PL398703A1 - Pochodne aromatycznych imidazolidynonów i ich zastosowanie - Google Patents

Pochodne aromatycznych imidazolidynonów i ich zastosowanie

Info

Publication number
PL398703A1
PL398703A1 PL398703A PL39870312A PL398703A1 PL 398703 A1 PL398703 A1 PL 398703A1 PL 398703 A PL398703 A PL 398703A PL 39870312 A PL39870312 A PL 39870312A PL 398703 A1 PL398703 A1 PL 398703A1
Authority
PL
Poland
Prior art keywords
formula
aromatic
derivatives
imidazolidinones
substituted
Prior art date
Application number
PL398703A
Other languages
English (en)
Other versions
PL223830B1 (pl
Inventor
Jadwiga Handzlik
Katarzyna Kieć-Kononowicz
Ewa Otrębska
Maria Kaleta
Original Assignee
Uniwersytet Jagiellonski
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Uniwersytet Jagiellonski filed Critical Uniwersytet Jagiellonski
Priority to PL398703A priority Critical patent/PL223830B1/pl
Priority to PCT/PL2013/000044 priority patent/WO2013151450A1/en
Publication of PL398703A1 publication Critical patent/PL398703A1/pl
Publication of PL223830B1 publication Critical patent/PL223830B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/96—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Wynalazek ujawnia pochodne aromatycznych imidazolidynonów, o ogólnym wzorze I oraz ich farmaceutyczne formy odpowiednich soli addycyjnych z kwasami, w którym to wzorze I, R1 oznacza fenyl podstawiony jednym lub wiecej podstawnikami alkilowymi, fluorowcowymi, alkoksylowymi lub naftalen, fluoren, fenantren, antracen, pyren, R2 oznacza (nie)podstawiona piperazyna, (nie)podstawiona piperydyna, morfolina, amina I rzedowa. Wynalazek obejmuje tez srodek leczniczy i zastosowanie zwiazków o wzorze I do wytwarzania leku uzytecznego do zapobiegania lub leczenia chorób o podlozu bakteryjnym.
PL398703A 2012-04-03 2012-04-03 Pochodne aromatycznych imidazolidynonów i ich zastosowanie PL223830B1 (pl)

Priority Applications (2)

Application Number Priority Date Filing Date Title
PL398703A PL223830B1 (pl) 2012-04-03 2012-04-03 Pochodne aromatycznych imidazolidynonów i ich zastosowanie
PCT/PL2013/000044 WO2013151450A1 (en) 2012-04-03 2013-04-02 Aromatic imidazolidinone derivatives and their use in the treatment of diseases of bacterial nature

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PL398703A PL223830B1 (pl) 2012-04-03 2012-04-03 Pochodne aromatycznych imidazolidynonów i ich zastosowanie

Publications (2)

Publication Number Publication Date
PL398703A1 true PL398703A1 (pl) 2013-10-14
PL223830B1 PL223830B1 (pl) 2016-11-30

Family

ID=48428591

Family Applications (1)

Application Number Title Priority Date Filing Date
PL398703A PL223830B1 (pl) 2012-04-03 2012-04-03 Pochodne aromatycznych imidazolidynonów i ich zastosowanie

Country Status (2)

Country Link
PL (1) PL223830B1 (pl)
WO (1) WO2013151450A1 (pl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL231082B1 (pl) * 2013-10-28 2019-01-31 Univ Jagiellonski N3-aminoalkilowe pochodne 5-arylidenohydantoiny i ich zastosowanie do hamowania wyrzutu leków
CN109942555A (zh) * 2019-04-24 2019-06-28 扬州工业职业技术学院 一种苄基取代的苯并呋喃-咪唑啉类抗水稻纹枯病化合物及其制备方法
CN109942554B (zh) * 2019-04-24 2021-06-04 扬州工业职业技术学院 一种新型杂环低毒高效农药及其制备方法与应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE910913A1 (en) 1990-03-20 1991-09-25 Sanofi Sa N-substituted heterocyclic derivates, their preparation¹and pharmaceutical compositions containing them
PL198993B1 (pl) * 1998-11-13 2008-08-29 Univ Jagiellonski Collegium Me Nowe aminowe i hydrazydowe pochodne 5-arylideno-hydantoiny
DE102004003811A1 (de) 2004-01-25 2005-08-11 Aventis Pharma Deutschland Gmbh Substituierte N-Cyclohexylimidazolinone, Verfahren ihrer Herstellung und ihre Verwendung als Arzneimittel
FR2903695B1 (fr) 2006-07-13 2008-10-24 Merck Sante Soc Par Actions Si Utilisation de derives d'imidazole activateurs de l'ampk, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
WO2013151450A1 (en) 2013-10-10
PL223830B1 (pl) 2016-11-30

