MD675Z - Method for prevention of pathological reflexes during surgical manipulations - Google Patents

Method for prevention of pathological reflexes during surgical manipulations Download PDF

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Publication number
MD675Z
MD675Z MDS20130051A MDS20130051A MD675Z MD 675 Z MD675 Z MD 675Z MD S20130051 A MDS20130051 A MD S20130051A MD S20130051 A MDS20130051 A MD S20130051A MD 675 Z MD675 Z MD 675Z
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Moldova
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prevention
dose
pathological
manipulations
during surgical
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MDS20130051A
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Romanian (ro)
Russian (ru)
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Виктор ГИКАВЫЙ
Янош КОРЕЦКИЙ
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Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова
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Priority to MDS20130051A priority Critical patent/MD675Z/en
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Abstract

The invention relates to medicine, namely to clinical pharmacology, anesthesiology and resuscitation, and may be used to prevent pathological reflexogenic disorders during surgical operations and other traumatic interventions.Summary of the invention consists in that at the stage of carrying out the surgical operations and other traumatic manipulations additionally to the appropriate anesthesia is intravenously administered azamethonium bromide in a dose of 3 mg/kg, then profetur in a dose of 5 mg/kg.

Description

Invenţia se referă la medicină, şi anume la farmacologia clinică, anesteziologie şi reanimare, şi poate fi utilizată pentru prevenirea dereglărilor patologice reflexogene în cadrul intervenţiilor chirurgicale şi a altor manipulări traumatizante. The invention relates to medicine, namely to clinical pharmacology, anesthesiology and resuscitation, and can be used to prevent pathological reflexogenic disorders during surgical interventions and other traumatic manipulations.

În diverse stări patologice (traume, arsuri) şi intervenţii chirurgicale masive, la executarea anumitor tehnici şi manipulări pe parcursul intervenţiilor chirurgicale, în special în regiunile reflexogene, pe fondalul anesteziilor (generale, regionale) se poate produce activarea locală patologică a sistemului nervos vegetativ şi somatic. Metodele de limitare a posibilităţilor de dezvoltare a reflexelor patologice şi, respectiv, de protejare a sistemului cardiovascular cu dirijare hemodinamică rămân a fi actuale. In various pathological conditions (trauma, burns) and massive surgical interventions, when performing certain techniques and manipulations during surgical interventions, especially in reflexogenic regions, against the background of anesthesia (general, regional), pathological local activation of the vegetative and somatic nervous system may occur. Methods of limiting the possibilities of developing pathological reflexes and, respectively, protecting the cardiovascular system with hemodynamic guidance remain relevant.

Este cunoscută metoda blocării ganglionare fără hipotensiune, care permite prevenirea dezvoltării reflexelor patologice cardiovasculare prin utilizarea ganglioblocantelor cu corijarea modificărilor nedorite şi stabilizarea parametrilor hemodinamici cu adrenomimetice (norepinefrină) [1]. The method of ganglionic blockade without hypotension is known, which allows preventing the development of pathological cardiovascular reflexes by using ganglionic blockers with correction of unwanted changes and stabilization of hemodynamic parameters with adrenomimetics (norepinephrine) [1].

De asemenea, este cunoscută metoda blocării ganglionare fără hipotensiune, care permite prevenirea dezvoltării reflexelor patologice cardiovasculare prin administrarea asociată a ganglioblocantelor cu etiron [2]. The method of ganglionic blockade without hypotension is also known, which allows the prevention of the development of pathological cardiovascular reflexes by the combined administration of ganglionic blockers with etirone [2].

Dezavantajele acestor metode constau în durata mică de acţiune a adrenomimeticelor şi necesitatea administrării intravenoase continue în perfuzie cu dereglări vădite ale microcirculaţiei, iar în cazul utilizării pentru premedicaţie şi a medicamentelor cu acţiune alfa-adrenoblocantă, acestea pot fi ineficace sau să manifeste o acţiune inversă. The disadvantages of these methods are the short duration of action of adrenomimetics and the need for continuous intravenous administration in infusion with obvious microcirculation disorders, and in the case of premedication and the use of drugs with alpha-adrenoblocking action, they may be ineffective or have the opposite effect.

De asemenea, medicamentele adrenergice pot provoca dereglări metabolice (hiperglicemie, hiperlactacidemie, acidoză metabolică, majorarea consumului de oxigen de către organism), aritmii etc. Also, adrenergic drugs can cause metabolic disorders (hyperglycemia, hyperlactacidemia, metabolic acidosis, increased oxygen consumption by the body), arrhythmias, etc.

Problema pe care o rezolvă invenţia constă în elaborarea unei metode de prevenire a dereglărilor hemodinamice şi metabolice, precum şi de protejare a sistemului cardiovascular faţă de reflexele patologice prin suplimentarea anesteziei generale cu profetur şi azametoniu pentru intervenţiile chirurgicale şi/sau alte manipulări traumatizante în zonele reflexogene. The problem solved by the invention consists in developing a method for preventing hemodynamic and metabolic disorders, as well as protecting the cardiovascular system from pathological reflexes by supplementing general anesthesia with prophethurium and azamethonium for surgical interventions and/or other traumatic manipulations in reflexogenic areas.

