MX2022013793A - Composicion de liberacion prolongada novedosa de 2-(2-aminotiazol-4-il)-n-[4-(2-{[(2r)-2-hidroxi2-feniletil]amino} etil)fenil]acetamida. - Google Patents

Composicion de liberacion prolongada novedosa de 2-(2-aminotiazol-4-il)-n-[4-(2-{[(2r)-2-hidroxi2-feniletil]amino} etil)fenil]acetamida.

Info

Publication number
MX2022013793A
MX2022013793A MX2022013793A MX2022013793A MX2022013793A MX 2022013793 A MX2022013793 A MX 2022013793A MX 2022013793 A MX2022013793 A MX 2022013793A MX 2022013793 A MX2022013793 A MX 2022013793A MX 2022013793 A MX2022013793 A MX 2022013793A
Authority
MX
Mexico
Prior art keywords
extended release
release composition
hydroxy2
aminothiazol
phenylethyl
Prior art date
Application number
MX2022013793A
Other languages
English (en)
Inventor
Anwar Daud
Chandrashekhar Mainde
Uttam Kedar
Kuldeep Gangawat
Original Assignee
Zim Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zim Laboratories Ltd filed Critical Zim Laboratories Ltd
Publication of MX2022013793A publication Critical patent/MX2022013793A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2813—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/288—Compounds of unknown constitution, e.g. material from plants or animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Zoology (AREA)
  • Botany (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

La presente invención se refiere a una composición de Mirabegron de liberación prolongada y al proceso de fabricación de la misma. La composición de liberación prolongada de Mirabegron que comprende un excipiente hidrofóbico no polimérico como agente de control de la liberación junto con uno o más excipientes farmacéuticamente aceptables se usa en el tratamiento de los síntomas asociados con la vejiga hiperactiva.
MX2022013793A 2020-05-17 2021-05-15 Composicion de liberacion prolongada novedosa de 2-(2-aminotiazol-4-il)-n-[4-(2-{[(2r)-2-hidroxi2-feniletil]amino} etil)fenil]acetamida. MX2022013793A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN202021020771 2020-05-17
PCT/IB2021/054184 WO2021234526A1 (en) 2020-05-17 2021-05-15 Novel extended release composition of 2-(2-aminothiazol-4-yl)-n-[4-(2-{[(2r)-2-hydroxy2-phenylethyl] amino} ethyl) phenyl] acetamide

Publications (1)

Publication Number Publication Date
MX2022013793A true MX2022013793A (es) 2023-02-22

Family

ID=78708181

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022013793A MX2022013793A (es) 2020-05-17 2021-05-15 Composicion de liberacion prolongada novedosa de 2-(2-aminotiazol-4-il)-n-[4-(2-{[(2r)-2-hidroxi2-feniletil]amino} etil)fenil]acetamida.

Country Status (6)

Country Link
US (1) US20230157962A1 (es)
EP (1) EP4153153A4 (es)
AU (1) AU2021274958A1 (es)
BR (1) BR112022022283A2 (es)
MX (1) MX2022013793A (es)
WO (1) WO2021234526A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114983956B (zh) * 2022-05-20 2025-06-10 海南普利制药股份有限公司 一种米拉贝隆缓释片及其制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5849946B2 (ja) * 2010-03-29 2016-02-03 アステラス製薬株式会社 放出制御医薬組成物
US20170128379A1 (en) * 2014-06-30 2017-05-11 Rubicon Research Private Limited Modified release pharmaceutical preparations
KR20180104259A (ko) * 2017-03-10 2018-09-20 (주)동구바이오제약 미라베그론을 포함하는 방출 제어 의약 조성물
KR20180106238A (ko) * 2017-03-17 2018-10-01 주식회사 네비팜 방출 제어 약학 조성물
EP3292864A1 (en) * 2017-10-12 2018-03-14 Synthon B.V. Modified release tablet composition comprising mirabegron
EP3694492A1 (en) * 2017-10-12 2020-08-19 Synthon B.V. Modified release tablet composition comprising mirabegron
KR20190089758A (ko) * 2018-01-22 2019-07-31 (주)동구바이오제약 미라베그론 또는 이의 약제학적으로 허용가능한 염을 함유하는 지속 방출 제제
KR102067261B1 (ko) * 2018-03-13 2020-01-16 충북대학교 산학협력단 미라베그론을 유효 성분으로 포함하는 서방형의 약학 조성물 및 이의 제조방법

Also Published As

Publication number Publication date
AU2021274958A1 (en) 2023-01-05
EP4153153A4 (en) 2024-07-03
WO2021234526A1 (en) 2021-11-25
US20230157962A1 (en) 2023-05-25
EP4153153A1 (en) 2023-03-29
BR112022022283A2 (pt) 2022-12-20

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