PE20011093A1 - MALE CONTRACEPTIVE FORMULATION INCLUDING NORETISTERONE - Google Patents

MALE CONTRACEPTIVE FORMULATION INCLUDING NORETISTERONE

Info

Publication number
PE20011093A1
PE20011093A1 PE2001000152A PE2001000152A PE20011093A1 PE 20011093 A1 PE20011093 A1 PE 20011093A1 PE 2001000152 A PE2001000152 A PE 2001000152A PE 2001000152 A PE2001000152 A PE 2001000152A PE 20011093 A1 PE20011093 A1 PE 20011093A1
Authority
PE
Peru
Prior art keywords
noretisterone
progestin
male contraceptive
formulation including
contraceptive formulation
Prior art date
Application number
PE2001000152A
Other languages
Spanish (es)
Inventor
Alexander Druebig
Ursula-Friederike Habenicht
Ekkerhard Schillinger
Eberhard Nieschlag
Michael Oettel
Axel Kamischke
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of PE20011093A1 publication Critical patent/PE20011093A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE PROGESTINA CON PROPIEDADES ANDROGENICAS COMO ESTROGENICAS TAL COMO NORETISTERONA (NET) O SUS DERIVADOS COMO ESTERES CARBOXILICOS. LA DOSIS DE NET ES DE 1 mg A 10mg Y LA DOSIS DURANTE 6 SEMANAS ES DE 100mg A 500mg. LA PROGESTINA SUPRIME LA ESPERMATOGENESIS E INDUCE LA OLIGOZOOSPERMIA O LA AZOOSPERMIA . LA PROGESTINA SE ADMINISTRA EN CANTIDADES SUFICIENTES COMO PARA DISMINUIR LA CONCENTRACION DEL ESPERMA EN MENOS DE 3 MILLONES/ml Y MANTENER LOS NIVELES POR LO MENOS UNA SEMANA. LA FORMULACION ANTICONCEPTIVA MASCULINA SUPRIME LA ESPERMATOGENESIS Y ES UTIL PARA PREVENIR LA CONCEPCION MASCULINAIT REFERS TO A PHARMACEUTICAL COMPOSITION THAT INCLUDES PROGESTIN WITH ANDROGENIC AND ESTROGENIC PROPERTIES SUCH AS NORETISTERONE (NET) OR ITS DERIVATIVES AS CARBOXYL ESTERS. THE DOSE OF NET IS FROM 1mg TO 10mg AND THE DOSE FOR 6 WEEKS IS FROM 100mg TO 500mg. PROGESTIN SUPPRESSES SPERMATOGENESIS AND INDUCES OLIGOZOOSPERMIA OR AZOOSPERMIA. PROGESTIN IS ADMINISTERED IN SUFFICIENT AMOUNTS TO REDUCE THE CONCENTRATION OF THE SPERM TO LESS THAN 3 MILLION / mL AND MAINTAIN THE LEVELS FOR AT LEAST ONE WEEK. MALE CONTRACEPTIVE FORMULATION SUPPRESSES SPERMATOGENESIS AND IS USEFUL TO PREVENT MALE CONCEPTION

PE2001000152A 2000-02-15 2001-02-12 MALE CONTRACEPTIVE FORMULATION INCLUDING NORETISTERONE PE20011093A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP00200493 2000-02-15

Publications (1)

Publication Number Publication Date
PE20011093A1 true PE20011093A1 (en) 2001-10-12

Family

ID=37515367

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2001000152A PE20011093A1 (en) 2000-02-15 2001-02-12 MALE CONTRACEPTIVE FORMULATION INCLUDING NORETISTERONE

Country Status (3)

Country Link
AR (1) AR027526A1 (en)
CO (1) CO5261637A1 (en)
PE (1) PE20011093A1 (en)

Also Published As

Publication number Publication date
CO5261637A1 (en) 2003-03-31
AR027526A1 (en) 2003-04-02

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Legal Events

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