NO20070502L - Azaindoles useful as inhibitors of protein kinases - Google Patents

Azaindoles useful as inhibitors of protein kinases

Info

Publication number
NO20070502L
NO20070502L NO20070502A NO20070502A NO20070502L NO 20070502 L NO20070502 L NO 20070502L NO 20070502 A NO20070502 A NO 20070502A NO 20070502 A NO20070502 A NO 20070502A NO 20070502 L NO20070502 L NO 20070502L
Authority
NO
Norway
Prior art keywords
inhibitors
protein kinases
azaindoles
useful
azaindoles useful
Prior art date
Application number
NO20070502A
Other languages
Norwegian (no)
Inventor
Michael Mortimore
Francoise Pierard
Juan-Miguel Jimenez
Ronald Kengtel
Guy Brenchley
Francesca Mazzei
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2005/011358 external-priority patent/WO2005103050A2/en
Priority claimed from PCT/US2005/023429 external-priority patent/WO2006004984A1/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20070502L publication Critical patent/NO20070502L/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)

Abstract

Foreliggende oppfinnelse vedrører azaindoler (I) som er nyttige som inhibitorer av proteinkinaser. Oppfinnelsen tilveiebringer også farmasøytisk akseptable sammensetninger omfattende nevnte forbindelser og metoder for å anvende sammensetningene i behandlingen av forskjellige sykdommer, tilstander eller forstyrrelser. Oppfinnelsen tilveiebringer også fremgangsmåter for å fremstille forbindelsene ifølge oppfinnelsen.The present invention relates to azaindoles (I) which are useful as inhibitors of protein kinases. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods for using the compositions in the treatment of various diseases, conditions or disorders. The invention also provides methods for preparing the compounds of the invention.

NO20070502A 2004-06-30 2007-01-26 Azaindoles useful as inhibitors of protein kinases NO20070502L (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US58472104P 2004-07-01 2004-07-01
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
PCT/US2005/023429 WO2006004984A1 (en) 2004-06-30 2005-06-29 Azaindoles useful as inhibitors of protein kinases

Publications (1)

Publication Number Publication Date
NO20070502L true NO20070502L (en) 2007-01-26

Family

ID=37801682

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20070502A NO20070502L (en) 2004-06-30 2007-01-26 Azaindoles useful as inhibitors of protein kinases

Country Status (4)

Country Link
JP (2) JP5122280B2 (en)
IL (1) IL180303A0 (en)
MX (1) MX2007000092A (en)
NO (1) NO20070502L (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5122280B2 (en) * 2004-06-30 2013-01-16 バーテックス ファーマシューティカルズ インコーポレイテッド Azaindoles useful as inhibitors of protein kinases
BRPI0515012A (en) * 2004-08-13 2008-07-01 Genentech Inc chemical substance, pharmaceutical composition and formulation, method of treatment, method of inhibiting at least one enzyme using atp and use
DE102008038221A1 (en) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-azaindole derivatives
DE102009058280A1 (en) * 2009-12-14 2011-06-16 Merck Patent Gmbh thiazole
JP5911470B2 (en) 2010-04-16 2016-04-27 エーシー・イミューン・エス・アー Novel compounds for treating diseases associated with amyloid or amyloid-like proteins
MX2013000103A (en) * 2010-06-23 2013-06-13 Vertex Pharma Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase.
DE102011105469A1 (en) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-azaindole derivatives
EA201791271A1 (en) * 2012-05-31 2018-01-31 Фенекс Фармасьютикалз Аг THIAZOLES, SUBSTITUTED BY CARBOXAMIDE OR SULPHONAMIDE AND RELATED DERIVATIVES AS MODULATORS FOR ORPHANIC NUCLEAR RORγ RECEPTOR
JP5938533B2 (en) 2014-02-04 2016-06-22 大鵬薬品工業株式会社 Azaindole derivatives
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
DE60136530D1 (en) * 2000-03-01 2008-12-24 Janssen Pharmaceutica Nv 2,4-DISUBSTITUTED THIAZOLYL DERIVATIVES
SE0202463D0 (en) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
AR049333A1 (en) * 2004-04-02 2006-07-19 Vertex Pharma INHIBITING AZAINDOLS OF ROCK PROTEINQUINASES AND OTHER KINASE PROTEINS. PHARMACEUTICAL COMPOSITIONS.
JP5122280B2 (en) * 2004-06-30 2013-01-16 バーテックス ファーマシューティカルズ インコーポレイテッド Azaindoles useful as inhibitors of protein kinases

Also Published As

Publication number Publication date
JP5122280B2 (en) 2013-01-16
JP2012012417A (en) 2012-01-19
IL180303A0 (en) 2007-06-03
MX2007000092A (en) 2007-03-07
JP2008513352A (en) 2008-05-01

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