ toi.atá: d U χΡ ;: .30: .1.¾ iní: OÍ: θόρια; Soc. Cit. Gtt; adó. , ························································ 01 'ΡΡΐΧ:' 'st.:S tf? ooot; : X, X, X, X, X, X, X, m.p. -a-Vk. . the catastrophe of the catastrophe is the same as that of the catfish. (a), (b), (d), (c)

Qaar ta f aaa &quot; In the case of the above-mentioned claims, the invention relates to the use of a compound of formula (I): wherein: X is SO, and X is SO, and X is SO; 1 to 2: 1 to 1: 1 to 1: 1 to 1: 1 to 1: 1 to 1: 1 to 1: X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X- ), And (6), (6), (6), (6), (6) and (6). X: 'ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã ã t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t. ........................ :. The . ·. .: SS: ana ato v PP CP; Î'C; A sis of the s f fass osssaai.r o f: ar GG GG ias a: a is. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • •. at.;:;.; the VPP: X Vi \ 'ã M i and P iV san se si to 0 :: to; ia CPP P Ti VPVi of the dCs 0C V .. 1 X assay to 0: this PAGGV. Pi χ Χ Χ Χ Χ Χ PP PP PP PP la M M. s May 0: Ci SSip. &lt;: &lt;: &gt;:; · Yp .o: ... MãXã · '·' &gt; M:. c. Xt Mã PP iorxp ce &lt;: SOs: da vÃ:: lã 1 and pg n. Iat p ti V. if dat a tatasa aaa: at CP Ci i.: ·. Οχ ..................... ;; v v ..... ..... ..... • • • • • • • • • • • • • • j j j j j j j j j j j j j j j j j j. ; . : Î'p: i '&gt; Std i nnt sPasts dad: a pot s PP panao; s a aa; 'isitsasitst 1 ···· st; : ·· · a tas jfatad .; a d; a s; χ · .χ; .. Ρ> ν GC &gt; TP:% VCVHPP C: PP to G. of P (4) and a. i.Van • Ο; v • 1 s Cv pXiXp p. ssas; tOs; The·; (Μ;:: P ((((((((((((((((((((((PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI PI (2), and (2), and (2), (2), (2) and (4). (a), (b), (b), (b), (b), (b), (b) and (b) IpM 0P> rias of the CPV: C: Cx Cx: St: t: p; aaf 1 Pi ss v v Pa Pa: cs: pd :: -a. : S: S: S: CS: S: S: S: S: S: S: S: S: S: S: S: S: SM: M:::::::::::::::::::::::::::::::::::::::::::. ; • PP nsto f ãP: d 1 p: X ;. d. ma s,., d d 's p dst sosass s st:' s y ·· '' '' '' anosra V .c. dst ) in the same manner as in Example 1, in which X is as defined in claim 1, (X), and P is the same as that described above. A 'PO 0510: &quot; A &quot;. Eooaaa do: q &lt; q 1 st asia of θ: θθ5'ρ «Μ; 5. . . . . . : P: s: .5. 5 5; The invention also relates to a method for the preparation of a compound of the general formula (II): wherein R 1 is as defined in formula (I): wherein R 1 is hydrogen; : ii50 idillli vai> · '; G: · 'S: CÍG Et μ ·; . q a- È '. : Î »max 55500: 5 05.50. 5: 0 is: 5: ST 0 55; 1: 5: 1: 5: 1: 1: 1: 1: 1: 1: 1: 1: : 0; Ei, t v;. ': T: d &gt; \ 1 · \> 00: 00 wing. . -I: pATIA 00 i :: ·. 3: 3 00: 0: Ώ 5: θ: ΡΟΟ, s s ·. the Ilidi and Ea. dsV? P?>: &gt; . A ': y.': ·. '· Õ; A A A A '. (a), (b), (b), (b) and (b) and (c) 055'p 0: 5: 5: 0: 1. i.e. 05: 00: p: 55. 5 &quot; 55: 0: 0: 33: VA) G: 3. W. o ·: d: · 1 Sl m; q. q; a..aO: 0: 0:.: 5050 ::. and the 0: 0: 0: 0: 0: 0: Fig. p. EOEE HO} laic oc pp pp XKWO; c.í.aic dpsoipotsoa ieehadpa Εοο. c. (I.e. Î'-.i; 00θ · &quot; 0 is. aa:; A compound according to any of the preceding claims, wherein: 555 connected to the power supply. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • The ; ooOOo Π r .: i aoiOd ;; 5á idogi -i? : Loflig Aid o: 10 ° F 550 ° F: 0.8% H 1.1% C3.3. a0: 0: 0: 0 0: 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 to &quot;'.; 3aA '; al., Cl. to give the title compound as a colorless oil. &lt;<lt; &lt; or 5; (I.e. 50 BODY 0: o5 to 3'3.ci 50: .50000.0 içl: a po: q p. δ 5 Γ .or CG; oleie 5'-O '&lt; â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ · The GOO of the archipelago: 3 d - aoo • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • GO, as the X-Γ Γ '1 1 1 1 d d d d d d d d d d d d d d. gxq: idj. thiyo: IdOi} praeánta aaO Mv: ....... id ola ld GIG ..3, .3 ... ...... OEM: ... a: | 0d: 5C: to q.avd qi t r. ': Oto ...... porea: oeoa íoaola ο? ;; Ca Ca Ca Ca Ca Ca Ca Ca Ca Ca Ca Ca Ca Ca Ca. 13 i Ea a · · · iq a .Td. A. to;; 0050 v 550 c.l: 0 5 ..: 0? 05: 0: 055 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 ·. · .. · s · .. c: pao: os.ir gives:: qa oi 05; Ooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooo i.e. 1: 1: 1: 1: 1: 3: 1: 3. 55: 0.550: Î'-O-Câ, Î'.05 &quot; t GC: s05000 and d- &gt; The AsV AdV 3 ............................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................................... 1a, 2a, 3a, 4a, 5a, 7a, 10a, 10a, 10a, 10a, 10a, 10a, 10a, 10a, G 'Gà 1 3 CG C. . A · .N Ο-αΌ,,, Ό Ό A A A A A A: 5: 10-15: 5 to 10: 5: 5: 10-15: 1 to 3: 1 to 3: 1 to 3: 1 to 5: (1) and (2) and (3), and (3) and (4) and (5) and (5) 5: 5: 55: 1: 1: 3: 3: 33: 5: 1: 1: 1: 1: 1

(1): 8: 1: 8.45: 5: 53808: 53340: 00 BB-Cyleil X 53 334 0 0 3. 5: p; S 0:44 55 0:58 8- GO 8: 1.300303: 0 03.3 8: 585 0 58 llScope 300 8-8 8300: «443 OD 8: 0088; 8> 538: 08430: Ei .; 3:: 3 3:: 1S3C: 8888888883 83:83; 383 :, 838: ¾: .3,3383 01,030: 8333 Od.G $ 8tCOCO 08: 838 85: 8 535.53,3,1,83883 : -: 838:: 3: J3: 8; 830 83303: 38, 550, 88883, 03: 833, 88045, 1, 581, 818, 1011,0353, 0: 0053045: .f : 8: 83: 1: 8: 8: 38 83 810838 -8 and 88838338 888 383833888: 383 888 0 38 0 0 1055: 00 8,418,88: 830: 1,830 03 8300 83 3: 8: 8. 8.88.88; 8.88.88; 088.88.8; 08.88.8; 08: 38.88; 83.8; 8.888888 838; 838808.38.3: 335383 8388 8; 8 '; 83.08; 8.88.88.88 '08 08; ..

Biphenyl-3-yl-propionylamino) -benzenesulfonyl] -amide: 1 H-NMR (CDCl3, 300 MHz)? d® C03d3S8S £ d8 83 ddittSGlDl CC '(4 5) 33 83 8 5500: 53 Itl V8' &gt; 88: 0-38; 83.8830 and 85101 .1408: 3: 8; .8. 33 88Olp: 33883 .8 3385. 3: 33: 8,838: 3 EO r'n. 830: 8 3.3 38 3388: 33: 8: 3 3380883 1 .80 588.8, 0, a-80, 455, 5; Sp: 0a: 5.58, 83383, 5,300. -0.0.0 v- V l.vd 0: 8. 551: 0 838: 388? 0: 11: 8: 8 8.3 0308 5 0: Ò: 0. ; 000 li i. 3 0 θ8 ?? 8ΐθ 00; 0: 008050. &gt; · 'sl ò · &gt; 5.500 '0'0; and g 3 8:. . C- to V? C: 0.11: 3.0 p3 8.3818; N, 5.51: 80; 55088 ': 5885 30 153 O 588803; at 0 ° C. p 08 OiO θ ': Ο :; ; d d; 83 0 0: 00083 88 8: ν''1 1 N.0. . . . 0058 ..... 0: 10). C0 .i. 0 380: 0 ': .1. &lt;% 8853 5338 0: 0: ..... 3355 00 ;: 838:: .1 :: 8 0: 1: 0-0 :): &gt; &gt; '- a 88: 3.3 38.3.8; 8 ;: 3 0.8: 3: '; : Î'8:38 333? 033 P; 3: 001 0 8 1 0:83 5 3 8 PIE; 1 v 1 i. 55358: 5 '··' s ··· 'lp; 3 2 8: 0 38: -; · · - · -: pp. ·. &Quot;. · I. ii) 0: 3: 8833,8,8308: &lt; 0 0 0 0.001 1: 0 8388; (1) and (2) and (3) and (4) and (4) and (4) C0.838.38; I-6B s. (I.e. 383 V · 0.100 a. 30 .0 '3: 3.v'0:: 0 :; 0:83 0 353533 :: 3,330: 33 83: 533: 110: 5: 1: 8: 883: 838: 338; 8388 33 3.8: 1-io-0i,: o 0 ·: '0: 0 01.'; : 8883: 3 .038 p i l;? '&Quot; 08388 5111 s ..... 83, DE-4 C6. -; 0.83 (s, 3H); 3.83 (s, 3H); 06.00COC. ·. .0 0: 0 300 '0000: 0050 i.d, at &lt; 3 &gt; 88 &gt; ·· &gt; 0.0001 Âμ: 88300 0 to 00; 3, 880, 0380, 1080: 38; an: 5: 5.3: 1 8'C; &gt;1-ΙΟΙ; , &gt;: &gt; 11 808 00 &gt;:88;s; &gt; 8, V 8.81: 0 0.3: OCE • C 0.1. 0.3 8: 3 or 30:?. &Gt; γ ··: 08353 0-008 0 to 43353 δ 1: 1.03: 1.03 (β3: β3: 3033) 0, 333, 83, 3, 3 in 8, 1,8,3, 8, 0, 0, 0, 3, 8330, 0033, 0.58.5.388.3 .14538453 0 ΪΕ / 88 88.: 3: 333: 333: 383383 3 38 33.88: 3 (i). 83 83.33. 0 11 80 35: 03 to 03.5: .5535: 33483 3,830 535530.S; .53 3 O 43; 8 838 Op: 88 a. 111.33; 0 8: 3: 8: 8: 8: 8: 8: 1.88 CO.I: i.taa. 3.83: 0 :: a .00 lotion 5: C;  € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ3: 3.88: 00.008888 00: s ..... 0: 33: 5 ?: to; 33: 30.83.13; Ò 0 0 00 ..... i. Example 083.1: Et.5: 8; .031.050,4. , 1: 53.83. 700 ·: Y00; ϊ. of estrus 83: 0 :: 3: 8 o; 03: 308-300 05; 838-333: 5 :, 1: 83-0; P: 33: 00 3 "V'8?: 8.0 to such 0.83? X8? 8338:. ΐ-, -8 3 3 '10 Ç · 1.3. 3, · 4 p: .388 s ...... ·: 3 0 0.00.: 1 01.030 3. 0. LOS 85333; 0 5,058,35: 0,001,003,353 gip. ·: 8338: 8,0000. 8,333, 8,383,808 O / y to p3,3; : 11o.u. 01-01 poo ΐοιρρ .pipi 58 '008 30530'43 5 l: C 83 83 0 0538 55: .3.35: 0 3.0 ii0: 53 0; 35: 4.335: 35 8.353 35? 8 3' ( i ........ 'vi: 0.0: 11.0 34033: 3? ..... 8.0 ·: ··························································· ... (w / w) 01: 30: 4.3.1 55 S0: .5 / .38 0, 80350035 5 08.5 3: 3: 3 00.3 .830: 8? .00 '4.1 COE 11.1, 05444: 10 · 0 0 3 31! 0 4.43: 0.5; 00: 1 55 8585 07: 40 CaptO D-: V00) 1.05: 5, 85, 11, 10, 10, 10, 10, 10, 10, 10, 10, 10, 11, -5.5: â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ4701 (30: 53 1 3 5.55 dO? 553? 00: 11 43.81530: 3.3: 3.3 33. 5, 855: 5.5: 533: 0 5 3 5. 818408 0? C: 8 300, and 00 -0 0 o -o 3: 583 0 5 :: 453: 335 55,843 5; 43,0-0: 53,335 3: 553,3553: .3,353.1 838,: 85: 345 38-8: 3 1: 1: 84: 1: 84: 1: 1: 84: 1: 1: 84: 1: 84: : 033,000 DD to (; .0 0: 0 .s. tb______________________________________ tbC 335040 tb______________________________________ tb 0: OCI- 11.11. .0 0 0 i: Ό 000'0 0 aa :. 88 355 C00.40 0.8 0.0001. 000. 0040 03531: 30: --- 8403 --- 83 35 p 34:: O? 4 5 from 9: 01: 05: Ò83. 4 4: 3-1 a g ÚC 0043 43: -p- or i-00 · 1.1185 0.855: 5.8: 11; 0: 1: 0: 0: 0: 1: 0: 1: 0: 1 0: 1 0: 1 0: 00: 8 EO-088 5; 0000: ia 3450 ::? 11 '.....: 0 7 · 483 ..... 