PA8567601A1 - B3-ADRENERGIC RECEPTOR AGONIST SALT, ITS FORMULATIONS AND ITS USES - Google Patents

B3-ADRENERGIC RECEPTOR AGONIST SALT, ITS FORMULATIONS AND ITS USES

Info

Publication number
PA8567601A1
PA8567601A1 PA20038567601A PA8567601A PA8567601A1 PA 8567601 A1 PA8567601 A1 PA 8567601A1 PA 20038567601 A PA20038567601 A PA 20038567601A PA 8567601 A PA8567601 A PA 8567601A PA 8567601 A1 PA8567601 A1 PA 8567601A1
Authority
PA
Panama
Prior art keywords
salt
monohidrate
formulations
procedures
receptor agonist
Prior art date
Application number
PA20038567601A
Other languages
Spanish (es)
Inventor
Jennifer Anne Lafontaine
Joseph Francis Krzyzaniak
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PA8567601A1 publication Critical patent/PA8567601A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

LA PRESENTE INVENCION PROPORCIONA LA SAL TOSILATO DE (R)-2-(2-(4-OXAZOL-4-ILFENOXI)ETILAMINO)-1-PIRIDIN-3-ILETANOL), EL MONOHIDRATO DE DICHA SAL, PROCEDIMIENTOS UTILES EN LA PREPARCION DE DICHA SAL Y DICHO MONOHIDRATO, COMPOSICIONES FARMACEUTICAS QUE COMPRENDE DICHA SAL, O DICHO MONOHIDRATO, PROCEDIMIENTOS PARA TRATAR ENFERMEDADES, AFECCIONES Y TRASTORNOS EN UN MAMIFERO MEDIADOS POR EL RECEPTOR BETA 3 ADRENERGICO UTILIZANDO DICHA SAL, DICHO MONOHIDRATO O DICHAS COMPOSICIONES FARMACEUTICAS; Y PROCEDIMIENTOS PARA AUMENTAR EL CONTENIDO DE CARNE MAGRA EN ANIMALES COMESTIBLES UTILIZANDO DICHA SAL, DICHO MONOHIDRATO O DICHAS COMPOSICIONES FARMACEUTICAS.THIS INVENTION PROVIDES THE TOSILATE SALT OF (R) -2- (2- (4-OXAZOL-4-ILFENOXI) ETHYLAMINE) -1-PIRIDIN-3-ILETANOL), THE SALT MONOHIDRATE, USEFUL PROCEDURES IN THE PREPARATION OF SUCH SALT AND SUCH MONOHIDRATE, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE SUCH SALT, OR SUCH MONOHIDRATE, PROCEDURES TO TREAT DISEASES, AFFECTIONS AND DISORDERS IN A MAMIFIER MEDIATED BY THE BETA 3 ADRENERGIC RECEIVER USING DICHAICHO DICHAICHO COMPACT AND PROCEDURES TO INCREASE THE CONTENT OF MEAT MEAT IN EDIBLE ANIMALS USING SUCH SALT, SUCH MONOHIDRATE OR SUCH PHARMACEUTICAL COMPOSITIONS.

PA20038567601A 2002-02-27 2003-02-26 B3-ADRENERGIC RECEPTOR AGONIST SALT, ITS FORMULATIONS AND ITS USES PA8567601A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US36024802P 2002-02-27 2002-02-27

Publications (1)

Publication Number Publication Date
PA8567601A1 true PA8567601A1 (en) 2003-12-10

Family

ID=27766205

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20038567601A PA8567601A1 (en) 2002-02-27 2003-02-26 B3-ADRENERGIC RECEPTOR AGONIST SALT, ITS FORMULATIONS AND ITS USES

Country Status (8)

Country Link
AR (1) AR038603A1 (en)
AU (1) AU2003248355A1 (en)
GT (1) GT200300044A (en)
PA (1) PA8567601A1 (en)
PE (1) PE20030900A1 (en)
TW (1) TW200305414A (en)
UY (1) UY27678A1 (en)
WO (1) WO2003072571A1 (en)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9812709D0 (en) * 1998-06-13 1998-08-12 Glaxo Group Ltd Chemical compounds
CA2423792A1 (en) * 2000-10-20 2002-04-25 Pfizer Products Inc. Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists

Also Published As

Publication number Publication date
AR038603A1 (en) 2005-01-19
PE20030900A1 (en) 2003-10-25
UY27678A1 (en) 2003-10-31
AU2003248355A1 (en) 2003-09-09
GT200300044A (en) 2003-09-22
WO2003072571A1 (en) 2003-09-04
TW200305414A (en) 2003-11-01

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PA8567601A1 (en) B3-ADRENERGIC RECEPTOR AGONIST SALT, ITS FORMULATIONS AND ITS USES
PA8567701A1 (en) B3-ADRENERGIC RECEIVER AGONISTS
PA8567501A1 (en) CRYSTAL FORMS OF B3-ADRENERGIC RECEIVER AGONISTS, PROCEDURES FOR THEIR PREPARATION, AND THEIR USES