Similar Documents

Publication Publication Date Title
DOP2017000081A (es) NUEVOS COMPUESTOS ANTAGONISTAS DE INTEGRINA aVß6
CR20140519A (es) Derivados de benzamida para la inhibición de la actividad de abl 1, abl 2 y bcr-abl 1
CR20140332A (es) Inhibidores de bromodominios
EA201490949A1 (ru) Ингибиторы киназ
UY35998A (es) 1-(3-(tert-BUTIL)1-(p-TOLIL)-1H-PIRAZOL-5-IL)-3-(4-((2-((6-ETILPIRAZIN-2-IL)AMINO)PIRIDIN-4-IL)METOXI)NAFTALEN-1-IL) UREA Y SUS SALES DERIVADAS FARMACÉUTICAMENTE ACEPTABLES, COMO INHIBIDORES DE P38 M AP QUINASA
PH12015502036A1 (en) Inhibitors of the kynurenine pathway
CY1121677T1 (el) Ενωσεις διμεθυλοβενζοϊκου οξεος
RS54526B1 (en) USE OF PIRAZOLOSPIROKETONE DERIVATIVES AS ACETYL-COA CARBOXYLASE INHIBITORS
MA40059A (fr) Inhibiteurs de la phosphatidylinositol 3-kinase
RS54730B1 (sr) Inhibitori beta sekretaze
UY34451A (es) Derivados de uracilo como inhibidores de la quinasa axl y c-met
CU20150084A7 (es) Derivados del ácido 4-((1,1) bisfenil -4-il)-3-(3-fosfonopropanamido)butanoico,activo como inhibidores de nep(endopeptidasa neutral)
IN2014DN07509A (pl)
CR20150244A (es) Trans-4-{2-[4-(2,3-diclorofenil)-piperazin-1-il]-etil}-n,n-dimetilcarbamoil-ciclohexilamina para el tratamiento de síntomas negativos de la esquizofrenia
RS54899B1 (sr) Jedinjenja tetrahidropirolotiazina
AR085308A1 (es) Formas solidas del inhibidor de girasa (r)-1-etil-3-[6-fluoro-5-[2-(1-hidroxi-1-metil-etil)pirimidin-5-il]-7-(tetrahidrofuran-2-il)-1h-benzimidazol-2-il]urea
PH12016500322A1 (en) Amide derivatives as lysophosphatidic acid receptor antagonists
PL398703A1 (pl) Pochodne aromatycznych imidazolidynonów i ich zastosowanie
CO7160116A2 (es) Derivados de pirimidinona como agentes antimalaricos
EA201391793A1 (ru) Новый способ синтеза 7-хлор-4-(пиперазин-1-ил)-хинолина
EA201301136A2 (ru) Новый способ синтеза (2e)-3-(3,4-диметоксифенил)проп-2-еннитрила, применение в синтезе ивабрадина и его фармацевтически приемлемых кислотно-аддитивных солей
EA201301235A1 (ru) Новый способ синтеза 3-(2-бром-4,5-диметоксифенил)пропаннитрила и применение в синтезе ивабрадина и его фармацевтически приемлемых кислотно-аддитивных солей
AR082766A1 (es) Derivados de quinolizidina e indolizidina
DOP2014000116A (es) Inhibidores de la péptido desformilasa
CO6680616A2 (es) Compuestos de tiofeno 2.3.5- trisustituidos y usos de los mismos