111 33 0: 85853 a e ..... p?: 48; 838333 ( (ii): 53 5 '010 XX 3.3, p 0: 0: 00 00 · 0000001 0 aa 5388935 5-A, 831 t 0-0 ': β3 · Î'· 3581 380: 0803 3.0: â J ¥ 500: 0: 0 1.0 01 00-0 8840.00 0..i 53: 7501: 1: 4 OO: / 35 8: 8S5: A compound according to any of the preceding claims, characterized in that the compound of the formula (I) is prepared by reacting the compound of formula (I) with the compound of formula (I). ΧΧ ΧΧ ΧΧ Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí Sí: (x, t), where x is the number of x, x, y, x, - - - - • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - , 0 1> gt; 4 tt: D · SS &quot; XiXisOTriSi X..1. X-X. C f-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L-C L a a. , X ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ ΐΓΐ. X-ray diffraction pattern. r iVss v a v 0 ta .; XX xP0s: X 00.00. Of the aisb> · Pxxx i 12 ix: X 8 £ :::. t g S.C <5 [v 19 tb cit acid d) MC X td i a et. wherein X, X and X are as defined above; The present invention relates to a process for the preparation of a compound of formula (III): A compound of the formula: ## STR4 ## wherein: s ······················································································································ ΧΧΧΐΧΧΐΧΧΪΛΧΪΛ Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í Í (a), (b), (b), (b), (b) and (c), and (b) (CDCl 3)? there; (I.e. i ff at 9: ·· < X-ray diffraction curve. TL • χχ • it χ Ρ β). apd: x. x ': X <xxi tat' 0 adi; fst of ..... to XXi:; 5: good ta X: i! idctl po.L f tf. X a is X a; the saga 'f; X-ray diffraction pattern of the X-ray diffraction pattern. N. ogo · a i.t 4 d i pp · 10 Xt • X X: X: a- Φ a rio ·. ; Sd:: .ia. · · · P it. sso ia de cii olot .... ·>, x Sr or X X'p. the O and V \ f N: ·. d; ra t2 4 < X; Λ à Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ. ici di 'SO Xv r ·. V ', .. · v &lt; P: aaa. and a · · · · · gt; : Î »max. C) v p 1 a · '' L-t ·· '' i &quot; i................. The title compound was prepared from the title compound as a white powder. p V &gt; X: N; Xa Xa Xaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa vsài at. (1), (2), (2) and (4). 1a-1a-1a-1a-1a-1a-1a-1a-1a tb______________________________________ tb______________________________________ tb: X 1, X 2, X 2, X 2, X 2, X 2, X 2, X 2; ft. .· P; \ f. ΟΡΧΧΧ i:; · ...... C ...... UC CU X cat: vi T: X: t ...... dl c;: afi pCft X ..X. .X: ....... (i- x,; ........... Lota tfp &lt;: &gt; SX ..... &gt;:::: • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • (a) X-ray diffraction pattern: X-ray diffraction pattern X-ray diffraction pattern X-ray diffraction pattern X-ray diffraction pattern X-ray diffraction pattern X- The title compound was prepared from the title compound as a white solid, mp 218-221øC. 1 H NMR (DMSO-d 6):? X, X, X, X, X, X, X, X, X, Y, X, X, (1), (2), (2), (2), (4) and (4). X-1 X &lt;: i of ffOf. . XXX X already a; C 't tH o tO SSi Cf; therein i: t; X'-V1 0 r.i; X-ray diffraction (X-ray) X is -CH2-; XX: Fig. i. i. i. SdxS '; This pdx '$ ιό :: togada .iil La it 6: X j c | V: l>'; &lt; 1, 2, 3, 4, 5, 6, 7, 8, 10, 10, 10, 10, 10, A compound of the formula: ## STR1 ## wherein X is as defined in formula (I). 1 ···>: ···································. to ; X: Sr snaga: pp t 'Pb SK; (1): L 65 5:; I am going to do it. .......................... L · a ..... 11 · Β v .; ' D. i. XXI, Si Si .1.00 'ortil. r a. (i.e., X-X-X) to: cu> X p Xp tlia X't &quot; NMR (CDCl3):? Mr. sfób. tf. X, X, XX, XX, X, X, X, X, X, X, to: &lt; tt &gt; X Sr aec: S i a% a ff. to i XSXi! U a j a bsqbte r; :. : 9 61 ···. ··. V fiat:: ··· ata dt The FCM ti), s t. : S, i: i'X Ott:

c. (I.e. P PP · -. (B) and (b), and (b). P: T · t. d ax: P'i &gt; '&gt; Γ Γ C X X X X X X X X X X X X X X X X X X X X X X X X X X edCii; 0 and "; x <&lt; as to Ot. only. CD. at t of; to the basket Ppp. d 'd. et d te pP · rd a fixidC; &lt; B and e .00 d of S-P: fluid C: CCC d ea easa OCC-Cd C i e b c e; a CA; Ireic i. 0 ° C. xa faacd.Cia 3: 000 ': EcoC. • át 'p; P PV '? P; &gt; cP aosiocipa ·; and you Sd. (a) (b) (c) (d) PoJ • P e c e c c e c t i n tio n Optio n; (i 2.) &gt; ϊΡ t; ΓΡ &gt; P (ΡΡΡΡ) Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ. CCiS; 4 5d • b Ó &lt; y xtx.xi.4 of this saxã qapl; ICC d 135; donates dc -1. The reaction was carried out in a similar manner to that described in Example 1, except that the reaction mixture was stirred at -20 ° C for 1 hour. X o -. ··: - ·· PP p pp 0. dociduç da oc saaote Ιοορν P ·. and the exo d: · d d; P; Pd · .aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa ssidcsiae pC? P and d d:? .0. C 1 -C 4 -alkyl, C 1 -C 4 -alkyl, C 1 -C 4 -alkyl, C 1 -C 4 -alkyl, for example. CC ei d dc: s & iiSdSC. ............... P-i CpCCiCCC iaaa tt t 0 c · 4 ·. ···; P &lt; v, 'a x.a SiC Sd: ex.So pp. p P; Ό U ÍU DO :; ; Î ± X. axepa to 1.1 and f: easacoi. C:-C:-C:-C:-C:-C:-C:-C:-C:-C:-C:-C:-C :- as well as the <P iecad. The present invention relates to a method for the preparation of a medicament for the treatment of a condition in the form of a medicament. X &gt; d d; ·. da saioeas &gt; (cc): 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, . Vc C: id (pit: .C ;. i.e. Cc:: 0- C C C C: iii, c, d, c, c, c, c, c, c, c, c, c, c, c, c, C PPC: P: PP · P PdC d · gt; PtP: PdP ts a ta 'ct: (S), S (S), S (S), (S), (S), (S) P: PP: PP: PP: PP: PP: PP: PP: PP: PP: PP: PP: PP: : &gt; of the following: XiSSX lo B0 3 â € ƒâ € ƒâ € ƒ3 â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ (a) 0: 1: 0: 1: Cp Cp XD BelC cc 00 'C CCivC if Xrc It; S,; Ό Ό': Cl The compounds of the present invention may be prepared by the following methods: (a) to provide a compound of the formula: ## STR1 ## wherein X is as defined above; e 'is at 0 d o..c 3 if' (d): C (O) C (O) C (O) C (O) C (O) C (O) dfp ;: C a eaea falls. e4. CS T: C S taitaxíev a diVC fi ck S a.p: a X. C P Ide .. -... a ...... p.t CC p: C; The title compound was prepared according to the procedure described in Example 1, which is incorporated herein by reference in its entirety. pppPp. PP &gt; 10i dd et. • • • • • • • • • • • • • • • • • • • • • • • • * Γ 0 S; Î ± β-CÎ ± -cyclohexylcarbodiimide. : P: -E 'P..C. 4): â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒC. SC, Six: CS • If donated to c • P. v. V: a Pd Pd O ei χ.ΙΡ; p; PP T vi.pd, fC; '. P C <Pve; dr, P :; gives the parent and ec: Se d O: v < .asxtaid teaseiade P:: P: da> 'N ···; PP, 0 d p.X avS.c. xsacsx SOS; &gt; • • • • • • • • • • • • .PPP: .C P ·. P ·, · p. Ot '· .ps Sii i. S B 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 PP: .i; P 1 d ia s a: this. ' of aaraad. T: -C \ ei &quot; 1 ........ ps p · ': &gt;; ... 1 pp tcpp it. x and y are as defined above. w: C cl c C c ia Pdla apar sd ar, i acíbdiS :. . p .. · &gt;. the s x &gt; t cicev lo a /p.t;i. for example, 1: 1: 1: 1: 1: 1: 1: ; (a) and (b) (c): (a) to (c) to (d): Crystalline Crystalline Crystalline Crystalline Crystalline Crystalline Sodium 14 P a, a U PP ss xS; (C) -C (O) -C (O) C (O) C (O) C (O) • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - . ooe. r v ·· PPP sat If you want to ... from 0 or < P d: ti.O: X peace. P'P 'c-dXi: 3, d de ce ce., Cd Pa o n Ç> you. èdt ppp tdv &gt;C1-6alkyl; C a Ti: TiO: 0;

Disinfection is expected to fall &amp; PCBC fIP) caadrcP.oasds poeee bed px .0 · 00 'its if qat i Ci i ICE; IP 0 • ··. ............ x 0; '>: 0.V t'00 • d P' VÃ C i.C.s: la a t a er des &gt; &gt;; : 00 00000 1 d casiaçds 0 she piis. The reaction mixture is cooled to 0 ° C. air: so does CO0I; ca rr ia 1; • DiC, 1. 0 Ã £ l &gt; C 0-C do-C 0-C 0-C 0-C 0-C 0-C 0-C acca Ca cac ca: acs 1¾ ssà • 00 0: 0 .ρΟ0 0: y 0 0 i: 0: l OOl.iài. , 0.1 g of the title compound was prepared. ; a Pliac at c 000 vO .0000 0 Ϊ.00 · .; C '00 pXvl &quot;OK; p Γ as:; r: are testa 0 are ase: 10 'a. V c ib, t .Pr &lt;;·; : o '· &gt; 15, 15 to 20: P is from -O-s. the CS; · »: Soa S ;; iir; d csaa 010. straight. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • The present invention relates to a process for the preparation of a compound of the formula: ## STR1 ## in which R 1 is hydrogen; the dials; d-thiazole; x :: 0 B &gt; 1 000: 0 times; s: aa: a a r ip &gt; 0 i paa oo < '1' and ': * - &gt; x ······························· A set to: .seu. those r: 00ii àidii clac c $ a; (a) 0 0 0 0 0 0 0 0 1 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Eca; skirt; : 0.001 1.00 010 0.: D.y '· c this' 0.0' .001 Vi 0010 · .1. i.Csc§ sàapav ar &gt; .alpha., .alpha., .alpha., .alpha., .alpha., .alpha., .alpha., .alpha. It will be possible to carry out the flight to the airport at any time of the day. e-eo; C a ·· P -1-> ··· aa-c 0x1 ··· p -x- v. The compounds of formula (I) · :. PH: 0. C: 's p-0-V: -,:;': 10:. 0, 0 r ... · · ,. i.e., 000100 C1'0 0. - • • • • • • • • • • • • • • • • • • • 5: vv. Qi si ti aae C. s • Ss; &gt; v '; 'P': X &lt; c tart :. (1: 1): 1: 1: 1: 1: 1: ai i a ti 51 Ti 00 ..... Vã 'pppp d ;; scdè • Ç; . .. - x v; ............... &quot; of the 5 'to 1' will be calculated as follows: (a) (b) (c) (b) 0 ° C. . . and X'tl P '00: i P-i. It sounds like sprucing up to Oic0 caa s. 00 cc: Dry air is dry c a0 0 o a 5 //; P a c e 121 a. a iesa ia a &gt; % 0: 0.1 tet: tt: &gt; &gt; of the R & D = 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, ..., ..atl sa &lt; 000. I am aware of the following: air to Si :: est < going to the c. 010 &gt; Pos 0 10 pac rp caa ied at da: t {i; The invention relates to a method for the preparation of a pharmaceutical composition comprising a pharmaceutical composition comprising a pharmaceutically acceptable carrier and a pharmaceutically acceptable carrier. r-0 -: 00. P Ò0 1; 5cesPsti.t. : V ó ó ó ó ó ó ó Ã ó::::::::::::. Households are available at: 0 to .011 Households at 1.1 iv. to: r, o n IP '. &quot;.'. '.'! r a 'Cs ·. Fr: ati aars access to the 0 .0 CSC cctrs::::::::::::::: 6: head 0.0 scaticlt; ,-s ·:·. The product of the present invention comprises the steps of: (a) providing a sewing machine with a sewing machine; (b) sewing a sewing machine; or 0. V: V0 010 c and a: a as; p 00 '1'; hunt • 0. : 0.000-a. (C) l of the handle ··; ..... .st: 00-00 .I-OIOIO; (B) and (b). 000 &quot; acss: ccaaria · \ · Ã x · '·: /.......0. &lt; / RTI &gt; 0: 1: 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 ' ò 1. 11 • Peeleeep telplte of the UCEC f) Fishing: K0.05. 1; P = 0.01¾ Pt = 0.001. : O ;;;;;;;;;;;; 0 aaa t .10. C-1-C-1-C-1. (1), and (2), and (2), and (2), and (2) (1) and (2) and (2) are as follows: (a) a) 0.01 0.01 taca t ase> 0001 .01-0.0 0: 6 Sara as - 0000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000000 , And in the case of a dry powder, the dry powder was dried in vacuo at -20 ° C. : S iso ce tioo S / 10 .epsilon 1: 1: 1: 1. : &gt; x 0 ... d; eeaa: .pi.t pe ... srstppip rrsesr Ι Ι Ι Ι Ι Ι Ι Ι Ι Ι se se se: 1 &lt;t; 1 &lt; tb &gt; &lt; tb &gt; dl> sco sco sco sco Q Q Q Q Q Q Q Q Q Q Q Q Q U U U U U U U U U U U U.

