NO943101L - 2,6-metano-2H-kinolizinderivat som 5-HT3-reseptorantagonist - Google Patents

2,6-metano-2H-kinolizinderivat som 5-HT3-reseptorantagonist

Info

Publication number
NO943101L
NO943101L NO943101A NO943101A NO943101L NO 943101 L NO943101 L NO 943101L NO 943101 A NO943101 A NO 943101A NO 943101 A NO943101 A NO 943101A NO 943101 L NO943101 L NO 943101L
Authority
NO
Norway
Prior art keywords
treatment
methano
receptor antagonist
quinolizine derivative
hallucinatory
Prior art date
Application number
NO943101A
Other languages
English (en)
Norwegian (no)
Other versions
NO943101D0 (no
Inventor
Maurice Ward Gittos
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of NO943101L publication Critical patent/NO943101L/no
Publication of NO943101D0 publication Critical patent/NO943101D0/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO943101A 1992-02-24 1994-08-23 2,6-metano-2H-kinolizinderivat som 5-HT3-reseptorantagonist NO943101D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP92400474 1992-02-24
PCT/US1993/000880 WO1993017019A1 (en) 1992-02-24 1993-02-03 2,6-methano-2h-quinolizin derivative as 5-ht3-receptor antagonist

Publications (2)

Publication Number Publication Date
NO943101L true NO943101L (no) 1994-08-23
NO943101D0 NO943101D0 (no) 1994-08-23

Family

ID=8211614

Family Applications (1)

Application Number Title Priority Date Filing Date
NO943101A NO943101D0 (no) 1992-02-24 1994-08-23 2,6-metano-2H-kinolizinderivat som 5-HT3-reseptorantagonist

Country Status (14)

Country Link
EP (1) EP0628043A1 (de)
JP (1) JPH07504192A (de)
KR (1) KR100287933B1 (de)
AU (1) AU675060B2 (de)
CA (1) CA2130563C (de)
FI (1) FI105917B (de)
HU (1) HU216831B (de)
IL (1) IL104821A (de)
MX (1) MX9300948A (de)
NO (1) NO943101D0 (de)
NZ (1) NZ249346A (de)
TW (1) TW226374B (de)
WO (1) WO1993017019A1 (de)
ZA (1) ZA931146B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000048597A1 (en) 1999-02-18 2000-08-24 Novartis Ag Systemic use of 5-ht3 receptor antagonists against rheumatic inflammatory processes
US8518962B2 (en) 2005-03-07 2013-08-27 The University Of Chicago Use of opioid antagonists
US8524731B2 (en) 2005-03-07 2013-09-03 The University Of Chicago Use of opioid antagonists to attenuate endothelial cell proliferation and migration
US9662325B2 (en) 2005-03-07 2017-05-30 The University Of Chicago Use of opioid antagonists to attenuate endothelial cell proliferation and migration
CN101171010B (zh) 2005-03-07 2014-09-17 芝加哥大学 阿片样物质拮抗剂用于减少内皮细胞增殖和迁移的用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2080727T3 (es) * 1988-02-23 1996-02-16 Merrell Pharma Inc Uso de quinolizina y derivados de quinolizinona en la fabricacion de medicamentos.
EP0517984A1 (de) * 1991-06-11 1992-12-16 Merrell Dow Pharmaceuticals Inc. Amidanaloge-Derivate von methanoverbrückten Chinolizinen

Also Published As

Publication number Publication date
ZA931146B (en) 1993-09-14
HU216831B (hu) 1999-09-28
HUT68249A (en) 1995-06-28
IL104821A (en) 1997-01-10
KR950700297A (ko) 1995-01-16
CA2130563A1 (en) 1993-09-02
EP0628043A1 (de) 1994-12-14
FI943872A (fi) 1994-08-23
FI943872A0 (fi) 1994-08-23
IL104821A0 (en) 1993-06-10
WO1993017019A1 (en) 1993-09-02
MX9300948A (es) 1993-08-01
HU9402436D0 (en) 1994-10-28
NZ249346A (en) 1995-10-26
AU675060B2 (en) 1997-01-23
KR100287933B1 (ko) 2001-05-02
FI105917B (fi) 2000-10-31
NO943101D0 (no) 1994-08-23
AU3603493A (en) 1993-09-13
JPH07504192A (ja) 1995-05-11
TW226374B (de) 1994-07-11
CA2130563C (en) 1997-11-11

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