MX9605426A - Derivados de acidos aminosulfonicos, utilizacion de los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion. - Google Patents

Derivados de acidos aminosulfonicos, utilizacion de los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion.

Info

Publication number
MX9605426A
MX9605426A MX9605426A MX9605426A MX9605426A MX 9605426 A MX9605426 A MX 9605426A MX 9605426 A MX9605426 A MX 9605426A MX 9605426 A MX9605426 A MX 9605426A MX 9605426 A MX9605426 A MX 9605426A
Authority
MX
Mexico
Prior art keywords
pseudopeptides
synthesis
derivatives
preparation
chains
Prior art date
Application number
MX9605426A
Other languages
English (en)
Other versions
MXPA96005426A (es
Inventor
Cesare Gennari
Donatella Potenza
Barbara Salom
Original Assignee
Pharmacia & Upjohn Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Spa filed Critical Pharmacia & Upjohn Spa
Publication of MX9605426A publication Critical patent/MX9605426A/es
Publication of MXPA96005426A publication Critical patent/MXPA96005426A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
    • C07C309/69—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a carbon skeleton substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
    • C07C311/47—Y being a hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

Derivados de ácidos sulfonicos gamma-amino-alfa,beta insaturados de la formula (I), donde: R se elige entre hidrogeno; fragmentos correspondientes a las cadenas laterales de aminoácidos naturales, sustituidos o sin sustituir; cadenas alquilo lineales, ramificadas o cíclicas; cadenas arilalquilo; grupos arilo o heteroaromáticos; Y indica hidrogeno, incluyendo las posibles formas salinas de la amina correspondiente; o cualquier grupo protector comunmente utilizado para la proteccion del grupo amina; X indica Cl, OH, OCH2CH3, OCH3, ONBu4, NHCH2Ph; proceso para la preparacion de los mismos y su utilizacion en la síntesis de seudopéptidos, caracterizados por la presencia de por lo menos un enlace de tipo sulfonamida conjugado a un doble enlace.
MXPA/A/1996/005426A 1994-05-17 1996-11-07 Derivados de acidos aminosulfonicos, utilizacionde los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion MXPA96005426A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
MIMI94A000989 1994-05-17
ITMI940989A IT1269511B (it) 1994-05-17 1994-05-17 Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione
PCT/EP1995/001788 WO1995031433A1 (en) 1994-05-17 1995-05-11 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation

Publications (2)

Publication Number Publication Date
MX9605426A true MX9605426A (es) 1998-05-31
MXPA96005426A MXPA96005426A (es) 1998-10-23

Family

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Also Published As

Publication number Publication date
AU2526895A (en) 1995-12-05
ITMI940989A0 (it) 1994-05-17
EP0759902A1 (en) 1997-03-05
WO1995031433A1 (en) 1995-11-23
DE69506540D1 (de) 1999-01-21
JP4023554B2 (ja) 2007-12-19
FI964582A0 (fi) 1996-11-15
CA2189896A1 (en) 1995-11-23
ATE174329T1 (de) 1998-12-15
US5869725A (en) 1999-02-09
NZ285763A (en) 1997-10-24
IT1269511B (it) 1997-04-01
AU691292B2 (en) 1998-05-14
ES2125617T3 (es) 1999-03-01
KR970703307A (ko) 1997-07-03
DE69506540T2 (de) 1999-06-02
ITMI940989A1 (it) 1995-11-17
NO964861L (no) 1997-01-16
NO964861D0 (no) 1996-11-15
HUT76483A (en) 1997-09-29
CN1148847A (zh) 1997-04-30
EP0759902B1 (en) 1998-12-09
FI964582A (fi) 1996-11-15
JPH10500123A (ja) 1998-01-06
HU9603128D0 (en) 1997-01-28
PL317258A1 (en) 1997-04-01

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal