NO20065783L - Pyridin-4-yl-ethyl imidazoles and pyrazoles as MGLU5 receptor antagonists - Google Patents

Pyridin-4-yl-ethyl imidazoles and pyrazoles as MGLU5 receptor antagonists

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Publication number
NO20065783L
NO20065783L NO20065783A NO20065783A NO20065783L NO 20065783 L NO20065783 L NO 20065783L NO 20065783 A NO20065783 A NO 20065783A NO 20065783 A NO20065783 A NO 20065783A NO 20065783 L NO20065783 L NO 20065783L
Authority
NO
Norway
Prior art keywords
pyrazoles
pyridin
receptor antagonists
mglu5 receptor
ethyl imidazoles
Prior art date
Application number
NO20065783A
Other languages
Norwegian (no)
Inventor
Sabine Kolczewski
Bernd Buettelmann
Georg Jaeschke
Eric Vieira
Simona Maria Ceccarelli
Richard Hugh Phillip Porter
Paul Spurr
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2004/005881 external-priority patent/WO2004108701A1/en
Priority claimed from PCT/EP2005/005559 external-priority patent/WO2005118568A1/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO20065783L publication Critical patent/NO20065783L/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Foreliggende oppfinnelse angår diazolderivater med den generelle formel (I) hvor A, E, R1, R2 og R3 er som definert i krav og beskrivelse, anvendelse av dem for fremstilling av medikamenter for behandling av sykdommer og fremgangsmåter for fremstilling av dem.The present invention relates to diazole derivatives of the general formula (I) wherein A, E, R 1, R 2 and R 3 are as defined in claim and description, their use in the manufacture of medicaments for the treatment of diseases and methods of preparing them.

NO20065783A 2004-06-01 2006-12-13 Pyridin-4-yl-ethyl imidazoles and pyrazoles as MGLU5 receptor antagonists NO20065783L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/EP2004/005881 WO2004108701A1 (en) 2003-06-05 2004-06-01 Imidazole derivatives as glutmate receptor antagonists
PCT/EP2005/005559 WO2005118568A1 (en) 2004-06-01 2005-05-23 Pyridin-4-yl-ethynyl-imidazoles and pyrazoles as mglu5 receptor antagonists

Publications (1)

Publication Number Publication Date
NO20065783L true NO20065783L (en) 2006-12-13

Family

ID=37781937

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20065783A NO20065783L (en) 2004-06-01 2006-12-13 Pyridin-4-yl-ethyl imidazoles and pyrazoles as MGLU5 receptor antagonists

Country Status (2)

Country Link
NO (1) NO20065783L (en)
UA (1) UA85094C2 (en)

Also Published As

Publication number Publication date
UA85094C2 (en) 2008-12-25

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application