NZ333760A - Processes and intermediates in the synthesis of 5-(3-[exobicyclo[2.2.1]hept-2-yloxy]-4methoxyphenyl)-3,4,5,6-t etrahydropyrimidin-2(1h)-one - Google Patents

Processes and intermediates in the synthesis of 5-(3-[exobicyclo[2.2.1]hept-2-yloxy]-4methoxyphenyl)-3,4,5,6-t etrahydropyrimidin-2(1h)-one

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Publication number
NZ333760A
NZ333760A NZ333760A NZ33376099A NZ333760A NZ 333760 A NZ333760 A NZ 333760A NZ 333760 A NZ333760 A NZ 333760A NZ 33376099 A NZ33376099 A NZ 33376099A NZ 333760 A NZ333760 A NZ 333760A
Authority
NZ
New Zealand
Prior art keywords
hept
yloxy
synthesis
processes
etrahydropyrimidin
Prior art date
Application number
NZ333760A
Inventor
Thomas G Lacour
Charles W Murtiashaw
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NZ333760A publication Critical patent/NZ333760A/en

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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

This application relates to processes for preparing the pharmaceutically active compound 5-(3-[(2S)-exo-bicyclo[2.2.1]hept-2-yloxy]-4-methoxyphenyl)-3,4,5,6-tetrahydropyrimidin-2(1H)-one and its corresponding 2R enantiomer and for preparing certain intermediates used in the synthesis of these compounds. The intermediates used are of the formula (II) where X and Y are CO2(1-6)alkyl, CONH2 and CONHOH or can be taken together to form a group of the formula (a).
NZ333760A 1994-08-05 1999-01-15 Processes and intermediates in the synthesis of 5-(3-[exobicyclo[2.2.1]hept-2-yloxy]-4methoxyphenyl)-3,4,5,6-t etrahydropyrimidin-2(1h)-one NZ333760A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28657994A 1994-08-05 1994-08-05
NZ28414499 1999-01-15

Publications (1)

Publication Number Publication Date
NZ333760A true NZ333760A (en) 2000-03-27

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Family Applications (1)

Application Number Title Priority Date Filing Date
NZ333760A NZ333760A (en) 1994-08-05 1999-01-15 Processes and intermediates in the synthesis of 5-(3-[exobicyclo[2.2.1]hept-2-yloxy]-4methoxyphenyl)-3,4,5,6-t etrahydropyrimidin-2(1h)-one

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NZ (1) NZ333760A (en)

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