PE20040723A1 - BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES - Google Patents
BENZOFURAN AND BENZOTHIOPHENE DERIVATIVESInfo
- Publication number
- PE20040723A1 PE20040723A1 PE2003000745A PE2003000745A PE20040723A1 PE 20040723 A1 PE20040723 A1 PE 20040723A1 PE 2003000745 A PE2003000745 A PE 2003000745A PE 2003000745 A PE2003000745 A PE 2003000745A PE 20040723 A1 PE20040723 A1 PE 20040723A1
- Authority
- PE
- Peru
- Prior art keywords
- benzofuran
- phenyl
- alkyl
- methanone
- amino
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Furan Compounds (AREA)
Abstract
SE REFIERE A UN COMPUESTO DE FORMULA I DONDE X ES O, S; R1 ES H, ALQUILO C1-C6, C(O)ALQUILO(C1-C6), BENZOILO; R2 ES FENILO Y NAFTILO OPCIONALMENTE SUSTITUIDOS CON 1, 2, o 3 SUSTITUYENTES, HETEROCICLO, ENTRE OTROS; R3 ES H, OH, CN, ALQUILO C1-C3, ENTRE OTROS; R4 ES PIPERONILO, HETEROCILCLO OPCIONALMENTE SUSTITUIDO; R5 Y R6 SON CADA UNO H, OH, CN, ALQUILO C1-C3, ENTRE OTROS. SON COMPUESTOS PREFERIDOS: (3-AMINO-6-FENIL-BENZOFURAN-2-IL)-(2,4-DICLORO-FENIL)-METANONA Y [3-AMINO-6-(3-NITRO-FENIL)-BENZOFURAN-2-IL]-(2,4-DICLOROFENIL)-METANONA; ENTRE OTROS. SE REFIERE TAMBIEN A UNA COMPOSICION FARMACEUTICA. DICHOS COMPUESTOS SON UTILES EN EL TRATAMIENTO O PREVENCION DE DESORDENES HIPER-PROLIFERATIVOSREFERS TO A COMPOUND OF FORMULA I WHERE X IS O, S; R1 IS H, C1-C6 ALKYL, C (O) (C1-C6) ALKYL, BENZOYL; R2 IS PHENYL AND NAPHTHYLUS OPTIONALLY SUBSTITUTED WITH 1, 2, or 3 SUBSTITUTES, HETEROCICLO, AMONG OTHERS; R3 IS H, OH, CN, C1-C3 ALKYL, AMONG OTHERS; R4 IS PIPERONYL, OPTIONALLY SUBSTITUTED HETEROCYCLE; R5 AND R6 ARE EACH H, OH, CN, C1-C3 ALKYL, AMONG OTHERS. PREFERRED COMPOUNDS ARE: (3-AMINO-6-PHENYL-BENZOFURAN-2-IL) - (2,4-DICHLORO-PHENYL) -METHANONE AND [3-AMINO-6- (3-NITRO-PHENYL) -BENZOFURAN-2 -IL] - (2,4-DICHLOROPHENYL) -METHANONE; AMONG OTHERS. IT ALSO REFERS TO A PHARMACEUTICAL COMPOSITION. SUCH COMPOUNDS ARE USEFUL IN THE TREATMENT OR PREVENTION OF HYPER-PROLIFERATIVE DISORDERS
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39988602P | 2002-07-31 | 2002-07-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20040723A1 true PE20040723A1 (en) | 2004-10-29 |
Family
ID=38812802
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2003000745A PE20040723A1 (en) | 2002-07-31 | 2003-07-30 | BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES |
Country Status (7)
| Country | Link |
|---|---|
| AR (1) | AR040669A1 (en) |
| GT (1) | GT200300158A (en) |
| HN (1) | HN2003000228A (en) |
| MY (1) | MY135649A (en) |
| PE (1) | PE20040723A1 (en) |
| TW (1) | TW200413343A (en) |
| UY (1) | UY27916A1 (en) |
-
2003
- 2003-07-23 AR ARP030102641 patent/AR040669A1/en unknown
- 2003-07-29 MY MYPI20032853 patent/MY135649A/en unknown
- 2003-07-29 GT GT200300158A patent/GT200300158A/en unknown
