NZ588104A - Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof - Google Patents

Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof

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Publication number
NZ588104A
NZ588104A NZ588104A NZ58810408A NZ588104A NZ 588104 A NZ588104 A NZ 588104A NZ 588104 A NZ588104 A NZ 588104A NZ 58810408 A NZ58810408 A NZ 58810408A NZ 588104 A NZ588104 A NZ 588104A
Authority
NZ
New Zealand
Prior art keywords
solid forms
acetylaminoisoindoline
methylsulfonylethyl
methoxyphenyl
ethoxy
Prior art date
Application number
NZ588104A
Inventor
George W Muller
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40043076&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ588104(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corp filed Critical Celgene Corp
Priority to NZ588104A priority Critical patent/NZ588104A/en
Publication of NZ588104A publication Critical patent/NZ588104A/en

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/4035—Isoindoles, e.g. phthalimide
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Abstract

The disclosure relates to solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2- methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione represented by structural formula (I), compositions comprising the solid forms, methods of making the solid forms and methods of their use are disclosed. These solid forms are suitable for treating and/or preventing disorders ameliorated by the reduction of levels of TNF-a or the inhibition of PDE4.
NZ588104A 2008-03-27 2008-03-27 Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof NZ588104A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NZ588104A NZ588104A (en) 2008-03-27 2008-03-27 Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NZ588104A NZ588104A (en) 2008-03-27 2008-03-27 Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof
PCT/US2008/004021 WO2009120167A1 (en) 2008-03-27 2008-03-27 Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof

Publications (1)

Publication Number Publication Date
NZ588104A true NZ588104A (en) 2012-11-30

Family

ID=40043076

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ588104A NZ588104A (en) 2008-03-27 2008-03-27 Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof

Country Status (21)

Country Link
EP (2) EP2695616A1 (en)
JP (1) JP5474043B2 (en)
KR (3) KR20150038547A (en)
CN (1) CN102046167A (en)
AU (1) AU2008353468B2 (en)
BR (1) BRPI0822398B8 (en)
CA (1) CA2718601A1 (en)
CY (1) CY1115361T1 (en)
DK (1) DK2276483T3 (en)
ES (1) ES2476252T3 (en)
HR (1) HRP20140609T1 (en)
IL (3) IL208216A0 (en)
MX (2) MX2010010454A (en)
NO (1) NO2015017I1 (en)
NZ (1) NZ588104A (en)
PL (1) PL2276483T3 (en)
PT (1) PT2276483E (en)
RU (1) RU2471782C2 (en)
SI (1) SI2276483T1 (en)
WO (1) WO2009120167A1 (en)
ZA (1) ZA201006663B (en)

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