KR900008168B1 - Novel radio pharmaceuticals and chelating agents useful in their preparation - Google Patents
Novel radio pharmaceuticals and chelating agents useful in their preparationInfo
- Publication number
- KR900008168B1 KR900008168B1 KR8505136A KR850005136A KR900008168B1 KR 900008168 B1 KR900008168 B1 KR 900008168B1 KR 8505136 A KR8505136 A KR 8505136A KR 850005136 A KR850005136 A KR 850005136A KR 900008168 B1 KR900008168 B1 KR 900008168B1
- Authority
- KR
- South Korea
- Prior art keywords
- preparation
- chelating agents
- agents useful
- novel radio
- radio pharmaceuticals
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/53—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F13/00—Compounds containing elements of Groups 7 or 17 of the Periodic System
- C07F13/005—Compounds without a metal-carbon linkage
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
Abstract
Pyridinium, quinolinium and isoquinolinium salts of formula (I) are prepared. In (I), A= residue of a chelating agent capable of chelating with ametallic radiomucleotide and having at least one p-, s- or t-amino functional gp., this gp. not being essential for the complexing properties; the residue is characterized by the absence of at least one of the p-, s-, t-amino functional gp.; y= 1 or 2; B= gp. of formula (II), (III) or (IV), each attached through the N atom; n, p, q= 0, 1 or 2; R= halogen, C1-7 alkyl, C1-7 alkoxy, C2-8 alkoxycarbonyl, etc.; X= anion of inorgainc acid; t= valence of the anion; S= integer; and S times t=y.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63238384A | 1984-07-19 | 1984-07-19 | |
US632383 | 1984-07-19 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR870000935A KR870000935A (en) | 1987-03-10 |
KR900008168B1 true KR900008168B1 (en) | 1990-11-05 |
Family
ID=24535323
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR8505136A KR900008168B1 (en) | 1984-07-19 | 1985-07-18 | Novel radio pharmaceuticals and chelating agents useful in their preparation |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP0191788A1 (en) |
JP (1) | JPS61112054A (en) |
KR (1) | KR900008168B1 (en) |
AU (1) | AU4632085A (en) |
CA (1) | CA1266864A (en) |
DK (1) | DK124686A (en) |
ES (2) | ES8700236A1 (en) |
FI (1) | FI861119A0 (en) |
GR (1) | GR851793B (en) |
IL (1) | IL75845A0 (en) |
NO (1) | NO860980L (en) |
PT (1) | PT80842B (en) |
WO (1) | WO1986000897A1 (en) |
ZA (1) | ZA855477B (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5071636A (en) * | 1987-12-29 | 1991-12-10 | Nihon Medi-Physics Co., Ltd. | Chelating compounds and their use |
SE526214C2 (en) * | 2003-02-28 | 2005-07-26 | Amersham Biosciences Ab | One way to generate metal chelating affinity ligands |
KR101033209B1 (en) * | 2004-12-31 | 2011-05-06 | 주식회사 효성 | A process for preparing polyester multifilamant for yarn diving having injection |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4444690A (en) * | 1982-02-25 | 1984-04-24 | University Patents, Inc. | Technetium chelates |
EP0222425A3 (en) * | 1982-05-18 | 1988-09-21 | University Of Florida | Brain-specific drug delivery |
-
1985
- 1985-07-15 AU AU46320/85A patent/AU4632085A/en not_active Abandoned
- 1985-07-15 EP EP85903750A patent/EP0191788A1/en not_active Withdrawn
- 1985-07-15 WO PCT/US1985/001333 patent/WO1986000897A1/en not_active Application Discontinuation
- 1985-07-18 KR KR8505136A patent/KR900008168B1/en active IP Right Grant
- 1985-07-18 GR GR851793A patent/GR851793B/el unknown
- 1985-07-18 IL IL75845A patent/IL75845A0/en unknown
- 1985-07-19 ZA ZA855477A patent/ZA855477B/en unknown
- 1985-07-19 CA CA000487166A patent/CA1266864A/en not_active Expired - Fee Related
- 1985-07-19 PT PT80842A patent/PT80842B/en unknown
- 1985-07-19 JP JP60160039A patent/JPS61112054A/en active Pending
- 1985-07-19 ES ES545395A patent/ES8700236A1/en not_active Expired
-
1986
- 1986-02-17 ES ES552090A patent/ES8705389A1/en not_active Expired
- 1986-03-14 NO NO860980A patent/NO860980L/en unknown
- 1986-03-18 FI FI861119A patent/FI861119A0/en not_active Application Discontinuation
- 1986-03-18 DK DK124686A patent/DK124686A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL75845A0 (en) | 1985-11-29 |
ES8700236A1 (en) | 1986-10-01 |
PT80842B (en) | 1987-05-27 |
ES8705389A1 (en) | 1987-05-01 |
ES545395A0 (en) | 1986-10-01 |
PT80842A (en) | 1985-08-01 |
NO860980L (en) | 1986-05-06 |
FI861119A (en) | 1986-03-18 |
KR870000935A (en) | 1987-03-10 |
ZA855477B (en) | 1987-03-25 |
EP0191788A1 (en) | 1986-08-27 |
AU4632085A (en) | 1986-02-25 |
GR851793B (en) | 1985-11-26 |
JPS61112054A (en) | 1986-05-30 |
ES552090A0 (en) | 1987-05-01 |
WO1986000897A1 (en) | 1986-02-13 |
DK124686D0 (en) | 1986-03-18 |
CA1266864A (en) | 1990-03-20 |
DK124686A (en) | 1986-05-20 |
FI861119A0 (en) | 1986-03-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
A201 | Request for examination | ||
E902 | Notification of reason for refusal | ||
G160 | Decision to publish patent application | ||
E701 | Decision to grant or registration of patent right | ||
NORF | Unpaid initial registration fee |