- 2003-07-30 TW TW92120734A patent/TW200413343A/en unknown
- 2003-07-30 PE PE2003000745A patent/PE20040723A1/en not_active Application Discontinuation
- 2003-07-30 HN HN2003000228A patent/HN2003000228A/en unknown
- 2003-07-31 UY UY27916A patent/UY27916A1/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AR040669A1 (en) | 2005-04-13 |
| MY135649A (en) | 2008-06-30 |
| GT200300158A (en) | 2004-06-08 |
| TW200413343A (en) | 2004-08-01 |
| UY27916A1 (en) | 2003-12-31 |
| HN2003000228A (en) | 2004-08-02 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20052493L (en) | Selected CGRP antagonists, processes for their preparation and their use as pharmaceutical compositions. | |
| PT863136E (en) | AZETIDINE AND PYRROLIDINE DERIVATIVES | |
| NO20021358L (en) | Alkylenediamine-substituted heterocycles | |
| IS6565A (en) | The tropane derivatives are useful in the treatment | |
| TW200510405A (en) | Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors | |
| WO2003039451A3 (en) | Thiazole pyridazinones as adenosine antagonists | |
| PE20030226A1 (en) | ARYLIC COMPOUNDS SUBSTITUTED WITH QUINUCLIDINES FOR THE TREATMENT OF DISEASES | |
| MXPA03011638A (en) | 4-piperazinylindole derivatives with 5-ht6 receptor affinity. | |
| FR2805817B1 (en) | PHARMACEUTICAL COMPOSITIONS CONTAINING AZETIDINE DERIVATIVES, NOVEL AZETIDINE DERIVATIVES AND THEIR PREPARATION | |
| RS20050469A (en) | Pyrrolopyrimidine derivatives | |
| NO20071642L (en) | N-Benzenesulfonyl-substituted anilino-pyrimidine analogs | |
| AR025225A1 (en) | PHYSYLOXAZOLIDINONES HETEROCICLIC BICYCLIC REPLACED ANTIBACTERIAL AND PHARMACEUTICAL COMPOSITIONS | |
| DE60222775D1 (en) | ANALOGUE AS ANTITUMORAL COMPOUNDS | |
| AR056321A1 (en) | THERAPEUTIC COMBINATIONS FOR THE TREATMENT OR PREVENTION OF PSYCHOTIC DISORDERS | |
| ATE540928T1 (en) | ISOQUINOLINE COMPOUNDS AND THEIR MEDICAL USES | |
| DK289888D0 (en) | 2-SUBSTITUTED-E-CONDENSED OE1,2,4, AATRIAZOLOOE1,5-CAAPYRIMIDINES, PHARMACEUTICAL PREPARATIONS AND APPLICATIONS THEREOF | |
| DK0759919T3 (en) | Azolidinediones as antihyperglycemic agents | |
| TR200102789T2 (en) | 1-Arenesulfonyl-2-aryl-pyrrolidine and piperidine derivatives for the treatment of Cns disorders | |
| EA200000614A1 (en) | 2,3-SUBSTITUTED INDO COMPOUNDS AS SOH-2 INHIBITORS | |
| MY128241A (en) | Substituted tetracyclic pyrroloquinolone derivatives useful as phosphodiesterase inhibitors | |
| DE69022744D1 (en) | PIPERIDINE AND PYRROLIDINE DERIVATIVES. | |
| TW200420292A (en) | Benzofuran derivative | |
| CY1108837T1 (en) | New aminopyridine derivatives as mGluR5 antagonists | |
| TW347389B (en) | Taxoids, their preparation and pharmaceutical compositions containing them | |
| EP0787725A4 (en) | Quinoline derivative |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration | ||
| FD | Application declared void or lapsed |