1c {(f: X P | p; ., 1 can> d d .d; 0000-3- pp: ia PP: OOO- d 33 in the aat.tl: i aacM: P 00 0 PI::::. 0 0 COO- •• Pd 'a da te ;; , SV Ss i; d p s; · D ··· _ trOOid gives D to DP CPPi t> Î ± a. 33.3 d 3 A 3 'D ·: · 03: 0 to 3: 1): 3 P 3' 33; the 3,3'-CiPI was 30% in the range of 1% to 3%; PM &gt;PP;dla; aaa PP: 'Ç; : 3: 1 to 3: 1: 3: 1: The results of the present work are summarized in the following table: PP-gt; d, 0; '&lt; /. 0; i3. 3 Ov dCS. : 'v. ·: d; (a) (b) (b) (b) (b) (b) (b) (b) In order to achieve this goal, the results are shown in Table 3. Table 3 shows the results obtained in Table 3. · A · · t t t · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · P P P P P P P P P P P P P P P P , 3-hydroxypropyl-3-hydroxypropyl-3-pyridyl] -3-hydroxypropyl] -3- (3) (3) (3) (4) (4) (4) (4) ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ ΡΟ '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' ' 'Ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ P: : 0- dacC: 3ΐ · 3: the OP is defined as ... P Q QOP e ·: · · P P P P P P P P P P P P. here; n &lt;. Par: PE; aaa ç ·; nact Q Π ':.;. t PO o ra C3 · day. Pd 'Dtta p -Idii; ii-030' '0 · O id p. : dc pd :: d apep 1 t IdÇ P | thio-O-CPC; st i: -vi d s-M 0.3 0. ooç 'dODi': 3 3 30, s: · d.dvv ..... U3: V &quot; Ot ::: Sp: 1.3. Amino-3-oxo-3-oxazolidin-1-yl] -amide; 301 0: 3 d &quot; , &Lt; tb &gt;ppí; : .t. pp ; aaa 3i: 'ss aaa rare .P .p' àd 3: ataa. (a) (b) (b) (b) (b) and (b). Pd 1 3) ai.v .t &gt; The rationale is as follows: (a) pppa ta dO 'd i di 3', OOi s s c; age of the child. p Pt v3 panai; DP P .; . .3: • p: 1 ãã aa; d-O-p-1,3-aza-1,3-dione. P; :: ç3d; aaa; r: OAidi. i..aa &lt; a a a 0 3. V èa a; _id; aaa i P: &quot; T · C. ·. (A) (b) (c) (b) (c) (b) (b) Yes P. J. '; Ppc is still at. 3aO3a ?; pi acca .ta ai o a ...... 3: ti 3 vi iaa < ........................ pm iappi .d; d \ 1 ata :; rsaa .iid · .; i OPIP 3 :: i: ta in P *: .p. ; 3 0 ai a aa a aaa: 3.3 · C xd '': PP.PÍ ··: ·>. (i.e. : 7.9 (d, 1H). • P = 0.01; P = 0.01; P = 0.01; P = 0.01; iO < at 0 Ό. iPPCPPP wrath; P O '&gt; &amp; aes' .ΓνΟ ·· .ν.Λ'ΛΡ i P; ts aa Si pz 03 O p ··; , p ': ..., &gt; ·· ,. 3 ..... 03; PP: ^ 1 .s.d; ... v'v ························································································: a a II p CD; P 03 aor :: a Cd =: Sd 30d: 030 0 ra P V '· pd; 1; (β-β-β-isopropyl-2-pyridyl) -piperazine-2-carboxylic acid tert-butyl ester - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - (a) and (b), (b) and (b) are as defined in claim 1, d Pd Pca pPa v-Pàt · CP; nial Puo ....... d:: V '0a or d ai' P; (1), (2), (2) and (3), and (3) to the following equation: In a preferred embodiment of the present invention, the present invention relates to a process for the preparation of a compound of formula (I) to (a) to (d): tat .1 ta; .003 N.N. · X. X., yyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyyy (a), (b), (b), (b) and (c) and (c) V: • • • • • • • • • • • • • • • • • • • •

ajs-sda:; asparagus sauce it aaa of aatrts 000000: 1.0010 astdPtasda for. PtOsltPO a.X tprnat.s. I do not know. s: ssi. ap: OPitÒPP Síls iTu C ay t asssdi gT ;. G? GG: aPt sips. sssa.sst: lrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrppyrrpyrrpyrnaphyride, moas: s .d; t a asadaassstadac sss dí.çKp-id asssd.pap pro •••: r.ld < i iissa: apiops iGia ç GOB 't t Pi - GGGG to as - ::: i G iiiiiiti GcC ·; GG CG ssops Ç GoiCG the sOdj to the Cspi: Γ 7'ps, fsaneia ias air: - ii: fs rrh OP P o Mb spts s pp. P 'W (is a ssi-ta sidi al P PC PC; k k pa pa pa pa pa pa pa pa pa pa pa pa pa pa pa pa pa pa S S S S S S S S S S;;;;;. 9 to be the same as those of the CG, and the CG is the same as the CG. , Which is the same as that of the GCC, and the GCC, 3 sopp pis v P isa assSPpri assa i 'i' · · b bb) pps a pa :; (a), (b) and (b). Dsaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa dN i 3 -) -id-it βΓί-CO Pi rc · < iCGG .G.y? ; 7dspppx; you; ; A mixture of the compounds of formula (I) and (II) ipiti i fidi IdapippitpddP ià; SS a p ar b.G; d ... si: ii · xiiii s.d i 7 G} G sac -: b tV &quot;: ντο sppss; to the sd pi to the dp ..... f saa oai aa t iii &gt; ..... dC a &lt; lisiaa: P. ·: ·. 1 ii '· b.y &lt;.·; ....... pG ·. G. } -> Pt dt. Vtp.:. d. i, :: s.SO spdp t; G-TG. s-p for GcHg Q. gá to aocoa: V; P. PIS: lisa pppbssi P ps; ............ ips CG; there ':? DiSiSi &gt; ia D s: st; Gi ': Cg; the op;: ;;, cs; G: t. G G: G GG :; will be discussed at the end of this section. '· &gt; The ? It was the assis tation, that is, if it was not possible to do so. 110 aa = 01: PP: Op s · ;; ppi, Xi.rp ici.6 · IPSISps; gt; gt; gt; gt; gt; gt; (1), (2) and (2), and (3) to provide the compounds of the formula ': Gd gg; &quot; GGG &gt; &gt; &gt; &gt; &gt; s. .3 G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G G GG GG GGGGGGGGGGGGGGGGGGGGGGGGGGGGGGG 3 (d), the bandwidth: aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa the first of the years of the AIDS pandemic, the AIDS pandemic was the first phase of the epidemic epidemic, and the pandemic epidemic was the first phase of the pandemic. aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa · S: sx.b.ts. Asr oroo UCECs Π. 1 r In the case of the present invention,

Oatroa arpai taetnsssae aaaari.aaa .d tdili.C fld asada apesa sit aitsaaaPdaa è daaaasaçda psa a feri. from the year to the year of the year, the year in which the year was at the end of the year. .5itsepto.ra paraleiopipédica; A ssistent for the sake of action, the capo of the spossessed: ono bssoo ac. 000: 105.0 sial. od or the pop doba. fido i watches the following questions: Sa: sisa; ss: ss. ss: ss sssssssssss ss: · - drying · a r aa .. a. aa-pr atasao asi '' '- &quot; '-. 1 ; . poses cosso n dorsal air a psssrae ror lati sssa r lassa is bta per aso a a pi. Pa 01. ca: d taba, from roast to fssei.iita.t -a sssps.i; A method according to any of the preceding claims, characterized in that: r.isiPípsai., práa aaaOa.afaa: &quot; Sa: dosar téop apaaad arb. a. In the case of the ss ii il sa t; d a ss d. a to E 3 (st), as shown in Fig. and p 'dC. , P è ;. p. ipc-i "; 'OO &quot;;d.r; : 3 3: 'N id- tide) 4 (7) ,, 0 sed 0 0: 3 33033: χ θ θ χ χ χ è è è è è è è è è è è è è è è te te te . . (I.e. : y · .. and 33133 0.3.33O0: s:. ·: Ί · • Ç CC. ··> (b) and (b). ic C, and t. i.e. 330: 033). and (b) and (b) of the compound of the invention. 33333 and 333, and p: OS 33333: 33. 0; 3X333 0 3 0 and 333) - ρο d d ': - PPPPP. Pedat: p i d p < Article 3313 of the Treaty establishing the European Coal and Steel Community. 3T: t leerieitl tpde, 1. t &lt;; and tit 3 X 3 yacht 3300 pc P &gt; F 3); ,> P>: can be made OO &quot; d is 0; 1: 1; Cp d. Vdc C 3.33: 33333. tt &lt; &gt; that X and Cp 11 are per i.C; PP; and COC '' C C dil dil eo C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. C. eo C. C. eo eo eo eo eo eo eo C. eo C. eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo eo et &gt; P d '&quot;' : m.p. V '· 0 cc = 33333 · 333 is 33 0333: Taxi' !. 3.3. CaCp: CV · eid.ai and ea: powa. 3 3 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 d C: .i Ci; td &quot;d;. d Cp. 0: 30033:: p 7 '; P: 1: 1: 2: oolacada: 1: C 1 et al. tdd {a-: • C '· .c or ·. d, 3, 4, 3, 4, 5, 6, 8, 9, 10, 12, 13, 13, 13, 13, from ea to i. Oteee P, et al., pp. Cp pp. Cp 33333 and A3; (Î ± O to Î ± 0.03.3), axet: : 0 0.8% 3: VO, '0': i ..e 0 &gt; P .3333 1; 33 33 333 p 10 33 3: 333 3 fltO.) 3: 3337 \ p.ra Pp 1 cc cp ·· pt · 'ip, p% s &quot; C '. &lt; v &gt; i: d: d: 0333 &quot; ipt .1 ea) 3303 eagete 133.033.3 Ílot) .1. Ç &gt; fCpC drt: ··: .a hapt; 33 ° C; 30: 3: 33,000 333: 33 33 3330330.0 3: 33000. , P • p Cp pC pCi ct p ct d d-d cr. ioe de dtr P '· ΪΡ .... 07.3 ..; .....; d; : where the ; C ip t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t: of the eatetete f Cp-0 ii itad Pd; -S < 0333 (i) to (e): (a) (b) (c) C 0 '· &gt; . C3-C5-C6-alkyl; P &quot;yCP; Γ :; Praça;; Pi. The present invention relates to a process for the preparation of a compound of the formula: ## STR1 ## in which R 3 is as defined above. (i.e., i.e., i.e., i.e., i.e., i.e., 3 c ···· and 333 CF 31) 03.3 3: 3: you can not. i.e. or d icid 3 i .; i.e. 0, 3, 4, 3, 4, 5, 6, 7, 8, Pi: r; xo te Pa.ie Da x, c; c 3: a tipi 00: 3! of 3,333,333; (3,3) 3: b.) 33 pyrrocycline cc. .P. ··;.; A compound according to any one of the preceding claims wherein: i.PP: ç r 0.0 CC'ip .3 Ο ΟΟχΟ Οίο ia ia 3: 3dotei die 1> ο a d eata: Cea C Γ s. to; you. and c. 3.30333: Ostde da; 3: 1). Λ Λ Λ Λ Λ Λ Λ 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30 30. 0 v ρρ.: Ϊ Ç Ç Ç Ç 330 330 330 330 330 330 330 330 330 330 330 330 330 330 330 330/3, d dr / ': (I), which is in the form of a compound of formula (I). from ç ..... rol XXò.ÍVí. .iip i '? OK; i. -23). I-a: jdd 3? Ot e raie ..... gives:, P Cp O of aetdete: eit.0 C; P;; (1) and (3) and (3). The results are shown in Fig. eeoate 3 40 d: OAc: dCCO: pC C tN of HC: P IP V 0 pd 1 P: d-oat 0 i.-eo -mt • i p. v \ quot; \ * '. ·' *:: p. to aà pOpO li < ..; cp believe dt P: ····· ·. ·; from the Ptd pd-dd to the test. P i:. &Quot; P C p p ip e t;.: ΊΡϊί: 03 | 333; td pN ·: t: a; 33; 3, 10, 10, 13, 13, 13, 13, 13, 13, 13, 13, 13, 13, 13, 13; o! : 1 A nc.:^ ...... N A ...... and d i Ò &gt; ep: does., d d. 33; s p: 0330 0 i 0333 gives i 0. deoiooifce &gt; i e 'v a t! e Pesedé d da lee Í3; tc 33 p O O c. , β3,3: 4.3 Î'0.0: 4): â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ33 ° C 333 x 333 30: 0. eat and 013 i 3 ed a ei dt: Pd% 'peei? 333: 0 33: 030,; &lt; tb &gt; Pt ed o. and, Often Ovieaae · '; 4 Pi ·. i.e. Cp ρ ·· 3 3 303 CO cd of the king and ooordadit; a d.e e d CC Cp · .. O i &quot;; Pt ·· '. 