MY101854A - Improvements in and relating to pyrimido-(4,5-g) quinolines and intermediates - Google Patents

Improvements in and relating to pyrimido-(4,5-g) quinolines and intermediates

Info

Publication number
MY101854A
MY101854A MYPI87001872A MYPI19871872A MY101854A MY 101854 A MY101854 A MY 101854A MY PI87001872 A MYPI87001872 A MY PI87001872A MY PI19871872 A MYPI19871872 A MY PI19871872A MY 101854 A MY101854 A MY 101854A
Authority
MY
Malaysia
Prior art keywords
quinolines
trans
intermediates
pyrimido
relating
Prior art date
Application number
MYPI87001872A
Inventor
Carl Kornfeld Edmund
Mehnert Schaus John
Taiwai Wong David
Nolan Booher Richard
Lynn Nichols Cynthia
Mortensen Foreman Mark
Lynn Huser Diane
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/535,503 external-priority patent/US4501890A/en
Priority claimed from US06/535,474 external-priority patent/US4521421A/en
Priority claimed from US06/575,126 external-priority patent/US4528290A/en
Priority claimed from EP84305684A external-priority patent/EP0139393B1/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MY101854A publication Critical patent/MY101854A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

TRANS-(?)-2-AMINO (OR SUBSTITUTED AMINO)-4-(PERMISSIBLY-SUBSTITUTED) -6-C1-C3 ALKYL (OR ALLYL)-5, 5A, -6, 7, 8, 9, 9A, 10-OCTAHYDROPYRIMIDO [4, 5-G] QUINOLINES, THE CORRESPONDING TRANS-(-) AND TRANS-(?)-STEREOISOMERS AND SALTS THEREOF, USEFUL IN TREATING PARKINSON'S SYNDROME, SEXUAL DYSFUNCTION, DEPRESSION, HYPERTENSION, AND PROLACTIN RELATED DISEASES, AND INTERMEDIATES USEFUL FOR THE SYNTHESIS THEREOF, ARE DISCLOSED. THE PRODUCTS ARE PREPARED BY CONDENSING AN APPROPRIATE KETONE WITH THE APPROPRIATELY SUBSTITUTED GUANIDINE.
MYPI87001872A 1983-09-26 1987-09-22 Improvements in and relating to pyrimido-(4,5-g) quinolines and intermediates MY101854A (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US53551983A 1983-09-26 1983-09-26
US06/535,503 US4501890A (en) 1983-09-26 1983-09-26 Trans-(±)-2,4,6-substituted-5,5a,6,7,8,9,9a,10-octahydro-pyrimido[4,5-g]quinolines
US06/535,474 US4521421A (en) 1983-09-26 1983-09-26 Treatment of sexual dysfunction
US06/575,126 US4528290A (en) 1984-01-30 1984-01-30 Stimulating dopamine D-1 receptors
US60609184A 1984-05-02 1984-05-02
EP84305684A EP0139393B1 (en) 1983-09-26 1984-08-21 Pyrimido(4,5-g)quinolines, process for their preparation, and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
MY101854A true MY101854A (en) 1992-01-31

Family

ID=27545340

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI87001872A MY101854A (en) 1983-09-26 1987-09-22 Improvements in and relating to pyrimido-(4,5-g) quinolines and intermediates

Country Status (2)

Country Link
AT (1) ATE63552T1 (en)
MY (1) MY101854A (en)

Also Published As

Publication number Publication date
ATE63552T1 (en) 1991-06-15

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