MX2014007398A - 2, 4-diamine-pyrimidine derivative as serine/threonine kinase inhibitors. - Google Patents
2, 4-diamine-pyrimidine derivative as serine/threonine kinase inhibitors.Info
- Publication number
- MX2014007398A MX2014007398A MX2014007398A MX2014007398A MX2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A
- Authority
- MX
- Mexico
- Prior art keywords
- serine
- diamine
- kinase inhibitors
- threonine kinase
- pyrimidine derivative
- Prior art date
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Compounds having the formula I wherein A, R1a, R1b, R2, R3, R4, R5, R6, R7, R8, Ra, Rb, X1, X2, X3 and n are as defined herein are inhibitors of PAK1. Also disclosed are compositions and methods for treating cancer and hyperproliferative disorders.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP61579227 | 2011-12-22 | ||
PCT/EP2012/076531 WO2013092940A1 (en) | 2011-12-22 | 2012-12-21 | 2, 4-diamine-pyrimidine derivative as serine/threonine kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2014007398A true MX2014007398A (en) | 2014-08-08 |
Family
ID=52130938
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2014007398A MX2014007398A (en) | 2011-12-22 | 2012-12-21 | 2, 4-diamine-pyrimidine derivative as serine/threonine kinase inhibitors. |
Country Status (1)
Country | Link |
---|---|
MX (1) | MX2014007398A (en) |
-
2012
- 2012-12-21 MX MX2014007398A patent/MX2014007398A/en unknown
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