MA38838B1 - Piperidinylindole derivatives and their use as complement factor b inhibitors - Google Patents

Piperidinylindole derivatives and their use as complement factor b inhibitors

Info

Publication number
MA38838B1
MA38838B1 MA38838A MA38838A MA38838B1 MA 38838 B1 MA38838 B1 MA 38838B1 MA 38838 A MA38838 A MA 38838A MA 38838 A MA38838 A MA 38838A MA 38838 B1 MA38838 B1 MA 38838B1
Authority
MA
Morocco
Prior art keywords
inhibitors
piperidinylindole
derivatives
complement factor
factor
Prior art date
Application number
MA38838A
Other languages
French (fr)
Other versions
MA38838A1 (en
Inventor
Takeru Ehara
Rajeshri Ganesh Karki
Chun Zhang
Christopher Adams
Michael Paul Capparelli
Nello Mainolfi
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Priority claimed from PCT/US2014/046515 external-priority patent/WO2015009616A1/en
Publication of MA38838A1 publication Critical patent/MA38838A1/en
Publication of MA38838B1 publication Critical patent/MA38838B1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Cette invention concerne un composé de formule i : (i), un procédé de production des composés selon l'invention, et leurs utilisations thérapeutiques en tant qu'inhibiteurs de la voie alternative du complément, en particulier, du facteur b. Une combinaison d'agents pharmaceutiquement actifs et une composition pharmaceutique sont en outre décrites.This invention relates to a compound of formula I: (i), a process for producing the compounds of the invention, and their therapeutic uses as inhibitors of the alternative complement pathway, in particular, factor b. A combination of pharmaceutically active agents and a pharmaceutical composition are further described.

MA38838A 2013-07-15 2014-07-14 Piperidinylindole derivatives and their use as complement factor b inhibitors MA38838B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361846355P 2013-07-15 2013-07-15
PCT/US2014/046515 WO2015009616A1 (en) 2013-07-15 2014-07-14 Piperidinyl indole derivatives and their use as complement factor b inhibitors

Publications (2)

Publication Number Publication Date
MA38838A1 MA38838A1 (en) 2017-03-31
MA38838B1 true MA38838B1 (en) 2017-11-30

Family

ID=56125325

Family Applications (1)

Application Number Title Priority Date Filing Date
MA38838A MA38838B1 (en) 2013-07-15 2014-07-14 Piperidinylindole derivatives and their use as complement factor b inhibitors

Country Status (2)

Country Link
AR (1) AR096904A1 (en)
MA (1) MA38838B1 (en)

Also Published As

Publication number Publication date
MA38838A1 (en) 2017-03-31
AR096904A1 (en) 2016-02-03

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