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Application filed by Almirall Prodesfarma SafiledCriticalAlmirall Prodesfarma Sa
Priority to MYPI20013708priorityCriticalpatent/MY122986A/en
Publication of MY122986ApublicationCriticalpatent/MY122986A/en
THE INVENTION RELATES TO NEW THERAPEUTICALLY USEFUL 8-(DISUBSTITUTED) PHENYL-6,9-DIHYDRO-5H-PYRROLO[2,3-e][1,2,4]TRIAZOLO<4,3-c]PYRIMIDINE-5-ONE DERIVATIVES OF FORMULA (1): WHEREIN: -X-C-Y- REPRESENTS I OR I TO PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, TO PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND TO THEIR MEDICAL USES AS POTENT AND SELECTIVE INHIBITORS OF PHOSPHODIESTERASE 5 (PDE 5).
Novel imidazo [4,5 -b] pyridine derivatives as inhibitors of glycogen synthase kinase 3 for use in the treatment of dementia and neurodegenerative disorders
5,7-diaminopyrazolo[4,3-d]pyrimidines with pde-5 inhibitory activity, compositions containing such derivatives and the use of such derivatives in the treatment of hypertension and other disorders