NL190775C - Pharmaceutical preparations with a psychotropic action containing an ester of substituted [(4-hydroxy-4-phenyl) piperidino] butyrophenones, and a method for preparing these preparations. - Google Patents

Pharmaceutical preparations with a psychotropic action containing an ester of substituted [(4-hydroxy-4-phenyl) piperidino] butyrophenones, and a method for preparing these preparations.

Info

Publication number
NL190775C
NL190775C NL8003583A NL8003583A NL190775C NL 190775 C NL190775 C NL 190775C NL 8003583 A NL8003583 A NL 8003583A NL 8003583 A NL8003583 A NL 8003583A NL 190775 C NL190775 C NL 190775C
Authority
NL
Netherlands
Prior art keywords
preparations
butyrophenones
piperidino
hydroxy
phenyl
Prior art date
Application number
NL8003583A
Other languages
Dutch (nl)
Other versions
NL8003583A (en
NL190775B (en
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NL8003583A publication Critical patent/NL8003583A/en
Publication of NL190775B publication Critical patent/NL190775B/en
Application granted granted Critical
Publication of NL190775C publication Critical patent/NL190775C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
NL8003583A 1979-06-28 1980-06-20 Pharmaceutical preparations with a psychotropic action containing an ester of substituted [(4-hydroxy-4-phenyl) piperidino] butyrophenones, and a method for preparing these preparations. NL190775C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP8082679A JPS568318A (en) 1979-06-28 1979-06-28 Non oral long acting composition of haloperidol and bromperidol derivative
JP8082679 1979-06-28

Publications (3)

Publication Number Publication Date
NL8003583A NL8003583A (en) 1980-12-30
NL190775B NL190775B (en) 1994-03-16
NL190775C true NL190775C (en) 1994-08-16

Family

ID=13729223

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8003583A NL190775C (en) 1979-06-28 1980-06-20 Pharmaceutical preparations with a psychotropic action containing an ester of substituted [(4-hydroxy-4-phenyl) piperidino] butyrophenones, and a method for preparing these preparations.

Country Status (9)

Country Link
JP (1) JPS568318A (en)
BE (1) BE883994A (en)
CY (1) CY1255A (en)
DE (1) DE3024305A1 (en)
FR (1) FR2460932A1 (en)
GB (1) GB2054371B (en)
HK (1) HK83384A (en)
KE (1) KE3427A (en)
NL (1) NL190775C (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8621892D0 (en) * 1986-09-11 1986-10-15 Lundbeck & Co As H Organic compound
DK238190D0 (en) * 1990-10-03 1990-10-03 Lundbeck & Co As H DEPOT DERIVATIVES
DK0669128T3 (en) * 1992-11-17 2000-06-19 Yoshitomi Pharmaceutical Sustained-release microsphere containing antipsychotics and method of producing same
WO1998018769A1 (en) * 1996-10-31 1998-05-07 The United States Of America, Represented By The Secretary, Department Of Health And Human Services Sustained-release derivatives of hydroxylated analogs of substituted 1-[2[bis(aryl)methoxy]ethyl]-piperazines and -homopiperazines and their use as noncompetitive antagonists of dopamine reuptake
JP2008519840A (en) 2004-11-10 2008-06-12 ジェンザイム・コーポレイション How to treat diabetes
WO2007134086A2 (en) 2006-05-09 2007-11-22 Genzyme Corporation Methods of treating fatty liver disease comprising inhibiting glucosphingolipid synthesis
WO2008150486A2 (en) 2007-05-31 2008-12-11 Genzyme Corporation 2-acylaminopropoanol-type glucosylceramide synthase inhibitors
BRPI0817864A2 (en) 2007-10-05 2012-12-25 Genzyme Corp use of a ceramide-derived compound
CA2731685A1 (en) 2008-07-28 2010-02-04 Genzyme Corporation Glucosylceramide synthase inhibition for the treatment of collapsing glomerulopathy and other glomerular disease
EP3078373A1 (en) 2008-10-03 2016-10-12 Genzyme Corporation 2-acylaminopropanol-type glucosylceramide synthase inhibitor
FI3156056T3 (en) 2011-03-18 2024-03-01 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising sorbitan esters
CN103301461B (en) * 2012-03-08 2018-09-07 江苏豪森药业集团有限公司 A kind of long acting injection and its preparation method and application
CA2867123C (en) 2012-03-19 2021-02-16 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising water-insoluble antipsychotic agents and glycerol esters
EP2827868B8 (en) 2012-03-19 2019-12-18 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
ES2950418T3 (en) 2012-03-19 2023-10-09 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising benzyl alcohol
JP6654042B2 (en) 2012-09-19 2020-02-26 アルカームス ファーマ アイルランド リミテッド Pharmaceutical composition with improved storage stability
CA2943213C (en) 2014-03-20 2022-07-05 Alkermes Pharma Ireland Limited Aripiprazole formulations having increased injection speeds
EP3761983A1 (en) 2018-03-05 2021-01-13 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
CN113117092A (en) * 2020-01-14 2021-07-16 中国科学院上海药物研究所 Non-aqueous sustained-release drug delivery system
HUP2100259A1 (en) 2021-07-07 2023-01-28 Richter Gedeon Nyrt Controlled release injectable cariprazine formulation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3408356A (en) * 1965-08-31 1968-10-29 Squibb & Sons Inc Long chain esters of 4'-fluoro-4-[4-hydroxy-4-(alpha, alpha, alpha-trifluorotolyl)piperi-dino]butyrophenone and the like
DE1695194A1 (en) * 1966-07-11 1971-03-18 Hoffmann La Roche Process for the preparation of piperidine derivatives
US3850935A (en) * 1971-10-16 1974-11-26 Sumitomo Chemical Co Process for producing piperidine derivatives by degrading quaternary piperidinium salts

Also Published As

Publication number Publication date
JPS568318A (en) 1981-01-28
DE3024305A1 (en) 1981-01-22
FR2460932B1 (en) 1984-11-16
KE3427A (en) 1984-08-10
NL8003583A (en) 1980-12-30
GB2054371A (en) 1981-02-18
BE883994A (en) 1980-12-29
CY1255A (en) 1984-08-31
DE3024305C2 (en) 1989-12-07
HK83384A (en) 1984-11-09
FR2460932A1 (en) 1981-01-30
NL190775B (en) 1994-03-16
GB2054371B (en) 1983-08-03

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
V4 Lapsed because of reaching the maximum lifetime of a patent

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