Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries LtdfiledCriticalTakeda Chemical Industries Ltd
Priority to MYPI9603156priorityCriticalpatent/MY117985A/en
Publication of MY117985ApublicationCriticalpatent/MY117985A/en
A GONADOTROPIN-RELEASING HORMONE ANTAGONISTIC COMPOSITION, WHICH COMPRISES AN OPTIONALLY SUBSTITUTED CONDENSED-BICYCLIC COMPOUND CO.NSISTING OF A HOMO OR HETERO 5 TO 7 MEMBERED RING AND A HOMO OR HETERO 5 TO 7 MEMBERED RING IS EFFECTIVE AS A PROPYLACTIC OR THERAPEUTIC AGENT FOR THE PREVENTION OR TREATMENT OF SEVERAL HORMONE DEPENDENT DISEASES, FOR EXAMPLE, A SEX HORMONE DEPENDENT CANCER (E.G. PROSTATIC CANCER, CANCER OF UTERINE CERVIX, BREAST CANCER, PITUITARY ADENOMA), BENIGN PROSTATIC HYPERTROPHY, MYOMA OF THE UTERUS, ENDOMETRIOSIS, PRECOCIOUS PUBERTY, AMENORRHEA, PREMENSTRUAL SYNDROME, POLYCYSTIC OVARY SYNDROME AND ACNE VULGARIS; IS EFFECTIVE AS A FERTILITY CONTROLLING AGENT IN BOTH SEXES (E.G. A PREGNANCY CONTROLLING AGENT AND A MENSTRUAL CYCLE CONTROLLING AGENT); CAN BE USED AS A CONTRACEPTIVE OF MALE OR FEMALE, AS AN OVULATION-INDUCING AGENT OF FEMALE; CAN BE USED AS AN INFERTILITY TREATING AGENT BY USING A REBOUND EFFECT OWING TO A STOPPAGE OF ADMINISTRATION THEREOF; IS USEFUL AS MODULATING ESTROUS CYCLES IN ANIMALS IN THE FIELD OF ANIMAL HUSBANDRY, .AS AN AGENT FRO IMPROVING THE QUALITY OF EDIBLE MEAT OR PROMOTING THE GROWTH OF ANIMALS; IS USEFUL AS AN AGENT OF SPAWNING PROMOTION IN FISH.
MYPI96031561996-08-011996-08-01Condensed-ring thiophene derivatives, their production and use.
MY117985A
(en)