PH12007502373B1 - Polycyclic carbamoylpyridone derivative having inhibitory activity on HIV integrase - Google Patents

Polycyclic carbamoylpyridone derivative having inhibitory activity on HIV integrase

Info

Publication number
PH12007502373B1
PH12007502373B1 PH12007502373A PH12007502373A PH12007502373B1 PH 12007502373 B1 PH12007502373 B1 PH 12007502373B1 PH 12007502373 A PH12007502373 A PH 12007502373A PH 12007502373 A PH12007502373 A PH 12007502373A PH 12007502373 B1 PH12007502373 B1 PH 12007502373B1
Authority
PH
Philippines
Prior art keywords
inhibitory activity
hiv integrase
polycyclic carbamoylpyridone
carbamoylpyridone derivative
derivative
Prior art date
Application number
PH12007502373A
Inventor
Kawasuji Takashi
Taishi Teruhiko
Taoda Yoshiyuki
Yoshida Hiroshi
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of PH12007502373B1 publication Critical patent/PH12007502373B1/en

Links

PH12007502373A 2005-10-27 2007-10-25 Polycyclic carbamoylpyridone derivative having inhibitory activity on HIV integrase PH12007502373B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005312076 2005-10-27

Publications (1)

Publication Number Publication Date
PH12007502373B1 true PH12007502373B1 (en) 2013-03-25

Family

ID=40247951

Family Applications (1)

Application Number Title Priority Date Filing Date
PH12007502373A PH12007502373B1 (en) 2005-10-27 2007-10-25 Polycyclic carbamoylpyridone derivative having inhibitory activity on HIV integrase

Country Status (3)

Country Link
CN (1) CN101346376A (en)
PH (1) PH12007502373B1 (en)
ZA (1) ZA200803423B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR201808501T4 (en) * 2009-06-15 2018-07-23 Shionogi & Co Substituted polycyclic carbamoylpyridone derivative.
RU2012140961A (en) * 2010-02-26 2014-04-10 Джапан Тобакко Инк. DERIVATIVE OF 1,3,4,8-TETRAHYDRO-2H-PYRIDO [1,2-a] PYRAZINE AND ITS APPLICATION AS AN HIV INTEGRASE INHIBITOR
WO2012039414A1 (en) * 2010-09-24 2012-03-29 塩野義製薬株式会社 Substituted polycyclic carbamoyl pyridone derivative prodrug
AR094311A1 (en) * 2012-12-27 2015-07-22 Japan Tobacco Inc DERIVATIVES OF TETRAHYDROESPIRO-CICLOPROPIL-PIRIDO [1,2-A] PIRAZINA INHIBITORS OF HIV INTEGRASE
WO2017113288A1 (en) * 2015-12-31 2017-07-06 Merck Sharp & Dohme Corp. Fused tricyclic heterocyclic compounds as hiv integrase inhibitors
WO2020221294A1 (en) * 2019-04-30 2020-11-05 上海拓界生物医药科技有限公司 Bridge ring-3,4-dihydro-pyrido[1,2-a]pyrazine-1,8-dione compound and pharmaceutical use thereof
CN114426540B (en) * 2020-10-29 2024-04-26 上海拓界生物医药科技有限公司 Pyrido [1,2-a ] pyrazine-1, 8-dione prodrug derivatives, preparation method and application thereof
WO2023006087A1 (en) * 2021-07-30 2023-02-02 南京明德新药研发有限公司 Macrocyclic pyridone compound and application thereof
WO2024061257A1 (en) * 2022-09-20 2024-03-28 吉斯凯(苏州)制药有限公司 Polycyclic n-heterocyclic ketone compound and use thereof

Also Published As

Publication number Publication date
CN101346376A (en) 2009-01-14
ZA200803423B (en) 2009-08-26

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