NO20053313L - Antiparasitic terpene alkaloids. - Google Patents

Antiparasitic terpene alkaloids.

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Publication number
NO20053313L
NO20053313L NO20053313A NO20053313A NO20053313L NO 20053313 L NO20053313 L NO 20053313L NO 20053313 A NO20053313 A NO 20053313A NO 20053313 A NO20053313 A NO 20053313A NO 20053313 L NO20053313 L NO 20053313L
Authority
NO
Norway
Prior art keywords
terpene
antiparasitic
disclosed
antiparasite
alkaloids
Prior art date
Application number
NO20053313A
Other languages
Norwegian (no)
Other versions
NO20053313D0 (en
Inventor
Nigel Derek Arthur Walshe
Graham Lunn
Douglas James Critcher
Nathan Anthony Logan Chubb
James John Eshelby
Andrew John Rudge
Paul Heinrich Wiedenau
David Howard Williams
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/IB2004/000320 external-priority patent/WO2004072086A2/en
Application filed by Pfizer filed Critical Pfizer
Publication of NO20053313D0 publication Critical patent/NO20053313D0/en
Publication of NO20053313L publication Critical patent/NO20053313L/en

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Abstract

Det er beskrevet nye terpenalkaloider og anvendelse derav som antiparasittmidler. Det er videre beskrevet et antiparasittmiddel som omfatter en terpenalkaloidforbindelse som en effektiv ingrediens i en antiparasittformulering. Foreliggende oppfinnelse vedrører spesielt derivater av terpenalkaloid (1S,2R,4aS,5R,8R,8aR)-2-(acetyloksy)-8a-hydroksy3,8-dimetyl-5-(1-metyletenyl)-1,2,4a,5,6,7,8,8a- oktahydronaftalen-1-yl (2S,3aR,9bR)-6-klor-9b-hydroksy-5-metyl-1,2,3,3a,5,9b-heksahydropyrrol[2,3-c] [2,1]benzoksazin-2-karboksylat. Det er beskrevet farmasøytiske sammensetninger som omfatter disse.New terpene alkaloids and their use as antiparasitic agents have been described. Further, an antiparasite agent is disclosed which comprises a terpene alkaloid compound as an effective ingredient in an antiparasite formulation. The present invention relates in particular to derivatives of terpene alkaloid (1S, 2R, 4aS, 5R, 8R, 8aR) -2- (acetyloxy) -8a-hydroxy3,8-dimethyl-5- (1-methylethenyl) -1,2,4a, 5 , 6,7,8,8a-octahydronaphthalen-1-yl (2S, 3aR, 9bR) -6-chloro-9b-hydroxy-5-methyl-1,2,3,3a, 5,9b-hexahydropyrrole [2, 3-c] [2,1] benzoxazine-2-carboxylate. Pharmaceutical compositions are disclosed which comprise these.

NO20053313A 2003-02-14 2005-07-06 Antiparasitic terpene alkaloids. NO20053313L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30343903A 2003-02-14 2003-02-14
PCT/IB2004/000320 WO2004072086A2 (en) 2003-02-14 2004-02-03 Antiparasitic terpene alkaloids

Publications (2)

Publication Number Publication Date
NO20053313D0 NO20053313D0 (en) 2005-07-06
NO20053313L true NO20053313L (en) 2005-08-08

Family

ID=35295146

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20053313A NO20053313L (en) 2003-02-14 2005-07-06 Antiparasitic terpene alkaloids.

Country Status (1)

Country Link
NO (1) NO20053313L (en)

Also Published As

Publication number Publication date
NO20053313D0 (en) 2005-07-06

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