Esenţa metodei constă în aceea că la etapa efectuării intervenţiilor chirurgicale sau a altor manipulări traumatizante la anestezia respectivă suplimentar se administrează intravenos bromură de azametoniu în doză de 3 mg/kg, apoi profetur în doză de 5 mg/kg. The essence of the method is that at the stage of performing surgical interventions or other traumatic manipulations, azamethonium bromide is additionally administered intravenously in a dose of 3 mg/kg, then profetur in a dose of 5 mg/kg.

Rezultatul constă în obţinerea blocării ganglionare cu prevenirea dezvoltării reflexelor patologice ca rezultat al denervării farmacologice şi perturbărilor hemodinamice şi metabolice, care se pot dezvolta pe parcursul anesteziei în intervenţiile chirurgicale şi manipulările traumatizante datorită stabilizării medicamentoase a nivelului tensiunii arteriale sistemice, ceea ce în final micşorează frecvenţa apariţiei complicaţiilor nedorite şi, respectiv, reduce costul tratamentului efectuat. The result is to achieve ganglionic blockade with the prevention of the development of pathological reflexes as a result of pharmacological denervation and hemodynamic and metabolic disturbances, which can develop during anesthesia in surgical interventions and traumatic manipulations due to drug stabilization of the level of systemic blood pressure, which ultimately reduces the frequency of unwanted complications and, respectively, reduces the cost of the treatment performed.

Avantajele metodei constau în aceea că la administrarea unimomentană a profeturului pe fondalul acţiunii azametoniului se obţine restabilirea îndelungată (mai mult de o oră) a valorilor tensiunii arteriale cu păstrarea concomitentă a acţiunii ganglioblocante specifice a azametoniului, care se manifestă prin lipsa modificărilor parametrilor respectivi la excitarea sistemului nervos vegetativ şi somatic. Spre deosebire de adrenomimetice, profeturul nu provoacă hiperglicemie şi acidoză, micşorează consumul de oxigen de către organism, posedă o durată de acţiune mai lungă, care se manifestă prin stabilizarea îndelungată a valorilor tensiunii arteriale, este mai inofensiv şi nu necesită administrarea îndelungată în perfuzie (are durată lungă de acţiune la administrarea unimomentană i/m şi i/v). The advantages of the method are that with a single administration of profetur against the background of the action of azamethonium, a long-term (more than an hour) restoration of blood pressure values is achieved with the simultaneous preservation of the specific ganglioblocking action of azamethonium, which is manifested by the lack of changes in the respective parameters upon excitation of the vegetative and somatic nervous systems. Unlike adrenomimetics, profetur does not cause hyperglycemia and acidosis, reduces oxygen consumption by the body, has a longer duration of action, which is manifested by the long-term stabilization of blood pressure values, is more harmless and does not require long-term administration in infusion (it has a long duration of action with a single i/m and i/v administration).

Metoda propusă se efectuează în felul următor: la etapa efectuării intervenţiilor chirurgicale sau a altor manipulări traumatizante la anestezia respectivă suplimentar se administrează intravenos bromură de azametoniu în doză de 3 mg/kg, apoi profetur în doză de 5 mg/kg. The proposed method is carried out as follows: at the stage of performing surgical interventions or other traumatic manipulations, azamethonium bromide is additionally administered intravenously to the respective anesthesia in a dose of 3 mg/kg, then profetur in a dose of 5 mg/kg.

Exemplu de realizare a invenţiei Example of embodiment of the invention

Acţiunea de prevenire a dereglărilor hemodinamice şi de protejare a sistemului cardiovascular faţă de reflexele patologice la utilizarea combinată a profeturului şi azametoniului a fost cercetată experimental la pisici anesteziate cu uretan (1...1,2 g/kg intraperitoneal). S-au determinat valorile iniţiale ale tensiunii arteriale, apoi cele obţinute la electrostimularea nervilor (segmentul central al nervului ischiatic şi segmentul periferic al nervului vag). Ulterior s-a administrat intravenos azametoniu (3 mg/kg) şi profetur (5 mg/kg) şi, din nou, s-au determinat valorile tensiunii arteriale până şi după excitarea nervilor respectivi. The action of preventing hemodynamic disorders and protecting the cardiovascular system from pathological reflexes with the combined use of profetur and azamethonium was experimentally investigated in cats anesthetized with urethane (1...1.2 g/kg intraperitoneally). Initial blood pressure values were determined, then those obtained during nerve electrostimulation (central segment of the sciatic nerve and peripheral segment of the vagus nerve). Subsequently, azamethonium (3 mg/kg) and profetur (5 mg/kg) were administered intravenously and, again, blood pressure values were determined until and after the excitation of the respective nerves.

