MXPA05010521A - Inhibidores de cinasa de amida de bifenilcarboxilica p38. - Google Patents

Inhibidores de cinasa de amida de bifenilcarboxilica p38.

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Publication number
MXPA05010521A
MXPA05010521A MXPA05010521A MXPA05010521A MXPA05010521A MX PA05010521 A MXPA05010521 A MX PA05010521A MX PA05010521 A MXPA05010521 A MX PA05010521A MX PA05010521 A MXPA05010521 A MX PA05010521A MX PA05010521 A MXPA05010521 A MX PA05010521A
Authority
MX
Mexico
Prior art keywords
kinase inhibitors
carboxylic amide
biphenyl carboxylic
biphenyl
amide
Prior art date
Application number
MXPA05010521A
Other languages
English (en)
Spanish (es)
Inventor
Ann Louise Walker
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of MXPA05010521A publication Critical patent/MXPA05010521A/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
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    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Psychology (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Vascular Medicine (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
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MXPA05010521A 2003-04-09 2004-04-07 Inhibidores de cinasa de amida de bifenilcarboxilica p38. MXPA05010521A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0308186.6A GB0308186D0 (en) 2003-04-09 2003-04-09 Novel compounds
PCT/EP2004/003774 WO2004089874A1 (en) 2003-04-09 2004-04-07 Biphenyl carboxylic amide p38 kinase inhibitors

Publications (1)

Publication Number Publication Date
MXPA05010521A true MXPA05010521A (es) 2005-12-14

Family

ID=9956478

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05010521A MXPA05010521A (es) 2003-04-09 2004-04-07 Inhibidores de cinasa de amida de bifenilcarboxilica p38.

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US (1) US7572790B2 (US07652168-20100126-C00055.png)
EP (1) EP1608616A1 (US07652168-20100126-C00055.png)
JP (1) JP2006523194A (US07652168-20100126-C00055.png)
AU (1) AU2004228199A1 (US07652168-20100126-C00055.png)
BR (1) BRPI0408727A (US07652168-20100126-C00055.png)
CA (1) CA2521228A1 (US07652168-20100126-C00055.png)
GB (1) GB0308186D0 (US07652168-20100126-C00055.png)
MX (1) MXPA05010521A (US07652168-20100126-C00055.png)
WO (1) WO2004089874A1 (US07652168-20100126-C00055.png)
ZA (1) ZA200506919B (US07652168-20100126-C00055.png)

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TWI263497B (en) * 2002-03-29 2006-10-11 Lilly Co Eli Pyridinoylpiperidines as 5-HT1F agonists
GB0217757D0 (en) 2002-07-31 2002-09-11 Glaxo Group Ltd Novel compounds
GB0308201D0 (en) 2003-04-09 2003-05-14 Smithkline Beecham Corp Novel compounds
ES2315703T3 (es) * 2003-07-25 2009-04-01 Novartis Ag Inhibidores de la quinasa p-38.
GB0318814D0 (en) 2003-08-11 2003-09-10 Smithkline Beecham Corp Novel compounds
GB0402137D0 (en) * 2004-01-30 2004-03-03 Smithkline Beecham Corp Novel compounds
GB0402140D0 (en) * 2004-01-30 2004-03-03 Smithkline Beecham Corp Novel compounds
GB0402143D0 (en) * 2004-01-30 2004-03-03 Smithkline Beecham Corp Novel compounds
CA2574600C (en) * 2004-07-23 2010-08-31 Pfizer Inc. Pyridine derivatives
TW200628153A (en) * 2004-10-05 2006-08-16 Smithkline Beecham Corp Novel compounds
RU2452729C2 (ru) * 2005-09-16 2012-06-10 Арроу Терапьютикс Лимитед Бифенильные производные и их применение при лечении гепатита с
CA2621364A1 (en) * 2005-09-16 2007-03-22 Arrow Therapeutics Limited Biphenyl derivatives and their use in treating hepatitis c
EP2038253A1 (en) * 2006-05-30 2009-03-25 Arrow Therapeutics Limited Biphenyl derivatives and their use in treating hepatitis c
GB0612026D0 (en) 2006-06-16 2006-07-26 Smithkline Beecham Corp New use
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CA2521228A1 (en) 2004-10-21
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