PE20040948A1 - METHOD OF TREATMENT WITH NELFINAVIR - Google Patents

METHOD OF TREATMENT WITH NELFINAVIR

Info

Publication number
PE20040948A1
PE20040948A1 PE2004000146A PE2004000146A PE20040948A1 PE 20040948 A1 PE20040948 A1 PE 20040948A1 PE 2004000146 A PE2004000146 A PE 2004000146A PE 2004000146 A PE2004000146 A PE 2004000146A PE 20040948 A1 PE20040948 A1 PE 20040948A1
Authority
PE
Peru
Prior art keywords
nelfinavir
fat
once
refers
pharmaceutical composition
Prior art date
Application number
PE2004000146A
Other languages
Spanish (es)
Inventor
Edward Fu Ceayong Pun
Carolyn Petersen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PE20040948A1 publication Critical patent/PE20040948A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/7056Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/30Dietetic or nutritional methods, e.g. for losing weight
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23VINDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2002/00Food compositions, function of food ingredients or processes for food or foodstuffs

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Chemistry (AREA)
  • Mycology (AREA)
  • Nutrition Science (AREA)
  • Engineering & Computer Science (AREA)
  • Food Science & Technology (AREA)
  • Polymers & Plastics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

SE REFIERE A UN METODO PARA TRATAR EL VIRUS DE INMUNODEFICIENCIA HUMANA (HIV) QUE COMPRENDE ADMINISTRAR NELFINAVIR, O SUS ESTEREOISOMEROS, SOLVATOS, SALES O PROFARMACOS, CONTENIDO EN UNA COMPOSICION FARMACEUTICA AL MENOS UNA VEZ AL DIA DURANTE AL MENOS DOS SEMANAS CONJUNTAMENTE CON ALIMENTOS QUE CONTIENEN MAS DE 800 KCAL Y MAS DE 40% DE GRASA POR CONTENIDO ENERGETICO. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE CONTIENE NELFINAVIR Y GRASA EN UNA RELACION EN PESO DE AL MENOS 25:1 DE GRASA Y NELFINAVIR. ESTE METODO PERMITE UNA MEJOR BIODISPONIBILIDAD DEL NELFINAVIRREFERS TO A METHOD TO TREAT THE HUMAN IMMUNODEFICIENCY VIRUS (HIV) THAT INCLUDES ADMINISTERING NELFINAVIR, OR ITS STEREOISOMERS, SOLVATES, SALTS OR PRO-DRUGS, CONTAINED IN A PHARMACEUTICAL COMPOSITION AT LEAST ONCE ONCE AT LEAST ONCE A DAY. THEY CONTAIN MORE THAN 800 KCAL AND MORE THAN 40% OF FAT BY ENERGY CONTENT. ALSO REFERS TO A PHARMACEUTICAL COMPOSITION CONTAINING NELFINAVIR AND FAT IN A WEIGHT RATIO OF AT LEAST 25: 1 OF FAT AND NELFINAVIR. THIS METHOD ALLOWS A BETTER BIOAVAILABILITY OF NELFINAVIR

PE2004000146A 2003-02-10 2004-02-09 METHOD OF TREATMENT WITH NELFINAVIR PE20040948A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US44644403P 2003-02-10 2003-02-10
US52425803P 2003-11-21 2003-11-21

Publications (1)

Publication Number Publication Date
PE20040948A1 true PE20040948A1 (en) 2004-12-27

Family

ID=32853430

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2004000146A PE20040948A1 (en) 2003-02-10 2004-02-09 METHOD OF TREATMENT WITH NELFINAVIR

Country Status (13)

Country Link
EP (1) EP1605942A1 (en)
JP (1) JP2006517221A (en)
AR (1) AR043133A1 (en)
BR (1) BRPI0407174A (en)
CA (1) CA2515095A1 (en)
CL (1) CL2004000202A1 (en)
MX (1) MXPA05008425A (en)
NL (1) NL1025449C2 (en)
PA (1) PA8595301A1 (en)
PE (1) PE20040948A1 (en)
TW (1) TW200423922A (en)
UY (1) UY28183A1 (en)
WO (1) WO2004069251A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7157455B2 (en) 2003-02-10 2007-01-02 Hoffmann-La Roche Inc. 4-Aminopyrimidine-5-one derivatives

Also Published As

Publication number Publication date
CL2004000202A1 (en) 2005-03-18
JP2006517221A (en) 2006-07-20
EP1605942A1 (en) 2005-12-21
NL1025449C2 (en) 2005-03-15
UY28183A1 (en) 2004-09-30
CA2515095A1 (en) 2004-08-19
NL1025449A1 (en) 2004-08-12
PA8595301A1 (en) 2005-08-04
AR043133A1 (en) 2005-07-20
TW200423922A (en) 2004-11-16
BRPI0407174A (en) 2006-02-07
WO2004069251A1 (en) 2004-08-19
MXPA05008425A (en) 2005-10-19

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal