NO20012099D0 - Process for the preparation of 4-arylpiperidine-3-carbinols and related compounds - Google Patents

Process for the preparation of 4-arylpiperidine-3-carbinols and related compounds

Info

Publication number
NO20012099D0
NO20012099D0 NO20012099A NO20012099A NO20012099D0 NO 20012099 D0 NO20012099 D0 NO 20012099D0 NO 20012099 A NO20012099 A NO 20012099A NO 20012099 A NO20012099 A NO 20012099A NO 20012099 D0 NO20012099 D0 NO 20012099D0
Authority
NO
Norway
Prior art keywords
arylpiperidine
carbinols
preparation
related compounds
compounds
Prior art date
Application number
NO20012099A
Other languages
Norwegian (no)
Other versions
NO20012099L (en
Inventor
Theodorus Hendricus Ant Peters
Franciscus Bernardus Benneker
Hans Jan Hoorn
Frantisek Picha
Original Assignee
Synthon Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthon Bv filed Critical Synthon Bv
Publication of NO20012099D0 publication Critical patent/NO20012099D0/en
Publication of NO20012099L publication Critical patent/NO20012099L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C07D211/76—Oxygen atoms attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
NO20012099A 1998-11-02 2001-04-27 Process for Preparation of 4-Arylpiperidine-3-Carbinols and Related Compounds NO20012099L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10667398P 1998-11-02 1998-11-02
PCT/IB1999/001762 WO2000026187A1 (en) 1998-11-02 1999-11-01 Process for producing 4-arylpiperidine-3-carbinols and related compounds

Publications (2)

Publication Number Publication Date
NO20012099D0 true NO20012099D0 (en) 2001-04-27
NO20012099L NO20012099L (en) 2001-07-02

Family

ID=22312658

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20012099A NO20012099L (en) 1998-11-02 2001-04-27 Process for Preparation of 4-Arylpiperidine-3-Carbinols and Related Compounds

Country Status (5)

Country Link
EP (1) EP1124802A1 (en)
AU (1) AU6360999A (en)
CZ (1) CZ20011465A3 (en)
NO (1) NO20012099L (en)
WO (1) WO2000026187A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE279393T1 (en) 1997-05-29 2004-10-15 Smithkline Beecham Corp NEW PROCEDURE
US20010053862A1 (en) * 1998-12-22 2001-12-20 Bruce Ronsen Process for preparing arylpiperidine carbinol intermediates and derivatives
WO2000037443A1 (en) * 1998-12-22 2000-06-29 Pentech Pharmaceuticals, Inc. Process for preparing arylpiperidine carbinol intermediates and derivatives
EP1280775A1 (en) * 2000-05-12 2003-02-05 Synthon B.V. TOSYLATE SALTS OF 4-(p-FLUOROPHENYL)-PIPERIDINE-3-CARBINOLS
WO2002053537A1 (en) 2001-01-04 2002-07-11 Ferrer Internacional, S.A. Process for preparing (±) trans-4-p-fluorophenyl-3-hydroxymethyl-1-methylpiperidine
EP1440067B1 (en) 2001-10-22 2004-12-22 Synthon B.V. N-formyl derivatives of paroxetine
WO2007089193A1 (en) * 2006-02-02 2007-08-09 Astrazeneca Ab A process for preparing 2-hydroxy-3- [5- (morpholin-4-ylmethyl)pyridin-2-yl] lh-indole-5-carbonitrile as a free base or salts thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI792076A (en) * 1978-07-05 1980-01-06 Ciba Geigy Ag FOERFARANDE FOER FRAMSTAELLNING AV NYA FENYLPIPERIDINDERIVAT
DE3680184D1 (en) * 1985-08-10 1991-08-14 Beecham Group Plc METHOD FOR PRODUCING ARYLPIPERIDINE CARBINOL.
US5258517A (en) * 1992-08-06 1993-11-02 Sepracor, Inc. Method of preparing optically pure precursors of paroxetine
GB9526645D0 (en) * 1995-12-28 1996-02-28 Chiroscience Ltd Stereoselective synthesis
JP3446468B2 (en) * 1996-04-15 2003-09-16 旭硝子株式会社 Method for producing piperidine carbinols
ATE279393T1 (en) * 1997-05-29 2004-10-15 Smithkline Beecham Corp NEW PROCEDURE

Also Published As

Publication number Publication date
EP1124802A1 (en) 2001-08-22
WO2000026187A1 (en) 2000-05-11
CZ20011465A3 (en) 2001-08-15
NO20012099L (en) 2001-07-02
AU6360999A (en) 2000-05-22

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application