NO169125C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 10-SUBSTITUTED 9-FLUOR-7-OXO-2,3-DIHYDRO-7H-PYRIDO (3.2.1-IJ) -1,3,4-BENZOXADIAZINE-6-CARBOXYLSYL - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 10-SUBSTITUTED 9-FLUOR-7-OXO-2,3-DIHYDRO-7H-PYRIDO (3.2.1-IJ) -1,3,4-BENZOXADIAZINE-6-CARBOXYLSYL

Info

Publication number
NO169125C
NO169125C NO873816A NO873816A NO169125C NO 169125 C NO169125 C NO 169125C NO 873816 A NO873816 A NO 873816A NO 873816 A NO873816 A NO 873816A NO 169125 C NO169125 C NO 169125C
Authority
NO
Norway
Prior art keywords
carboxylsyl
benzoxadiazine
pyrido
fluor
dihydro
Prior art date
Application number
NO873816A
Other languages
Norwegian (no)
Other versions
NO169125B (en
NO873816L (en
NO873816D0 (en
Inventor
Masahiro Aoki
Miyako Kamata
Tatsuo Ohtsuka
Nobuo Shimma
Kazuteru Yokose
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO873816D0 publication Critical patent/NO873816D0/en
Publication of NO873816L publication Critical patent/NO873816L/en
Priority to NO894108A priority Critical patent/NO171162C/en
Priority to NO894109A priority patent/NO174926C/en
Publication of NO169125B publication Critical patent/NO169125B/en
Publication of NO169125C publication Critical patent/NO169125C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/58—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO873816A 1986-09-12 1987-09-11 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 10-SUBSTITUTED 9-FLUOR-7-OXO-2,3-DIHYDRO-7H-PYRIDO (3.2.1-IJ) -1,3,4-BENZOXADIAZINE-6-CARBOXYLSYL NO169125C (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
NO894108A NO171162C (en) 1986-09-12 1989-10-13 Pyrido BENZOKSADIAZINDERIVATER
NO894109A NO174926C (en) 1986-09-12 1989-10-13 Hydroxyamino oksodihydrokinolinderivater

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP86112619 1986-09-12

Publications (4)

Publication Number Publication Date
NO873816D0 NO873816D0 (en) 1987-09-11
NO873816L NO873816L (en) 1988-03-14
NO169125B NO169125B (en) 1992-02-03
NO169125C true NO169125C (en) 1992-05-13

Family

ID=8195410

Family Applications (1)

Application Number Title Priority Date Filing Date
NO873816A NO169125C (en) 1986-09-12 1987-09-11 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 10-SUBSTITUTED 9-FLUOR-7-OXO-2,3-DIHYDRO-7H-PYRIDO (3.2.1-IJ) -1,3,4-BENZOXADIAZINE-6-CARBOXYLSYL

Country Status (22)

Country Link
JP (3) JPH0696578B2 (en)
KR (1) KR960002857B1 (en)
CN (1) CN1017800B (en)
AT (1) AT389119B (en)
AU (1) AU602534B2 (en)
CA (1) CA1336905C (en)
CZ (1) CZ281195B6 (en)
DK (1) DK173330B1 (en)
DZ (1) DZ1124A1 (en)
FI (1) FI86428C (en)
HU (1) HU199481B (en)
IE (1) IE61624B1 (en)
IL (1) IL83814A (en)
MC (1) MC1850A1 (en)
MX (1) MX8302A (en)
NO (1) NO169125C (en)
NZ (1) NZ221681A (en)
PH (1) PH23930A (en)
PT (1) PT85686B (en)
SK (1) SK278990B6 (en)
ZA (1) ZA876636B (en)
ZW (1) ZW16387A1 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW16387A1 (en) * 1986-09-12 1988-05-25 Hoffmann La Roche Tricyclic compounds
EP1757598A4 (en) 2004-05-13 2010-07-21 Daiichi Seiyaku Co Substituted pyrrolidine derivative
US7563805B2 (en) * 2005-05-19 2009-07-21 Daiichi Pharmaceutical Co., Ltd. Tri-, tetra-substituted-3-aminopyrrolidine derivative
CN101443314B (en) 2006-03-13 2014-04-09 杏林制药株式会社 Aminoquinolones as GSK-3 inhibitors
JP5426552B2 (en) 2007-09-11 2014-02-26 杏林製薬株式会社 Cyanoaminoquinolones and tetrazoloaminoquinolones as GSK-3 inhibitors
MX2010002662A (en) 2007-09-12 2010-04-09 Activx Biosciences Inc Spirocyclic aminoquinolones as gsk-3 inhibitors.
FR2928150A1 (en) * 2008-02-29 2009-09-04 Vetoquinol Sa Sa NOVEL 7-SUBSTITUTED 3-CARBOXY-OXADIAZINO-QUINOLONES DERIVATIVES, THEIR PREPARATION AND APPLICATION AS ANTI-BACTERIANS
EP2145891A1 (en) * 2008-07-09 2010-01-20 Vetoquinol S.A. 9-substituted-5-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials
WO2010104205A1 (en) 2009-03-11 2010-09-16 Kyorin Pharmaceutical Co., Ltd. 7-cycloalkylaminoquinolones as gsk-3 inhibitors
CN107522718B (en) * 2017-09-14 2019-11-08 浙江国邦药业有限公司 A kind of synthetic method of Marbofloxacin

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW16387A1 (en) * 1986-09-12 1988-05-25 Hoffmann La Roche Tricyclic compounds

Also Published As

Publication number Publication date
KR960002857B1 (en) 1996-02-27
ATA263887A (en) 1989-03-15
SK660487A3 (en) 1998-05-06
DK173330B1 (en) 2000-07-24
NO169125B (en) 1992-02-03
FI86428C (en) 1992-08-25
MC1850A1 (en) 1988-09-30
IL83814A (en) 1991-09-16
IE872444L (en) 1988-03-12
CN87106838A (en) 1988-05-11
HUT47294A (en) 1989-02-28
DK477287A (en) 1988-03-13
JPH07138262A (en) 1995-05-30
FI86428B (en) 1992-05-15
JPH0826030B2 (en) 1996-03-13
NO873816L (en) 1988-03-14
PT85686B (en) 1990-05-31
KR880003954A (en) 1988-06-01
NO873816D0 (en) 1987-09-11
HU199481B (en) 1990-02-28
SK278990B6 (en) 1998-05-06
JPS63132891A (en) 1988-06-04
AU602534B2 (en) 1990-10-18
CN1017800B (en) 1992-08-12
AU7811487A (en) 1988-03-17
ZA876636B (en) 1988-07-27
CZ660487A3 (en) 1996-04-17
CA1336905C (en) 1995-09-05
IE61624B1 (en) 1994-11-16
JPH07138256A (en) 1995-05-30
ZW16387A1 (en) 1988-05-25
DK477287D0 (en) 1987-09-11
FI873940A (en) 1988-03-13
CZ281195B6 (en) 1996-07-17
PH23930A (en) 1990-01-23
JPH0819120B2 (en) 1996-02-28
PT85686A (en) 1987-10-01
AT389119B (en) 1989-10-25
FI873940A0 (en) 1987-09-11
JPH0696578B2 (en) 1994-11-30
NZ221681A (en) 1990-12-21
DZ1124A1 (en) 2004-09-13
MX8302A (en) 1993-12-01

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