MX2016005092A - Composiciones farmaceuticas de estradiol insertadas en la vagina y metodos. - Google Patents

Composiciones farmaceuticas de estradiol insertadas en la vagina y metodos.

Info

Publication number
MX2016005092A
MX2016005092A MX2016005092A MX2016005092A MX2016005092A MX 2016005092 A MX2016005092 A MX 2016005092A MX 2016005092 A MX2016005092 A MX 2016005092A MX 2016005092 A MX2016005092 A MX 2016005092A MX 2016005092 A MX2016005092 A MX 2016005092A
Authority
MX
Mexico
Prior art keywords
methods
pharmaceutical compositons
vaginal
estradiol pharmaceutical
vaginal inserted
Prior art date
Application number
MX2016005092A
Other languages
English (en)
Inventor
A Bernick Brian
Louise Cacace Janice
M Amadio Julia
H R Persicaner Peter
Thorsteinsson Thorsteinn
D Sanscilio Frederick
Irani Neda
Original Assignee
Therapeuticsmd Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US14/099,562 external-priority patent/US8987237B2/en
Application filed by Therapeuticsmd Inc filed Critical Therapeuticsmd Inc
Publication of MX2016005092A publication Critical patent/MX2016005092A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4875Compounds of unknown constitution, e.g. material from plants or animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Botany (AREA)
  • Zoology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

De conformidad con varias modalidades de la presente descripción, se proporcionan composiciones farmacéuticas que comprenden estradiol solubilizado. En varias modalidades, dichas composiciones se encapsulan en cápsulas blandas que pueden insertarse en la vagina para el tratamiento de la atrofia vulvovaginal.
MX2016005092A 2013-10-10 2014-10-22 Composiciones farmaceuticas de estradiol insertadas en la vagina y metodos. MX2016005092A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361889483P 2013-10-10 2013-10-10
US201361894411P 2013-10-22 2013-10-22
US14/099,562 US8987237B2 (en) 2011-11-23 2013-12-06 Natural combination hormone replacement formulations and therapies
US201461932140P 2014-01-27 2014-01-27
PCT/US2014/061811 WO2015073177A1 (en) 2013-10-10 2014-10-22 Vaginal inserted estradiol pharmaceutical compositons and methods

Publications (1)

Publication Number Publication Date
MX2016005092A true MX2016005092A (es) 2016-08-17

Family

ID=53140634

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016005092A MX2016005092A (es) 2013-10-10 2014-10-22 Composiciones farmaceuticas de estradiol insertadas en la vagina y metodos.

Country Status (3)

Country Link
CA (1) CA2926342A1 (es)
MX (1) MX2016005092A (es)
WO (1) WO2015073177A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
EP3936133A1 (en) 2011-11-23 2022-01-12 TherapeuticsMD, Inc. Natural combination hormone replacement formulations and therapies
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
AU2020397648B2 (en) 2019-12-06 2022-03-24 Prathima Chowdary Sustained release estrogen vaginal ring pessary for treatment of atrophy, cystitis and uterovaginal prolapse

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU1300799A (en) * 1997-11-03 1999-05-24 Deschutes Medical Products, Inc. Pessary with medicated cartridge
MX367596B (es) * 2012-01-26 2019-08-27 Therapeuticsmd Inc Tratamientos transdermicos de sustitucion hormonal.
US20130224268A1 (en) * 2012-02-27 2013-08-29 Newgen Biopharma Corp. Topical delivery of hormonal and non hormonal nano formulations, methods of making and using the same

Also Published As

Publication number Publication date
WO2015073177A8 (en) 2016-07-07
CA2926342A1 (en) 2015-05-21
WO2015073177A1 (en) 2015-05-21

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