OA06794A - 2-Nitroimidazoles, et procédés pour leur préparation. - Google Patents

2-Nitroimidazoles, et procédés pour leur préparation.

Info

Publication number
OA06794A
OA06794A OA57385A OA57385A OA06794A OA 06794 A OA06794 A OA 06794A OA 57385 A OA57385 A OA 57385A OA 57385 A OA57385 A OA 57385A OA 06794 A OA06794 A OA 06794A
Authority
OA
OAPI
Prior art keywords
nitroimidazoles
processes
preparation
Prior art date
Application number
OA57385A
Other languages
English (en)
Original Assignee
Hoffmann La Roche & Cie S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche & Cie S A filed Critical Hoffmann La Roche & Cie S A
Publication of OA06794A publication Critical patent/OA06794A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/91Nitro radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
OA57385A 1980-05-23 1981-04-23 2-Nitroimidazoles, et procédés pour leur préparation. OA06794A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH405780 1980-05-23

Publications (1)

Publication Number Publication Date
OA06794A true OA06794A (fr) 1982-12-31

Family

ID=4269011

Family Applications (1)

Application Number Title Priority Date Filing Date
OA57385A OA06794A (fr) 1980-05-23 1981-04-23 2-Nitroimidazoles, et procédés pour leur préparation.

Country Status (11)

Country Link
US (2) US4366166A (fr)
EP (1) EP0040761A1 (fr)
JP (1) JPS5711969A (fr)
AU (1) AU541912B2 (fr)
BR (1) BR8103216A (fr)
GB (1) GB2076402B (fr)
IN (1) IN155338B (fr)
MW (1) MW1681A1 (fr)
OA (1) OA06794A (fr)
PH (1) PH16858A (fr)
ZW (1) ZW8781A1 (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3362868D1 (en) * 1982-02-19 1986-05-15 Ciba Geigy Ag Microbicidal and plant-growth regulating agents
US4568111A (en) * 1983-08-29 1986-02-04 The United States Of America As Represented By The United States Department Of Energy Detachable connection for a nuclear reactor fuel assembly
AU4327585A (en) * 1984-06-21 1986-01-02 Imperial Chemical Industries Plc Antifungal azole compounds
CA1329206C (fr) * 1987-06-10 1994-05-03 Tsutomu Kagiya Derives nitroazole fluores et radiosensibilisant en contenant
FR2684382B1 (fr) * 1991-12-02 1994-10-21 Rhone Merieux Medicaments et preparations pures de dichlorhydrate de melarsomine, leur procede d'obtention et produits intermediaires obtenus.
JP3577079B2 (ja) * 1992-12-18 2004-10-13 ポーラ化成工業株式会社 光学活性2−ニトロイミダゾール誘導体
WO1995009844A1 (fr) * 1993-10-04 1995-04-13 Board Of Regents, The University Of Texas System Synthese rapide et utilisation de 18f-fluoromisonidazole et d'analogues
US5700825A (en) * 1995-03-31 1997-12-23 Florida State University Radiosensitizing diamines and their pharmaceutical preparations
US6060604A (en) * 1995-03-31 2000-05-09 Florida State University Pharmaceutical compounds comprising polyamines substituted with electron-affinic groups
US6423707B1 (en) 2000-08-28 2002-07-23 California Pacific Medical Center Nitroimidazole ester analogues and therapeutic applications
WO2005041853A2 (fr) * 2003-10-28 2005-05-12 Ems S.A. Composes derives de nitroimidazole antibacteriens et/ou antiprotozoaires a activite inhibitrice d'urease, procede de preparation desdits composes et utilisation dans des compositions pharmaceutiques et dans des medicaments

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3255201A (en) * 1965-04-09 1966-06-07 Hoffmann La Roche 2-nitroimidazoles
US3505349A (en) * 1966-04-18 1970-04-07 Hoffmann La Roche 2-nitro-imidazolyl-1-acetamides
US3641047A (en) * 1970-08-05 1972-02-08 Hoffmann La Roche 2-nitroimidazole derivatives substituted in the 1-position with a 2-oxo-propyl or semicarbazone group
CA1034126A (fr) * 1974-01-17 1978-07-04 Alden G. Beaman Nitroimidazoles -2
IE47132B1 (en) * 1977-08-19 1983-12-28 Roche Products Ltd Novel nitroimidazoles and pharmaceutical preparations containing these as well as their manufacture

Also Published As

Publication number Publication date
AU541912B2 (en) 1985-01-31
GB2076402A (en) 1981-12-02
AU7064081A (en) 1981-11-26
IN155338B (fr) 1985-01-19
EP0040761A1 (fr) 1981-12-02
US4456610A (en) 1984-06-26
JPS5711969A (en) 1982-01-21
MW1681A1 (en) 1982-08-11
US4366166A (en) 1982-12-28
ZW8781A1 (en) 1981-12-16
BR8103216A (pt) 1982-02-16
PH16858A (en) 1984-03-22
GB2076402B (en) 1984-05-02

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