MX9401080A - HETEROAROMATIC COMPOUNDS. - Google Patents
HETEROAROMATIC COMPOUNDS.Info
- Publication number
- MX9401080A MX9401080A MX9401080A MX9401080A MX9401080A MX 9401080 A MX9401080 A MX 9401080A MX 9401080 A MX9401080 A MX 9401080A MX 9401080 A MX9401080 A MX 9401080A MX 9401080 A MX9401080 A MX 9401080A
- Authority
- MX
- Mexico
- Prior art keywords
- heteroaromatic compounds
- piperazine
- therapy
- processes
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a un grupo de derivados de piperacina y piperidina, a procedimientos para su preparación, a composiciones farmacéuticas que los contienen, y a su uso en terapia, en particular, en el tratamiento de desórdenes psicóticos.The present invention relates to a group of piperazine and piperidine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their use in therapy, in particular, in the treatment of psychotic disorders.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB939302622A GB9302622D0 (en) | 1993-02-10 | 1993-02-10 | Heteroaromatic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
MX9401080A true MX9401080A (en) | 1994-08-31 |
Family
ID=10730183
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX9401080A MX9401080A (en) | 1993-02-10 | 1994-02-10 | HETEROAROMATIC COMPOUNDS. |
Country Status (15)
Country | Link |
---|---|
EP (1) | EP0683778A1 (en) |
JP (1) | JPH08506337A (en) |
CN (1) | CN1117731A (en) |
AU (1) | AU6005194A (en) |
BG (1) | BG99839A (en) |
CA (1) | CA2155758A1 (en) |
CZ (1) | CZ204495A3 (en) |
FI (1) | FI953777A (en) |
GB (1) | GB9302622D0 (en) |
HU (1) | HUT73654A (en) |
IL (1) | IL108601A0 (en) |
MX (1) | MX9401080A (en) |
SK (1) | SK99195A3 (en) |
WO (1) | WO1994018196A1 (en) |
ZA (1) | ZA94891B (en) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5776963A (en) * | 1989-05-19 | 1998-07-07 | Hoechst Marion Roussel, Inc. | 3-(heteroaryl)-1- (2,3-dihydro-1h-isoindol-2-yl)alkyl!pyrrolidines and 3-(heteroaryl)-1- (2,3-dihydro-1h-indol-1-yl)alkyl!pyrrolidines and related compounds and their therapeutic untility |
US5364866A (en) | 1989-05-19 | 1994-11-15 | Hoechst-Roussel Pharmaceuticals, Inc. | Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analetics |
GB9420521D0 (en) * | 1994-10-12 | 1994-11-30 | Smithkline Beecham Plc | Novel compounds |
JP3274579B2 (en) * | 1995-01-12 | 2002-04-15 | 住友製薬株式会社 | Agent for treating psychiatric symptoms associated with cerebrovascular disorders |
EP0732332B1 (en) * | 1995-03-17 | 2001-12-19 | Aventis Pharmaceuticals Inc. | Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation |
UA73981C2 (en) | 2000-03-10 | 2005-10-17 | Merck Patent Gmbh | (r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane for treatment of extrapyramidal movement disorders (variants), pharmaceutical composition and kit |
WO2002039988A2 (en) * | 2000-11-14 | 2002-05-23 | Merck Patent Gmbh | Novel uses of combined selective dopamine d2 receptor antagonists and 5-ht1a receptor agonists |
WO2002066469A2 (en) * | 2001-02-16 | 2002-08-29 | Aventis Pharmaceuticals Inc. | Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands |
ES2280602T3 (en) | 2001-07-26 | 2007-09-16 | Merck Patent Gmbh | USE OF 2- (5- (4-FLUOROPHENYL) -3-PIRIDYLMETHYLAMINOME) -CROMANO AND ITS PHYSIOLOGICALLY ACCEPTABLE SALTS. |
GB0222909D0 (en) | 2002-10-03 | 2002-11-13 | Astrazeneca Ab | Novel process and intermediates |
GB0222912D0 (en) | 2002-10-03 | 2002-11-13 | Astrazeneca Ab | Novel process and intermediates |
AU2005263592A1 (en) * | 2004-07-20 | 2006-01-26 | Siena Biotech S.P.A | Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof |
TW200901974A (en) | 2007-01-16 | 2009-01-16 | Wyeth Corp | Compounds, compositions, and methods of making and using them |
EP2736905A4 (en) * | 2011-07-28 | 2015-07-29 | Mapi Pharma Ltd | Intermediate compounds and process for the preparation of lurasidone and salts thereof |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0625181B2 (en) * | 1985-03-27 | 1994-04-06 | 住友製薬株式会社 | New imide derivative |
JP2660407B2 (en) * | 1986-09-26 | 1997-10-08 | 住友製薬株式会社 | New imide derivatives |
US5143923B1 (en) * | 1991-04-29 | 1993-11-02 | Hoechst-Roussel Pharmaceuticals Incorporated | Benzoisothiazole-and benzisoxazole-3-carboxamides |
AU645681B2 (en) * | 1991-05-02 | 1994-01-20 | John Wyeth & Brother Limited | Piperazine derivatives |
-
1993
- 1993-02-10 GB GB939302622A patent/GB9302622D0/en active Pending
-
1994
- 1994-02-09 ZA ZA94891A patent/ZA94891B/en unknown
- 1994-02-09 IL IL10860194A patent/IL108601A0/en unknown
- 1994-02-10 CZ CZ952044A patent/CZ204495A3/en unknown
- 1994-02-10 AU AU60051/94A patent/AU6005194A/en not_active Abandoned
- 1994-02-10 JP JP6517819A patent/JPH08506337A/en active Pending
- 1994-02-10 MX MX9401080A patent/MX9401080A/en unknown
- 1994-02-10 CN CN94191142A patent/CN1117731A/en active Pending
- 1994-02-10 HU HU9501881A patent/HUT73654A/en unknown
- 1994-02-10 CA CA002155758A patent/CA2155758A1/en not_active Abandoned
- 1994-02-10 EP EP94906290A patent/EP0683778A1/en not_active Withdrawn
- 1994-02-10 WO PCT/GB1994/000265 patent/WO1994018196A1/en not_active Application Discontinuation
- 1994-02-10 SK SK991-95A patent/SK99195A3/en unknown
-
1995
- 1995-08-02 BG BG99839A patent/BG99839A/en unknown
- 1995-08-09 FI FI953777A patent/FI953777A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
HUT73654A (en) | 1996-09-30 |
CA2155758A1 (en) | 1994-08-18 |
WO1994018196A1 (en) | 1994-08-18 |
CZ204495A3 (en) | 1996-03-13 |
EP0683778A1 (en) | 1995-11-29 |
SK99195A3 (en) | 1995-12-06 |
FI953777A0 (en) | 1995-08-09 |
HU9501881D0 (en) | 1995-08-28 |
JPH08506337A (en) | 1996-07-09 |
GB9302622D0 (en) | 1993-03-24 |
BG99839A (en) | 1996-02-28 |
IL108601A0 (en) | 1994-05-30 |
AU6005194A (en) | 1994-08-29 |
ZA94891B (en) | 1995-08-10 |
CN1117731A (en) | 1996-02-28 |
FI953777A (en) | 1995-08-09 |
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