PE20030732A1 - USE OF ALKYLPHOSPHOCOLINS IN THE PREVENTIVE TREATMENT OF DISEASES CAUSED BY PROTOZOARIANS - Google Patents

USE OF ALKYLPHOSPHOCOLINS IN THE PREVENTIVE TREATMENT OF DISEASES CAUSED BY PROTOZOARIANS

Info

Publication number
PE20030732A1
PE20030732A1 PE2003000061A PE2003000061A PE20030732A1 PE 20030732 A1 PE20030732 A1 PE 20030732A1 PE 2003000061 A PE2003000061 A PE 2003000061A PE 2003000061 A PE2003000061 A PE 2003000061A PE 20030732 A1 PE20030732 A1 PE 20030732A1
Authority
PE
Peru
Prior art keywords
diseases caused
protozoarians
alkylphosphocolins
treatment
preventive treatment
Prior art date
Application number
PE2003000061A
Other languages
Spanish (es)
Inventor
Jurgen Engel
Original Assignee
Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Gmbh filed Critical Zentaris Gmbh
Publication of PE20030732A1 publication Critical patent/PE20030732A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/683Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols
    • A61K31/685Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols one of the hydroxy compounds having nitrogen atoms, e.g. phosphatidylserine, lecithin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA PARA EL TRATAMIENTO EN MAMIFEROS, DE ENFERMEDADES CAUSADAS POR PROTOZOARIOS, EN PARTICULAR LEISHMANIASIS, LA CUAL CONTIENE a)ALQUILFOSFOCOLINA, EN PARTICULAR HEXADECILFOSFOCOLINA (MILTEFOSINA) o FOSFATO DE OCTADECIL-(1,1-DIMETIL-PIPERIDINIO-4-ILO) (PERIFOSINA); b)UN ANTIEMETICO Y/O UN ANTIDIARREICO. SE REFIERE TAMBIEN AL EMPLEO DE ALQUILFOSFOCOLINAS PARA LA PREPARACION DE UN MEDICAMENTO PARA EL TRATAMIENTO YA DESCRITO Y A UN ESQUEMA DE DOSIFICACION DE LA COMPOSICION PARA DICHO TRATAMIENTOREFERS TO A PHARMACEUTICAL COMPOSITION FOR THE TREATMENT IN MAMMALS, OF DISEASES CAUSED BY PROTOZOARIES, IN PARTICULAR LEISHMANIASIS, WHICH CONTAINS a) ALKYLPHOSPHOCOLINE, IN PARTICULAR HEXADECILPHOSPHOCOLINE (1,1-PHYPTEPHOSADETILE-4-OXYPTEPHOSADETILE-DIMETHYL-4-MILTHYPTEPHOSADE -ILO) (PERIPHOSINE); b) AN ANTIEMETIC AND / OR AN ANTIDIARRHEAL. IT ALSO REFERS TO THE USE OF ALKYLPHOSPHOCOLINES FOR THE PREPARATION OF A DRUG FOR THE TREATMENT ALREADY DESCRIBED AND TO A DOSAGE SCHEME OF THE COMPOSITION FOR SUCH TREATMENT

PE2003000061A 2002-01-25 2003-01-20 USE OF ALKYLPHOSPHOCOLINS IN THE PREVENTIVE TREATMENT OF DISEASES CAUSED BY PROTOZOARIANS PE20030732A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10203195A DE10203195A1 (en) 2002-01-25 2002-01-25 Use of alkylphosphocholines in the preventive treatment of protozoal diseases

Publications (1)

Publication Number Publication Date
PE20030732A1 true PE20030732A1 (en) 2003-09-27

Family

ID=7713213

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2003000061A PE20030732A1 (en) 2002-01-25 2003-01-20 USE OF ALKYLPHOSPHOCOLINS IN THE PREVENTIVE TREATMENT OF DISEASES CAUSED BY PROTOZOARIANS

Country Status (16)

Country Link
EP (1) EP1467742A1 (en)
JP (1) JP2005515244A (en)
CN (1) CN1622811A (en)
AR (1) AR038224A1 (en)
AU (1) AU2003236787B2 (en)
BR (1) BR0307021A (en)
CA (1) CA2470185A1 (en)
CO (1) CO5601024A2 (en)
DE (1) DE10203195A1 (en)
IL (2) IL162492A0 (en)
MX (1) MXPA04007193A (en)
NZ (1) NZ548040A (en)
PE (1) PE20030732A1 (en)
TW (1) TWI339582B (en)
WO (1) WO2003061669A1 (en)
ZA (1) ZA200404690B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT501545B1 (en) * 2005-02-23 2007-10-15 Obwaller Andreas Dr CLEANING AGENT FOR CONTACT LENSES
EP1800684A1 (en) * 2005-12-20 2007-06-27 Zentaris GmbH Novel alkyl phospholipid derivatives and uses thereof
AU2006328479B2 (en) * 2005-12-19 2012-03-08 Aeterna Zentaris Gmbh Alkyl phospholipid derivatives with reduced cytotoxicity and uses thereof
CN104473941A (en) * 2014-12-20 2015-04-01 长沙佰顺生物科技有限公司 Miltefosine-containing medicine preparation and preparation method thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4132344A1 (en) * 1991-09-27 1993-04-01 Max Planck Gesellschaft METHOD FOR PRODUCING A MEDAL FOR ORAL OR TOPICAL ADMINISTRATION IN THE TREATMENT OF LEISHMANIASIS
DE4132345A1 (en) * 1991-09-27 1993-04-01 Max Planck Gesellschaft Medicament compsns. for intravenous admin. of lytic agents - used for treatment of tumours, auto-immune disorders, multiple sclerosis, etc.
AU682464B2 (en) * 1992-03-06 1997-10-09 Lica Pharmaceuticals A/S Treatment and prophylaxis of diseases caused by parasites, or bacteria
PT1051159E (en) * 1998-01-22 2002-09-30 Zentaris Ag SOLID PHARMACEUTICAL COMPOSITIONS CONTAINING MILTEFOSIN FOR ORAL ADMINISTRATION IN THE TREATMENT OF LEISHMANIOSE
DE10020812C2 (en) * 2000-04-20 2003-06-26 Robert Koch Inst Use of naphthindazole-4,9-quinones as antiparasitic agents
AU2002232400A1 (en) * 2000-11-06 2002-05-15 U.S. Army Medical Research And Materiel Command Reversed amidines and methods of using for treating, preventing, or inhibiting leishmaniasis

Also Published As

Publication number Publication date
TWI339582B (en) 2011-04-01
WO2003061669A1 (en) 2003-07-31
JP2005515244A (en) 2005-05-26
AU2003236787B2 (en) 2007-03-22
MXPA04007193A (en) 2004-10-29
TW200302103A (en) 2003-08-01
IL162492A (en) 2009-12-24
IL162492A0 (en) 2005-11-20
DE10203195A1 (en) 2003-08-07
ZA200404690B (en) 2004-09-27
CN1622811A (en) 2005-06-01
EP1467742A1 (en) 2004-10-20
NZ548040A (en) 2007-06-29
CA2470185A1 (en) 2003-07-31
AR038224A1 (en) 2005-01-05
CO5601024A2 (en) 2006-01-31
BR0307021A (en) 2004-11-03

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