10; . d &quot; Peta o.ic Ό ...... .3.3; it's the; eda; 33 of o. 330000: 0 BQ: t; -P -¾ ·· - &gt; ·· eça e Ov C &quot; COO d fie; et; te 30 att: dltt &gt;0; r or cm-3: OEO: p33 xylene 3303 .pp P1; . cc to sed% nlcg ..P ... ... d 03 '·'>. tpi 3333.3. 3, 4, 5, 6, 7, 8, 9, 10, 10, o ·· íitt € P. PC ppCp of dedd dl d; : · Ί Ϊ. ; d i pe :; p = i -bet x.te 1.3: 33: 303 pot 3X30 s; and d Çi pt Pi * F • P &gt; i.e. titi: ie, and C.P v, UPed · e; 33 tiK d.) pot 3.3: 333 3X33330: 133; t. p- en.t- and p. (i.e. to: P OLICY OF THE OCCUPATION, P; &lt; / RTI &gt; &lt; / RTI &gt; &lt; / RTI &gt; 30X33: 3: 1 isotherm pP: PPPO PP P ..... pCeoCaC: V: dP: P: P; t) e33i.et.os oíte et: Ote o:; · .; , UIP Cv! : V \ pd and e and d 31 P < &gt; ro &gt; · 'd &lt; tep 3001 &lt; &gt;pi; ): t.sub.330 c: 37371; pC V; he. . xeat et al. i.P. 314 i 0 l Pd.) ot 03. 333 30 efoieo dt; . ·. · .; ,· \ : day ; ion 0333 · 401 0 4? 3333.33? '3033a 333? 3 ': aa: · .i. 3p3: iild:: 4.1.1 T: Go: 35: 2: 3; 3330 j. 011: 4.4 co 33: 033 &gt; '' ''; . · ;; ; Ctia dali. ·. Eur-lex.europa.eu eur-lex.europa.eu .·: -.·· .O. (I.e. c 0 33 mt 44. 033 a.3.0 3.3 S33 530 03 ?:; ó), 0: p? 33?; 1: 1 33? OoasSSd? li-aa? 41.004 1..0.1.1: 4. ; \? Î'3.3.3. 3 :. i-d-dl-i-i-i-i-333: .: 3333 pd, 3 tb______________________________________ tb1: L d., R;.; â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ340 - 33 d 03- r ;. to 46.6 ° C. βAPP: aaap ·: 4 P-4d 1 =. 4: air: -0 soasss 03? 1.4 'i 1 03 3 33 3: 33330 Τ; 33 ° 33 'P; 1 and <. '1' '' ': 3: 3a '11' '1' '. 4 33.0; LO: ??? The; : 11011 11.1.0 pt: t '0.0C p. ;, · &Lt; .1. - n. &lt; 3 0 33-33 3333333 053 3,33: 3: 3: 3: - MC; The title compound was prepared from the title compound as a white solid, mp 218-224øC. The title compound was obtained from the title compound as a white solid. ··. (I.e. ·; par 1: 0? 3 {â € ƒâ € ƒâ € ƒ1,44 leaves 40.1:. 041: 4 dl 0..010 -d- ri ;? (1: 1): 1 H-NMR (CDCl3):? 11-10130 ° C. Iddl: 13: 3: 33: 1. id 3; 4d. 4 a? 1: .d 1.1 pdl.14 :. &gt; p TIG; CEP '303; C-O3? d; dC-3S: d &gt; of the title compound. (C) 0: 1: 1: 1: 1: 1: 1: 1: 1: As a result of this, it is clear from the results that the results of this study are shown in the following table. i gives CU 3 4 1 2 3 4 5 6 7 8 9 10 10 10 10 20 20 25 30 35 40 45 50 55 60 3 4 5 6 7 8 9 10 11 12 13 14 15 20 20 20 25 30 35 40 45 50 55 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 60 50 100 [ 333-3: 3: 4,433,333: 0-333: 1 to 3:?: Aa?:? 1 to 3: 1 to 3: 1 to 3: 1 to 3: 1 to 3: 1 to 3: 3333: 30: 30: 30.3: 3: 1 powder: from 0: 05: 1: 3 to 3: 1: a - Ρ: 01110 0101: 14 - d X: 1 to if MCS € · · ·: ··· 03330 S3Í t 1.3S'S3 ': ....... 01 55 ::. 53,330 1'4 ... asa? 3 3 333 30: .30 ':? 1 i-.Vyí.d. ...... .pdf: .pd: 1, 2, 3, 4, 3, 4, 5, 6, 7, 8, 9, 10, d rd Xv: ¾ r 33? : â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ3: 3: d 0. di P 3.3: 0: í> d.G.i3.33: 333-333: . ll 33.3 :: 33 1.1.1 cl

ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ ΟΟ. the donation.:. d ο d a a a: 9 i 35 pt .3. 33 am to 1 am ; aar: a 35.0-1.

Caa? The compound of formula (I) ?:? 3t; 0-3 ° C. Ο?: Ρ30 li. a aa 101 f a.aa 1,100 1,04 0 3305,1 0r a: 3 33 3303. d. dl to &quot; -. 33:30 0.1. : c .1 vtrpa ?. , 33333:: 3: 33 :: r 3? 0.1 0.1 to 1; 114 1 3 33.0.1.11:; ?? 0a 003;: 0: 1 40-0 the blade 3: 3 i 0.0 J 44:: -4 01: 1 :: 4. ; ?. to t :: 33 :: 3; :; 41401: 3 a? . 5 3: 33353 ::? 5000 00: 3 Ο; &quot;. '. . : 'IP' ·· a 033.0 3033.:., Aa. dapo. ?? 0ili cri 0 il :-p: aioa? d 3.3. 3: 333: 3.5 dl poo Iv 1 v a 1 0 33.53.00 0? d. 1-: 01. 0 sd Ò 0 d: ti.a.? 3 141040 aie 0.0 4 4 40t: 0, &gt; dPtòd. or; from 5 to 11, from 0 to 33 3300 ..... a to 0: 0: 1. i.e. now at the same time: ip.oa · -: &lt; &gt; 3 h to a, a: a di t a 1 4 1¾ .1141.10 4: 0 ar: 33? 4 0 11 3: 3 3? : 3: 3330 3 1: 1: 3: 33: J, 2:33 0 3 .3. A? (I.e. are 4 4: 4 i 300: a 530 333 3 3 335 adi? 0- to 4:: a φ. Ss ap ap ap::::::::::::::: s s s s s s s s s s. d p .1 iiii: a da 333? rd; d: a day of Cd 4 L 5 a a d d o a 04 .0101,110; 1 &gt; 00 4.1.14; 0. 333: 025.33; ratify ata. IC 11 11 - s - 1. : 0: 0 dv0 0 'd: d: i .1 &quot; li 010? ; i aio d: θ3:? ί? : 3: 3: 1: 1: 1: -4: ids aa ??? ' The invention also relates to a process for the preparation of a compound of formula (I): ?:? 04? 3 to 3: 3: 3: 1: 1: 1: 1: 1: 1: 1: 1: ; 10: 1010: 11: 1: 1. 3 to .0 '. 'i. . i.e., â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ- 0 to: 3333.: ¾? 3: 3-33: 333: 33. x: y i a Id: .1.11101 'a la i a 400'i'lóld 330. •. &lt; id: d; C-d-3 00 'C; .'Λ. . ·. • 1 30 '3': 0: 3 ad.P: aa 1.10 ..... -0.00 '0-10-ti: d 33: ta. The title compound was prepared from the title compound as a white solid, mp 218 DEG-285 DEG. \>. · · &Gt; t. od: Ρ'Ρ-ν rá Ί1 a ????: ?? 3033 3:20 would attract 03; 3? 5,333,333 104 1, 1, 2, 3, 4, 5, ; βθ3? Î ±: 110 Pd 33 4: 4? 35.3.0 33 '' .lilill, d P 3 33da 0 411 4d: i: 333: 1.30 00 · 40 dll'lp -: d 0101 0141 aã; .1 .. 1 5.3: 33 da. &gt; 5 '':: 0: 411114 11 'to 5': 3aa.?docs 33333: 31111 d: ??? laughed at ?. The ? &gt; the formula: &lt; / RTI &gt; 0? of Abras. 1 of 2011

Claims (2)

Mx? IPDicm? C yi?: O ν? ·? ΊΥ ti; (i.e. X X X c &gt; was: to cie itl s P-; :. gie; kinetics bUO; ···; - X; R. The present invention also provides a method for the preparation of a compound of the formula: ## STR1 ## wherein X is as defined in formula (I). ia 01: CXOX &quot;.X; 1, C: X · Ο -:. ;; s, P: OR and r is the parent of the child. apo:; X X. O * C. CdbX U XXX; 'C rés ΟΠ 1; :: ¾¾¾¾ es ors; P; &lt; v sael ai y darei pee: Pae: p x.> rc i: ·: ΧΧ. d:. · .. Pi \ 7. • / Ορ. ΧΧΧΧΧ are are are are are are are are are are are are are are a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a (A) (b) (b) (b) and (b) and (b). _ &gt; '··· oseed ar; OO U t b e. pi V · 'p ip · ί'Ρ; '; &gt; ae. OR rr. (a) XO: X of UCUxUX; (X): X: X: X: X: X X: X X: X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - (1) and (2) and (2), and (3) and (4) and (4) and (4) and X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X- Π Π ea Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π:::::::::::::::::::::::: , which is the same as that of the X-axis, and the X-axis of the X-axis. In the case of the present invention, the present invention relates to a method for preparing a compound of the formula: ## STR2 ## wherein X is as defined in claim 1, X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X Y ieaaaaaaaaaaaaaaaaaaaaaaaaaa X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X - , And in the case of a number of factors, such as: (a) (b), (b), (c) (5), and (5) to (5) and (5) to (5) and (5) to (5). of the following equation: X: X: X: X: X: X: X: X: X: X: (X), X (X), X (X), X (X) '' - ·: P h - O i rear aa OeP X'-: Pd- ;. b X ': X i; pd: w X &lt; r ae o; &lt;. and (b) the amount of a compound of formula (I) ouesee e..a do è; X; ... ·: -s erpa until X: i x p; (X) X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X - and X is the same as X and X is X and X is X and X is X and X is X, and then to the X-axis, X, X, X, X, X, X, X, X; X-ray absorptiometry, X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X-ray diffraction, X- and X is a region where X and Y are the same as those of X and X; As shown in FIGS. 1 and 2, there is shown a cross-sectional view of a cross- • '': '': '' '' '' '' '' '' '' '' '' '' '' '' / Pear xx; ...... XpX; C ...... (eteear; '0'XU s flee ....... Ι'5 / · ....... r .. ..... or UeO: a Pa ab arrrerr x. / x. ae · · · · · · · · · · · · · · · · · · · · · · · s the acre c: ο; Eur-lex.europa.eu eur-lex.europa.eu and cet Pr rode. : Cell; (1) and (2) and (3) and (4). given by Captions: '' '': '': '', '' ''; ; i arétie, P; r; Scratch back. eg, a and a are are X; X redirele X P &gt; ..... X 'C ;; x: a a s s? :, X 'C. .............. : P Re (pee raçse aaa; P re: rrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrrr X-ray diffraction pattern (X-ray diffraction pattern), and X-ray diffraction (X-ray diffraction) The reaction is carried out in a manner similar to that described in Reaction Scheme 1, which is incorporated herein by reference in its entirety. : ex ex ex ex ex ex ip ip ip ip ip::::::::::::................................. aa: ad G1 t; X dg d; • &g;; S, .gif: dd e ra.Caa dl). p &lt; 3 &gt; of o d; ··; d &quot; day.- . Δ: i i; d epa ferra Q.p. X and y are C :: Poa :: dP'.elet Ò CdG hl of: dd. 1 nlsox caad; Q li: '; A solution of: XaXS here: mp: 100: 1. oe eoa-recipe. dP to a Cd d- and cg:; d; d id. d aipeaG :; Id .;. cag O X: g 1 and d. w, n. or the like, or the like; = 3 C.v ·:: 5 Ct acd · Ga a dS / dO and / dv G: 'j tdai: ΡΡ' XO; Oi i. . ·. The title compound was prepared according to the procedure described in Example 1. c. ivi-ii-dans f '· ta X. f Lxxx x 0:; (1), (2) and (2), and (2), and (2), and (3). The invention relates to a process for the preparation of a compound of the formula: ## STR1 ## wherein X is as defined in claim 1, and the present invention relates to a process for the preparation of a compound of the formula: ## STR2 ## wherein X is as defined in claim 1, (a) and (b), and (b) in the same manner as in the present invention. (a) and (b) are as defined in claim 1, characterized in that the polypeptide of formula (I) A PC of the PC of the day of the day is set forth in the accompanying drawings, in which: FIG. aedaa d ': ..... Xaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa d 3; p aap oat • 3 • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • : a.: 3 P tace i &quot; aa: OS '3': apo afe yi; e and P: ò v.iOX ££ .d and the sink network; al 00 t:. G'V and P • d d i e: d i and j .duS i.d. powder: 3 X.. a / d d £ 10 :: d of the stock of G at the beginning of the year. Hi 0: 3: 1 and qqqqqqqq 3; 3.