NO20053313L - Antiparasitic terpene alkaloids. - Google Patents

Antiparasitic terpene alkaloids.

Info

Publication number
NO20053313L
NO20053313L NO20053313A NO20053313A NO20053313L NO 20053313 L NO20053313 L NO 20053313L NO 20053313 A NO20053313 A NO 20053313A NO 20053313 A NO20053313 A NO 20053313A NO 20053313 L NO20053313 L NO 20053313L
Authority
NO
Norway
Prior art keywords
terpene
antiparasitic
disclosed
antiparasite
alkaloids
Prior art date
Application number
NO20053313A
Other languages
Norwegian (no)
Other versions
NO20053313D0 (en
Inventor
Nigel Derek Arthur Walshe
Graham Lunn
Douglas James Critcher
Nathan Anthony Logan Chubb
James John Eshelby
Andrew John Rudge
Paul Heinrich Wiedenau
David Howard Williams
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/IB2004/000320 external-priority patent/WO2004072086A2/en
Application filed by Pfizer filed Critical Pfizer
Publication of NO20053313D0 publication Critical patent/NO20053313D0/en
Publication of NO20053313L publication Critical patent/NO20053313L/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Det er beskrevet nye terpenalkaloider og anvendelse derav som antiparasittmidler. Det er videre beskrevet et antiparasittmiddel som omfatter en terpenalkaloidforbindelse som en effektiv ingrediens i en antiparasittformulering. Foreliggende oppfinnelse vedrører spesielt derivater av terpenalkaloid (1S,2R,4aS,5R,8R,8aR)-2-(acetyloksy)-8a-hydroksy3,8-dimetyl-5-(1-metyletenyl)-1,2,4a,5,6,7,8,8a- oktahydronaftalen-1-yl (2S,3aR,9bR)-6-klor-9b-hydroksy-5-metyl-1,2,3,3a,5,9b-heksahydropyrrol[2,3-c] [2,1]benzoksazin-2-karboksylat. Det er beskrevet farmasøytiske sammensetninger som omfatter disse.New terpene alkaloids and their use as antiparasitic agents have been described. Further, an antiparasite agent is disclosed which comprises a terpene alkaloid compound as an effective ingredient in an antiparasite formulation. The present invention relates in particular to derivatives of terpene alkaloid (1S, 2R, 4aS, 5R, 8R, 8aR) -2- (acetyloxy) -8a-hydroxy3,8-dimethyl-5- (1-methylethenyl) -1,2,4a, 5 , 6,7,8,8a-octahydronaphthalen-1-yl (2S, 3aR, 9bR) -6-chloro-9b-hydroxy-5-methyl-1,2,3,3a, 5,9b-hexahydropyrrole [2, 3-c] [2,1] benzoxazine-2-carboxylate. Pharmaceutical compositions are disclosed which comprise these.

NO20053313A 2003-02-14 2005-07-06 Antiparasitic terpene alkaloids. NO20053313L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30343903A 2003-02-14 2003-02-14
PCT/IB2004/000320 WO2004072086A2 (en) 2003-02-14 2004-02-03 Antiparasitic terpene alkaloids

Publications (2)

Publication Number Publication Date
NO20053313D0 NO20053313D0 (en) 2005-07-06
NO20053313L true NO20053313L (en) 2005-08-08

Family

ID=35295146

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20053313A NO20053313L (en) 2003-02-14 2005-07-06 Antiparasitic terpene alkaloids.

Country Status (1)

Country Link
NO (1) NO20053313L (en)

Also Published As

Publication number Publication date
NO20053313D0 (en) 2005-07-06

Similar Documents

Publication Publication Date Title
MXPA05008618A (en) Antiparasitic terpene alkaloids.
YU49898A (en) Chemical compounds
HUP0303271A2 (en) Use of rapamycin for preparation of pharmaceutical composition suitable for cancer treatment
UY26258A1 (en) DERIVATIVES OF 8-PHENYL-6,9-DIHYDRO- [1,2,4] TRIAZOLO [3,4-I] PURIN-5-ONA.
HUT77667A (en) Imidazo[4,5-c]quinoline amines, their use and pharmaceutical compositions containing them
DE69231522T2 (en) 1-SUBSTITUTED-4-AMINO-1H-IMIDAZO 4,5-C CHINOLINE, INTERMEDIATE PRODUCTS AND MEDICINAL PRODUCTS
WO2006107771A3 (en) PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS
WO2004037212A3 (en) Compositions comprising zopiclone derivatives and methods of making and using the same
NO961136L (en) Pharmaceutical formulation basis for nano-suspensions
DE69226537T2 (en) ANTIVIRAL 2-ETHYL-1H-IMIDAZO (4,5-C) CHINOLIN-4-AMINE
NO20062019L (en) Β-Glycoprotein Inhibitor, Methods of Preparation thereof, and Pharmaceutical Preparations Containing the Same
WO2006016067A3 (en) Pyrido-pyrido pyrimidine derivatives, preparation thereof, therapeutic use thereof for treating cancer
WO2002048148A3 (en) Pyrazolopyridine derivatives
TNSN07485A1 (en) N- (ARYLALKYL) -1H-PYRROLOPYRIDINE -2-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE
ES2328496T3 (en) 1,4,8-TRIAZA-ESPIRO (4,5) DECAN-2-ONA SUBSTITUTED COMPOUNDS.
WO2005044818A3 (en) Imidazo[1,2-a]pyridine anxiolytics
HUP9900438A2 (en) Use of pyrazolo[4,3-d]pyrimidin-7-one derivatives for the preparation of pharmaceutical compositions treaing impotence due to spinal cord injury
HUP0500028A2 (en) Drugs comprising combination of triazaspiro[5,5]undecane derivative with cytochrome p450 isozyme 3a4 inhibitor and/or p-glycoprotein inhibitor
NO20053313L (en) Antiparasitic terpene alkaloids.
PT880520E (en) DERIVATIVES OF BENZOICHINOLIZIN ITS PREPARATION AND USE AS 5-ALPHA-REDUCTASE INHIBITORS
WO2005013935A3 (en) Composition for releasing a weak base for an extended period of time
CA2438813A1 (en) Alkoxycarbonylamino heteroaryl carboxylic acid derivatives as ip antagonists
CA2445189A1 (en) Carboline derivatives as pdev inhibitors
WO2002000656A3 (en) Pirazino '1$m(1)2$m(1) :1, 6! pyrido '3,4-b! indole derivatives
WO2004085436A3 (en) Pyrido[2,3-d]pyrimidin-7-carboxylic acid derivatives, their manufacture and use as pharmaceutical agents

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application