MC1332A1 - NEW QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS - Google Patents

NEW QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS

Info

Publication number
MC1332A1
MC1332A1 MC801454A MC1454A MC1332A1 MC 1332 A1 MC1332 A1 MC 1332A1 MC 801454 A MC801454 A MC 801454A MC 1454 A MC1454 A MC 1454A MC 1332 A1 MC1332 A1 MC 1332A1
Authority
MC
Monaco
Prior art keywords
pharmaceutical preparations
quinazoline derivatives
new quinazoline
new
derivatives
Prior art date
Application number
MC801454A
Other languages
French (fr)
Inventor
A Kaiser
M Chodnekar
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/050,395 external-priority patent/US4256748A/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1332A1 publication Critical patent/MC1332A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
MC801454A 1979-06-20 1980-06-18 NEW QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS MC1332A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/050,395 US4256748A (en) 1977-07-25 1979-06-20 Imidazo[2,1-b]quinazolin-2(3H)-ones and pharmaceutical compositions for treatment and prophylaxis of cardiac insufficiency and cardiac failure
CH360080 1980-05-08

Publications (1)

Publication Number Publication Date
MC1332A1 true MC1332A1 (en) 1981-04-21

Family

ID=25693404

Family Applications (1)

Application Number Title Priority Date Filing Date
MC801454A MC1332A1 (en) 1979-06-20 1980-06-18 NEW QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS

Country Status (14)

Country Link
EP (1) EP0021338B1 (en)
AU (1) AU538119B2 (en)
CA (1) CA1131631A (en)
DE (1) DE3065273D1 (en)
DK (1) DK259380A (en)
ES (3) ES8105321A1 (en)
FI (1) FI66870C (en)
IL (1) IL60325A (en)
MC (1) MC1332A1 (en)
NO (1) NO801843L (en)
NZ (1) NZ194046A (en)
PH (1) PH16369A (en)
PT (1) PT71411B (en)
YU (1) YU161580A (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0054180A3 (en) * 1980-12-16 1982-12-01 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Process for the preparation of imidazoquinazoline derivatives
US4783467A (en) * 1985-06-05 1988-11-08 Pfizer Inc. Tetrahydroimidazoquinazolinone inotropic agents
US6388073B1 (en) * 2000-07-26 2002-05-14 Shire Us Inc. Method for the manufacture of anagrelide
US7700608B2 (en) 2004-08-04 2010-04-20 Shire Holdings Ag Quinazoline derivatives and their use in the treatment of thrombocythemia
US8436006B2 (en) 2004-08-06 2013-05-07 Jansssen Pharmaceutica N.V. 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE)
US8383637B2 (en) 2004-08-06 2013-02-26 Jansssen Pharmaceutica N.V. 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE)
US8426429B2 (en) 2004-08-06 2013-04-23 Jansssen Pharmaceutica N.V. 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE)
US7910597B2 (en) 2006-11-28 2011-03-22 Shire Llc Substituted quinazolines
GB0623750D0 (en) * 2006-11-28 2007-01-10 Shire Llc Substituted quinazolines
US8304420B2 (en) 2006-11-28 2012-11-06 Shire Llc Substituted quinazolines for reducing platelet count

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE794964A (en) * 1972-02-04 1973-08-02 Bristol Myers Co NEW HYPOTENSING AGENTS AND METHOD FOR PREPARING THEM
US3932407A (en) * 1973-11-19 1976-01-13 Bristol-Myers Company Optionally substituted 1,2,3,5-tetrahydroimidezo(2,1-b)-quinazolin-2-ones and 6(H)-1,2,3,4-tetrahydropyimido(2,1-b)quinazolin-2-ones
US3988340A (en) * 1975-01-23 1976-10-26 Bristol-Myers Company 6-Alkoxymethyl-1,2,3,5-tetrahydroimidazo[2,1-b]quinazolin-2-ones and 7-alkoxymethyl-6-[H]-1,2,3,4-tetrahydropyrimido[2,1-b]quinazolin-2-ones
NL7807507A (en) * 1977-07-25 1979-01-29 Hoffmann La Roche TRICYCLICAL CONNECTIONS.
US4146718A (en) * 1978-04-10 1979-03-27 Bristol-Myers Company Alkyl 5,6-dichloro-3,4-dihydro-2(1h)-iminoquinazoline-3-acetate hydrohalides

Also Published As

Publication number Publication date
IL60325A0 (en) 1980-09-16
AU538119B2 (en) 1984-08-02
AU5933980A (en) 1981-01-08
ES499455A0 (en) 1982-08-16
FI66870C (en) 1984-12-10
ES492573A0 (en) 1981-06-01
DK259380A (en) 1980-12-21
DE3065273D1 (en) 1983-11-17
ES499454A0 (en) 1981-12-01
ES8206524A1 (en) 1982-08-16
ES8201164A1 (en) 1981-12-01
YU161580A (en) 1983-04-30
FI801910A (en) 1980-12-21
PT71411B (en) 1981-12-11
PH16369A (en) 1983-09-14
FI66870B (en) 1984-08-31
CA1131631A (en) 1982-09-14
EP0021338A1 (en) 1981-01-07
EP0021338B1 (en) 1983-10-12
ES8105321A1 (en) 1981-06-01
NZ194046A (en) 1982-05-25
IL60325A (en) 1983-06-15
NO801843L (en) 1980-12-22
PT71411A (en) 1980-07-01

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