Ç àXC; dv-3. ΐ da. e: idd v 00 Hi from peepea:.;. d ode of theta to et ea- · · ... ·>: yidXè; V.sup. ; Λ di: __ __ __ __ __ __ __ __ __ __ __ __ __ __ __. X.G.G.C.P.P.P.P.C.G.C.C.G.C.G.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C.C. : GÍ. O and p is the same as O and p is the same. d rd; pd: pp to c ....... ·; i .f. \ y: l. ΐ'Ρ and /C.i; V of X ..... 1 O 2, and eci apeai: t: i: eq Ρ: Ρ0001 / 00 is Ga raefPe ipedC: · ΡΟΓί 3. tfvid.aap dP CGptGGSO 00 E; :: Gí ::: VG .GC.G.étlOG. (1) Pair of PP 10:00 PP: 101 PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PPP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP PP > the ceaec euaa ptafgdes d'Ietdeeee Frost that is ee-ee ee ee ee ee e ee e e: e: e: e: e: e: of the population and of the population and of the population and of the population. (13) and the geography of the errarpaçdo p G r ρ G Od od: 1 ar ρ ρ pb il iq: ad í e qa 1. aa I. g: dv, P to Pos1 gadde ceepo a The date of the completion of the drilling and drilling of the fluid is as follows: (a) The drilling of the drilling rig and the drilling rig and the drilling rig. in the case of the X-ray diffraction curve of the X- (a) (b), (b) and (c). a tatra: aot d. (i) and (b). apo r.cX atta aoru arti-ar lor 01 p 80. traia: c; XPiV: S d: 8 rave ppa õ P; X ara 'Xr'p. ddX ': νX: cd-18 -X: B. d.-X Ρ Ó tut e fie CSf X) .89: Λ:; : X s &gt;; 9 B X P:, XXa o aatt rtf.:ur:),ò8:fUfo ta V ;. W; ) p i ·· '· < '' '' '' '' '' '' '' '' '' '' '' '' vai: d 8 Xi itt. &lt; 8.8 Pd 8: 98 of 88: 1: 8: 8: 8: 1: 8: 1. 8-aorta: from Pg. X-ray diffraction: X-ray diffraction; X-ray diffraction; X-ray diffraction; X-ray diffraction; BCBi to Cluster PO. at ra ρ sp. ' X; d. X'DXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXX i-ttpo: aX, DXXXXX-5, 1). &quot; VX. Cl Oit. t, f (L)) and d), (a) f Pg 1190-p 11;: P: &gt; Ρ 'Χ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π Π (A), (b), (c), (b) and (c) and (b). Cd X i:, χΧ, ρrt8: OdOdlUitl; / 88 eight X; 8 οΐοΐοόοο i á; X'X 'P: i.J. i, 8; β;. 8 iv. ; Xci; The reaction mixture is allowed to cool to room temperature and then evaporated to dryness. p Ο.Γ Vi .d; ; i i. X t: 8 Ρ 1 atorphoretic and O: vl: p < :  € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ 91 Χ Χ i i i Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Χ Χ Χ Χ Χ Χ Χ Χ Χ: : P:) 9 c tape; (A) the temperature in the range from 0 ° C to 60 ° C (° C); χχ.χχ. (a) and (b) and (d), and (d) to (d) and (c) to (d). 9 OOtip is t 'tas' St: t::::: oi d. f B) a · to XX: X to P &lt; the X-ray diffraction pattern is shown in Fig. 0080 8808;: 1 ···· 9 O: y \ a. donate to: p. X: X: p.BX: X-ray diffraction angle X: X o. ylp Q X X. X X X.X BC! ) 7) Because Ρ.ΐ CP pp: • 'PP; mp. pXX 'ooadoa tt.a tstta tt O X: pC d' ó P.X a a rea rea s s ·· / S. .. ύ · \ 8 ;; sink ; afi 08; (a) and (b), and (b), and (b). v d :; oui; a. x or X.X. X Pip .V.-s S1 ... 8PP &gt; 8S9: 88: 080: 80; 8: 90 from 8 C-8; P a r tf, at trave i: XX Pftcr; pr r 8 at V pi-pip i.Çd pcò d odpC dp PC d yP B · - v Xc: BX: i. of the X and the one of ae: -r: · UfU: XX / d 80) 88 d.sX d 'XXc'i XX t &quot; over there. (1): 9) 08; 8: PC. of the ceaipt r: X ·): i; d: X iO .f X. · ta 'a ta r: Pi: pffi ·. i X Cy 88 Poupor would d) .2) .cpB ·: ·· o d ': 0 and \% · o air; aobob X C: XX; and ... XXV; XXXX: X,: X: I actPf C: - 0: 8 X :, 088 'x. -XB B. piterart 8: Î »P 8; 89 χ. B Ò; &gt; 8 · 00008 /: Ρ; CH 2 O: 8080; X: XX X: X 88 X 9; The title compound was prepared according to the procedure described in Example 1. p r 6 rd r: a of t. f 881 X of berrrtra / feoirCí doa C O m O X Parry; .s &gt; &lt; p &gt; (C = 1%); uu; or; 80 48 a, ai.au Pt; •, • &gt; · '. &Lt; : p: .aP: ata qtf 9; P dd: (ddd..f. 880 oaraodorlati CX X 1: · 08 d iniaaf: a 8 f.Od; X · X 8 if 9 9 'PVP · (a), (b) and (c) and (b). X &quot; &lt; v · '· V.voX-pN; U.s 1 &quot; X &gt; at itf; 8fft. -X ·· B / X t X; · χ · ϊ 'Β · Χ V d ia V. ·; pc d 'X ata italy ida sf.t: s Isrer; te o X ·. The title compound was prepared from the title compound as a white solid, mp 218-888.8 ° C. (Xi), Xi (Xi), Xi (Xi), Xi (Xi), Xi (Xi), and Xi (Xi). (2), (2), (2), (2) and (4), respectively. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • X.XB was ti9 9 8,988: ooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooooo . •••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• (a) (b)) 88: otiorlobor; (b) (b) (c) p. &lt; itrobi :). the: aó ip · &gt; tb 8 i a P t U i. The compounds of formula (I) (Cd), qoartdo a X, X fe SBi iUBXc i SOS: pear; air baif: ftitr Ϊ actutor f.t8: d: or egrod ata oXp, d &quot; i 1 X 1 eap a fe aai ··. X. ar t; irri8 s · '; u ff of P sC ·. pP x. the &gt;. i.e. ai oibt .pB; .p P: ·: &quot; · c 4 go to dota r 8 &lt; t &gt; s 8 a ·. *. n! *. ; U f .. P. yà irra da &lt; Cl P or '88 d p. 9 ptip: atirtiuoco ::; ; iooPi.) Î ±, Î ± Î »Î» Î »ia rap X. λ 1: ats Cp. a &lt; The title compound was prepared as described in Example 1. O: 0b 8 'XB-XB X: XXX. d; 800; mp: 8.8 (d, 1); X X. Xc t.X.9 9 tr or o:? T ?;; 0: a8ta c ': <B s. : ¾ P a. 8 · '·; From the point of view of the letter to the letter to the letter, X bay X: XXÍ'XpB: 'ρΧΪ.'ο' Çd d p; (s); 1 (d) (d): 4; porf: the XV ;: x .c vc X :: < C: 1 rutreria.;. 1.08 B: VX a .1 dnadod or O.Pd; : p; XX-; to XXX. and d: X d. you will see: ti Β · ΐ o-: · &lt; 4 &quot;J; • χβ: art ecaar. gold &gt; Pi · <a · atair iPi.ti p. Federal Police; (i.e., Xavier et al., J. Biol., Vol. sb cs o c s o c c r r i c c c c c d c c c c c c d c c c c d c c c c d c c c c d c c c c c d c c c c d c c c c d c c c c d c c c c d c c c c c d f: 1 been · nét1 ca (12) DC: h :. CI.CGG / OCGG: A 6 X'i: i. ·: 15: ......... ·>:. ,  € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒD. di C d d r 1.5: ®5: o pair; 45: 4 CaCl2: 1: C: 1: C: 1; C a-C q; \ rir Γίν &gt; 5: iS 55555: ¾ d ad ad ara® / ta®®® Q0 / l d; C ': Sdp: tasting; ; C 6 · 00: alataca of the .2.2.21 q® - a / d® ® acructure 1 l: b cated: decàd boa Ca 5 :: 5r ®5.® &gt; : .P &lt; · .; -.1. (a) and (b) (b) and (b) and (b) and (b). polo or .55 lac® d® a®. 00555 Ϊ .co 1, 3 '4) i ·. · 1 · · · ·. 5 to 10: 1 to 5: 1 to 2: 1 to 2: 1 to 2: 1 to 2: 1 to 2: ¹H-NMR (CDCl do): δ = 1.05; d; .1120: Î ± 5: Î ± 1; CG; G of the errata 50-. THE . t d; 12 aaa p;: &gt; â € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒX: The compound of the present invention comprises a compound of the formula: wherein R 1 is as defined for formula (I): wherein R 1 is as defined in formula (I). C ltϊ st ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO ISO Òϊ · · · (b): (1: 1): (1: 1): (1: 1). ; 55aa pos 0:55 ® bi: V: '' '': 555: h: 'ÇC 42 ....... · 3' 2; S 505 ': 5: 1: 5: 5: 5: 5: 5: 5: - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - - (1), (2), (2) and (2) and (2). ¾ ursa ®; s s s s ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ ¾ 21 ¾ ¾ ¾ ¾ ¾ The following table shows the results obtained from the following table: (a) (b) (c) 55.5 If 5 ......... qslO S ; 5: 1: 5: 5: 5: 5: 5: 5: 1: 5: 1: 5: 1: 5: 1: 5. S: S. Hi c. 555 as:.: 1: to si5: 551: .5: 55 &gt; 1: ® rs: batone®; ® &gt; Γ dd 5/5 3 Cd OO y: ·. ;;;. 1 (2: 1): S: C and Ct 0; (a) and (b) (c) and (c) (c) and (b). (1): XC1 415 C 2 0 - Id / iC-CcC C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C 1: 5: 5: 1: 5: 1: 5: 1: 1: 1: (21 g. &Gt;): 5: C03 st s: a C-3 ssis GDCX ataiososa: ao®® (3 s · bato ®) (s) (c): (a) (b): (a) (b): (i) x x a d 5 0 0 '&quot;5; 512 &quot; CSC' &quot; 4: 5 'c'l ;:' cCc C &gt; &quot; 1-1 1 · Ρ / '0' ... 1: 55: 1: 55: 1: 1: 00: 25 to 5: .12.1 The reaction mixture is cooled to -78 ° C and the solvent is evaporated under reduced pressure to give the title compound as a white powder. C: d ou ou ou ou ou ou ou i PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC PC (24:25 o'clock). The following table shows the results of the present study. Ic d 'd &gt; ... 3: 1: 1 -: 0: 1: 1: 1: 5a: aqa 1:55 &gt; ·· a ... f c &gt; tb______________________________________ tb______________________________________ tb______________________________________ tb______________________________________ tb 50 tb______________________________________ tb 50% 'p.apS' '; bi CG. RTI ID = 0.0 &gt; 1 to 2: 1: 1: 1: 1 to 5: 1: 1: 1 to 5: 1 to 5: (I.e. (B) 5- 5 a> cd O; , fb silk ® ad qba bC · cio p: S: t C511 iCCS- v. u. GC 1 to bc. ir 5: a .5: 1. (2): 2, 3, 4, 5, 6, 5, 6, 7, 8, 9, 10, 1: 5 to:: 1: 1: 1: 5: 5: 5: 1: 1: (1: 1), and (2): O21 ipO-Ci 3iOaa dbb ss® ai;., •••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• dl i 4 &quot;: &quot;: &lt; v: ·. d;: - ';' ';; ai \ / 2' · 5 SC r.V Λ Λ V id C 'S5 sara i &quot; &quot; &quot; 0 if you attach to it; (22§ ® ® d.; s: C55i: p 5a 5 to 2.: 555 2 rcici: b ΡοΟ: '2 c: sii- i' Ον (5: 5): 5: 5: 5: 5: C: 5: 1: 1: 1: • 5: 5: 055: 555-: 5: 55 :: c ΐϊ: 55 bl bl bl bl bl bl bl bl bl bl bl bl bl bl bl bl bl bl ΐϊ ΐϊ ΐϊ ΐϊ ΐϊ (C) (15.5 5: 0: 0.5: 55). The reaction mixture was concentrated in vacuo to give the title compound as a white solid. I55C: d:: S2b / 2: ®: dbb (: - 'a ..j: s® ri.5: 1 ibtd ..... \. · Aba}: 0: 0552: ® b: í: Ç (5: 55: 0), and the reaction mixture was cooled to 0 ° C. 1: 2: 5: 55: 5: 5: 5: 5: 5 5505 of the unidirectional rate of rotation is: (22), 11, according to the present invention; and (b) the cyclodextrin (1), if 10, the temperature of the ice is more or less constant. (3), received in step (144), which engages in a reciprocating mechanism, generating the yoke (33) to the upwardly movable (53b) , enter: on. (4c) engages a position sensed by the sensor, so as to make it easier to move the drive wheel (49) to the blade of the blade. - (51). The city was aioal. ds comande (43), this one asks to be elecUromagnéeo, guando O: mounts " (30), in its movable portion (S6b), enters the contactor with the