KR960037661A - Silkworm bioactive modulator - Google Patents

Silkworm bioactive modulator Download PDF

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Publication number
KR960037661A
KR960037661A KR1019950010135A KR19950010135A KR960037661A KR 960037661 A KR960037661 A KR 960037661A KR 1019950010135 A KR1019950010135 A KR 1019950010135A KR 19950010135 A KR19950010135 A KR 19950010135A KR 960037661 A KR960037661 A KR 960037661A
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KR
South Korea
Prior art keywords
compound
formula
silkworms
heptadienyl
fluorobenzyl
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Application number
KR1019950010135A
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Korean (ko)
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KR0173436B1 (en
Inventor
강석구
설광열
Original Assignee
김광희
농촌진흥청
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Application filed by 김광희, 농촌진흥청 filed Critical 김광희
Priority to KR1019950010135A priority Critical patent/KR0173436B1/en
Publication of KR960037661A publication Critical patent/KR960037661A/en
Application granted granted Critical
Publication of KR0173436B1 publication Critical patent/KR0173436B1/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

본 발명은 신규한 1-(4-플루오로벤질)-5-〔(E) 또는 (Z)-2,6-디메틸-1,5-헵타디에닐〕이미다졸 화합물, 및 그의 제조방법, 그를 함유하는 누에의 생리활성 조절 조성물 및 누에의 생리활성 조절 방법을 제공한다.The present invention provides a novel 1- (4-fluorobenzyl) -5-[(E) or (Z) -2,6-dimethyl-1,5-heptadienyl] imidazole compound, and a preparation method thereof Provided are a physiological activity regulating composition of silkworms containing and a method of controlling physiological activity of silkworms.

상기 본 발명의 화합물은 종래의 화합물들과는 달리 (E) 형태와 (Z) 형태가 모두 누에의 3면화(眠化)를 유도할 수 있는 생리활성을 갖기 때문에 이들을 서로 분리할 필요가 없어 제조방법이 간단하고, 나아가 종래 화합물에 비해 생리활성이 높다.Unlike the conventional compounds, the compounds of the present invention do not need to be separated from each other because the (E) form and the (Z) form have physiological activities that can induce tricotylation of silkworms. It is simple and furthermore has higher physiological activity as compared with the conventional compound.

Description

누에 생리활성 조정제Silkworm bioactive modulator

본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음As this is a public information case, the full text was not included.

Claims (5)

하기 일반식(1A) 또는 (1B)로 나타내지는 1-(4-플루오로벤질)-5-〔(E) 또는 (Z)-2,6-디메틸-1,5-헵타디에닐〕이미다졸.1- (4-fluorobenzyl) -5-[(E) or (Z) -2,6-dimethyl-1,5-heptadienyl] imidazole represented by the following general formula (1A) or (1B) . 하기 일반식(3)의 화합물과 하기 일반식(4)의 화합물을 반응시켜 하기 일반식(5)의 화합물을 수득하고, 이어 일반식(5)의 화합물을 하기 일반식(2)의 화합물과 반응시켜 하기 일반식 (1A)의 화합물(E-형태)과 하기 일반식(1B)의 화합물(Z-형태)의 혼합물의 형태로서 1-(4-플루오로벤질)-5-〔2,6-디메틸-1,5-헵타디에닐〕이미다졸을 수득함을 특징으로 하는 1-(4-플루오로벤질)-5-〔(E) 또는 (Z)-2,6-디메틸-1,5-헵타디에닐〕이미다졸의 제조방법.The compound of formula (3) is reacted with the compound of formula (4) to obtain a compound of formula (5), and the compound of formula (5) is then reacted with the compound of formula (2) 1- (4-fluorobenzyl) -5- [2,6 in the form of a mixture of the compound of formula (1A) (E-form) and the compound of formula (1B) (Z-form) -Dimethyl-1,5-heptadienyl] imidazole, characterized in that 1- (4-fluorobenzyl) -5-[(E) or (Z) -2,6-dimethyl-1,5 A process for preparing -heptadienyl] imidazole. 제1항의 화합물(1A), (1B)도는 이들의 혼합물을 유효성분으로서 함유함을 특징으로 하는 누에를 3면화(眠化)하기 위한 생리활성 조절제 조성물.The compounds (1A) and (1B) of claim 1, which contain a mixture thereof as an active ingredient, are bioactive modulator compositions for triangulation of silkworms. 제3항에 있어서, 화합물 (1A), (1B) 또는 이들의 혼합물은 10∼20중량%이 양으로 함유됨을 특징으로 하는 조성물.The composition according to claim 3, wherein the compound (1A), (1B) or a mixture thereof is contained in an amount of 10 to 20% by weight. 제3항의 조성물을 3령 또는 4령의 누에에 경구 투여함을 특징으로 하는 누에를 조기변태시켜 3면화를 유도하는 방법.A method of inducing tricot by premature transformation of silkworms, characterized by orally administering the composition of claim 3 to silkworms of 3 or 4 years of age. ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.※ Note: The disclosure is based on the initial application.
KR1019950010135A 1995-04-27 1995-04-27 Silkworm bioactivity regulator KR0173436B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019950010135A KR0173436B1 (en) 1995-04-27 1995-04-27 Silkworm bioactivity regulator

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1019950010135A KR0173436B1 (en) 1995-04-27 1995-04-27 Silkworm bioactivity regulator

Publications (2)

Publication Number Publication Date
KR960037661A true KR960037661A (en) 1996-11-19
KR0173436B1 KR0173436B1 (en) 1999-02-01

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ID=19413117

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019950010135A KR0173436B1 (en) 1995-04-27 1995-04-27 Silkworm bioactivity regulator

Country Status (1)

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KR (1) KR0173436B1 (en)

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Publication number Publication date
KR0173436B1 (en) 1999-02-01

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