PH25389A - Novel thiazole derivatives active on the cholinergic system, process for obtention, pharmaceutical compositions - Google Patents
Novel thiazole derivatives active on the cholinergic system, process for obtention, pharmaceutical compositionsInfo
- Publication number
- PH25389A PH25389A PH36616A PH36616A PH25389A PH 25389 A PH25389 A PH 25389A PH 36616 A PH36616 A PH 36616A PH 36616 A PH36616 A PH 36616A PH 25389 A PH25389 A PH 25389A
- Authority
- PH
- Philippines
- Prior art keywords
- obtention
- pharmaceutical compositions
- thiazole derivatives
- cholinergic system
- derivatives active
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/84—Naphthothiazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8703398A FR2612187B1 (en) | 1987-03-12 | 1987-03-12 | THIAZOLE DERIVATIVES ACTIVE IN THE CHOLINERGIC SYSTEM, THEIR PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH25389A true PH25389A (en) | 1991-06-03 |
Family
ID=9348897
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH36616A PH25389A (en) | 1987-03-12 | 1988-03-09 | Novel thiazole derivatives active on the cholinergic system, process for obtention, pharmaceutical compositions |
Country Status (27)
| Country | Link |
|---|---|
| EP (1) | EP0283390B1 (en) |
| JP (1) | JPS63243080A (en) |
| KR (1) | KR880011135A (en) |
| AR (1) | AR243515A1 (en) |
| AT (1) | ATE86249T1 (en) |
| AU (1) | AU612350B2 (en) |
| DD (1) | DD274028A5 (en) |
| DE (1) | DE3878708T2 (en) |
| DK (1) | DK170162B1 (en) |
| ES (1) | ES2053778T3 (en) |
| FI (1) | FI881152A (en) |
| FR (1) | FR2612187B1 (en) |
| HU (1) | HU198916B (en) |
| IE (1) | IE60173B1 (en) |
| IL (1) | IL85704A (en) |
| MA (1) | MA21207A1 (en) |
| MY (1) | MY103233A (en) |
| NO (1) | NO170081C (en) |
| NZ (1) | NZ223845A (en) |
| OA (1) | OA08871A (en) |
| PH (1) | PH25389A (en) |
| PL (1) | PL151889B1 (en) |
| PT (1) | PT86952B (en) |
| SU (1) | SU1604157A3 (en) |
| TN (1) | TNSN88020A1 (en) |
| YU (1) | YU49688A (en) |
| ZA (1) | ZA881764B (en) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6440474A (en) * | 1987-08-04 | 1989-02-10 | Hisamitsu Pharmaceutical Co | Novel 2-substituted aminothiazole derivative |
| JPH0753666B2 (en) * | 1987-09-14 | 1995-06-07 | 久光製薬株式会社 | Anti-inflammatory agent consisting of substituted diphenylthiazole derivative |
| FR2656610B1 (en) * | 1989-12-29 | 1992-05-07 | Sanofi Sa | DERIVATIVES OF 2-AMINO PHENYL-4 THIAZOLE, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION. |
| EP0535227A4 (en) * | 1990-05-29 | 1993-08-18 | Nippon Soda Co., Ltd. | N-substituted heterocyclic amidine derivative |
| FR2677021B1 (en) * | 1991-05-31 | 1993-10-01 | Upsa Laboratoires | NOVEL THIAZOLE DERIVATIVES ANTAGONISTS OF ANGIOTENSIN II RECEPTORS; THEIR PREPARATION METHODS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. |
| WO1992021666A1 (en) * | 1991-05-31 | 1992-12-10 | Laboratoires Upsa | Angiotensin ii receptor antagonist thiazole devivatives |
| FR2692893B1 (en) * | 1992-06-24 | 1994-09-02 | Sanofi Elf | Branched alkylamino thiazole derivatives, processes for their preparation and pharmaceutical compositions containing them. |
| AU4982293A (en) * | 1993-03-02 | 1994-09-26 | Fujisawa Pharmaceutical Co., Ltd. | Novel heterocyclic compound |
| FR2714059B1 (en) * | 1993-12-21 | 1996-03-08 | Sanofi Elf | Branched amino derivatives of thiazole, processes for their preparation and pharmaceutical compositions containing them. |
| FR2735777B1 (en) * | 1995-06-21 | 1997-09-12 | Sanofi Sa | 4-PHENYLAMINOTHIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| FR2754258B1 (en) * | 1996-10-08 | 1998-12-31 | Sanofi Sa | AMINOTHIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| GB9705428D0 (en) * | 1997-03-15 | 1997-04-30 | Knoll Ag | Therapeutic agents |
| ES2237919T4 (en) * | 1998-06-18 | 2007-05-01 | Bristol-Myers Squibb Company | AMINOTIAZOL INHIBITORS REPLACED WITH CARBON OF CYCLINE DEPENDENT KINASES. |
| US6218408B1 (en) | 1999-06-30 | 2001-04-17 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
| DE60034783T2 (en) | 1999-04-22 | 2008-01-31 | H. Lundbeck A/S, Valby | SELECTIVE NPY (Y5) ANTAGONISTS |
| US6989379B1 (en) | 1999-04-22 | 2006-01-24 | H. Lundbick A/S | Selective NPY (Y5) antagonists |
| US6340683B1 (en) | 1999-04-22 | 2002-01-22 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (triazines) |
| US7273880B2 (en) | 1999-06-30 | 2007-09-25 | H. Lunbeck A/S | Selective NPY (Y5) antagonists |
| US6225330B1 (en) | 1999-06-30 | 2001-05-01 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (tricyclics) |
| US6214853B1 (en) | 1999-06-30 | 2001-04-10 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
