MXPA03003233A - Formas de cristal de 1-[6-cloro -5-(trifluorometil) -2-piridinil) piperazina .hidrocloruro. - Google Patents
Formas de cristal de 1-[6-cloro -5-(trifluorometil) -2-piridinil) piperazina .hidrocloruro.Info
- Publication number
- MXPA03003233A MXPA03003233A MXPA03003233A MXPA03003233A MXPA03003233A MX PA03003233 A MXPA03003233 A MX PA03003233A MX PA03003233 A MXPA03003233 A MX PA03003233A MX PA03003233 A MXPA03003233 A MX PA03003233A MX PA03003233 A MXPA03003233 A MX PA03003233A
- Authority
- MX
- Mexico
- Prior art keywords
- pyridinyl
- piperazine
- trifluoromethyl
- hydrochloride
- chloro
- Prior art date
Links
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical compound Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 title 1
- 239000013078 crystal Substances 0.000 title 1
- QZYYPQAYSFBKPW-UHFFFAOYSA-N org 12962 Chemical compound N1=C(Cl)C(C(F)(F)F)=CC=C1N1CCNCC1 QZYYPQAYSFBKPW-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
- A61B17/00—Surgical instruments, devices or methods, e.g. tourniquets
- A61B17/34—Trocars; Puncturing needles
- A61B17/3403—Needle locating or guiding means
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
- A61B5/00—Measuring for diagnostic purposes; Identification of persons
- A61B5/48—Other medical applications
- A61B5/4887—Locating particular structures in or on the body
- A61B5/489—Blood vessels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
- A61B17/00—Surgical instruments, devices or methods, e.g. tourniquets
- A61B17/34—Trocars; Puncturing needles
- A61B17/3403—Needle locating or guiding means
- A61B2017/3405—Needle locating or guiding means using mechanical guide means
- A61B2017/3409—Needle locating or guiding means using mechanical guide means including needle or instrument drives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
- A61B17/00—Surgical instruments, devices or methods, e.g. tourniquets
- A61B17/34—Trocars; Puncturing needles
- A61B17/3403—Needle locating or guiding means
- A61B2017/3413—Needle locating or guiding means guided by ultrasound
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M5/00—Devices for bringing media into the body in a subcutaneous, intra-vascular or intramuscular way; Accessories therefor, e.g. filling or cleaning devices, arm-rests
- A61M5/44—Devices for bringing media into the body in a subcutaneous, intra-vascular or intramuscular way; Accessories therefor, e.g. filling or cleaning devices, arm-rests having means for cooling or heating the devices or media
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Surgery (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pathology (AREA)
- Heart & Thoracic Surgery (AREA)
- Molecular Biology (AREA)
- Medical Informatics (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Physics & Mathematics (AREA)
- Biophysics (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00203528 | 2000-10-13 | ||
| PCT/EP2001/011714 WO2002030902A1 (en) | 2000-10-13 | 2001-10-09 | Crystal forms of 1-[6-chloro-5-(trifluoromethyl)-2-pyridinyl]piperazine.hydrochloride |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03003233A true MXPA03003233A (es) | 2003-09-10 |
Family
ID=8172124
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03003233A MXPA03003233A (es) | 2000-10-13 | 2001-10-09 | Formas de cristal de 1-[6-cloro -5-(trifluorometil) -2-piridinil) piperazina .hidrocloruro. |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20040038985A1 (es) |
| EP (1) | EP1326837A1 (es) |
| JP (1) | JP2004512282A (es) |
| KR (1) | KR20030060906A (es) |
