KR960000860A - Phenyl Benzoyl Urea Derivative - Google Patents

Phenyl Benzoyl Urea Derivative Download PDF

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Publication number
KR960000860A
KR960000860A KR1019940012553A KR19940012553A KR960000860A KR 960000860 A KR960000860 A KR 960000860A KR 1019940012553 A KR1019940012553 A KR 1019940012553A KR 19940012553 A KR19940012553 A KR 19940012553A KR 960000860 A KR960000860 A KR 960000860A
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KR
South Korea
Prior art keywords
benzoyl
formula
urea
compound
bromo
Prior art date
Application number
KR1019940012553A
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Korean (ko)
Inventor
이정구
우제완
김승희
신용우
황공현
Original Assignee
이진우
주식회사 한 화
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Publication date
Application filed by 이진우, 주식회사 한 화 filed Critical 이진우
Priority to KR1019940012553A priority Critical patent/KR960000860A/en
Priority to PCT/KR1995/000072 priority patent/WO1995033711A1/en
Publication of KR960000860A publication Critical patent/KR960000860A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/34—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the groups, e.g. biuret; Thio analogues thereof; Urea-aldehyde condensation products
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C273/00—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C273/02—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of urea, its salts, complexes or addition compounds
    • C07C273/06—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of urea, its salts, complexes or addition compounds from cyanamide or calcium cyanamide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/46—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylureas
    • C07C275/48—Y being a hydrogen or a carbon atom
    • C07C275/54—Y being a carbon atom of a six-membered aromatic ring, e.g. benzoylureas

Abstract

본 발명은 강력한 살충작용을 갖는 다음 일반식(I)로 표시되는 신규한 N-페닐-N'-벤조일 우레아 유도체에 관한 것이다.The present invention relates to novel N-phenyl-N'-benzoyl urea derivatives represented by the following general formula (I) with potent insecticidal action.

상기 식(I)에서 X는 탄소 또는 질소이고, R1,R2,R3,R5는 플로오르, 염소, 브롬 중에서 선택되는 1개 이상의 할로겐 원자, 또는 수소원자이며, R4는 X가 탄소인 경우에는 플로오르, 염소, 브롬, 또는 수소원자 중의 하나를 나타낸다.In formula (I), X is carbon or nitrogen, R 1 , R 2 , R 3 , R 5 is at least one halogen atom selected from fluorine, chlorine, bromine, or a hydrogen atom, and R 4 is X In the case of carbon, it represents one of fluorine, chlorine, bromine or hydrogen atoms.

Description

페닐 벤조일 우레아 유도체Phenyl Benzoyl Urea Derivative

본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음As this is a public information case, the full text was not included.

Claims (10)

