MA30013B1 - PIRAZOLE-ISOQUINOLEINE UREA DERIVATIVES AS INHIBITORS OF KINASE P38 - Google Patents

PIRAZOLE-ISOQUINOLEINE UREA DERIVATIVES AS INHIBITORS OF KINASE P38

Info

Publication number
MA30013B1
MA30013B1 MA30968A MA30968A MA30013B1 MA 30013 B1 MA30013 B1 MA 30013B1 MA 30968 A MA30968 A MA 30968A MA 30968 A MA30968 A MA 30968A MA 30013 B1 MA30013 B1 MA 30013B1
Authority
MA
Morocco
Prior art keywords
inhibitors
kinase
isoquinoleine
pirazole
urea derivatives
Prior art date
Application number
MA30968A
Other languages
French (fr)
Inventor
Dios Alfonso De
Cristina Garcia-Paredes
De Uralde Garmendia Beatriz Lopez
Mary Margaret Mader
Mark Andrew Pobanz
Chuan Shih
Boyu Zhong
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MA30013B1 publication Critical patent/MA30013B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des inhibiteurs de kinase représentés par la formule (I) ou un sel pharmaceutiquement acceptable de ces inhibiteurs. Dans la formule (I), R1, R2 et X sont tels que décrits dans le descriptif.The invention relates to kinase inhibitors represented by the formula (I) or a pharmaceutically acceptable salt of these inhibitors. In formula (I), R1, R2 and X are as described in the specification.

MA30968A 2005-10-28 2008-05-27 PIRAZOLE-ISOQUINOLEINE UREA DERIVATIVES AS INHIBITORS OF KINASE P38 MA30013B1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP05380240 2005-10-28
US75020005P 2005-12-14 2005-12-14
EP06380097 2006-04-26
US82196406P 2006-08-10 2006-08-10

Publications (1)

Publication Number Publication Date
MA30013B1 true MA30013B1 (en) 2008-12-01

Family

ID=37735293

Family Applications (1)

Application Number Title Priority Date Filing Date
MA30968A MA30013B1 (en) 2005-10-28 2008-05-27 PIRAZOLE-ISOQUINOLEINE UREA DERIVATIVES AS INHIBITORS OF KINASE P38

Country Status (4)

Country Link
EC (1) ECSP088399A (en)
IL (1) IL190062A0 (en)
MA (1) MA30013B1 (en)
NO (1) NO20082419L (en)

Also Published As

Publication number Publication date
NO20082419L (en) 2008-07-07
IL190062A0 (en) 2008-08-07
ECSP088399A (en) 2008-05-30

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