suctioning ring (SNA) (41) and the position and position of the catcher, acknowledging that the same transmission is accepted, if possible. the semitransmittance of the test is performed in accordance with the method of the present invention in accordance with the method of the present invention. upper amortocedes (4 2) to eom. (41), 13, according to the accompanying drawings 1, 6, 0 and 10, the description of the subject (s) in which the head of the head (4) is connected d Unit of Energy Capture Kinetics (1) at the branches of the aan system of abortion / fact of the components jumped dl) to pen to: from oer.e.são:: (25), point: oecerde - If you are not satisfied with the stock market, you should assume that the stock market is at the same time as the stock market, (2 5b V, with the following steps being taken: (4) (1) (b) (b) (b) of the Kinetic Energy Collecting Unit ( X), by means of the eyepiece (23) goe etsanes if the st st and eaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa ad comb of being. (4) is connected to the other end (4) of the connecting cable (4), the pulling cable (4) being wound on the connecting piece (4c) the feet. (1), and (2), (2) and (3) above, if necessary, to determine whether the head of the head of the head of the head of the head of the head (4) 33), in Fig. siotaPa. (43) and the length of the traction gauge (4), the length of the traction cable (4), and the length (3), and if it is in the middle of the mouth and in the mouth of the Oaxies (35), it shall belong to the Governing Council of ............ - - - - - - - - - - - - - - - - - 00.001, roca: ..... 12), ................................. .................................................. .................................................. (I.e. 13, according to the rationale of X, 5, 5, 5, 5, 5, 5, 5, 5, 5, 5, 5, 5, isaa ísdsv •: 0 3.XXX: sic 3ars ;.a xx: xdx: xxz, xxz, xx, xx, x, : X0.> X: X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X- · Χοο ο 11 11 11 o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o o 11 11 11 11 11 11 11 X X X X X X X X t Stdn t .33: 3 00't: oia t XX. Xi .., v ·> tag: g:> X: 'Ssqss CSl ita assas sc a 0θΧό ·: adi OOO: (3 P / d.: Z.XXO.XXO.XXO.XXO.XXO.XXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXX / Χ 'ao 0 X / OK> 0: i csess / cd X &lt;The; . : ddas; . ';'. &Gt; Xy. ': S: gpid and ace. ΧίΌ X! X ': sdoata COZO yl isaises X 0X': X 3. . IOS SSI skirt 30 i a · t -X. s. 1 tdtstsasd. YES: from 0X0 X / sau Ϊ: tv. XiX-dO: i.e. 0 and p.p. d Cap td; Aaaaaaaaaaaaaaaaaaaaaaaaaaaaaa (3) and (4) and (4). &gt; y and fiaaid: · s à / xo; s touch. .xoo: • d '· /. <X V XO d titi cscaa i. ? at;.; ; SiO 2 salt: SCS: c. Hexane (4: 1); of ÇQI .ttdSttd &lt; G-XX agi. the saccharide is added to the saccharide buffer at -0.3 ° C. 1: 0: 3 /; 0.; ^ dass sasap ΧΌ 0: sds tao; t: 0 X 00 / 0.3 0 / Ç UP 0 /: · attvld: ¾ \ Z.;. : X1. d datta; d ata da cl a ti X · ': O idt.! SSiS 0 0: cs asa ta; OOitXXX sr; 3. to the .X // z cable; And X-OXY-OXY-OXY-OXY-OXY-OXY. ca dst a si rd Si d gives V: X do. rt a:; XX ': 3 XX' scds-sao scda? dl. 1 0 '0. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • •. 1 -X ssda-3-one esterase; • 0 0 (:) :) :) :) r r r r r r r r r r r r a a a a a a a a a a a. d y 'd% / // · &gt; / OZ.CPZZXX dssdlsdsta. ρβ 3 ld 5 Sdt dst :; apdt dsdp '/ /./' tX: 0 .X / p ;. / roz wing to 4) Xt: XXXI XZX; 1: 2 · oxy 3: X X; .X Xi asserts .cXXk; the sacristan to ãp &quot; a t • x a d d;) ted 00 Z VCd i g: aa f t- ;; (X, y, z). Γ / ./ΧΟ 0; / v / v / v / v / vv. 3 v t spyfc j :. OiOOa s acipacsias o o SS Opa v 'XXX. laat: s risccsa a da ...... d ddtii i: X'X &gt; XXdX stt idap 0v 0: sdts ..... a; X ;; X; 0 X eoo Zi d · '; d; d to 3 &lt; ta X / XZ XXX &quot; O X 0 0 'O' S 'S SS SS: idt 3 &quot; . X? XX: sC st. 0 'x ;. ei 0X0 'of X ·. . a: yv.v 0 &gt;. 0. ttd. &gt; litd s: S ta.ndO &quot; d......... • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - i ibc 1 · '* &gt;. Z oxxxx of X.tOZ- t s. to 11 XXOCOXO Proo Sd.s t .dst 00 | X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X a d d o o o o o o o o o o o o o o o o o o o o o o o o o. SSTI 'ΡΧΧΐΧΧ ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... ... I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I I SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS SS X 0: 00x0X30 .ot d &gt; t tsa '• • • • • • • • • • • • • • &lt; X-X-. C: a χχχχ Σ SIS dst Sib.scetd · o 15 tas dd a: 1 a: 3 /. • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • scs: ta a scdte ··: &lt; '&gt; s &gt;, 1 pacs at XX; be be be Γ Γ Γ Γ Γ Γ be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be be. (1), (2), (2) and (2), and (2) and (2) ) ad: a tb a ca X: X / st if ti s ss. tSiCy X: &gt; d is SSS 00 / ds dss. p: X: 'X 00:03 x / d x: xo / ·' sd. a further 1 oz οχο .0. ta tssassisi 2 &gt; P. a. (1), (2), (2), (2) and (2), and (2), and (2) PO 00 / a ta ac o o o o 0 ·. (3): S03s dSS 11i S0 O0XXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXX ................... st t i 0 0 to X i srai; X .X / 3 ', X00' p / Ϊ · ' &lt;Sil; siassic Z each. S Yes ii 0 '· Ϊ; S., i.e., q.sub.a, di.sub.it: a ¢: 30, a cs ss X./: x. 1 ...: 0 ........ X / d: id..t t X.t vs .........% edim ... c itatç .Code. ........ J., 1/1 / 's d-: ddt.rsstsird cs v.-pt 0 f; : Ο, Χ Χ Χ Χ Χ Χ Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò <03 t / c: / 3 · · · · · · · · If sti assairs s cpsa S3Ss.ss SSS ascbsi sS 0 /: / 0 /: ... ·>: ..: fCC:; ..;;.,; &Gt; XX 3. aad t esatssa da .L 0. t dst d 1 çlp): f ib; cslta t: pi.g.y 0: 0 '-: ./,/ 3: s; 1 d. tasess · dii. · &lt; ... • 1.3 •: • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • - and. ·: &quot; / X / XOO. Amino Acids were prepared according to the procedure described in Example 1. .0 0: X /: .X: d pl //.0; of 3b s r 2θ. ΟΡΟ X · · /. 1-one of the compounds of the invention. Cit; tia Si: 1 ii. at: a.s I Siti p 1 0: bii CiOP / 0 p'X'p.3, Χ / ΟΪ / 0 ρΧΧ.Χ. 3X &lt;: X 00./1 staa ataages 3 p 0. .x &gt; .00 // 0 i'iaX ti v »gt: / p t.X.V / spt. Ci ibi. 1. 1 - Ο · / 0 ': / OXpO / pO XXX /: 3 X; d isss st. cl. •: 0 sssic siss XO tt Z Z ct bX / p2b t: ss rel: IdS / X &gt; d / 03 S.SSSCSSSS SiS S.Satat:: 0 r; The baits of the &gt; cstigapa ϋ '' ta isasitid V. · s.ii idt: .// ': / 00' csstdss 3/00 ': /. s .ca. 3 xd 'isscclsca. ...: .Cd X at 14 o'clock o'clock "it this: 000 / :: d. ·. d. X; d: fvf.si: 1c ss ar s d SS a 3 times: &lt; p.sa dappsd. : t i t BGia i 0.1 6 Ca \ C ÇTG P. xlÇ vp :; 1 0 'p: \ vb CG of BB GCC-G Bd; 0-0 0 0 5BdB.Ç: d: G ' <3 BBg :: C.l b 0. J. lt. : 1 g. . (B) G B G B G G G P d Gb d Gb Gb Gb Gb Gb Gb Gb Gb Gb Gb Gb .GPBCíBG X, ·· \ PB- 1ΐ ϊ} ·. 1: GfGBpB B; G. G. OcOlpO: dl. G · .. · BBC: ••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• &lt; BtBGP: is OO · G ························································. d 'tVp: bPP: .GOB: βΡ' g Pp I; 'b; 0 0:, Β qu'B; pO-; G: B; S B 010 • p% d p ·. · '.1 h ld: d ·. l.l:; r &amp; s PPY 'p Çp · Ç1 ϊ:' p GP G. : 0: ·; 0 ITBxBcGC, ρΟρρΒ pd-d ·; G s, dp; .., ΟΟ'οΟΟ'ΐΙ 'CBG ΡΌ &quot; Px1: 0 CiPGt .1 G: p 11.) Gd: Oa-> '·; &Gt; V, .. · Ρ · Α rpOiOOiiiO! , 0: 0.0001 (10: 1). XBtB-GpG Op. GCCBC V -p. !. (GB 00: 00100 cg Pb: 0) V •••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••••• GBDBCBGO '0 0 0: B' SOGICB B ': GB' '' '' '' '' '' '' ''. &lt;. dioc PpGiB; C; 1 Âμl · CG; P βΡϊβ O ': · &gt; PN: BGG 1B, BGCG 0. pCGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGG In a preferred embodiment of the present invention, the present invention relates to a compound of the general formula: ## STR1 ## wherein: Cd pB: Binding to Compound B: Compound B: Compound B: Compound B: Compound B: Compound B: bgPb; bxy BB: B Cd O '0 OO' X. ············································································ <B: G \ ·· -i CfCBBido pp 0. OGB.B 'Β.ί.ί): ·: BB. BGCBC :. BGp. r &gt;. i. : 0t - ·. XV · -P ..; ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ ΒΒ BBBCpG: CÍB: CGSÍG: ÍBBGG: GB: BG: 1. CCBG B; 0 0 0.0.0:: 0 ·: * &lt; u: IcGldc &gt; &lt; pBBCCBG: GGG 1-: 1Bbbg; (I.e. .B ': BC .BC; C: CB CBG. : G: C, B; (1): Gd cCdBBxd BdG tBdG 1 d: vldadGj sp CBd &quot;: CdGCpdBBi 0 B x.-gp: xd:. &gt; ..... p; 00 G Ir; BCG. .ClGBB; BB C CBGCS; ; B: 0 BB B B C; W; 0, pPr: 0, pPr: 0, • • • • • • • • • • • • • • • • • • • • • • • • • • • • • " BdGC ¥: Y: d: B GiBdd G .GGBBC pp'-0 0: 0CU i ooí: &quot;'1; . & PP i> 0K &gt; C G G:: C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C ΒΡΒΒΒΒΒ li li li C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C C li li C C C C C C C C C C li li li li li li li li li li C li C li C li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li li BB BB BB: 0t B GB ..... G G; GB BBã d PB ........ BG ΠΡΟ - B B · 1. BG GG; G BB ΒΟΟΡΠG € B pilo OG GBP G 4. GC 1 GO GntBCB OGdB CbBtBGl GB vllGGiSPg G COGCBOlO (40) OOP B (ΙΡίΡΟΒΡ: OG: Còttgbcccbsc 'GB ρΒυΟυΤ'Β Ι-Β; ΠΙτοτΗβΙρβ (-G) G Gb: GGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgGgG g BGCbbuBGyB BCC GBGGI B d®: P1: T; B. , lp &lt; B. 1. GO® GO.yy: CPOCd H1 CBGC pQGC, ()) G; G,. G: G ΠΒϋΒ, Βυ T. Q B GB.CB BBBBÇBGPyGCí ·; B.Dl scb.C: B: XBBB.B: BG GGCCBB BCGCGPG CdGibBBG 1 GB: Bpt; B: BGB GB: .dTBBBBPBG CCBBGG .B CG (1) pBCBgGG &gt; B 0 · νΧ.Οί '; 0 ppg. &lt; P pP. ; B Β.ΒΓΒΛ? Β'Β BCG psB. B BPGGGG PB PGGGP.B 1.BiCipb: B The PPO; . (1), (2), (1), (2), (2), (3) and (6) (BGB BCB: GB) C: OG CBG BiaGBGOB / GGBCBpGGGr ('4.6) SituPdO PB PiB BBGBc CbCGPB GBCB · :; Od BGddCí: BC® P :. pi B •• Cd (0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, xd \ B · x CCG ···. d ·> B; OOO B> <0 -dCCB ..... 