NO20063380L - Triazole derivatives as vasopressin antagonists - Google Patents
Triazole derivatives as vasopressin antagonistsInfo
- Publication number
- NO20063380L NO20063380L NO20063380A NO20063380A NO20063380L NO 20063380 L NO20063380 L NO 20063380L NO 20063380 A NO20063380 A NO 20063380A NO 20063380 A NO20063380 A NO 20063380A NO 20063380 L NO20063380 L NO 20063380L
- Authority
- NO
- Norway
- Prior art keywords
- triazole derivatives
- vasopressin antagonists
- ring
- vasopressin
- antagonists
- Prior art date
Links
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- C07—ORGANIC CHEMISTRY
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Abstract
Forbindelser med formel (I) eller farmasøytisk akseptable derivater derav, hvori: V representerer en direkte binding eller -O-; Ring A representerer en eventuelt substituert 5- til 7-leddet mettet heterosyklisk ring, eller en fenylengruppe.Compounds of formula (I) or pharmaceutically acceptable derivatives thereof, wherein: V represents a direct bond or -O-; Ring A represents an optionally substituted 5- to 7-membered saturated heterocyclic ring, or a phenylene group.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0329693A GB0329693D0 (en) | 2003-12-22 | 2003-12-22 | Compounds useful in therapy |
GB0408789A GB0408789D0 (en) | 2004-04-20 | 2004-04-20 | Triazole derivatives |
PCT/IB2004/004059 WO2005063754A1 (en) | 2003-12-22 | 2004-12-09 | Triazole derivatives as vasopressin antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20063380L true NO20063380L (en) | 2006-09-22 |
Family
ID=34740750
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20063380A NO20063380L (en) | 2003-12-22 | 2006-07-21 | Triazole derivatives as vasopressin antagonists |
Country Status (25)
Country | Link |
---|---|
EP (1) | EP1701959A1 (en) |
JP (1) | JP4698604B2 (en) |
KR (1) | KR100854872B1 (en) |
AP (1) | AP2331A (en) |
AR (1) | AR047340A1 (en) |
AU (1) | AU2004309164B2 (en) |
BR (1) | BRPI0417267A (en) |
CA (1) | CA2551038C (en) |
CR (1) | CR8481A (en) |
DO (1) | DOP2004001062A (en) |
EA (1) | EA010132B1 (en) |
EC (1) | ECSP066647A (en) |
GE (1) | GEP20084571B (en) |
HK (1) | HK1095822A1 (en) |
IL (1) | IL176349A (en) |
IS (1) | IS8472A (en) |
MA (1) | MA28393B1 (en) |
NL (1) | NL1027833C2 (en) |
NO (1) | NO20063380L (en) |
OA (1) | OA13347A (en) |
PA (1) | PA8620501A1 (en) |
PE (1) | PE20051051A1 (en) |
TW (1) | TWI287541B (en) |
UY (1) | UY28693A1 (en) |
WO (1) | WO2005063754A1 (en) |
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EP1830837B1 (en) | 2004-09-20 | 2013-09-04 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes |
MX2007003325A (en) * | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors. |
AU2005286648A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors |
AU2005286728A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as mediators of stearoyl-CoA desaturase |
BRPI0515482A (en) | 2004-09-20 | 2008-07-22 | Xenon Pharmaceuticals Inc | heterocyclic derivatives and their uses as therapeutic agents |
AR051094A1 (en) | 2004-09-20 | 2006-12-20 | Xenon Pharmaceuticals Inc | HETEROCICLIC DERIVATIVES AND THEIR USE AS INHIBITORS OF ESTEAROIL-COA DESATURASA |
DE602005019602D1 (en) | 2004-10-26 | 2010-04-08 | Eisai R&D Man Co Ltd | AMORPHIC FORM OF A CINEMA ACID AMID CONNECTION |
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WO2019081303A1 (en) | 2017-10-24 | 2019-05-02 | Bayer Pharma Aktiengesellschaft | Substituted triazole derivatives and uses thereof |
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US4481360A (en) * | 1983-08-26 | 1984-11-06 | The Upjohn Company | 4H-1,2,4-Triazol-3-yl compounds |
AU2000223275A1 (en) * | 2000-02-08 | 2001-08-20 | Yamanouchi Pharmaceutical Co..Ltd. | Novel triazole derivatives |
BR0110961A (en) * | 2000-05-19 | 2004-06-29 | Merck Patent Gmbh | Triazole derivatives |
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DOP2004001062A (en) | 2005-06-30 |
MA28393B1 (en) | 2007-01-02 |
JP2007515468A (en) | 2007-06-14 |
IL176349A (en) | 2011-11-30 |
PE20051051A1 (en) | 2005-12-17 |
BRPI0417267A (en) | 2007-04-17 |
EA200600925A1 (en) | 2006-12-29 |
GEP20084571B (en) | 2008-12-25 |
AP2331A (en) | 2011-12-05 |
WO2005063754A1 (en) | 2005-07-14 |
NL1027833C2 (en) | 2006-03-06 |
IS8472A (en) | 2006-05-18 |
AU2004309164B2 (en) | 2007-11-15 |
NL1027833A1 (en) | 2005-06-23 |
UY28693A1 (en) | 2005-07-29 |
CR8481A (en) | 2007-12-04 |
PA8620501A1 (en) | 2005-08-04 |
AU2004309164A1 (en) | 2005-07-14 |
EP1701959A1 (en) | 2006-09-20 |
TWI287541B (en) | 2007-10-01 |
HK1095822A1 (en) | 2007-07-06 |
AR047340A1 (en) | 2006-01-18 |
KR100854872B1 (en) | 2008-08-28 |
OA13347A (en) | 2007-04-13 |
CA2551038A1 (en) | 2005-07-14 |
TW200528099A (en) | 2005-09-01 |
JP4698604B2 (en) | 2011-06-08 |
AP2006003631A0 (en) | 2006-06-30 |
IL176349A0 (en) | 2006-10-05 |
CA2551038C (en) | 2010-04-27 |
ECSP066647A (en) | 2006-10-25 |
EA010132B1 (en) | 2008-06-30 |
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