다음 일반식(I)로 표시되는 생리활성을 갖는 벤조일 우레아 유도체.Benzoyl urea derivatives having a physiological activity represented by the following general formula (I). 상기 식(I)에서 X는 탄소 또는 질소이고, R1,R2,R3,R5는 플로오르, 염소, 브롬 중에서 선택되는 1개 이상의 할로겐 원자, 또는 수소원자이며, R4는 X가 탄소인 경우에는 플로오르, 염소, 브롬, 또는 수소원자 중의 하나를 나타낸다.In formula (I), X is carbon or nitrogen, R 1 , R 2 , R 3 , R 5 is at least one halogen atom selected from fluorine, chlorine, bromine, or a hydrogen atom, and R 4 is X In the case of carbon, it represents one of fluorine, chlorine, bromine or hydrogen atoms. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2,6-디플루오르 벤조일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.The compound of claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2,6-difluoro benzoyl) urea Benzoyl urea derivative characterized by the above-mentioned. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2-플루오르 벤조일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.A compound according to claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2-fluoro benzoyl) urea. Benzoyl urea derivatives. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2-클로로 벤조일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.A compound according to claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2-chloro benzoyl) urea Benzoyl urea derivatives. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2-브로모벤조일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.A compound according to claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2-bromobenzoyl) urea Benzoyl urea derivatives. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2,6-디클로로 벤조일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.A compound according to claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2,6-dichloro benzoyl) urea Benzoyl urea derivatives. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2,4-디클로로 벤조일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.A compound according to claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2,4-dichloro benzoyl) urea Benzoyl urea derivatives. 제1항에 있어서, 상기 식(I)의 화합물이 1-[2-브로모-3,5-(비스트리플루오로메틸)페닐]-3-(2-클로로니코티노일)우레아인 것을 특징으로 하는 벤조일 우레아 유도체.A compound according to claim 1, wherein the compound of formula (I) is 1- [2-bromo-3,5- (bistrifluoromethyl) phenyl] -3- (2-chloronicotinoyl) urea Benzoyl urea derivatives. 다음 일반식(Ⅱ)로 표시되는 2-브로모-3,5-비스트리플루오로아닐린을 다음 일반식(Ⅲ)으로 표시되는 벤조일 이소시아네이트와 반응시켜서 다음의 구조식(I)로 표시되는 벤조일 우레아 유도체를 제조하는 방법.Benzoyl urea derivative represented by the following structural formula (I) by reacting 2-bromo-3,5-bistrifluoroaniline represented by the following general formula (II) with benzoyl isocyanate represented by the following general formula (III) How to prepare. 상기 식에서 X는 탄소 또는 질소이고, R1,R2,R3,R5는 플로오르, 염소, 브롬 중에서 선택되는 1개 이상의 할로겐 원자, 또는 수소원자이며, R4는 X가 탄소인 경우에는 플로오르, 염소, 브롬, 또는 수소원자 중의 하나를 나타낸다.Wherein X is carbon or nitrogen, R 1 , R 2 , R 3 , R 5 is at least one halogen atom selected from fluorine, chlorine, bromine, or a hydrogen atom, and R 4 is when X is carbon Fluorine, chlorine, bromine or hydrogen atoms. 다음 일반식(I)로 표시되는 벤조일 우레아 유도체가 유효성분으로 함유되어 있는 것을 특징으로 하는 농약 조성물.A pesticide composition, characterized in that the benzoyl urea derivative represented by the following general formula (I) is contained as an active ingredient. 상기 식(I)에서 X는 탄소 또는 질소이고, R1,R2,R3,R5는 플로오르, 염소, 브롬 중에서 선택되는 1개 이상의 할로겐 원자, 또는 수소원자이며, R4는 X가 탄소인 경우에는 플로오르, 염소, 브롬, 또는 수소원자 중의 하나를 나타낸다.In formula (I), X is carbon or nitrogen, R 1 , R 2 , R 3 , R 5 is at least one halogen atom selected from fluorine, chlorine, bromine, or a hydrogen atom, and R 4 is X In the case of carbon, it represents one of fluorine, chlorine, bromine or hydrogen atoms. ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.※ Note: The disclosure is based on the initial application.
KR1019940012553A 1994-06-03 1994-06-03 Phenyl Benzoyl Urea Derivative KR960000860A (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
KR1019940012553A KR960000860A (en) 1994-06-03 1994-06-03 Phenyl Benzoyl Urea Derivative
PCT/KR1995/000072 WO1995033711A1 (en) 1994-06-03 1995-06-02 Phenyl benzoyl(nicotinoyl) urea derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1019940012553A KR960000860A (en) 1994-06-03 1994-06-03 Phenyl Benzoyl Urea Derivative

Publications (1)

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KR960000860A true KR960000860A (en) 1996-01-25

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WO (1) WO1995033711A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100194535B1 (en) * 1995-12-27 1999-06-15 우종일 Aryl benzoyl urea derivative and pesticide composition containing the same
KR100194534B1 (en) * 1996-06-29 1999-06-15 우종일 2-Chloro-3,5-bis (tpyfluoromethyl) phenyl benzoyl urea derivative and preparation method thereof
CN102960356A (en) * 2012-12-12 2013-03-13 海利尔药业集团股份有限公司 Parasiticide composite containing bistrifluron and methoxyfenozide
CN102986700A (en) * 2012-12-18 2013-03-27 海利尔药业集团股份有限公司 Insecticide composition containing flutenzine and bistrifluron

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4148902A (en) * 1977-05-13 1979-04-10 The Dow Chemical Company N-[(optionally substituted phenylamino)carbonyl] pyridine carboxamides and insecticidal use thereof
HU184062B (en) * 1979-10-19 1984-06-28 Chinoin Gyogyszer Es Vegyeszet Process for producing substituted acyl urea
DE3217619A1 (en) * 1982-05-11 1983-11-17 Bayer Ag, 5090 Leverkusen 2,4-DIHALOGENBENZOYL (THIO) UREA, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A PEST CONTROL
DE3217620A1 (en) * 1982-05-11 1983-11-17 Bayer Ag, 5090 Leverkusen 2,5-DIHALOGENBENZOYL (THIO) UREA, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A PEST CONTROL
JPS6176452A (en) * 1984-09-20 1986-04-18 Nippon Soda Co Ltd Benzoylurea derivative, its preparation and insecticide
DE3607298A1 (en) * 1985-03-14 1986-09-18 Shell Internationale Research Maatschappij B.V., Den Haag/S'gravenhage Process for the preparation of benzoylureas
DD253614A1 (en) * 1986-11-13 1988-01-27 Paedagogische Hochschule N K K A NEW METHOD FOR THE PRODUCTION OF SUBSTITUTED N-PHENYL-N'-BENZOYL HARVES

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WO1995033711A1 (en) 1995-12-14

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