0. · 00 Oi: ^, χΡΒΡν -p vs ^ BB: G s { (b) BB (; dB: B Cc Γ; BBBClc 0 0 0 Cc. 5 ΒΓ K BG TBC! BBByC) GdB BBCGYi p 00; GB i 37; &lt; BC &gt; BBC 1: &lt; / RTI &gt; &gt; p <0 of the d .1; p ggbbg Δ: 0 c B 1: CiO OÒO: '· ·; (b) (b) CD ...; . ·; X-b.a x; · P.dxP dO-OCO it; . 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0: 1, : étc 000 \ ... d. : V. • PG: 0: 00: 0: 0: 0: 0: 0: 0: 0: cc i OOOí di pB 0 '.' Ο.ρ'χΐΡ iiv tO B d GBt • 0 .0: BBSdBa: (:: TB cbg PByb; gp.gg pi 0 pOBiddance: The results are summarized in the following table in which the results are shown in the following table. : C &gt; 0: CGGG GC 4: 0: '::::::::::: BCBdoa coo, ·· γ: 0 G.GBBG: BdBG of g Gr 0 B 0 t; Gd GByGy p -c 0.dpd: GBC G dec pG> d.lt.l GG m 0 Ο i 0 G v díscd • 1ΪΙ IddBBiB 0. Ge; P uc: 00000 0 · 01 G PG • x: & gt (1) and (2) and (2), and (3) and (4) and (4) and (6) x Β · · · · · · x x x x x x x x x x x x P P P P P P P P P P P P P P P P P P P A compound according to any of claims 1 to 4, characterized in that the compound of the formula (I): wherein R 1 is as defined in formula (I). 0 m CG ΒΪ CyBBCB.yBB CC CCGG 7 ' (4: Bd.) OU &gt; -vc Op ti BB x · Ό \ .d · the GBBBCt CBBdC \ 0 PG; GS'SG; PG BG 0: Ο ΟΙ Ι Ι Ι Ι i i Ι Ι Ι Ι Ι Ι Ι Ι Ι Ι Ι Ι &lt; x &gt; d BB ', · P BBCBBBGB: C BdTGBPB PPp; 100 B-0-00 X C'-B 'cmdc -0 5d: B G pp 00' • 0 v.7 V. ·· o. 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, .2; /. such as 2: -i 1 ... · &gt;: 11.0 :; 'Ii &gt; iq 16: 16 cU. : .00- · &lt; 0- &gt; &lt; tb &gt; &lt; tb &gt; .delta. = 0.01 g / mol. t is the same as in the previous section. t 0 or 3. p: 0; The results are shown in the following table in the following table: 4 11 i 1.1 00: 00: .00.0 ···: 1: 0. trlot. It has also been added to this subject; of Clt; 11C t ura / toco &gt; <4 to 1,111 rap dtco p:. i.e. 3 ''. the act and the ooto; te: iO: e | otdtl &lt; &gt; C · OO Xt; X-tr isad and 12 2 · n i: O OΟ; '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' ' and (d). / s; • 's, v vd: asac 1: te 2: d \ v dc v r; y: ppt 'ai cr 1; .2 1.1 Ot. When the doaoate of the C-; s .mryp O 5: 00.0, <0: o. ......... . the value of the value of the value of the equation is: tl &quot; -si d X dOCCÒ; 6 ··, .. c Π t .t: d, l tq. In addition, the results of the present work are summarized in the following table. i. X is O, X is O, X is O; X is O; X is O; X is O; X is 0; ; oo-pâOo of ioo &gt; The reaction mixture was cooled to -10 ° C / -0 ° C. (s), and (c) to (b) and (c) to (b) are as follows: • d: · ana a rásd: 2iol if ias idO OO 2 'I 11 o' ao ao XX XX xx ΟΟΟΐΟ act 10 · e Ό. 1: p: ·: 2 .0 d-4; 011 i dl ir .. • 4 d sv f -dic. - - · rs'sX dt or 00 td king atol (taaq 00: too seet: link 1; (A) and (b) and (b) of the compound of formula (II): wherein R 1 is hydrogen; ¾ t t Λ Λ Λ Λ Λ t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t t: &lt; ..... is; GSf! 2 ire gold X xx tdorl ladro 'ορθό tt o &quot; &quot; &quot; &quot; &quot; Ododo: see iiddi-idl ..... ei 0 d ata f ioo {1 ·· 3 ϊ o. At 6 o'clock, a doe of -4 to eaot gd te pote sac i. 1 to 0: 0 to 1: 1 to 4: 1 to 4: c dl a '], · .ii: t.l a d irdi ΐ t ii.ç J'l; &lt; / tb &gt; 10% &lt; / RTI &gt; Ot :. CQ XC r 0: 0: a a ... F rc to XX 2 r to οοΐϊ!.: * O. t 0 s' i &gt; 0% of allyla; tiq editss: llllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllllll In order to be able to do this, it is important to note that there is no such thing as a rule of thumb. .óe · ·; erl. The title compound was prepared from the title compound as a white solid (0.1 g). γ 14 o o V \. · '; p. ............... and in the presence of a compound of formula (I). eree 10 0s: d of: ededO &gt;: St ly 5 ... 6 et 16, is dl 0 or i d: ttx ls' '': aee. qÃ: 21 -s: l sa i oo d era ore this. all of them will be: and so on. Codt sro i. .Es: OO !. Ci will be tarará and 2 d 21 · l d -. ··; &lt; 'tae t apitt ttll d .; air is used as the solvent. read: to be read; asor. q ·· - this / d action; The composition of the present invention comprises the steps of: (a) preparing a compound of the formula: ## STR1 ## in which: ## STR1 ## is as defined hereinbefore. The compound of formula (I) s e e e e e Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ Ρ. • pp, 0 iaddl elasa roo reelesseèsest • ti es iersqS t o s i. tb______________________________________ tb______________________________________ . air is datoctodo 1: 2 o.t te rassaesea · \ i- q saoeseoísté .: oseeeso eeeess qs..s Ό .... pov: 00 • Ip; Ut: OsS: if quotients nc 1 -12 1 -t •• p S-. ·; . (s) of the eS: ret. to (d). W: . dl: S 'Ο, Ι'ΟΟΟΟ' '' '' '' '' '' '' '' '' 'a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a ΙΟΟ v v a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a a as i.e., et al., p. feet ....... .1: ¾ ρ: θ; 1:. p. pio · coptoçors dst Oh st: · d: L ϊ: i 3 3i ssét .1.0: ei. (11). The compounds of formula (I) are prepared by reacting the compound of formula (I) with the compound of formula (I). .: 1:: 1 &gt; tèo po.ro. .................. ; of the tara ·. :· a·. 1 1-. V is the ratio of the amount of the compound of the invention to the compound of the formula: There you are &lt; Ò 1; (i.e., tetramethoxyethoxyethane), and the like. The reaction was carried out for 2 hours. and the roesses are as follows: &gt;. (1) is the same as that of the other (2) and (2) is the same, • 1.11 .2. Sl &gt; eto reo eseqreto seed O 1. ·: 2 61) tors to the following: ss: oe.s dee Cs-tt: rt arae / seasecrsro doa 1 ..- 02 o .v .; 2: 2 té tea. 21: 1: 1: 1: 1: 1: 0 to 0; 0 to 0; (1) (1): (1) (1) (1) (1) (1) Td ma ta &lt; s &gt; oot if a-q: idldl o C t il o aerao ·: ·. (D) ISO / IEC ISO / IEC Directives. ti α and t i t i t i t i n t 1 to 0.1: 0. S 2 tfc:: erse toa seer t ·; dt;. Î ± βâ, † â, † â, € â, € â,ƒâ, € â,,â, : - ·· ν a C 1.: See N ·. · '1: 1; : o = 2,1,2. atoeto l. &lt;The.;' 1, 2, 3, 4, 5, 6, 8, 10, 10, 10, 10, 10, 10, 10, 10, 10, :. tt -ϊ,: ···. The 5 'to 5 diastereoisomers give the compound of the formula: Spitting: aq. the i.CP.CrO v -C ea of &gt; r ertareate C :; (1) and (2) and (3) and (4) and (4) and (4) and (4). Pit, and the pit to be squeezed; &lt; / RTI &gt; 0: Oc (i) p. Cd. (14) of COOΝ \ a to et. to be cleaned; e: pe? - r 0: 0 elt: è. ·· PC açor.d; &gt; 0 OOP 0 0 re .0 V 0 ·: i v- \ y. ), • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • • · Sa ee.ie re 1. dsa 1,0 ae CP Οχ · 'Ό Co. C O H O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O O! The compound of formula (I) ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ ΌΟΐ. aeedaia r C i iia) ni> 0c CCpv 0; p .1. PP, for capping. .Alpha., .Alpha., .Alpha., .Alpha., .Alpha., .Alpha., .Alpha., .Alpha. pc d O-l.Cpé.p ç ta tal.) qaa ee S ··· sV there; &lt; / RTI &gt; &lt; / RTI &gt; &lt; / RTI &gt; &lt; / RTI &gt; , for example, to be able to be able to do the same thing, and to do the following: .............................. .................. air and CdP; aedo 0 ner: ple 0 · 0 1 Peai ... ... ee of eate; j>. t is the p ooe eaaaaaaaaaa. yl ester; C: K &gt;tas;). and gave birth to CP. 0 d 1 of the tapeie .. '; aqae (tOa r ΡΡϊΐί 0 c e; dr t; t 0 t; a e d 0 c <or the eco <or. Ratio of d; a and tirape • C &gt; O0 ', d0.tC:' 0Ò ': &gt; % p: V &gt; OOCOOO 0 iree. as · ρ \\ &gt; ' Pp .PPi a. i.e. 00.times.X.- et d 14 f and dl asue and i.t 1 and the aeedaieo c '. 0: 0). pe r; The reaction mixture is cooled to 0 ° C. - - - - - - • • • • • • • • • • • • • • • • • • • • • • C0. j.) ρee a; s aspf rer ad of t. OOOOOO ia ·; taree. to PPd. Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò Ò. laughed # v: rriaaeo ee pl; and a; d; and to the method of the invention. roa Ceateal; ie Coma and Ore. (to be followed by the day-to-day operations of the company) , Which is to be found in the following table: (a) (b) (c) (b) & numsp &numsp; &numsp; &numsp; &numsp; &numsp; &numsp; &numsp; (d) and (c), and (c) the reaction is carried out at a temperature of from 0 ° C to 0 ° C. &lt; d &gt; 0 &lt; / RTI &gt; The peptide is. •P &lt; \ d; ' . As such, there are many different types of compounds. C &gt; Oi &lt; / RTI &gt; ^ sOpd eers dd qráo. d sis: .v 'd ·. cpp. Atiríreàa i rrr: 1Ό ..... p .0. P and rios a .......... ir.): Ea.aea O O OCCO will be in the air and airspace; : it lies at the heart of the UYÍ: aeie; : The laughing one; P> 0, P <0.05, P <0.05. .............. ; s and s .0) P &lt; / RTI &gt; d-i lo qs.:e;adr, ne iia; (i.e. The invention relates to a method for preparing a compound of formula (I). the network and the Caa '.1::: P; &gt; amino acid; -v ', and qe ipiiiéi; lee · (5 4 | &lt; (a) (b) (c): (a) s 'a a \ Õ &quot;' 0 and a and et; to e: e | &gt; e for P0, 0, 0, 0, 0, 0; Eur-lex.europa.eu eur-lex.europa.eu C ·· &gt; · C O P c · ·; C (O) -alkyl; 0, '. . ·; i. i of this of: O0. tb______________________________________ tb tb______________________________________ tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb tb eme tt el and be: C qC q. &gt; 0 t; and (a) : i. p is 0, and p is 0, 0, 0, 0 and 0, respectively. ; and out of the way. 0 e>: a e d a te r a re a tica t.PCtCts X a dl s'.s dl s peeitirs ;; 010, 0 to 0, 0 to 0, 0 to 0; idr d \: ;; p: λaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa and the CP is going to &lt;v; &gt;remove; The reaction mixture was stirred at room temperature for 1 hour. d apt r ço C X: v .: a · air; Urania. d-a Χχ ·; XaP XX (a) to (d); (c) to (d); ax r: &gt; &lt; / RTI &gt; Gre isopropyl sulfate P 4 ki f: r 303 X 3 .etc a:, dd} &gt; 3: C: G: G33: X33 is ox Oxide. 1, 2, 3, 4, 5, 6, 7, 7, 8, 9, 10, and 10: aarGadra Td, ·: &gt; c c atr: Λ V · 'arr par' Λ 'V u: 3 x-dpã de pa-n.t 00 \' λ A c. 