KR930004282A - 1,2,4-oxadiazole-5-one derivatives and preparation methods thereof - Google Patents

1,2,4-oxadiazole-5-one derivatives and preparation methods thereof Download PDF

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KR930004282A
KR930004282A KR1019910014924A KR910014924A KR930004282A KR 930004282 A KR930004282 A KR 930004282A KR 1019910014924 A KR1019910014924 A KR 1019910014924A KR 910014924 A KR910014924 A KR 910014924A KR 930004282 A KR930004282 A KR 930004282A
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South Korea
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group
methyl
halogen atom
aminocarbonylmethyl
bromo
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KR1019910014924A
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Korean (ko)
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KR0183540B1 (en
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조광연
정인화
정영륜
김영섭
민용기
오영주
전근숙
김홍태
김병섭
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채영복
재단법인 한국화학연구소
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
    • A01N37/22—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof the nitrogen atom being directly attached to an aromatic ring system, e.g. anilides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

내용 없음.No content.

Description

1,2,4-옥사디아졸-5-온 유도체와 그의 제조방법1,2,4-oxadiazole-5-one derivatives and preparation methods thereof

본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음Since this is an open matter, no full text was included.

Claims (12)

하기 일반식(Ⅰ)로 표시되는 1,2,4-옥사디아졸-5-온 유호체.1,2,4-oxadiazole-5-one emulsion represented by the following general formula (I). 상기 식에서, X는 수소원자, 할로겐원자, C1-3알킬기 또는 C1-2알콕시기이고, Y는 수소원자, 할로겐원자, C1-4알킬기, C1-3알콕시기 또는 메틸티오기이며, Z는 수소원자, 할로겐원자, 메틸기 또는 메톡시기이고, R1는 수소원자, 할로겐원자, 메틸기, 트리플루오로메틸기 또는 메톡시기이며, R2는 수소원자 또는 할로겐원자이다.Wherein X is a hydrogen atom, a halogen atom, a C 1-3 alkyl group or a C 1-2 alkoxy group, Y is a hydrogen atom, a halogen atom, a C 1-4 alkyl group, a C 1-3 alkoxy group or a methylthio group , Z is a hydrogen atom, a halogen atom, a methyl group or a methoxy group, R 1 is a hydrogen atom, a halogen atom, a methyl group, a trifluoromethyl group or a methoxy group, R 2 is a hydrogen atom or a halogen atom. 제1항에 있어서, 상기 일반식(Ⅰ)에서 X가 할로겐원자, 메틸기 또는 메톡시기이고, Y가 할로겐원자, C1-2알킬기, 또는 C1-2알콕시기이며, Z가 할로겐원자 또는 메틸기이고, R1이 할로겐원자, 메틸기 또는 메톡시기이며, R2가 수수원자인 화합물.The compound of claim 1, wherein in the general formula (I), X is a halogen atom, a methyl group or a methoxy group, Y is a halogen atom, a C 1-2 alkyl group, or a C 1-2 alkoxy group, and Z is a halogen atom or a methyl group And R 1 is a halogen atom, a methyl group or a methoxy group, and R 2 is a canine atom. 제2항에 있어서, 상기 일반식(Ⅰ)에서 X가 클로로, 브로모 또는 메틸기이고, Y가 클로로, 브로모, 메틸기 또는 메톡시기이며, Z가 클로로, 브로모 또는 메틸기이고, R1이 클로로, 브로모, 메틸기 또는 메톡시기이며, R2가 수소원자인 화합물.A compound according to claim 2, wherein in formula (I), X is a chloro, bromo or methyl group, Y is a chloro, bromo, methyl or methoxy group, Z is a chloro, bromo or methyl group, and R 1 is chloro , A bromo, a methyl group or a methoxy group, wherein R 2 is a hydrogen atom. 3-(2′4′-디클로로페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2'4'-dichlorophenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(4′-브로모-2′,6′-디메틸페녹시)메틸-4-(3′-브로모페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (4′-bromo-2 ′, 6′-dimethylphenoxy) methyl-4- (3′-bromophenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(4′,-브로모-2′,6′-디메틸페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (4 ',-bromo-2', 6'-dimethylphenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(4′-브로모-2′-클로-6′-메틸페녹시)메틸-4-(3′-메톡시페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (4′-bromo-2′-chloro-6′-methylphenoxy) methyl-4- (3′-methoxyphenyl) aminocarbonylmethyl-1,2,4-oxadiazole-5- On. 3-(2′,4′,6′-트리메틸페녹시)메틸-4-(3′-클로로페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2 ', 4', 6'-trimethylphenoxy) methyl-4- (3'-chlorophenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(2′,4′,6′-트리메틸페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2 ', 4', 6'-trimethylphenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 3-(2′,4′,6′-트리클로로페녹시)메틸-4-(3′-메틸페닐)아미노카보닐메틸-1,2,4-옥사디아졸-5-온.3- (2 ', 4', 6'-trichlorophenoxy) methyl-4- (3'-methylphenyl) aminocarbonylmethyl-1,2,4-oxadiazol-5-one. 하기 일반식(Ⅱ)의 5-히드록시-1,2,4-옥사디아졸 유도체와 일반식(Ⅲ)의 클로아세트아미드 유도체를 반응시켜서 일반식(Ⅰ)의 1,2,4-옥사디아졸-5-온 유도체를 제조하는 방법.1,2,4-oxadia of general formula (I) by reacting the 5-hydroxy-1,2,4-oxadiazole derivatives of the general formula (II) with the cloacetamide derivatives of the general formula (III) Process for preparing sol-5-one derivative. 상기 식들에서 X, Y, Z, R1및 R2는 상기 제1항에서 정의한 바와같다.X, Y, Z, R 1 and R 2 in the above formulas are as defined in claim 1 above. 제1항에 따른 일반식(Ⅰ)의 1,2,4-옥사디아졸-5-온 유도체를 유효 성분으로 함유하는 살균제 조성물.A fungicide composition comprising the 1,2,4-oxadiazole-5-one derivative of formula (I) according to claim 1 as an active ingredient. ※ 참고사항 : 최초출원 내용에 의하여 공개되는 것임.※ Note: This is to be disclosed by the original application.
KR1019910014924A 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof KR0183540B1 (en)

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KR1019910014924A KR0183540B1 (en) 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof

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KR1019910014924A KR0183540B1 (en) 1991-08-28 1991-08-28 1,2,4-oxadiazole-5-one derivatives and preparation method thereof

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KR930004282A true KR930004282A (en) 1993-03-22
KR0183540B1 KR0183540B1 (en) 1999-05-01

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