MD117C2 - Replaced acyloaminobenzamides with fungicide activity and the method of their obtaining - Google Patents

Abstract

The invention relates to some new replaced acyloaminobenzamides with funghicidal activity and to the method of their obtaining and may be used in controlling agriculture administration, especially for the controlling of fungeous infections of plants.The substitution acyloaminobenxamides are of general formula:wherein: A and B represent independently H, fluorin, chlor, bromine, C14-alkyl, C14-aleoxy- or halo-(C1-4), alkyl provided that they together simultaneosly are not H;D and E independently represent H or fluorine;R1 represents H or C1-4-alkyl; R2 represents C1-4 alkyl, C1-4-aleoxy - or phenyl, or R1 and R2 together with nitrogen atom, which are coupled, form the morpholine, piperidine, pyrrolidine or axetidine cycle, perhaps substituted by C1-4-alkyl, R3 represents H; R4 represents trichlormetyl, C2-8-alkyl, (substituted by Halogen, C1-8-aleoxyl or R12S group (O)n, where R12 is C1-4-alkyl, n has the meaning of 0,1 or 2 cyclopropyl (substituted by halogen or C1-4-alkyl), C2-8-alkenyl, C2-alkinil, C1-8 alcoxygroup, mono- or di-(C1-4)- alkylamingroup or group of formula R13ON=C(CN), where R13 represents C1-4-alkyl or R3 and R4 together with C(O)N group which are coupled form azetidine cycle-2-onic,The substation acyloaminobenzamides are obtained by the interaction of compounds with general formula:where A,B,D,E have the above indicated meanings with a chloranhidrid with formula R4 COCL, where R4 had the above indicated meaning with the subsequent elimination of product with special destination.