'Πΐίϊ XO i; X3, d; .Gy ········································································· Ge V r ooo village r d a rrrr; 3 0. (a), (b) (b), (b), (b), (b), (b), (c) and (c) (a), (b) and (b) of the compound of the formula: (a) and (b) of the general formula (XX): ## STR1 ## in which X is a C and X, X: X: X: X: X: X: X: X: X: X: X: &lt; 1 X X X 3: aXT dd U-.GX XX X ra Ge. j adtae xi: 0 c. Xa 300 and 3 to Ur: XO (Xa): Xaaa: Xaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa Ox. 36-; parapPa X 3 to at least 1% to 0%; and Xa% to 3% to 3% to 3% to 3% to 3% to 3% to 3% 3 X 1: 3: 1 X 2 X 2 X 2 X 2 X 2 X 2 X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X (a) Xaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa : xx 3 =:: 0x Olad.] d.addr: e: &quot; .l3: = ad; U: GtX; : 3 to burn with er, G ........ U CÍ-a ii.ar i.adv s &quot;'····· X, Xi, Xr and ....... 22 X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X X 3 X X X X X X X X X X X X X X X X X X X X X X X X X X X X X 3 : 0 G · X XC d> gxx 133; axt. · '3 0 vara $; ata' X.pyG; aa adca XX yx &gt;;; &gt; a doderer is aaonà. X3 .: / Xr Al = 0: 0: 3 a.m. The X-ray is the X-axis of the X-ray diffraction curve.  € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ â € ‡ χ> Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0. &lt; (X: X), and (X) (X) (X), where X = 3.00 to 3.00 to 3.00 to 3.00 to 5.00 to 5.00 to 3.00 to 3.00 to 3.00 to 3.00 to 3.00 to 4.00 to 4.00 to 3.00 to 3.00 to 4.00. (a) and (b), (b) and (b), and (c) GXe ...... XXr rar a aaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaaa : Dxtar X &gt;. G 3 X "- ixrr 03 U 3X3 aid SX-G pa rie% i ν '. and Ο χ, 3: χ, Χχ3 for Ox .X · 0 'ot. ta dd v.dX UàX trai ar.bd 03 5 T.Ti Λ: 000c; Cir: Ca P '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' ' (Xd V Od a Χ:: dd dd dd X X X X X 0 0 0 0 0 0 0 0 0 0 Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο Ο C '' XX ç of the i-dralf: x. &lt; χ ... a d ar; X = 0, x 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, 0, DG V: :: d. X-ray powder. . X · X a daDr v '. &Gt; aaa aa atiti, CíUei 33: '' '' '' '' '' '' Χ XX 1 o 10, - O di spo. iaa ff a; The invention relates to a method for the preparation of a compound of formula (III). rr; it is rare to see the results of this study. &lt; Ϊ i radarae 03 Ò Ò aa aa aa aa aa aa aa aa aa & X> X is from 1 to 10; and X is 1 to 3; Ó 0 ap: a t a. tri. apa. -i '= ··· are ald ed Q S .Ti x QX · tid; .radeà 3 X1 te a. ·. Xytx i.aada &gt; "aoa: itXaa. 3 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 ' · P-O 0 30 ν 'si 3 V. 3: 0 d X: t; air d &lt; ............ pi.Vi; ; and X (3; Cr-X-C3 3 &quot; 3 .0: 0. Dy having the pear r &gt; 3 t 3 X X X X X X X X X X X X X X X X X X X X X X .1: 0 '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' '' • '3000' x XX. '. aaarru aaie roitGi etaa street: 'X: ···; the V w: X ee:. and ia ar, xry ··: r x; d XX ddaat. &gt; 0 'C3 :. HOLLOW. 3 · &quot; 0-A and 3-O- t xc d (3 aa, by plowing Οχ dve xx ip Gr a 1 Oiaa, • XX çp 0O; X and diaraatte d ΧΟΧΧΪ, ΟΧΧν, ΧΟΧοοΧΧ: O-: -O-0D.) CláXXC & NXXXX XXlOO: ΟΧΟΧΧΧΧΧΧ, ΟΧΧ Χ V V V...................... Ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ ϊ. aa C'i a s' oex% .... ... · &gt; .. s -d :, and ci d (d: i .0,) cc 1 a; (a) 0: 0: 0 or 90%; iles; (&quot; 7 &quot;), from the ad d air XXX, 1 ur 9: 00 to 1: 1, and 80: g '; OS: cs syria SSS SCO ssmcnmxx to 10 (; .d The dCO: • VV oee • V Civ, ··························· (1) to (2) to (3) to (5) to (5) to (5) to (6) (a) and (b) (c) and (b) are as follows: (a) The following table shows the results of the present study, which are summarized in the following table: 1. The method of claim 1, wherein: (a) X is: &lt;; &gt; 3 $ v: UX d turMn 0. sp vv: ·. &Gt; ia : to GC SUBSCO: C \ CtC; (X-ray diffraction). ΟΠ tssísrsd; Vi 6 ;: t; The reaction mixture was cooled to 0 ° C. The reaction mixture was cooled to 0 ° C. . ;: sap: aa da I lss: a: sst, a.r O dd Oa i &lt; l &gt;: &lt; / RTI &gt; &lt; / RTI &gt; s ds ssiadi cac 40 0 '1 v 3 c S,: 6, 3, 12 ... 13, aa to PP f õ dlapaa. Sla ao o vi \ .1: &lt; ΐ: ÍSj.d &lt; i &gt; Cd CO XX X 'X- 0 0 OdX · OCO ã d': Pa sd ò. OVA 0: 1: 1: 1: 3: 1 &lt; s {Pi may be assumed to be 1 ¾ ii 0 pa las pa pa pa pa pa pa pa pa pa pa pa; ; &quot; &lt;d; X-ray diffraction (X-ray), X-ray diffraction (X-ray) X çad O a dl orla la Ui; 1a to 1a; (Xa Ix XX: C V pCXc Sis Is issio argui taot ssra 0.1 x 0 sossiiís ds Idlli X ': lvi The law and Hl ddldi. i.e. 060 or lO4, &lt; 11 &quot; s d a sai g dl 4 .i a; f, <X1> X <x <X <X <X <X <3. λΡ ;,. 13........ ......................................... X is O; X is O; X is O; ssa par X çx ga 'dflssao ca ssto a Si V · v 0 salt: is ss a sis; Go to i i 'a &gt; V · 1 day s &gt; : i; ox 'S; et CCy sc; Γ Γ Γ Γ Γ su su su su su su su su su su su su su su su su su su su su su Γ su Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ Γ (s), and (c) to (c): (a) (b) (c): (a) 1 to 22: 1 to 22: 1: 1: 1: 0 to 0: 1: 0 to 1: a.14 ç.t.ç. 's sfa; &lt; (I.e. doo pal 3 '. Cl.:. Cl: 4 '. The. ss dS; the post 0 01 floor and 2ddi * Pf Çd; 1; X: X. i sar> 3 1. Φ solder pass SSSii v 0 of the jarsp d ·:. Cl '·························································································································································································· tb______________________________________ lio. (1) and (2) and (2) and (2) and (2) and (2) and (4). i aa a.ds al. (1), (f), 7.0 (s); (a) to (b) to (a) to (b) to (c) to (g) cl. I flew to Paris. ar sca, P ·; _. ·:: Ls • 0 OCSS.ddSS; The compounds of the present invention may be prepared by the following methods: V; : 11 Cl to X -; &quot;.: Λ o! 000 0 .........: 3dl ϊ ...... fdõ'd C 11: Xli 0: X: á rd ciea to sodoa ........ c. 0 to 1 of the cough. (a), (b) and (b) of the general formula (I): ## STR1 ## wherein X is as defined above. (1) and (2) and (2), and (3) and (4) and (4) and (4). 3. a oi cc &gt; ls 1331 4a4a ai iS dl diXoiCIO: ... D ...% · ········································· 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: 1: i 7 s, ses sars si a 0 s SSd 00SCO 1 gga Ss Cs &gt; 6S stafea ialC SO or tSSsS V. eagatdíslr 33 a dSi ga rd acsaa X:: X 4 ei; :  € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒâ € ƒ 1 to v., CvS 10 Pbx to Cyspc: X Cie-i, P c: 1 to be thus: · 0 c vP: 'a, s: \ v &quot; 1 orlo 1 dapar a, SIS1 OvrCtov Oo ssioa Ira: ssto (36 d_L P x .000 to i.e. of O-O-X1 to OT1 to acetoxy. 0: 0.1. sS Sid and ooopooo 0 Ό. &gt; 'li ... i. V 0. 3) i-P 0: ls Si acad.ossa .0; The title compound was prepared from the title compound as a white solid (0.8 g). 1 H NMR (DMSO-d 6):? is / pCl / 0 Odeagala ssa i. a. x t 611; &quot; &quot; Od Xo o.ttasss; / fd dlsd: ....... dOX.Xi OO ssa ar 1 ass ala C '' so so so so so Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol Ol eco rd;:.? &lt; tb &gt;2;, d: 10; lid 10; 21, 22 d 23; \; X l 21vM> of the d-, xo>, xi. 'Χ. ···· X i ??; c. &lt; 21 carat? aar, Ps ardei? to give; ΟΟ.ΐι.2. ............. .All of ΟΧΧΧΧ'Χ pi 10? X ' 0 eca: p? caa?, - Pard.? ; B Q d of the 2 acts at the same time? of the trait: · · · · · · · · · &lt; 21% to 25%. v .1 i v d ·; , 2.00.22. Cover agac dd: · IX TlídX XX. X x.v mát x .aa; · X'xgxogog at the air X nCOXO-a agia ÒX.lO d · .; The title of the present invention relates to a process for the preparation of a compound of formula (I): wherein R 1 is as defined in claim 1, Pd; ': t? D? P. 1. Staaa. d X 1; · bo; x taaa / r. acac from ao.aa? c x Pa to Η? sx / and icodx doo to: cd; dai CX (a -X tra &lt; ai a a a a a <? s tra a a? XX'-xo x · ρο-χο; .X Xi &lt; ν · ν \ d 1 V · '; d. 2 ": adx a i .d eai as a: p x?, Oapa.a tíd: .áaoP X t: <xx 1: 15¾¾; χχ ΧΡ'ΡΧΡΧοΡ C: 'i; X face the dal • s. -V:; U? the carpentry; xx or p.l.d •: 0x x d 0-dd o Gd d • ;. ptapídip; to 0 .OCX arca i.caa i Ί Xo-G a noa: td i rlsta X: XXi X an P; iC XdataPiPa gives PP s t 'O. IXX. a-a dlp; ·· X -XX spar Paa dta al; S &gt; il p:; to bring the support to the X-axis; X X t: aaadr y.P ar? adi Cia, aaadPd: d. .The. (a), (b) and (b) and (b). (CDCl3):. ; d. X · aa a? rar r; 1a; Xió apar ?: Γ. ' X. YXXXXXXXXX. a. alsira dl; 1 O2: appaat ^ arp Papp PiiaPiP a a h aatr? (1) and (2) and (3) and (4). a ddpsrppac ddédtc ...... Ο Ό ..... 1 O; . &lt; The composition of the present invention will be described in detail below. ; PX; • Xi Xaaaa P or XtXlpiXid Xaa? for air; X:; Xi in the appended Table X.2 XiXXXOXXX- i.id; , d. of the compounds of formula (I) and (III) of the compounds of formula (I). AX da ...... m ': d · *' espoa; . : ò: .s The CXXX 00 <1. XXiX ip; ..... X ra x a a x aa 'XX ϊχ.ιχ pasxxaa .....; the a? :: V.i: ad. X 1, X 1, X 1, X 1, X 1, X 2, X 1, OXX XXX idioxioo or la)? d 0: 0 .no OXi 1 'and d :; rp ·· '·· dl. \ 1 {I}; to the apiad; XiO a i 1. Pado P &gt; 0 X 0 00.1 d? x to ip. Remove ax; the chip of the lappaçaa ria iÒX and prol. to Cl. a? sp? (a), (b), (b), (b), (b) and (b) and (b). ??? d p? r i a i, .m i; P p Pa P p d d x D x D x D x D x D x D 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 : a? PpO PP a. the iia: to give: 1 d Ir 1 ΧίΟΧ ·:, or \ d: ld li \. · d ·. 11. CQSAD; AR I GO Box of Praoc: (4: 1 Χ Χ Χ i i aa aa aa aa aa aa aa aa aa aa aa aa aa aa aa aa). X-ray diffraction pattern of the X-ray diffraction pattern is shown in Fig. Tali ri Xi Xo, rxradta a &gt;;; d aft (1 Mia); ¹H-NMR d.i. iito a ?? C; S; a a. a a Pa) d C irrtarraatd p. Q? aPdilxa • vin a; of the ParaP .. ································ Exxo r gx to lidrpáx p. X · 222 aor? ΡΡχ Face ia 1 -V> d 1 V X a ·. ·:, S ...... d · · · ·. Fig. CiX: · aaap O Cv; and f; to XX. PidP? <p: dtl? .22 i attracted: xijaapao dr? bxxxxs d; S; gaaPPd. dd. ·:: v · ·. · ?. vgyd: &gt; a a t a a 0: ΧΧΧΧ: 0: 0: a ccpcpP. X XX: X: X '2 x p; p'P? Dda 0: 0 aa. • -.sà.i rivaaaal td &quot;,; was going to the action '·. Eur-lex.europa.eu eur-lex.europa.eu The? aa p .0? of Aard. 1 of 2: 01.1