Electrostimularea iniţială a nervilor a determinat modificarea corespunzătoare a valorilor tensiunii arteriale. Administrarea combinată a profeturului şi azametoniului a dus la stabilizarea indicilor hemodinamici şi la lipsa răspunsului reflector după electrostimularea nervilor. Initial nerve stimulation resulted in corresponding changes in blood pressure values. Combined administration of profetur and azamethonium led to stabilization of hemodynamic indices and lack of reflex response after nerve stimulation.

Comparativ cu utilizarea catecolaminelor în condiţii similare, profeturul nu necesită administrarea continuă în perfuzie, nu determină dereglări ale metabolismului (hiperglicemie, hiperlactacidemie, acidoză metabolică, tahiaritmii, majorarea consumului de oxigen de către organism). Compared to the use of catecholamines in similar conditions, profetur does not require continuous infusion administration, does not cause metabolic disorders (hyperglycemia, hyperlactacidemia, metabolic acidosis, tachyarrhythmias, increased oxygen consumption by the body).

1. Виноградов В.М. Новые пути лекарственной профилактики и терапии травматического и кардиогенного шока. Автрореф. диссертации. Ленинград, 1965 1. Vinogradov V.M. New ways of medicinal prevention and therapy of traumatic and cardiogenic shock. Autoref. dissertations. Leningrad, 1965

2. Гикавый В.И. Применение этирона при ганглионарном блоке без гипотонии в эксперименте. Здравохранение.Кишинёв, 1970, I, с. 47-50 2. Гикавый В.И. The use of ethirone in ganglionar block without hypotonia in an experiment. Здравохранение. Кишинёв, 1970, I, с. 47-50

Claims (1)

Metodă de prevenire a reflexelor patologice în manipulările operatorii care constă în aceea că la etapa efectuării intervenţiilor chirurgicale sau a altor manipulări traumatizante la anestezia respectivă suplimentar se administrează intravenos bromură de azametoniu în doză de 3 mg/kg, apoi profetur în doză de 5 mg/kg.Method of preventing pathological reflexes in surgical manipulations which consists in that at the stage of performing surgical interventions or other traumatic manipulations, azamethonium bromide is additionally administered intravenously in a dose of 3 mg/kg, then profetur in a dose of 5 mg/kg.
MDS20130051A 2013-03-15 2013-03-15 Method for prevention of pathological reflexes during surgical manipulations MD675Z (en)

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Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MD263C2 (en) * 1995-03-01 1995-12-31 Виктор ГИКАВЫЙ "Isoturon" means with antihypotensive activity
MD586C2 (en) * 1995-05-25 1997-03-31 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Remedy antihypotensif "Difetur"
MD1123F1 (en) * 1997-03-25 1998-12-31 Firma Svetskii & Co Drum mixer of reversible rotation
MD1138C2 (en) * 1997-02-17 1999-07-31 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Isopropylphosphite-S-isopropylisothiuronium - isothiourea derivative - possessing the hypertensive activity
MD1431G2 (en) * 1998-01-16 2001-02-28 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Antihypotensive remedies
RU2200552C1 (en) * 2001-07-18 2003-03-20 ГУ Научно-исследовательский институт экспериментальной медицины РАМН Method for protecting cardiovascular system during operation dealing with myocardial revascularization upon working heart
MD2066G2 (en) * 2002-07-10 2003-09-30 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Antihypertensive remedy
MD2228G2 (en) * 2003-01-21 2004-02-29 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова use of isothiouronic derivatives in the treatment and prophylaxis of intestinal atony
  • 2013

Patent Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MD263C2 (en) * 1995-03-01 1995-12-31 Виктор ГИКАВЫЙ "Isoturon" means with antihypotensive activity
MD586C2 (en) * 1995-05-25 1997-03-31 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Remedy antihypotensif "Difetur"
MD1138C2 (en) * 1997-02-17 1999-07-31 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Isopropylphosphite-S-isopropylisothiuronium - isothiourea derivative - possessing the hypertensive activity
MD1123F1 (en) * 1997-03-25 1998-12-31 Firma Svetskii & Co Drum mixer of reversible rotation
MD1431G2 (en) * 1998-01-16 2001-02-28 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Antihypotensive remedies
RU2200552C1 (en) * 2001-07-18 2003-03-20 ГУ Научно-исследовательский институт экспериментальной медицины РАМН Method for protecting cardiovascular system during operation dealing with myocardial revascularization upon working heart
MD2066G2 (en) * 2002-07-10 2003-09-30 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова Antihypertensive remedy
MD2228G2 (en) * 2003-01-21 2004-02-29 Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова use of isothiouronic derivatives in the treatment and prophylaxis of intestinal atony

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Виноградов В.М. Новые пути лекарственной профилактики и терапии травматического и кардиогенного шока. Автрореф. диссертации. Ленинград, 1965 *
Гикавый В.И. Применение этирона при ганглионарном блоке без гипотонии в эксперименте. Здравохранение.Кишинёв, 1970, I, с. 47-50 *

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