KR930004282A - 1,2,4-oxadiazole-5-one derivatives and preparation methods thereof - Google Patents

1,2,4-oxadiazole-5-one derivatives and preparation methods thereof Download PDF

Info

Publication number
KR930004282A
KR930004282A KR1019910014924A KR910014924A KR930004282A KR 930004282 A KR930004282 A KR 930004282A KR 1019910014924 A KR1019910014924 A KR 1019910014924A KR 910014924 A KR910014924 A KR 910014924A KR 930004282 A KR930004282 A KR 930004282A
Authority
KR
South Korea
Prior art keywords
group
methyl
halogen atom
aminocarbonylmethyl
bromo
Prior art date
Application number
KR1019910014924A
Other languages
Korean (ko)
Other versions
KR0183540B1 (en
Inventor
조광연
정인화
정영륜
김영섭
민용기
오영주
전근숙
김홍태
김병섭
Original Assignee
채영복
재단법인 한국화학연구소
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 채영복, 재단법인 한국화학연구소 filed Critical 채영복
Priority to KR1019910014924A priority Critical patent/KR0183540B1/en
Publication of KR930004282A publication Critical patent/KR930004282A/en
Application granted granted Critical
Publication of KR0183540B1 publication Critical patent/KR0183540B1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/18Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
    • A01N37/22Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof the nitrogen atom being directly attached to an aromatic ring system, e.g. anilides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/071,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

내용 없음.No content.

Description

1,2,4-옥사디아졸-5-온 유도체와 그의 제조방법1,2,4-oxadiazole-5-one derivatives and preparation methods thereof

본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음Since this is an open matter, no full text was included.

Claims (12)

하기 일반식(Ⅰ)로 표시되는 1,2,4-옥사디아졸-5-온 유호체.1,2,4-oxadiazole-5-one emulsion represented by the following general formula (I). 상기 식에서, X는 수소원자, 할로겐원자, C1-3알킬기 또는 C1-2알콕시기이고, Y는 수소원자, 할로겐원자, C1-4알킬기, C1-3알콕시기 또는 메틸티오기이며, Z는 수소원자, 할로겐원자, 메틸기 또는 메톡시기이고, R1는 수소원자, 할로겐원자, 메틸기, 트리플루오로메틸기 또는 메톡시기이며, R2는 수소원자 또는 할로겐원자이다.Wherein X is a hydrogen atom, a halogen atom, a C 1-3 alkyl group or a C 1-2 alkoxy group, Y is a hydrogen atom, a halogen atom, a C 1-4 alkyl group, a C 1-3 alkoxy group or a methylthio group , Z is a hydrogen atom, a halogen atom, a methyl group or a methoxy group, R 1 is a hydrogen atom, a halogen atom, a methyl group, a trifluoromethyl group or a methoxy group, R 2 is a hydrogen atom or a halogen atom. 제1항에 있어서, 상기 일반식(Ⅰ)에서 X가 할로겐원자, 메틸기 또는 메톡시기이고, Y가 할로겐원자, C1-2알킬기, 또는 C1-2알콕시기이며, Z가 할로겐원자 또는 메틸기이고, R1이 할로겐원자, 메틸기 또는 메톡시기이며, R2가 수수원자인 화합물.The compound of claim 1, wherein in the general formula (I), X is a halogen atom, a methyl group or a methoxy group, Y is a halogen atom, a C 1-2 alkyl group, or a C 1-2 alkoxy group, and Z is a halogen atom or a methyl group And R 1 is a halogen atom, a methyl group or a methoxy group, and R 2 is a canine atom. 제2항에 있어서, 상기 일반식(Ⅰ)에서 X가 클로로, 브로모 또는 메틸기이고, Y가 클로로, 브로모, 메틸기 또는 메톡시기이며, Z가 클로로, 브로모 또는 메틸기이고, R1이 클로로, 브로모, 메틸기 또는 메톡시기이며, R2가 수소원자인 화합물.A compound according to claim 2, wherein in formula (I), X is a chloro, bromo or methyl group, Y is a chloro, bromo, methyl or methoxy group, Z is a chloro, bromo or methyl group, and R 1 is chloro , A bromo, a methyl group or a methoxy group, wherein R 2 is a hydrogen atom. 3-(2′4′-디클로로페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2'4'-dichlorophenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(4′-브로모-2′,6′-디메틸페녹시)메틸-4-(3′-브로모페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (4′-bromo-2 ′, 6′-dimethylphenoxy) methyl-4- (3′-bromophenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(4′,-브로모-2′,6′-디메틸페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (4 ',-bromo-2', 6'-dimethylphenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(4′-브로모-2′-클로-6′-메틸페녹시)메틸-4-(3′-메톡시페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (4′-bromo-2′-chloro-6′-methylphenoxy) methyl-4- (3′-methoxyphenyl) aminocarbonylmethyl-1,2,4-oxadiazole-5- On. 3-(2′,4′,6′-트리메틸페녹시)메틸-4-(3′-클로로페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2 ', 4', 6'-trimethylphenoxy) methyl-4- (3'-chlorophenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(2′,4′,6′-트리메틸페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2 ', 4', 6'-trimethylphenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(2′,4′,6′-트리클로로페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2 ', 4', 6'-trichlorophenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 하기 일반식(Ⅱ)의 5-히드록시-1,2,4-옥사디아졸 유도체와 일반식(Ⅲ)의 클로아세트아미드 유도체를 반응시켜서 일반식(Ⅰ)의 1,2,4-옥사디아졸-5-온 유도체를 제조하는 방법.1,2,4-oxadia of general formula (I) by reacting the 5-hydroxy-1,2,4-oxadiazole derivatives of the general formula (II) with the cloacetamide derivatives of the general formula (III) Process for preparing sol-5-one derivative. 상기 식들에서 X, Y, Z, R1및 R2는 상기 제1항에서 정의한 바와같다.X, Y, Z, R 1 and R 2 in the above formulas are as defined in claim 1 above. 제1항에 따른 일반식(Ⅰ)의 1,2,4-옥사디아졸-5-온 유도체를 유효 성분으로 함유하는 살균제 조성물.A fungicide composition comprising the 1,2,4-oxadiazole-5-one derivative of formula (I) according to claim 1 as an active ingredient. ※ 참고사항 : 최초출원 내용에 의하여 공개되는 것임.※ Note: This is to be disclosed by the original application.
KR1019910014924A 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof KR0183540B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019910014924A KR0183540B1 (en) 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1019910014924A KR0183540B1 (en) 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof

Publications (2)

Publication Number Publication Date
KR930004282A true KR930004282A (en) 1993-03-22
KR0183540B1 KR0183540B1 (en) 1999-05-01

Family

ID=19319234

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019910014924A KR0183540B1 (en) 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof

Country Status (1)

Country Link
KR (1) KR0183540B1 (en)

Also Published As

Publication number Publication date
KR0183540B1 (en) 1999-05-01

Similar Documents

Publication Publication Date Title
KR840009092A (en) Method for preparing benzofuran- or benzopyran-carboxamide derivatives
KR910002800A (en) 4-acyloxyquinoline derivatives and pesticidal or acaricide compositions containing them
KR880000413A (en) Anti-allergic and anti-inflammatory preparations and preparation methods thereof
KR840004345A (en) A pyrazole derivative, a method for producing the same, and a selective herbicidal composition containing the same as an active ingredient, and a method for removing and inhibiting weeds using the same.
KR910015558A (en) Improved leukotriine antagonist
PH24355A (en) Macrolide compounds,composition said compound and method of use thereof
KR900016178A (en) 2-substituted N, N&#39;-ditrimethoxybenzoyl piperazine, preparation method thereof and therapeutic composition containing the same
KR930004282A (en) 1,2,4-oxadiazole-5-one derivatives and preparation methods thereof
KR880003932A (en) Heterocyclic Compounds, Preparations and Uses thereof
KR840004757A (en) Method for preparing cephalosporin derivative
KR900006316A (en) Benzo heterocyclic compound and preparation method thereof
KR860008983A (en) Method for preparing 4-benzoyl-1-alkyl (alkenyl) pyrazole
KR880002820A (en) Ether Derivatives and Acaricides or Pesticide Compositions Composed of These Derivatives
KR890012949A (en) O-acylamide oxime derivative
KR890002079A (en) 1- [2- (phenylmethyl) phenyl] piperazine and preparation method thereof
KR850000415A (en) Method for preparing quinazolinone derivatives
KR870004038A (en) Method for preparing herbicide compound
KR890005076A (en) Thiadiazine derivatives, preparation method thereof, and insecticide containing the compound
KR900001668A (en) Novel thiadiazines, preparations thereof, and pesticidal bases containing the compounds
SE8605458L (en) 4-HYDROXIKUMARING DERIVATIVES
KR910004573A (en) Imidazole derivatives, preparation method thereof and anti-ulcer agent containing the same
KR920006312A (en) 3,4-trans-4-ethyl-1- (substituted phenyl) -3- (substituted phenyl) pyrrolidin-2-one, preparation method thereof and herbicidal composition containing it as herbicidal active ingredient
KR830006285A (en) Method for preparing benzoquinolizine
KR840001151A (en) Method for preparing N-substituted-tetrahydrophthalimide derivative
KR920016428A (en) Novel pyrazole derivatives, preparation method thereof and herbicide composition containing the same

Legal Events

Date Code Title Description
A201 Request for examination
E701 Decision to grant or registration of patent right
GRNT Written decision to grant
FPAY Annual fee payment

Payment date: 20020927

Year of fee payment: 5

LAPS Lapse due to unpaid annual fee