NL144944B - PROCESS FOR THE PREPARATION OF 6-AMINOPENICILLAAN ACID DERIVATIVES. - Google Patents

PROCESS FOR THE PREPARATION OF 6-AMINOPENICILLAAN ACID DERIVATIVES.

Info

Publication number
NL144944B
NL144944B NL686804392A NL6804392A NL144944B NL 144944 B NL144944 B NL 144944B NL 686804392 A NL686804392 A NL 686804392A NL 6804392 A NL6804392 A NL 6804392A NL 144944 B NL144944 B NL 144944B
Authority
NL
Netherlands
Prior art keywords
aminopenicillaan
preparation
acid derivatives
derivatives
acid
Prior art date
Application number
NL686804392A
Other languages
Dutch (nl)
Other versions
NL6804392A (en
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of NL6804392A publication Critical patent/NL6804392A/xx
Publication of NL144944B publication Critical patent/NL144944B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
NL686804392A 1967-03-29 1968-03-28 PROCESS FOR THE PREPARATION OF 6-AMINOPENICILLAAN ACID DERIVATIVES. NL144944B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR100617A FR1525186A (en) 1967-03-29 1967-03-29 New penicillins and method of preparation
FR138141A FR7155M (en) 1967-03-29 1968-01-31

Publications (2)

Publication Number Publication Date
NL6804392A NL6804392A (en) 1968-09-30
NL144944B true NL144944B (en) 1975-02-17

Family

ID=26175147

Family Applications (1)

Application Number Title Priority Date Filing Date
NL686804392A NL144944B (en) 1967-03-29 1968-03-28 PROCESS FOR THE PREPARATION OF 6-AMINOPENICILLAAN ACID DERIVATIVES.

Country Status (8)

Country Link
US (1) US3494917A (en)
CH (1) CH491958A (en)
DE (1) DE1770062C3 (en)
DK (1) DK118021B (en)
FR (2) FR1525186A (en)
GB (2) GB1209669A (en)
IL (1) IL29661A (en)
NL (1) NL144944B (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8531615D0 (en) * 1985-12-23 1986-02-05 Zambeletti Spa L Compounds
HU212427B (en) * 1991-12-19 1996-06-28 Gyogyszerkutato Intezet Process for producing dl-, d- and l-1,2,3,4-tetrahydroisoquinoline-1-carboxylic acids and their derivatives containing urethane-type n-protecting groups
CN103987697B (en) 2011-10-14 2017-04-26 百时美施贵宝公司 Substituted tetrahydroisoquinoline compounds as factor XIA inhibitors
ES2579832T3 (en) 2011-10-14 2016-08-17 Bristol-Myers Squibb Company Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
SG11201401384UA (en) 2011-10-14 2014-09-26 Bristol Myers Squibb Co Substituted tetrahydroisoquinoline compounds as factor xia inhibitors
CN104837833B (en) 2012-10-12 2017-07-14 百时美施贵宝公司 The crystal formation of XIA factor inhibitors
EP2906552B1 (en) 2012-10-12 2017-11-22 Bristol-Myers Squibb Company Guanidine substituted tetrahydroisoquinoline compounds as factor xia inhibitors
WO2014059214A1 (en) 2012-10-12 2014-04-17 Bristol-Myers Squibb Company Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors
ES2712699T3 (en) 2013-03-25 2019-05-14 Bristol Myers Squibb Co Tetrahydroisoquinolines containing substituted azoles as inhibitors of factor XIa
CN116987080A (en) 2014-01-31 2023-11-03 百时美施贵宝公司 Macrocyclic compounds with heterocyclic P2' groups as factor XIA inhibitors
NO2760821T3 (en) 2014-01-31 2018-03-10
JP6526796B2 (en) 2014-09-04 2019-06-05 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company Diamide macrocycles that are FXIA inhibitors
US9453018B2 (en) 2014-10-01 2016-09-27 Bristol-Myers Squibb Company Pyrimidinones as factor XIa inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3174964A (en) * 1959-12-10 1965-03-23 Pfizer & Co C Derivatives of 6-aminopenicillanic acid
US3043831A (en) * 1960-07-18 1962-07-10 Doyle Frank Peter Synthetic penicillins

Also Published As

Publication number Publication date
FR7155M (en) 1969-08-04
DK118021B (en) 1970-06-29
DE1770062B2 (en) 1978-11-30
IL29661A (en) 1972-01-27
CH491958A (en) 1970-06-15
DE1770062C3 (en) 1979-08-02
US3494917A (en) 1970-02-10
FR1525186A (en) 1968-05-17
DE1770062A1 (en) 1971-09-16
GB1209668A (en) 1970-10-21
GB1209669A (en) 1970-10-21
NL6804392A (en) 1968-09-30

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Legal Events

Date Code Title Description
VJC Lapsed due to non-payment of the due maintenance fee for the patent or patent application