| CN (1) | CN1469863A (es) |
| AU (1) | AU2002220614A1 (es) |
| BR (1) | BR0114609A (es) |
| CA (1) | CA2425540A1 (es) |
| EC (1) | ECSP034549A (es) |
| HR (1) | HRP20030246A2 (es) |
| HU (1) | HUP0302842A2 (es) |
| IL (1) | IL154982A0 (es) |
| IS (1) | IS6758A (es) |
| MX (1) | MXPA03003233A (es) |
| NO (1) | NO20031698D0 (es) |
| PL (1) | PL366055A1 (es) |
| RU (1) | RU2003113536A (es) |
| SK (1) | SK4332003A3 (es) |
| WO (1) | WO2002030902A1 (es) |
| ZA (1) | ZA200302520B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008004945A1 (en) * | 2006-07-04 | 2008-01-10 | Astrazeneca Ab | Novel crystalline forms i and ii |
| WO2008004944A1 (en) * | 2006-07-04 | 2008-01-10 | Astrazeneca Ab | Novel crystalline form ii |
| CZ303950B6 (cs) * | 2011-12-12 | 2013-07-10 | Masarykova Univerzita | Zpusob prípravy 1-(pyridin-4-yl)piperazinu a jeho 1,1-dialkyl-1-ium derivátu |
| WO2015066344A1 (en) | 2013-11-01 | 2015-05-07 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists and compositions and methods of use |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2061953T3 (es) * | 1988-11-24 | 1994-12-16 | Akzo Nv | Un procedimiento para preparar una composicion farmaceutica. |
| WO1998033504A1 (en) * | 1997-02-03 | 1998-08-06 | Akzo Nobel N.V. | Treatment of urinary incontinence |
-
2001
- 2001-10-09 HU HU0302842A patent/HUP0302842A2/hu unknown
- 2001-10-09 WO PCT/EP2001/011714 patent/WO2002030902A1/en not_active Application Discontinuation
- 2001-10-09 IL IL15498201A patent/IL154982A0/xx unknown
- 2001-10-09 KR KR10-2003-7005122A patent/KR20030060906A/ko not_active Application Discontinuation
- 2001-10-09 MX MXPA03003233A patent/MXPA03003233A/es unknown
- 2001-10-09 CN CNA018172571A patent/CN1469863A/zh active Pending
- 2001-10-09 AU AU2002220614A patent/AU2002220614A1/en not_active Abandoned
- 2001-10-09 RU RU2003113536/04A patent/RU2003113536A/ru not_active Application Discontinuation
- 2001-10-09 CA CA002425540A patent/CA2425540A1/en not_active Abandoned
- 2001-10-09 SK SK433-2003A patent/SK4332003A3/sk unknown
- 2001-10-09 US US10/398,991 patent/US20040038985A1/en not_active Abandoned
- 2001-10-09 PL PL01366055A patent/PL366055A1/xx not_active Application Discontinuation
- 2001-10-09 EP EP01986679A patent/EP1326837A1/en not_active Withdrawn
- 2001-10-09 BR BR0114609-2A patent/BR0114609A/pt not_active Application Discontinuation
- 2001-10-09 JP JP2002534288A patent/JP2004512282A/ja not_active Withdrawn
-
2003
- 2003-03-27 IS IS6758A patent/IS6758A/is unknown
- 2003-03-31 ZA ZA200302520A patent/ZA200302520B/en unknown
- 2003-04-01 HR HR20030246A patent/HRP20030246A2/hr not_active Application Discontinuation
- 2003-04-08 EC EC2003004549A patent/ECSP034549A/es unknown
- 2003-04-11 NO NO20031698A patent/NO20031698D0/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IL154982A0 (en) | 2003-10-31 |
| CN1469863A (zh) | 2004-01-21 |
| SK4332003A3 (en) | 2003-10-07 |
| ZA200302520B (en) | 2004-06-30 |
| AU2002220614A1 (en) | 2002-04-22 |
| NO20031698D0 (no) | 2003-04-11 |
| CA2425540A1 (en) | 2002-04-18 |
| BR0114609A (pt) | 2003-12-23 |
| HUP0302842A2 (hu) | 2003-12-29 |
| WO2002030902A1 (en) | 2002-04-18 |
| JP2004512282A (ja) | 2004-04-22 |
| ECSP034549A (es) | 2003-05-26 |
| HRP20030246A2 (en) | 2003-06-30 |
| PL366055A1 (en) | 2005-01-24 |
| KR20030060906A (ko) | 2003-07-16 |
| US20040038985A1 (en) | 2004-02-26 |
| RU2003113536A (ru) | 2004-11-10 |
| EP1326837A1 (en) | 2003-07-16 |
| WO2002030902A8 (en) | 2004-02-26 |
| IS6758A (is) | 2003-03-27 |
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