| US6222040B1 (en) | 1999-06-30 | 2001-04-24 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (tricyclics) |
| US6699866B2 (en) | 2001-04-17 | 2004-03-02 | Sepracor Inc. | Thiazole and other heterocyclic ligands for mammalian dopamine, muscarinic and serotonin receptors and transporters, and methods of use thereof |
| WO2003061655A1 (en) * | 2002-01-16 | 2003-07-31 | University Of Virginia Patent Foundation | 2-aminothiazole allosteric enhancers of a1 adenosine receptors |
| DE10251513A1 (en) * | 2002-11-04 | 2004-05-19 | Basf Ag | Compounds with 5-membered heterocycle linked by amino- or phosphino-methyl to a benzene ring with an ortho-hydroxy, alkoxy, thiol or amino group, used as multidentate ligands in olefin polymerization catalysts |
| JP2007261945A (en) * | 2004-04-07 | 2007-10-11 | Taisho Pharmaceut Co Ltd | Thiazole derivative |
| EP1904491A2 (en) * | 2005-05-31 | 2008-04-02 | Vertex Pharmaceuticals Incorporated | Heterocycles useful as modulators of ion channels |
| KR20110137941A (en) * | 2010-06-18 | 2011-12-26 | (주) 에빅스젠 | Novel thiourea or urea derivative, process for preparing the same and pharmaceutical composition for preventing or treating aids comprising the same |
| RU2456284C1 (en) * | 2011-04-12 | 2012-07-20 | Федеральное государственное автономное образовательное учреждение высшего профессионального образования "Уральский федеральный университет имени первого Президента России Б.Н. Ельцина" | 2-aminopropylmorpholino-5-aryl-6h-1,3,4-thiadiazines, dihydrobromides and 2-aminopropylmorpholino-4-arylthiazoles, hydrobromides showing antiaggregant action |
| CN107438435B (en) * | 2014-11-10 | 2020-12-04 | 埃弗里斯生物有限责任公司 | anti-HCMV compositions and methods |
| CN115160207B (en) * | 2022-04-21 | 2023-09-26 | 烟台大学 | Benzoyl thiourea compound, preparation method thereof and application of red tide algae algicide |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2975182A (en) * | 1959-11-16 | 1961-03-14 | Paul A J Janssen | 1-(aroylalkyl)-4-(heterocyclyl) piperazines |
| FR2092714B1 (en) * | 1970-06-11 | 1974-03-22 | Melle Bezons | |
| CH583232A5 (en) * | 1973-02-02 | 1976-12-31 | Wander Ag Dr A | |
| DE3135250A1 (en) * | 1981-09-05 | 1983-03-17 | Basf Ag, 6700 Ludwigshafen | TRICYCLIC THIAZOLYLOXAMATES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM |
| US4552886A (en) * | 1982-06-07 | 1985-11-12 | Eli Lilly And Company | Fungicidal pyridylmethyl-amines |
| FR2581063B1 (en) * | 1985-04-30 | 1987-07-17 | Chauvin Blache Lab | AMINO-2 THIAZOLES N-SUBSTITUTED, THEIR PREPARATION PROCESS AND THEIR APPLICATION IN THERAPEUTICS |
| HUT43600A (en) * | 1985-06-22 | 1987-11-30 | Sandoz Ag | Process for production of new thiazole derivatives and medical compound containing those |
-
1987
- 1987-03-12 FR FR8703398A patent/FR2612187B1/en not_active Expired
-
1988
- 1988-03-03 AU AU12662/88A patent/AU612350B2/en not_active Ceased
- 1988-03-08 MA MA21448A patent/MA21207A1/en unknown
- 1988-03-08 DD DD88313502A patent/DD274028A5/en not_active IP Right Cessation
- 1988-03-09 DK DK128688A patent/DK170162B1/en not_active IP Right Cessation
- 1988-03-09 PH PH36616A patent/PH25389A/en unknown
- 1988-03-10 AR AR88310267A patent/AR243515A1/en active
- 1988-03-10 NZ NZ223845A patent/NZ223845A/en unknown
- 1988-03-11 OA OA59299A patent/OA08871A/en unknown
- 1988-03-11 DE DE8888400572T patent/DE3878708T2/en not_active Expired - Fee Related
- 1988-03-11 FI FI881152A patent/FI881152A/en not_active Application Discontinuation
- 1988-03-11 PT PT86952A patent/PT86952B/en not_active IP Right Cessation
- 1988-03-11 HU HU881190A patent/HU198916B/en not_active IP Right Cessation
- 1988-03-11 SU SU884355377A patent/SU1604157A3/en active
- 1988-03-11 MY MYPI88000258A patent/MY103233A/en unknown
- 1988-03-11 ZA ZA881764A patent/ZA881764B/en unknown
- 1988-03-11 IL IL85704A patent/IL85704A/en unknown
- 1988-03-11 AT AT88400572T patent/ATE86249T1/en not_active IP Right Cessation
- 1988-03-11 PL PL1988271132A patent/PL151889B1/en unknown
- 1988-03-11 ES ES88400572T patent/ES2053778T3/en not_active Expired - Lifetime
- 1988-03-11 TN TNTNSN88020A patent/TNSN88020A1/en unknown
- 1988-03-11 YU YU00496/88A patent/YU49688A/en unknown
- 1988-03-11 EP EP88400572A patent/EP0283390B1/en not_active Expired - Lifetime
- 1988-03-11 NO NO881093A patent/NO170081C/en unknown
- 1988-03-11 IE IE72188A patent/IE60173B1/en not_active IP Right Cessation
- 1988-03-12 KR KR1019880002614A patent/KR880011135A/en not_active Application Discontinuation
- 1988-03-12 JP JP63059223A patent/JPS63243080A/en active Pending
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