MA28308A1 - NOVEL DERIVATIVES OF PYRROLIDINES AND THIAZOLIDINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME - Google Patents
NOVEL DERIVATIVES OF PYRROLIDINES AND THIAZOLIDINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAMEInfo
- Publication number
- MA28308A1 MA28308A1 MA28252A MA28252A MA28308A1 MA 28308 A1 MA28308 A1 MA 28308A1 MA 28252 A MA28252 A MA 28252A MA 28252 A MA28252 A MA 28252A MA 28308 A1 MA28308 A1 MA 28308A1
- Authority
- MA
- Morocco
- Prior art keywords
- group
- thiazolidines
- pyrrolidines
- preparing
- pharmaceutical compositions
- Prior art date
Links
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NOUVEAUX DERIVES DE PYRROLIDINES ET DE THIAZOLIDINES, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES QUI LES CONTIENNENT Composé de formule (I): dans laquelle : - X1 représente un atome ou groupement choisi parmi CR4aR4b, O, S(O)q1 et NR5, où R4a, R4b, q1 et R5 sont tels que définis dans la description, - m1 représente zéro ou un entier compris entre 1 et 4 inclus, - m2 représente un entier compris entre 1 et 4 inclus, - n1 et n2, identiques ou différents, représentent chacun un entier compris entre 1 et 3 inclus, - R1 représente un atome d'hydrogène ou un groupement choisi parmi carboxy, alkoxycarbonyle, carbamoyle éventuellement substitué et alkyle éventuellement substitué, - R2 représente un atome d'hydrogène ou un groupement alkyle, - Ak représente une chaîne alkylène éventuellement substituée, - p représente zéro, 1 ou 2, - R3 représente un atome d'hydrogène ou un groupement cyano. - X2 et X3, identiques ou différents, représentent chacun, soit un groupement S(O)q2, soit un groupement CR6aR6b, où q2, R6a et R6b sont tels que définis dans la description, ses isomères optiques lorsqu'ils existent, ainsi que ses sels d'addition à un acide pharmaceutiquement acceptable. Médicaments.NOVEL DERIVATIVES OF PYRROLIDINES AND THIAZOLIDINES, PROCESS FOR PREPARING THEM AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM COMPOUND OF formula (I): in which: X1 represents an atom or a group chosen from CR4aR4b, O, S (O) q1 and NR5, where R4a, R4b, q1 and R5 are as defined in the description, - m1 represents zero or an integer between 1 and 4 inclusive, - m2 represents an integer between 1 and 4 inclusive, - n1 and n2, identical or different. , each represents an integer between 1 and 3 inclusive, - R1 represents a hydrogen atom or a group chosen from carboxy, alkoxycarbonyl, optionally substituted carbamoyl and optionally substituted alkyl, - R2 represents a hydrogen atom or an alkyl group, - Ak represents an optionally substituted alkylene chain, - p represents zero, 1 or 2, - R3 represents a hydrogen atom or a cyano group. X2 and X3, identical or different, each represent either a group S (O) q2 or a group CR6aR6b, where q2, R6a and R6b are as defined in the description, its optical isomers where they exist, and its addition salts with a pharmaceutically acceptable acid. Drugs.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MA28252A MA28308A1 (en) | 2005-05-02 | 2005-05-02 | NOVEL DERIVATIVES OF PYRROLIDINES AND THIAZOLIDINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MA28252A MA28308A1 (en) | 2005-05-02 | 2005-05-02 | NOVEL DERIVATIVES OF PYRROLIDINES AND THIAZOLIDINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA28308A1 true MA28308A1 (en) | 2006-12-01 |
Family
ID=43989709
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA28252A MA28308A1 (en) | 2005-05-02 | 2005-05-02 | NOVEL DERIVATIVES OF PYRROLIDINES AND THIAZOLIDINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
Country Status (1)
| Country | Link |
|---|---|
| MA (1) | MA28308A1 (en) |
-
2005
- 2005-05-02 MA MA28252A patent/MA28308A1/en unknown
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